GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.018 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(194 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5983 produits trouvés pour "GPCR/G-Protéine"
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Urotensin I acetate (83930-33-0 Free base)
Urotensin I acetate, CRF1/CRF2 agonist: pEC50s - hCRF1 11.46, hCRF2 9.36, rCRF2α 9.85; KIs - hCRF1 0.4 nM, rCRF2α 1.8 nM, mCRF2β 5.7 nM.Degré de pureté :95.44% - 99.73%Couleur et forme :SolidMasse moléculaire :N/ABevantolol hydrochloride
CAS :Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.Formule :C20H28ClNO4Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :381.9Alprenolol benzoate
CAS :Alprenolol benzoate is the benzoate salt of Alprenolol -- a beta blocker.Formule :C22H29NO4Couleur et forme :SolidMasse moléculaire :371.48SB-334867 free base
CAS :SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.Formule :C17H13N5O2Degré de pureté :99.67% - >99.99%Couleur et forme :SolidMasse moléculaire :319.32Ref: TM-T6140
2mg39,00€5mg66,00€10mg94,00€25mg152,00€50mg215,00€100mg319,00€200mg475,00€1mL*10mM (DMSO)73,00€Pancreatic Polypeptide (human) acetate
Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist.Degré de pureté :97.26%Couleur et forme :LiquidMasse moléculaire :N/ATC-G 1005
CAS :TC-G 1005 is a potent and selective GPBA agonist (EC50 :0.72 nM; hTGR5).Formule :C25H25N3O2Degré de pureté :98.60% - 99.78%Couleur et forme :SolidMasse moléculaire :399.48Ref: TM-T8818
1mg34,00€2mg43,00€5mg65,00€10mg90,00€25mg178,00€50mg269,00€100mg400,00€1mL*10mM (DMSO)72,00€Clozapine N-Oxide
CAS :View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.Formule :C18H19ClN4ODegré de pureté :98.65% - 99.94%Couleur et forme :SolidMasse moléculaire :342.82Guanethidine monosulfate
CAS :Guanethidine monosulfate is an antihypertensive drug that reduces the release of catecholamines.Formule :C10H24N4O4SDegré de pureté :99.61% - 99.74%Couleur et forme :SolidMasse moléculaire :296.39SCH-23390 hydrochloride
CAS :SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Formule :C17H19Cl2NODegré de pureté :98% - 99.83%Couleur et forme :SolidMasse moléculaire :324.24Ref: TM-T4369
1mg39,00€2mg50,00€5mg78,00€10mg97,00€25mg195,00€50mg369,00€100mg550,00€1mL*10mM (DMSO)78,00€SAX-187 hydrochloride
CAS :WAY-181187 is a potent, selective 5-HT6 agonist with high affinity (2.2-4.8 nM), and increases GABA in rat cortex at 3-30 mg/kg s.c.Formule :C15H14Cl2N4O2S2Couleur et forme :SolidMasse moléculaire :417.33Felypressin
CAS :Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.Formule :C46H65N13O11S2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :1040.22Ibutamoren Mesylate
CAS :Ibutamoren Mesylate (MK-0677) is a potent, non-peptide Growth hormone secretagogue receptor (GHSR) agonist.Formule :C28H40N4O8S2Degré de pureté :97.98% - ≥98%Couleur et forme :SolidMasse moléculaire :624.77FK962
CAS :FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.Formule :C14H17FN2O2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :264.3Ref: TM-T7829
2mg34,00€5mg52,00€10mg82,00€25mg144,00€50mg200,00€100mg278,00€200mg389,00€1mL*10mM (DMSO)57,00€Otenabant hydrochloride
CAS :Otenabant hydrochloride (Otenabant) (CP-945598) is a competitive, high affinity, selective antagonist of the CB1 receptor (Ki: 0.7 nM).Formule :C25H26Cl3N7ODegré de pureté :99.79% - ≥95%Couleur et forme :SolidMasse moléculaire :546.88Talnetant
CAS :Talnetant (SB 223412) is a selective NK3 receptor antagonist that can penetrate the brain and modulate dopamine.Formule :C25H22N2O2Degré de pureté :97.88%Couleur et forme :SolidMasse moléculaire :382.45Ref: TM-T7549
1mg40,00€2mg52,00€5mg87,00€10mg123,00€25mg251,00€50mg464,00€100mg705,00€1mL*10mM (DMSO)135,00€SB-200646
CAS :SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptorFormule :C15H14N4ODegré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :266.3Arformoterol Tartrate
CAS :Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.Formule :C23H30N2O10Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :494.49Ref: TM-T22245
5mg60,00€10mg87,00€25mg150,00€50mg221,00€100mg329,00€200mg487,00€1mL*10mM (DMSO)85,00€Seltorexant hydrochloride
