GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(251 produits)
- Récepteur adrénergique(3.028 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(218 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(36 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(195 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(42 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(61 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
6012 produits trouvés pour "GPCR/G-Protéine"
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Remoxipride hydrochloride
CAS :Remoxipride hydrochloride (Roxiam) is a selective antagonist of D2 receptor with IC50s of 1.57 μM, ＞100 μM and 42 μM for D2 receptor, D1 receptor and α1-Formule :C16H24BrClN2O3Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :407.73Rezatomidine
CAS :Rezatomidine (AGN203818) is a selective antagonist of α2-adrenergic receptor and can be used in studies about chronic pain, including neuropathic pain.Formule :C13H16N2SDegré de pureté :98.34%Couleur et forme :SolidMasse moléculaire :232.34Upacicalcet
CAS :Upacicalcet (AJT-240) is a calcium mimetic for SHPT in dialysis, reducing PTH by targeting parathyroid receptors.Formule :C11H14ClN3O6SDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :351.76Rocepafant
CAS :Rocepafant (LAU8080), a PAF antagonist, reduces neonatal rat brain damage and inhibits TNF-α toxicity in L929 cells.Formule :C26H23ClN6OS2Degré de pureté :97.31% - 98.95%Couleur et forme :SolidMasse moléculaire :535.08Rafabegron
CAS :Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of diabetes and obesity.Formule :C21H23ClN2O4Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :402.87SDZ-62-434
CAS :SDZ-62-434 is a platelet-activating factor inhibitor with antitumor activity and may be used in the study of leukemia.Formule :C23H27Cl2N3Degré de pureté :98.38%Couleur et forme :SolidMasse moléculaire :416.39Nonabine
CAS :Nonabine is a compound with strong antiemetic properties that can be used to prevent nausea and vomiting associated with cancer chemotherapy.Formule :C25H33NO2Degré de pureté :99.82% - 99.94%Couleur et forme :SolidMasse moléculaire :379.54FPL 55712
CAS :FPL 55712 is a leukotriene receptor and SRS-A antagonist that inhibits bronchoconstriction and can be used in studies of asthma and coronary artery thrombosis.Formule :C27H30O9Degré de pureté :98.15% - 99.8%Couleur et forme :SolidMasse moléculaire :498.52Antihistamine-1
CAS :Antihistamine-1 是能够渗透血脑屏障的 H1-抗组胺药 (Ki=6.9 nM), 它也是 CYP2D6 和 hERG 通道的抑制剂，其 IC50 值分别为 5.4 和 0.8 μM。Formule :C23H24FN5Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :389.47RG 7152
CAS :RG 7152 is a leukotriene D4 antagonist with anti-asthmatic properties and can be used in the study of asthma.Formule :C20H19N5O2Degré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :361.4RO3244794
CAS :RO3244794 is a selective prostacyclin (IP) receptor antagonist that can be used to study liver injury.Formule :C25H19F2NO5Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :451.42GS-9667
CAS :GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia viaFormule :C21H24FN5O4SDegré de pureté :99.77% - 99.96%Couleur et forme :SolidMasse moléculaire :461.51Lecozotan HCl
CAS :Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.
