GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.022 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(194 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5984 produits trouvés pour "GPCR/G-Protéine"
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Latrepirdine dihydrochloride
CAS :Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.Formule :C21H25N3·2HClDegré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :392.37Protein deglycase DJ-1 against-1
CAS :Protein deglycase DJ-1 against-1 penetrate the BBB and bind to DJ-1 protein,restoring neuronal cellular death in a neurotoxin MPTP-induced model of PD.Formule :C24H23N3O4Degré de pureté :97.23%Couleur et forme :SolidMasse moléculaire :417.46CGP 20712 A
CAS :CGP 20712 A (CGP 20712 mesylate) is a β1-adrenergic receptor antagonist with antihypertensive activity that reverses RKT-induced gastric relaxation.Formule :C24H29F3N4O8SDegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :590.57Fenoterol hydrobromide
CAS :Fenoterol hydrobromide is a beta2-adrenergic receptor agonist and bronchodilator used in the study of cardiovascular diseases such as asthma and bronchitis.Formule :C17H22BrNO4Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :384.27Bucindolol
CAS :Bucindolol (BMY 13105) is a novel and potent β1-adrenergic receptor blocker that mediates vasodilation and can be used to study chronic heart failure.Formule :C22H25N3O2Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :363.45Rolofylline
CAS :Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.Formule :C20H28N4O2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :356.46S1RA
CAS :S1RA (E-52862)(E-52862) is a potent, selective antagonist of the sigma-1 receptor (σ1R, Ki=17 nM), demonstrating significant selectivity over the sigma-2Formule :C20H23N3O2Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :337.42Ozanimod hydrochloride
CAS :Ozanimod (RPC-1063) HCl is a selective S1P1/S1P5 modulator with high affinity, used in relapsing MS research.Formule :C23H25ClN4O3Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :440.92Ref: TM-T62552
1mg47,00€5mg92,00€1mL*10mM (DMSO)101,00€10mg137,00€25mg268,00€50mg432,00€100mg620,00€200mg875,00€Poly-D-lysine hydrobromide (MW 30000-70000)
CAS :Poly-D-lysine hydrobromide (MW 30000-70000) (Poly-D-lysine HBr) is a peptide CaSR agonist that removes proteinase K-resistant PrP from SN56 neuroblastoma cells.Formule :(C6H14N2O2)x·xHBrCouleur et forme :SolidMasse moléculaire :227.102WAY-100635 maleate
CAS :WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).Formule :C25H34N4O2·xC4H4O4Degré de pureté :99.96%Couleur et forme :White SolidMasse moléculaire :538.645Ref: TM-T3453
2mg43,00€5mg63,00€1mL*10mM (DMSO)74,00€10mg89,00€25mg150,00€50mg215,00€100mg316,00€500mg765,00€Citalopram
CAS :Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.Formule :C20H21FN2ODegré de pureté :99.78% - 99.89%Couleur et forme :SolidMasse moléculaire :324.39Maropitant citrate
CAS :Maropitant citrate is a synthetic neurokinin-1 receptor antagonist and substance P inhibitor, used for controlling vomiting in cats and dogs.Formule :C38H50N2O9Degré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :678.81Alfuzosin
CAS :Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and urethral dysfunction.Formule :C19H27N5O4Degré de pureté :99.64%Couleur et forme :White Crystaline PowderMasse moléculaire :389.45ACT-462206
CAS :ACT-462206 is a Orexin 1/Orexin 2 receptor antagonist.ACT-462206 is highly potent and can be used to study sleep and anxiety.Formule :C20H24N2O4SDegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :388.48Ref: TM-T26559