CAS :Seltorexant hydrochloride is a selective, orally active and high-affinity antagonist of OX2R with pKi values of 8.0 and 8.1 for human and rat OX2R.Formule :C21H23ClFN7ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :443.91Decloxizine dihydrochloride
CAS :Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.Formule :C21H28N2O2·2ClHDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :413.39Talinolol
CAS :(±)-Talinolol is a selective β1 adrenoceptor antagonist well known for its cardioprotective and antihypertensive activity.Formule :C20H33N3O3Degré de pureté :98.8%Couleur et forme :SolidMasse moléculaire :363.49Ref: TM-T21640
2mg34,00€5mg52,00€10mg92,00€25mg178,00€50mg313,00€100mg535,00€200mg775,00€1mL*10mM (DMSO)52,00€Dimaprit dihydrochloride
CAS :Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.Formule :C6H15N3S·2HClDegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :234.19LML134
CAS :LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).Formule :C19H29N5O3Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :375.47Ref: TM-T8514
1mg34,00€5mg78,00€10mg112,00€25mg203,00€50mg299,00€100mg447,00€200mg600,00€1mL*10mM (DMSO)86,00€Neuropeptide Y (29-64), amide, human acetate
Neuropeptide Y (29-64), amide, human acetate is involved in Alzheimer's disease (AD) and protects rat cortical neurons against β-Amyloid toxicity.Degré de pureté :98.42%Couleur et forme :LiquidMasse moléculaire :N/ASB399885
CAS :SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.Formule :C18H21Cl2N3O4SDegré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :446.35Ref: TM-T19669
1mg67,00€5mg123,00€10mg177,00€25mg291,00€50mg393,00€100mg553,00€200mg743,00€1mL*10mM (DMSO)150,00€Pancreatic Polypeptide, rat acetate
Pancreatic Polypeptide, rat acetate is an agonist of NPY receptor, with high affinity at NPYR4.Degré de pureté :97.53%Couleur et forme :SolidMasse moléculaire :N/ARef: TM-TP1044L
1mg215,00€5mg510,00€10mg692,00€25mg1.009,00€50mg1.378,00€100mg1.863,00€200mg2.520,00€Neurokinin A(4-10) TFA(97559-35-8 free base)
Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].Formule :C36H55F3N8O12SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :880.93ML221
CAS :ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM inFormule :C17H11N3O6SDegré de pureté :97.74%Couleur et forme :SolidMasse moléculaire :385.35Ref: TM-T4390
2mg34,00€5mg50,00€10mg80,00€25mg137,00€50mg215,00€100mg349,00€200mg512,00€1mL*10mM (DMSO)52,00€Rotigotine-
CAS :Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.Formule :C19H25NOSDegré de pureté :98.08% - 99.59%Couleur et forme :SolidMasse moléculaire :315.47Ref: TM-T6647
5mg50,00€10mg73,00€25mg138,00€50mg241,00€100mg358,00€200mg523,00€500mg822,00€1mL*10mM (DMSO)52,00€Piperacetazine
CAS :Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.Formule :C24H30N2O2SDegré de pureté :99.9% - 99.92%Couleur et forme :SolidMasse moléculaire :410.57Ganirelix Acetate
CAS :Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonistFormule :C82H117ClN18O15Degré de pureté :96.05%Couleur et forme :SolidMasse moléculaire :1630.4Ritanserin
CAS :Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Formule :C27H25F2N3OSDegré de pureté :99.77% - 99.89%Couleur et forme :SolidMasse moléculaire :477.57Thonzylamine
CAS :Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy relief.Formule :C16H22N4ODegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :286.37Glucagon (19-29), human acetate
Glucagon (19-29), human acetate a COOH-terminal fragment processed from glucagon, is a potent and efficient inhibitor of insulin secretion.Formule :C63H93N15O20SDegré de pureté :98.11%Couleur et forme :SolidMasse moléculaire :1412.57SB297006
CAS :SB297006 is an antagonist of C-C chemokine receptor 3, which normally is activated by eotaxin, eotaxin-3, MCP-3, MCP-4, RANTES, and MIP-1δ.Formule :C18H18N2O5Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :342.35GW842166X
CAS :GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.Formule :C18H17Cl2F3N4O2Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :449.25ABT-724