Formule :C28H30ClN5O3Degré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :520.02SF-22
CAS :SF-22 is a Y2R antagonist with potential anti-inflammatory activity that can be used to study diseases associated with neurological disorders.Formule :C28H26N2O3SDegré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :470.58N 0861
CAS :N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.Formule :C13H17N5Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :243.31Ref: TM-T70722
1mg164,00€2mg234,00€5mg389,00€10mg532,00€25mg820,00€50mg1.063,00€100mg1.423,00€200mg1.945,00€Adoprazine
CAS :Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.Formule :C24H24FN3O2Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :405.46Ref: TM-T10249
1mg60,00€5mg130,00€1mL*10mM (DMSO)142,00€10mg205,00€25mg363,00€50mg580,00€100mg782,00€Eclazolast
CAS :Eclazolast (RHC 2871), a lipophilic anti-allergic, inhibits mast cell mediator release by affecting Fc(epsilon)RI-related processes, dose-dependently.Formule :C12H12ClNO4Degré de pureté :98.29% - 98.61%Couleur et forme :SolidMasse moléculaire :269.68Ref: TM-T25360
1mg112,00€1mL*10mM (DMSO)249,00€5mg261,00€10mg396,00€25mg655,00€50mg888,00€100mg1.251,00€500mg2.493,00€LTB4-IN-1
CAS :LTB4-IN-1 (Anti-inflammatory agent 2) with IC50 of 70 nM is an inhibitor of leukotriene synthesis (LTB4).Formule :C26H30N2O4SDegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :466.59Ref: TM-T10917
1mg261,00€5mg515,00€1mL*10mM (DMSO)653,00€10mg874,00€25mg1.288,00€50mg1.755,00€100mg2.358,00€Masupirdine free base
CAS :Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.Formule :C21H24BrN3O3SDegré de pureté :98.36% - 99.65%Couleur et forme :SolidMasse moléculaire :478.4MK-0686
CAS :MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.Formule :C22H19ClF4N2O4Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :486.84Safotibant
CAS :Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edemaFormule :C25H34N4O5SDegré de pureté :99.62% - 99.67%Couleur et forme :SolidMasse moléculaire :502.63JP1302
CAS :JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, renal issues.Formule :C24H24N4Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :368.47Itasetron
CAS :Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer treatments.Formule :C16H20N4O2Degré de pureté :98.58% - 99.68%Couleur et forme :SolidMasse moléculaire :300.36RS 67333 hydrochloride
CAS :RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.Formule :C19H30Cl2N2O2Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :389.36AZ-1355
CAS :AZ-1355 is a novel dibenzoxepine derivative with lipid-lowering properties.Formule :C17H17NO4Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :299.32Ref: TM-T13563
1mg78,00€1mL*10mM (DMSO)156,00€5mg170,00€10mg224,00€25mg338,00€50mg460,00€100mg600,00€200mg820,00€Regrelor disodium
CAS :Regrelor disodium (INS 50589) is a p2y12 receptor antagonist that prevents thrombosis, effectively inhibits vascular smooth muscle cell contraction, inhibitsFormule :C22H23N6Na2O8PDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :576.41LY-2624803
CAS :LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.Formule :C22H25N3O3Degré de pureté :99.78% - 99.97%Couleur et forme :SolidMasse moléculaire :379.45NE-100 hydrochloride
CAS :NE-100 hydrochloride (NE-100 HCl) is a potent and selective antagonist of σ1 (IC50 = 4.16 nM) with antipsychotic activity.Formule :C23H34ClNO2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :391.98Ref: TM-T20797
1mg43,00€2mg54,00€5mg87,00€10mg130,00€25mg210,00€50mg313,00€100mg465,00€200mg662,00€500mg982,00€L 674573
CAS :L 674573 is an inhibitor of leukotriene biosynthesis.Formule :C28H27NO3SDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :457.58Pimethixene maleate
CAS :Pimethixene maleate (Pimetixene maleate) is a 5-HT2B receptor antagonist with sedative activity that can be used to study dry cough in children.Formule :C23H23NO4SDegré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :409.5NNC 92-1687
CAS :NNC 92-1687 is a selective glucagon receptor antagonist that can be used to study type 2 diabetes.Formule :C15H12N2O3SDegré de pureté :98.70% - 99.96%Couleur et forme :SolidMasse moléculaire :300.33CB1R antagonist 1
CAS :CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.Formule :C18H23F3N2O3SDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :404.45Lorglumide sodium salt
CAS :Lorglumide sodium salt (CR-1409 sodium salt) is an antagonist of cholecystokinin receptors (CCK).Formule :C22H31Cl2N2NaO4Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :481.39Sitaxsentan
CAS :Sitaxsentan (TBC-11251), a selective ETA receptor antagonist, prevents vasoconstriction by blocking endothelin.Formule :C18H15ClN2O6S2Degré de pureté :97.99% - 98.71%Couleur et forme :SolidMasse moléculaire :454.9CYM50374
CAS :CYM50374 inhibits Sphingosine-1-phosphate receptor 4 (S1P4 ) with an IC50 of µM.Formule :C19H19NO3SDegré de pureté :98.35% - 98.96%Couleur et forme :SolidMasse moléculaire :341.42ABT-080
CAS :ABT-080 (VML 530), a leukotriene synthesis inhibitor, is used potentially for treatment of asthma.