1mg42,00€1mL*10mM (DMSO)87,00€5mg88,00€10mg130,00€25mg264,00€50mg423,00€100mg670,00€500mg1.341,00€KB-5492 free base
CAS :KB-5492 free base is an antiulcer agent that inhibits sigma receptors and can be used to study gastric lesions and gastric secretion.Formule :C23H30N2O6Degré de pureté :97.10% - 97.94%Couleur et forme :SolidMasse moléculaire :430.49Ref: TM-T62396
2mg39,00€5mg58,00€1mL*10mM (DMSO)64,00€10mg82,00€25mg119,00€50mg168,00€100mg249,00€500mg613,00€SID 7969543
CAS :SID 7969543 is a selective SF-1 inhibitor with potential anticancer activity, inhibits SF-1-triggered luciferase expression and can be used for cancer research.Formule :C24H24N2O7Degré de pureté :98.94%Couleur et forme :SolidMasse moléculaire :452.46Syk Inhibitor II
CAS :Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).Formule :C14H15F3N6ODegré de pureté :97.63%Couleur et forme :SolidMasse moléculaire :340.3(S)-Pramipexole-(N-Propyl-2,2,3,3,3-d5) Dihydrochloride
CAS :(S)-Pramipexole-(N-Propyl-2,2,3,3,3-d5) Dihydrochloride is a deuterated compound of (S)-Pramipexole Dihydrochloride. (S)-Pramipexole Dihydrochloride has a CAS number of 104632-25-9. Pramipexole dihydrochloride could be used to treat Parkinson disease.Formule :C10H14D5Cl2N3SCouleur et forme :SolidMasse moléculaire :289.28Hydroxyzine-d8 DiHCl
CAS :Hydroxyzine-d8 DiHCl is a deuterated compound of Hydroxyzine DiHCl. Hydroxyzine DiHCl has a CAS number of 2192-20-3.Formule :C21H21D8Cl3N2O2Couleur et forme :SolidMasse moléculaire :455.88L-745870
CAS :L-745870 is a D4 receptor antagonist that also inhibits D2 receptors, 5-HT2 receptors, and α-adrenergic receptors.Formule :C18H19ClN4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :326.82Ropinirole
CAS :Ropinirole, D2-like agonist, no D1 affinity, Ki 29 nM for D2, treats Parkinson's.Formule :C16H24N2ODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :260.38SR59230A hydrochloride
CAS :SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue thermogenesis.Formule :C21H28ClNO2Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :361.91R 59-022
CAS :R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.Formule :C27H26FN3OSDegré de pureté :98.55%Couleur et forme :SolidMasse moléculaire :459.58Ref: TM-T16709
1mg35,00€5mg74,00€1mL*10mM (DMSO)75,00€10mg119,00€25mg269,00€50mg447,00€100mg733,00€200mg973,00€Travoprost
CAS :Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.Formule :C26H35F3O6Degré de pureté :97.39% - 99.58%Couleur et forme :Colorless OilMasse moléculaire :500.55Ref: TM-T5841
1mg46,00€5mg88,00€1mL*10mM (DMSO)96,00€10mg120,00€25mg175,00€50mg255,00€100mg371,00€200mg507,00€Cyproheptadine hydrochloride
CAS :Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.
Formule :C21H21N·HClDegré de pureté :99.88% - 99.97%Couleur et forme :SolidMasse moléculaire :323.86PACAP (1-38), human, ovine, rat
CAS :PACAP (1-38), human, ovine, rat (Pituitary Adenylate Cyclase Activating Polypeptide 38) is a neuropeptide with 38 amino acid residues.Formule :C203H331N63O53SDegré de pureté :96.93% - 98.16%Couleur et forme :SolidMasse moléculaire :4534.26Blontuvetmab
CAS :Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].Couleur et forme :LiquidP2Y14R antagonist 1
CAS :P2Y14R antagonist 1 (compound I-17) is a selective oral that inhibits inflammatory response in acute gouty arthritis the NLRP3/GSDMD y and cellular pyroptosis.Formule :C15H12BrN3O2Degré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :346.18Rocatinlimab
CAS :Rocatinlimab (AMG 451) (KHK4083) is a fully human, non-fucosylated IgG1 anti-OX40 monoclonal antibody indicated for atopic dermatitis (AD) research [1].Couleur et forme :LiquidGLP-1 Receptor modulator 1