CAS :ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)Formule :C17H19N5Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :293.37Betaxolol
CAS :Betaxolol (Kerlone) is a selective beta1 adrenergic receptor blocker used in the treatment of hypertension and glaucoma.Formule :C18H29NO3Degré de pureté :99.01%Couleur et forme :White Crystalline SolidMasse moléculaire :307.43Ablukast
CAS :Ablukast (Ro 23-3544) is a leuktriene receptor antagonist. Ablukast acts as an anti-asthmatic.Formule :C28H34O8Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :498.56RTICBM-189
CAS :RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.Formule :C15H14Cl2N2ODegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :309.19Ref: TM-T9466
2mg34,00€5mg52,00€10mg84,00€25mg161,00€50mg250,00€100mg369,00€200mg522,00€1mL*10mM (DMSO)67,00€Bay 55-9837 acetate
Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.Degré de pureté :98.27%Couleur et forme :LiquidMasse moléculaire :N/ARelugolix
CAS :Relugolix (RVT-601) is an orally available, non-peptide gonadotropin-releasing hormone (GnRH or luteinizing hormone-releasing hormone (LHRH)) antagonist, withFormule :C29H27F2N7O5SDegré de pureté :98.64% - 99.97%Couleur et forme :SolidMasse moléculaire :623.63Ref: TM-T3630
2mg39,00€5mg58,00€10mg93,00€25mg167,00€50mg250,00€100mg408,00€200mg585,00€1mL*10mM (DMSO)81,00€BMS 182874 hydrochloride
CAS :BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.Formule :C17H20ClN3O3SDegré de pureté :97.01%Couleur et forme :SolidMasse moléculaire :381.88Ref: TM-T21790
1mg77,00€2mg92,00€5mg140,00€10mg205,00€25mg343,00€50mg477,00€100mg665,00€200mg897,00€1mL*10mM (DMSO)146,00€Liraglutide
CAS :Liraglutide (Liraglutida) is a synthetic analog of GLP-1, an agonist of the GLP-1 receptor. Liraglutide is an antidiabetic agent. Cost effective and quality assured.Formule :C172H265N43O51Degré de pureté :97.65% - 99.04%Couleur et forme :SolidMasse moléculaire :3751.25Ref: TM-T6876
1mg111,00€2mg197,00€5mg447,00€10mg527,00€25mg843,00€50mg1.144,00€100mg1.521,00€200mg2.052,00€HTMT dimaleate
CAS :HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.Formule :C27H33F3N4O9Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :614.57MK 571
CAS :MK 571 (L660711) is an orally active antagonist of CysLT1 receptor.Formule :C26H27ClN2O3S2Degré de pureté :98.69% - 99.65%Couleur et forme :SolidMasse moléculaire :515.09Ref: TM-T7841
2mg34,00€5mg50,00€10mg81,00€25mg165,00€50mg285,00€100mg432,00€200mg617,00€1mL*10mM (DMSO)59,00€GLP-1 receptor agonist 9
CAS :1H-Benzimidazole-6-carboxylic acid is a GLP-1 receptor agonist.Formule :C32H31ClFN3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :592.06Medetomidine hydrochloride
CAS :Medetomidine hydrochloride (MPV785) is a selective α2-adrenoceptor agonist, with Ki of 1.08 nM, exhibts 1620-fold selectivity over α1-adrenoceptor.Formule :C13H16N2·HClDegré de pureté :99.96%Couleur et forme :White Or Off White Crystalline PowderMasse moléculaire :236.74ACH-000143
CAS :ACH-000143 是一种可口服的褪黑素受体激动剂，对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。Formule :C13H16ClN3O3Degré de pureté :98.15%Couleur et forme :SolidMasse moléculaire :297.74Ref: TM-T9193
1mg50,00€5mg110,00€10mg172,00€25mg304,00€50mg424,00€100mg583,00€200mg785,00€1mL*10mM (DMSO)122,00€Linzagolix
CAS :Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by KisseiFormule :C22H15F3N2O7SDegré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :508.42Obestatin (rat) acetate
Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).Formule :C114H174N34O31Degré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :2516.81Ref: TM-TP2279L
1mg77,00€2mg97,00€5mg156,00€10mg225,00€25mg375,00€50mg535,00€100mg730,00€200mg938,00€HAEGTFT acetate(926018-95-3 free base)
HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.Formule :C35H51N9O14Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :821.84dasiglucagon acetate
Dasiglucagon acetate: new, stable glucagon for hypoglycemia with better absorption and longer half-life.Formule :C154H226N38O52Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :3441.67NAN-190 hydrobromide
CAS :NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.