Formule :C37H31N2NaO4Degré de pureté :98.42%Couleur et forme :SolidMasse moléculaire :590.64Camonagrel
CAS :Camonagrel is a compound that has inhibitory effects on Prostaglandin E2.Formule :C15H16N2O3Degré de pureté :98.71% - 99.25%Couleur et forme :SolidMasse moléculaire :272.3TC LPA5 4
CAS :TC LPA5 4 is a LPA5 receptor antagonist.Formule :C23H23ClN2O3Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :410.89Ref: TM-T23438
1mg49,00€5mg98,00€1mL*10mM (DMSO)107,00€10mg157,00€25mg324,00€50mg485,00€100mg713,00€200mg982,00€Egis-11150
CAS :Egis-11150 is a potent inhibitor of adrenergic alpha1, alpha2c, 5-HT2a, 5HT7 receptors.Formule :C19H21ClFN5O2Degré de pureté :97.49% - >99.99%Couleur et forme :SolidMasse moléculaire :405.85Milenperone
CAS :Milenperone (R 34009) is a novel anti-invasive compound for the control of behavioral disorders in patients with epilepsy and alcoholism.Formule :C22H23ClFN3O2Degré de pureté :98.09% - 99.84%Couleur et forme :SolidMasse moléculaire :415.89Spizofurone
CAS :Spizofurone (Espizofurona) has anti-ulcer activity, protective effect on the gastric mucosa of rats and can increase alkaline secretion.Formule :C12H10O3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :202.21Pirodomast
CAS :Pirodomast is a thromboxane A (TXA2) synthase inhibitor.Formule :C18H17N3O2Degré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :307.35PD 168568 dihydrochloride
CAS :PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).Formule :C22H29Cl2N3ODegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :422.39Ref: TM-T12383
5mg46,00€10mg55,00€1mL*10mM (DMSO)57,00€25mg111,00€50mg166,00€100mg235,00€200mg329,00€Ancriviroc
CAS :Ancriviroc (SCH-351125) is an orally bioavailable small molecule chemokine receptor CCR5 antagonist.Cost-effective and quality-assured.Formule :C28H37BrN4O3Degré de pureté :99.76% - 99.82%Couleur et forme :SolidMasse moléculaire :557.533GP2-114
CAS :GP2-114 is a catecholamine motility mimetic that produces current-dependent cardiovascular effects.Cost-effective and quality-assured.Formule :C19H24N2O4Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :344.4D18024
CAS :D18024 is a phthalazinonderivat with anti-allergic and anti-histamine effect.Formule :C29H31ClFN3ODegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :492.03Ref: TM-T10945
1mg349,00€5mg697,00€1mL*10mM (DMSO)880,00€10mg888,00€25mg1.395,00€50mg1.783,00€100mg2.530,00€Bedoradrine sulfate
CAS :Bedoradrine sulfate (MN-221 sulfate) is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.Formule :C24H32N2O5H2O4SDegré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :477.56SR144528
CAS :SR144528 is an antagonist of the CB2 receptor (Ki = 0.6 nM) and inhibits microsomal ACAT activity (IC50 = 3.6 μM).Formule :C29H34ClN3ODegré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :476.055-HT6/7 antagonist 1
CAS :5-HT6/7 antagonist 1 is a dual 5-HT6/7/2A and D2 receptor antagonist for the study of dementia and Alzheimer's disease.Formule :C22H20FN3O3Degré de pureté :98.78% - 99.26%Couleur et forme :SolidMasse moléculaire :393.41Bedoradrine
CAS :Bedoradrine (MN-221) free base is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.Formule :C24H32N2O5Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :428.52Irdabisant