CAS :GLP-1 Receptormodulator 1 (Compound 7) is an effective positive allosteric modulator of the GLP-1 receptor. It is utilized in the research of obesity and type 2 diabetes.Formule :C18H21NOSMasse moléculaire :299.43GPR183-IN-1
CAS :GPR183-IN-1 (compound 15) is an effective orally active inhibitor of GPR183. It inhibits Ca2+ mobilization with an IC50 value of 39.97 nM. GPR183-IN-1 holds potential for research in cancer, autoimmune diseases, pain, and osteoporosis.Formule :C16H19BrN2O2Couleur et forme :SolidMasse moléculaire :351.24Keto Ziprasidone
CAS :Ziprasidone, an antipsychotic agent, functions as a dual antagonist of 5-HT (serotonin) and dopamine receptors.Formule :C21H19ClN4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :426.92Carlumab
CAS :Carlumab is a high-affinity human monoclonal antibody that targets CCL2, suppressing the recruitment of monocytes/macrophages in the tumour microenvironment.Degré de pureté :95%Couleur et forme :LiquidMasse moléculaire :144.87 kDaN-Methyl amisulpride
CAS :N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.Formule :C18H29N3O4SCouleur et forme :SolidMasse moléculaire :383.51Methaphenilene hydrochloride
CAS :Methaphenilene hydrochloride is an H1 receptor antagonist with antihistaminic and anticholinergic activity, in allergic inflammation and autonomic research.Formule :C15H21ClN2SDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :296.86Metoxibutropate
CAS :Metoxibutropate is a biochemical.Formule :C20H24O3Couleur et forme :SolidMasse moléculaire :312.4PF-610355
CAS :PF-610355 is a long-acting and potent β2-adrenergic receptor agonist (EC50: 0.26 nM).PF-610355 can be used to study asthma and COPD.
Formule :C34H39N3O6SDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :617.76Risperidone Mesylate
CAS :Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.Formule :C24H31FN4O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :506.5917-phenyl trinor Prostaglandin F2α isopropyl ester
CAS :17-phenyl trinor PGF2α N-ethyl amide is an F-series prostaglandin analog which has been approved for use as an ocular hypotensive drug, sold under the AllerganFormule :C26H38O5Couleur et forme :SolidMasse moléculaire :430.58Tulobuterol
CAS :Tulobuterol is mainly used for the prevention and treatment of bronchial asthma, asthmatic bronchitis and chronic bronchitis. Research shows that it could inhibit rhinovirus infection in primary cultures of human tracheal epithelial cells.Formule :C12H18ClNOCouleur et forme :Crystalline SolidMasse moléculaire :227.73Olopatadine
CAS :Olopatadine is an antihistamine and anti-allergy medication for itchy eyes, also possibly treats red skin syndrome.Formule :C21H23NO3Degré de pureté :98%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :337.41Meticillin
CAS :Methicillin: Narrow-spectrum beta-lactam, penicillin-type antibiotic for certain gram-positive bacterial infections.Formule :C17H20N2O6SCouleur et forme :SolidMasse moléculaire :380.42Arazasetron HCl
CAS :Arazasetron is an antiemetic which acts as a 5-HT3 receptor antagonist, pKi = 9.27.Formule :C17H20ClN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :349.81Escitalopram
CAS :Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.Formule :C20H21FN2ODegré de pureté :99.82%Couleur et forme :White Or White Crystalline PowderMasse moléculaire :324.39Eptinezumab
CAS :Eptinezumab is a humanised monoclonal antibody targeting CGRP (calcitonin gene-related peptide), which prevents CGRP binding to its receptor, migraine.