Formule :C23H28BrN3O3Degré de pureté :95.20%Couleur et forme :SolidMasse moléculaire :474.39Spexin acetate(1370290-58-6 free base)
Spexin acetate: GAL2/GAL3 agonist. EC50: 45.7/112.2 nM. Inactive at GAL1. Reduces appetite, fat uptake, and food intake; lowers LH in fish; anxiolytic.Formule :C76H117N19O22SDegré de pureté :95.43%Couleur et forme :SolidMasse moléculaire :1680.94Cutamesine dihydrochloride
CAS :Cutamesine dihydrochloride is a σ1 receptor agonist, selective over σ2, combating cardiomyocyte hypertrophy and improving stroke recovery.Formule :C23H32N2O2·2HClDegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :441.43Ref: TM-T3597
2mg34,00€5mg50,00€10mg86,00€25mg167,00€50mg260,00€100mg401,00€200mg580,00€1mL*10mM (DMSO)55,00€Thrombin Receptor Activator for Peptide
Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.Formule :C32H51F3N8O9Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :748.79Mecamylamine
CAS :Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.Formule :C11H21NCouleur et forme :SolidMasse moléculaire :167.29Opiranserin hydrochloride
CAS :Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFormule :C21H35ClN2O5Degré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :430.97Ref: TM-T9833
1mg90,00€5mg215,00€10mg340,00€25mg618,00€50mg879,00€100mg1.224,00€500mg2.457,00€1mL*10mM (DMSO)236,00€Trimethobenzamide hydrochloride
CAS :Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.Formule :C21H29ClN2O5Degré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :424.92LGnRH-III, lamprey acetate(147859-97-0 free base)
LGnRH-III, lamprey acetate is an evolutionarily conserved member of the GnRH family, can stimulate the secretion of gonadotropins, it stimulates the secretionFormule :C61H78N18O16Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :1319.38L-368,899 hydrochloride
CAS :L-368,899 hydrochloride is an OXTR antagonist that prevents oxytocin-induced antiabnormal pain and anti-nausea, and may be used in the study of depression.Formule :C26H43ClN4O5S2Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :591.23Ref: TM-T11794
2mg105,00€5mg147,00€10mg230,00€25mg439,00€50mg685,00€100mg964,00€1mL*10mM (DMSO)200,00€WAY-100635 maleate
CAS :WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).Formule :C25H34N4O2·xC4H4O4Degré de pureté :99.96%Couleur et forme :White SolidMasse moléculaire :538.645Ref: TM-T3453
2mg43,00€5mg63,00€10mg89,00€25mg150,00€50mg215,00€100mg316,00€500mg765,00€1mL*10mM (DMSO)74,00€Trabodenoson
CAS :Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.Formule :C15H20N6O6Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :380.36Ref: TM-T34914
1mg40,00€5mg89,00€10mg116,00€25mg187,00€50mg285,00€100mg411,00€200mg577,00€1mL*10mM (DMSO)88,00€Fenoterol hydrobromide
CAS :Fenoterol hydrobromide is a beta2-adrenergic receptor agonist and bronchodilator used in the study of cardiovascular diseases such as asthma and bronchitis.Formule :C17H22BrNO4Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :384.27(R)-Mirtazapine
CAS :(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.Formule :C17H19N3Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :265.35Ozanimod hydrochloride
CAS :Ozanimod (RPC-1063) HCl is a selective S1P1/S1P5 modulator with high affinity, used in relapsing MS research.Formule :C23H25ClN4O3Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :440.92Ref: TM-T62552
1mg47,00€5mg92,00€10mg137,00€25mg268,00€50mg432,00€100mg620,00€200mg875,00€1mL*10mM (DMSO)101,00€Atogepant
CAS :Atogepant (MK-8031) is an orally available, selective and potent calcitonin gene-related peptide receptor (CGRP) antagonist for the study of migraine.Formule :C29H23F6N5O3Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :603.52Ref: TM-T26682
1mg147,00€5mg250,00€10mg313,00€25mg620,00€50mg1.108,00€100mg1.611,00€200mg2.178,00€1mL*10mM (DMSO)334,00€Dexpramipexole