CAS :Irdabisant (CEP-26401) is an H3R antagonist/inverse agonist, BBB permeable, with cognition-enhancing effects for schizophrenia/cognitive research.Formule :C18H23N3O2Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :313.39cis-Urocanic acid
CAS :cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).Formule :C6H6N2O2Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :138.12Goxalapladib
CAS :Goxalapladib（GSK 677116） is a small molecule compound that can be used to treat cardiovascular risks associated with atherosclerosis.Formule :C40H39F5N4O3Degré de pureté :99.64% - 99.93%Couleur et forme :SolidMasse moléculaire :718.75Xamoterol hemifumarate
CAS :Xamoterol hemifumarate is a potent and selective β1-adrenoceptor agonist.Xamoterol hemifumarate is a potential compound for the study of the relationshipFormule :C36H54N6O14Degré de pureté :99.79%Couleur et forme :White SolidMasse moléculaire :794.37A-437203
CAS :A-437203 (Lu201640), selective D3 antagonist with Ki: D2-71nM, D3-1.6nM, D4-6220nM; based on 1H-pyrimidin-2-one scaffold.Formule :C20H27F3N6OSDegré de pureté :98.80%Couleur et forme :SolidMasse moléculaire :456.53Ref: TM-T10213
1mg94,00€5mg188,00€1mL*10mM (DMSO)215,00€10mg264,00€25mg411,00€50mg532,00€100mg740,00€200mg982,00€Dimethindene
CAS :Dimethindene (Dimetindeno) is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects.Formule :C20H24N2Degré de pureté :98.3% - 98.99%Couleur et forme :SolidMasse moléculaire :292.42ORM-10921
CAS :ORM-10921 is an α2C-adrenoceptor antagonist that has shown antipsychotic and antidepressant activity in animal studies.Formule :C18H23NO2Degré de pureté :99.46% - 99.98%Couleur et forme :SolidMasse moléculaire :285.38Vadocaine
CAS :Vadocaine (Vadocaina) is a novel analgesic compound for local anaesthesia and can be used to study the central nervous system and cardiovascular system.Formule :C18H28N2O2Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :304.43CMF019
CAS :CMF019 is a potent agonist of the Apelin receptor (APJ) with G protein bias. CMF019 binds to APJ (pKis: 8.58, 8.49, and 8.71 for the human, rat, and mouse).Formule :C25H33N3O3SDegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :455.61NCGC00135472
CAS :NCGC00135472: DRV1 agonist with pro-catabolic effects, activates DRV1/GPR32, EC50: 0.37 uM (beta-blocker), 0.05 uM (cAMP), enhances phagocytosis.Formule :C20H14F2N4ODegré de pureté :99.41% - 99.48%Couleur et forme :SolidMasse moléculaire :364.35Ref: TM-T33613
1mg315,00€5mg745,00€10mg1.018,00€25mg1.431,00€50mg1.783,00€100mg2.250,00€500mg4.410,00€ST 91
CAS :ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.Formule :C13H20ClN3Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :253.77Ref: TM-T23397
5mg49,00€1mL*10mM (DMSO)50,00€10mg72,00€25mg142,00€50mg245,00€100mg354,00€200mg497,00€Benperidol
CAS :Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.Formule :C22H24FN3O2Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :381.44Ref: TM-T26360
1mg116,00€5mg276,00€1mL*10mM (DMSO)279,00€10mg410,00€25mg680,00€50mg938,00€100mg1.293,00€500mg2.593,00€BAY 60-6583
CAS :BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3Formule :C19H17N5O2SDegré de pureté :98.46% - 99.8%Couleur et forme :SolidMasse moléculaire :379.44Ref: TM-T14506
1mg39,00€2mg50,00€5mg84,00€1mL*10mM (DMSO)101,00€10mg116,00€25mg233,00€50mg376,00€100mg567,00€200mg797,00€Olorinab