Degré de pureté :95% - 95%Couleur et forme :LiquidTriflupromazine
CAS :Triflupromazine is a dopamine receptor D1/D2 antagonist and LHDA inhibitor that suppresses dopamine activity in (CNS)mental disorders, sedation, and antiemesis.Formule :C18H19F3N2SCouleur et forme :SolidMasse moléculaire :352.42Buflomedil
CAS :Buflomedil is a vasoactive compound. Buflomedil has been used for peripheral arterial diseases.Formule :C17H25NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :307.38DL-Phenylephrine HCl
CAS :DL-Phenylephrine HCl is a selective agonist of the alpha1-adrenergic receptor.Formule :C9H14ClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :203.67Dapagliflozin-d5
CAS :Dapagliflozin D5 (BMS-512148 D5) is deuterated Dapagliflozin. Dapagliflozin is a competitive SGLT2 inhibitor.Formule :C21H25ClO6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :413.9Mianserin-d3
CAS :Mianserin-d3 is a deuterated compound of Mianserin. Mianserin has a CAS number of 24219-97-4. Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, antianxiety, antiemetic, hypotrophic, hypnotic and antihistamine effects, and can be used as a combination of norepinephrine and specific serotonin to treat depression.Formule :C18H17D3N2Couleur et forme :SolidMasse moléculaire :267.38Cinnarizine D8
CAS :Cinnarizine D8 is a deuterium-labeled Cinnarizine which is an antihistamine and a calcium channel blocker.Formule :C26H28N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :376.573Amitriptyline-d6 Hydrochloride
CAS :Amitriptyline-d6 Hydrochloride is a deuterated compound of Amitriptyline Hydrochloride. Amitriptyline Hydrochloride has a CAS number of 549-18-8. Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.Formule :C20H18D6ClNCouleur et forme :SolidMasse moléculaire :319.9015-keto Prostaglandin F2α
CAS :15-keto Prostaglandin F2α is a metabolite of Prostaglandin F2α that lowers intraocular pressure in rabbits.Formule :C20H32O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.47Mirtazapine D3
CAS :Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .Formule :C17H19N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :268.37Brexpiprazole-d8
CAS :Brexpiprazole D8 is a deuterium-modified partial agonist of 5-HT1A and dopamine receptors, with Ki values of 0.12 nM and 0.3 nM respectively.Formule :C25H27N3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :441.62Hydroxy ziprasidone
CAS :Hydroxy ziprasidone is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a 5-HT and dopamine receptor antagonist.Formule :C21H21ClN4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :428.94Dopamine D4 receptor ligand 2
CAS :Compound 17, a dopamine D4 receptor ligand, exhibits high potency and selectivity with IC 50 values of 0.057 nM for D4, and >1000, 220, and 270 nM for D2, 5-HT1A, and α1 receptors, respectively [1].Formule :C20H24ClN3O2Couleur et forme :SolidMasse moléculaire :373.88Norreticuline
CAS :Norreticuline is a potential adrenoceptor-α/β agonist and CYP2D6 and D2 receptor inhibitor for the study of neurodegenerative diseases.Formule :C18H21NO4Couleur et forme :SolidMasse moléculaire :315.36Caerulein, desulfated
CAS :Caerulein, desulfated (FI-6934, desulfated) is a desulfated compound formed after caerulein hydrolysis, a neuropeptide with lower smooth muscle activity.Formule :C58H73N13O18SDegré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :1272.345-Methyltryptamine hydrochloride
CAS :5-Methyltryptamine hydrochloride is a high-affinity 5-HT1C receptor ligand and a partial agonist of 5-HT. 5-Methyltryptamine hydrochloride protects mice subjected to burn, tourniquet and endotoxin shock.Formule :C11H15ClN2Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :210.703Ketanserinol
CAS :Ketanserinol is a metabolite of the antihypertensive drug ketanserin, which blocks 5-HT2 receptors to treat protamine-induced pulmonary hypertension.Formule :C22H24FN3O3Couleur et forme :SolidMasse moléculaire :397.44Litorin
CAS :Litorin suppresses appetite and stimulates smooth muscle, gastrin, gastric acid, and pancreatic secretion.Formule :C51H68N14O11SCouleur et forme :White PowderMasse moléculaire :1085.24Diclofensine
CAS :Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.Formule :C17H17Cl2NODegré de pureté :97.01% - 98.13%Couleur et forme :SolidMasse moléculaire :322.23Roxatidine acetate
CAS :Roxatidine acetate: anti-ulcer, blocks histamine, reduces acid. Safer at lower doses.Formule :C19H28N2O4Degré de pureté :98%Couleur et forme :White Or Off-White PowderMasse moléculaire :348.44Itopride free base
CAS :Itopride HCl combats dyspepsia and GERD, inhibiting AChE and blocking D2 receptors.