CAS :Dexpramipexole ((R)-Pramipexole) is a mitochondrial protective agent that maintains mitochondrial function and energy production.Formule :C10H17N3SDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :211.33Clopidogrel thiolactone
CAS :Clopidogrel thiolactone (2-oxoclopidogrel), a P2Y12 receptor inhibitor, is an antiplatelet aggregation compound.Formule :C16H16ClNO3SDegré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :337.82Ref: TM-T5501
1mg96,00€5mg205,00€10mg326,00€25mg557,00€50mg803,00€100mg1.063,00€200mg1.459,00€1mL*10mM (DMSO)227,00€Setiptiline
CAS :Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.Formule :C19H19NDegré de pureté :98.05% - 98.07%Couleur et forme :SolidMasse moléculaire :261.36Levocetirizine Dihydrochloride
CAS :Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.Formule :C21H27Cl3N2O3Degré de pureté :99.89%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :461.81Benzylthiouracil
CAS :Benzylthiouracil (6-Benzyl-2-thiouracil) induces ANCA-associated glomerulonephritis in Graves' disease patients and is used to study hyperthyroidism.Formule :C11H10N2OSDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :218.28CB1/2 agonist 3
CAS :CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.Formule :C25H41NO2Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :387.6Poly-D-lysine hydrobromide (MW 30000-70000)
CAS :Poly-D-lysine hydrobromide (MW 30000-70000) (Poly-D-lysine HBr) is a peptide CaSR agonist that removes proteinase K-resistant PrP from SN56 neuroblastoma cells.Formule :(C6H14N2O2)x·xHBrCouleur et forme :SolidMasse moléculaire :227.102A2ti-1
CAS :A2ti-1 is an annexin A2/S100A10 heterotetramer (A2t) inhibitor that inhibits Src activation and can be used to study human papillomavirus type 16 infection.Formule :C20H22N4O2SDegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :382.48Ref: TM-T36432
1mg94,00€5mg200,00€10mg313,00€25mg620,00€50mg982,00€100mg1.341,00€500mg2.682,00€1mL*10mM (DMSO)286,00€Canagliflozin hemihydrate
CAS :Canagliflozin hemihydrate (TA 7284) treats type 2 diabetes by blocking SGLT2, leading to glucose excretion in urine.Formule :C48H52F2O11S2Degré de pureté :99.42% - 99.96%Couleur et forme :SolidMasse moléculaire :907.05Atipamezole
CAS :Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.Formule :C14H16N2Degré de pureté :99.88%Couleur et forme :Off-White To Light Yellow Crystal PowderMasse moléculaire :212.29SID 7969543
CAS :SID 7969543 is a selective SF-1 inhibitor with potential anticancer activity, inhibits SF-1-triggered luciferase expression and can be used for cancer research.Formule :C24H24N2O7Degré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :452.46CGP 20712 A
CAS :CGP 20712 A (CGP 20712 mesylate) is a β1-adrenergic receptor antagonist with antihypertensive activity that reverses RKT-induced gastric relaxation.Formule :C24H29F3N4O8SDegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :590.57S1RA
CAS :S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating significant selectivity over the sigma-2Formule :C20H23N3O2Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :337.42KB-5492 free base
CAS :KB-5492 free base is an antiulcer agent that inhibits sigma receptors and can be used to study gastric lesions and gastric secretion.Formule :C23H30N2O6Degré de pureté :97.10% - 97.94%Couleur et forme :SolidMasse moléculaire :430.49Ref: TM-T62396
2mg39,00€5mg58,00€10mg82,00€25mg119,00€50mg168,00€100mg249,00€500mg613,00€1mL*10mM (DMSO)64,00€Citalopram
CAS :Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.Formule :C20H21FN2ODegré de pureté :99.78% - 99.89%Couleur et forme :SolidMasse moléculaire :324.39INCB 3284
CAS :INCB 3284, a potent human CCR2 antagonist with an IC50 of 3.7 nM, is researchable for acute liver failure and inhibits MCP-1/hCCR2 binding.Formule :C26H31F3N4O4Degré de pureté :97.81% - 99.42%Couleur et forme :SolidMasse moléculaire :520.54Alfuzosin
CAS :Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and urethral dysfunction.Formule :C19H27N5O4Degré de pureté :99.64%Couleur et forme :White Crystaline PowderMasse moléculaire :389.45Opipramol