Formule :C20H26N2O4Couleur et forme :WhiteMasse moléculaire :358.43MK-447
CAS :MK-447 is a nonsteroidal antiinflammatory agent.Formule :C11H16INODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :305.16Ticlopidine
CAS :Ticlopidine (PCR 5332) is an antiplatelet drug in the thienopyridine family which is an adenosine diphosphate (ADP) receptor inhibitor.Formule :C14H14ClNSDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :263.797-Desmethyl-3-hydroxyagomelatine
CAS :7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.Formule :C14H15NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :245.27Amthamine
CAS :Compound AMTHAMINE DIHYDROBROMIDE is a useful organic compound for research related to life sciences.Formule :C6H11N3SCouleur et forme :SoildMasse moléculaire :157.24S 25585
CAS :S 25585 is a neuropeptide Y (NPY) Y5 receptor antagonist.Formule :C22H23F3N4O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :528.5AR244555
CAS :AR244555 is a bioactive chemical.Formule :C23H23ClF2N2OCouleur et forme :SolidMasse moléculaire :416.89Vanoxerine
CAS :Vanoxerine is an antagonist of dopamine transporter (Ki: 16.9nM).Formule :C28H32F2N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :450.56Amidephrine hydrochloride
CAS :Amidephrine hydrochloride is a biochemical.Formule :C10H17ClN2O3SCouleur et forme :SolidMasse moléculaire :280.776-hydroxy Buspirone
CAS :6-Hydroxy Buspirone, an active metabolite of the anxiolytic compound buspirone, is produced via the cytochrome P450 (CYP) isoform CYP3A4.Formule :C21H31N5O3Couleur et forme :SolidMasse moléculaire :401.50Ciproxifan
CAS :Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).Formule :C16H18N2O2Degré de pureté :98.00%Couleur et forme :SolidMasse moléculaire :270.33Dehydroabiethylamine
CAS :Dehydroabiethylamine (NSC-2955) boosts liver CYP2B, blocks PDKs & cholesterol transport, and has anti-tumor effects.Formule :C20H31NDegré de pureté :98.79%Couleur et forme :Pale Yellow Viscous Liquid /Technical Grade/ Viscous Colorless To Amber LiquidMasse moléculaire :285.47Penbutolol sulfate
CAS :Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.Formule :C18H29NO2H2O4SDegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :340.47Isoproterenol sulfate anhydrous
CAS :Isoproterenol sulfate anhydrous is a useful alkaloid. It is used for biological research.Formule :C22H36N2O10SDegré de pureté :98%Couleur et forme :CoaMasse moléculaire :520.597-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene
CAS :7-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene is a liver receptor homolog-1 (LRH-1) antagonist (IC50: 3.1 μM).Formule :C42H44N2O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :704.87Tivumecirnon
CAS :Tivumecirnon (FLX475) is a selective and oral CCR4 antagonist inhibits the infiltration and migration of Treg into the tumour microenvironment, antitumourFormule :C24H27Cl2F3N6ODegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :543.41Ref: TM-T69834
1mg171,00€5mg418,00€1mL*10mM (DMSO)500,00€10mg666,00€25mg1.334,00€50mg2.071,00€100mg2.879,00€R-138727
CAS :R-138727 is a novel P2Y12 receptor inhibitor.Formule :C18H20FNO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :349.42(RS)-ICI-118551 Hydrochloride
CAS :ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3Formule :C17H27NO2·HClDegré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :313.86Bethanidine sulfate
CAS :Bethanidine sulfate and its ortho-chloro derivative (BW 392C60) are potent adrenergic neuron blockers exhibiting sympathomimetic effects similar to those of bromobenzamine and guanethidine in various animal models, particularly in cats. These compounds inhibit the release of norepinephrine during neural stimulation and enhance the responsiveness of smooth muscle to epinephrine and norepinephrine. Notably, bethanidine sulfate increases the pressor response to tyramine, although this effect diminishes with higher doses. Unlike guanethidine, bethanidine sulfate does not deplete pressor amines in the iris of cats following administration. Additionally, it temporarily suppresses autonomic cholinergic mechanisms and can cause transient neuromuscular paralysis at large doses, contrasting its long-term adrenergic neuron blocking effects.Formule :C20H32N6O4SCouleur et forme :SolidMasse moléculaire :452.57Pardoprunox
CAS :Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.Formule :C12H15N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :233.27Proxyfan Oxalate
CAS :Proxyfan Oxalate is a potent antagonist of the histamine H3 receptor (histamine H3 receptor), with Ki values of 2.9 nM for rats and 2.7 nM for humans. Its inhibitory effect on H3 receptors is over 1000 times stronger than its effect on other histamine receptors.Formule :C15H18N2O5Couleur et forme :SolidMasse moléculaire :306.31Amidephrine
CAS :Amidephrine is an adrenergic agent.Formule :C10H16N2O3SCouleur et forme :SolidMasse moléculaire :244.31Ridazolol HCl
CAS :Ridazolol HCl (CAS 413) is a novel β-adrenoceptor (β-AR) blocker with α-adrenerolytic activity.Formule :C15H19Cl3N4O3Degré de pureté :99.48%Couleur et forme :SoildMasse moléculaire :409.7Atenolol Hydrochloride
CAS :Atenolol Hydrochloride is a selective antagonist of ß1 receptor.Formule :C14H23ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :302.80PSB-KK1445
CAS :PSB-KK1445 is a potent and selective agonist of GPR18, exhibiting EC50 values of 45.4 nM for humans and 124 nM for mice. The selectivity of PSB-KK1445 for GPR18 over the CB receptor subtypes GPR55 and GPR183 exceeds 200-fold.Formule :C24H23FN6O2Masse moléculaire :446.48SB 271046 hydrochloride
CAS :SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is > 200-fold selective over 55 other receptors, enzymes and ion channels.Formule :C20H22ClN3O3S2·HClDegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :488.45MCI-225 dehydratase
CAS :MCI-225 dehydratase is an oral, selective inhibitor of noradrenaline reuptake, and functions as a 5-HT3 antagonist, exhibiting antidepressant effects in vivo .Formule :C17H18ClFN4SCouleur et forme :SolidMasse moléculaire :364.87Dolasetron Mesylate
CAS :Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea followingFormule :C20H24N2O6SDegré de pureté :99.05%Couleur et forme :White PowderMasse moléculaire :420.48Lodoxamide tromethamine
CAS :Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergicFormule :C19H28ClN5O12Degré de pureté :98.8%Couleur et forme :SolidMasse moléculaire :553.91LY 344864
CAS :LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.Formule :C21H22FN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :351.42Paroxetine hydrochloride hemihydrate
CAS :Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).Formule :C38H44Cl2F2N2O7Degré de pureté :99.949%Couleur et forme :SolidMasse moléculaire :749.67MK-5046
CAS :MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).Formule :C20H18F6N4ODegré de pureté :98.56%Couleur et forme :SolidMasse moléculaire :444.37Guacetisal
CAS :Guacetisal, from acetylsalicylic acid and guaiacol, may treat chronic bronchitis.
Formule :C16H14O5Degré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :286.28Bifeprunox Mesylate
CAS :Bifeprunox: partial dopamine/serotonin agonist for schizophrenia; suppresses VTA neurons via D2; affects rat nicotine-seeking.Formule :C25H27N3O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :481.56Penbutolol
CAS :Penbutolol is a nonselective beta-blocker utilized as an antihypertensive and an antianginal.Formule :C18H29NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :291.43DMP 696
CAS :DMP 696 is a selective antagonist of corticotropin-releasing hormone receptor 1. It is used for the treatment of anxiety and depression.Formule :C18H21Cl2N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :410.3
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