CAS :Opipramol (Ensidon) is a compound with antidepressant activity, a sigma (σ) receptor agonist, and anxiolytic activity.Formule :C23H29N3ODegré de pureté :99.84% - 99.98%Couleur et forme :SolidMasse moléculaire :363.5Nebentan potassium
CAS :Nebentan potassium (YM598) is an ETA receptor antagonist that inhibits pulmonary arterial hypertension and is used in the study of neurologic diseases.Formule :C24H20KN5O5SDegré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :529.61Ref: TM-T36008
1mg52,00€2mg77,00€5mg111,00€10mg177,00€25mg313,00€50mg502,00€100mg680,00€200mg888,00€1mL*10mM (DMSO)133,00€Medetomidine
CAS :Medetomidine (MPV785 free base) is a selective α2-adrenoceptor agonist, with sedative and analgesic and vasoconstrictive hypoxic , in small animal anesthesia.Formule :C13H16N2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :200.28Ref: TM-T21492
2mg38,00€5mg57,00€10mg77,00€25mg128,00€50mg193,00€100mg290,00€200mg447,00€1mL*10mM (DMSO)62,00€WIN 51,708
CAS :WIN 51,708 is an antagonist of neurokinin-1 receptor.Formule :C29H33N3ODegré de pureté :99%Couleur et forme :SolidMasse moléculaire :439.59Trazpiroben
CAS :Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.Formule :C31H39N3O4Degré de pureté :99.41% - >99.99%Couleur et forme :SolidMasse moléculaire :517.66Rizatriptan
CAS :Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.Formule :C15H19N5Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :269.35Latrepirdine dihydrochloride
CAS :Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.Formule :C21H25N3·2HClDegré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :392.37Fenoprofen
CAS :Fenoprofen (LILLY-5385) is a non-steroidal anti-inflammatory compound and a modifier enhancer of the melanocortin receptor, increasing ERK1/2 activation.Formule :C15H14O3Degré de pureté :98.4%Couleur et forme :SolidMasse moléculaire :242.27CP-105696
CAS :CP-105696 is a potent and selective leukotriene B4 (LTB4) receptor antagonist for the study of allograft rejection.Formule :C28H28O4Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :428.52(S)-VU0637120
CAS :(S)-VU0637120 is a selective neuropeptide Y(4)R-mutant antagonist used in the study of metabolic disorders.Formule :C16H19N3O5S2Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :397.47Renzapride
CAS :Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.Formule :C16H22ClN3O2Degré de pureté :98.97% - 99.09%Couleur et forme :SolidMasse moléculaire :323.82Ref: TM-T38507
1mg93,00€2mg124,00€5mg200,00€10mg359,00€25mg692,00€50mg945,00€100mg1.279,00€200mg1.701,00€GRK6-IN-2
CAS :GRK6-IN-2 is a potent G protein-coupled receptor kinase 6 (GRK6) inhibitor with potential antitumor activity.GRK6-IN-2 has been studied in multiple myeloma.Formule :C21H21FN6Degré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :376.43LP-533401 hydrochloride
CAS :LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.Formule :C27H23ClF4N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :562.94Protein deglycase DJ-1 against-1
CAS :Protein deglycase DJ-1 against-1 penetrate the BBB and bind to DJ-1 protein,restoring neuronal cellular death in a neurotoxin MPTP-induced model of PD.Formule :C24H23N3O4Degré de pureté :97.23%Couleur et forme :SolidMasse moléculaire :417.46Rotigotine
CAS :Rotigotine (1-Naphthalenol, 5,6,7,8-tetrahydro-6-[propyl[2-(2-thienyl)ethyl]amino]-) is an antiparkinson agent and dopamine receptor agonist.Formule :C19H25NOSDegré de pureté :99.04% - 99.88%Couleur et forme :SolidMasse moléculaire :315.47ACT-462206
CAS :ACT-462206 is a Orexin 1/Orexin 2 receptor antagonist.ACT-462206 is highly potent and can be used to study sleep and anxiety.Formule :C20H24N2O4SDegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :388.48Ref: TM-T26559
1mg42,00€5mg88,00€10mg130,00€25mg264,00€50mg423,00€100mg670,00€500mg1.341,00€1mL*10mM (DMSO)87,00€