CAS :Olorinab (APD 371) (APD 371) is a highly potent, selective and fully efficacious cannabinoid receptor type 2 (CB2) agonist. With an EC50 of 6.2 nM for hCB2.Formule :C18H23N5O3Degré de pureté :97.67% - 98.47%Couleur et forme :SolidMasse moléculaire :357.41Runcaciguat
CAS :Runcaciguat, a soluble guanylate cyclase stimulator, aids in cardiovascular and renal research.Formule :C23H22Cl2F3NO3Degré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :488.33SPD-473 citrate
CAS :SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.Formule :C23H31Cl2NO8SDegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :552.47Enerisant hydrochloride
CAS :Enerisant HCl is a novel potent and selective histamine H3 receptor antagonist, a substrate for P-gp, mediated by cytochrome P450 (CYP) and transporter proteinsFormule :C22H31ClN4O3Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :434.96CCG 203769
CAS :CCG 203769 (Thiadiazolidinone (TDZD) deriv. 6) is a selective inhibitor of RGS4 with an IC50 of 17 nM for the RGS4-Gαo protein-protein interaction.Formule :C8H14N2O2SDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :202.27Ref: TM-T10705
1mg84,00€5mg177,00€1mL*10mM (DMSO)195,00€10mg250,00€25mg444,00€50mg622,00€100mg893,00€500mg1.783,00€Efletirizine
CAS :Efletirizine (UCB-28754), a histamine blocker and 5-LO inhibitor, aids in topical allergy treatment.Formule :C21H24F2N2O3Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :390.42SB 218795
CAS :SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM for hNK3 which is about 90-fold and 7000-fold selectivity over hNK2 and hNK1.Formule :C25H20N2O3Degré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :396.44Ref: TM-T23316
1mg49,00€2mg63,00€5mg90,00€1mL*10mM (DMSO)109,00€10mg160,00€25mg313,00€50mg505,00€100mg713,00€500mg1.504,00€KI-7
CAS :KI-7 is an adenosine A2B receptor positive allosteric modulator.Formule :C23H18N2O2Degré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :354.4Ref: TM-T9238
2mg35,00€5mg55,00€1mL*10mM (DMSO)62,00€10mg95,00€25mg172,00€50mg264,00€100mg399,00€200mg560,00€LAS38096
CAS :LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .Formule :C17H12N6ODegré de pureté :99.18% - 99.95%Couleur et forme :SolidMasse moléculaire :316.32Besipirdine
CAS :Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic activity and cardiovascular activity.Formule :C16H17N3Degré de pureté :97.15% - 98.85%Couleur et forme :SolidMasse moléculaire :251.332'-MeCCPA
CAS :2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.Formule :C16H22ClN5O4Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :383.83DF-1111301
CAS :DF-1111301 is a novel anti-allergic compound with anti-histamine H1 and anti-PAF activity.Formule :C15H25Cl2N3ODegré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :334.29Antalarmin hydrochloride
CAS :Antalarmin hydrochloride, a CRF1 antagonist, offers anti-inflammatory benefits and prevents stress ulcers in IBS.Formule :C24H35ClN4Degré de pureté :99.84% - 99.85%Couleur et forme :SolidMasse moléculaire :415.02Nexopamil
CAS :Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.
Formule :C24H40N2O3Degré de pureté :97.87% - >99.99%Couleur et forme :SolidMasse moléculaire :404.59CyPPA
CAS :CyPPA enhances SK channels, reducing firing rate and extending apamin-sensitive afterhyperpolarization.Formule :C16H23N5Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :285.39Ref: TM-T20968
2mg42,00€5mg62,00€1mL*10mM (DMSO)66,00€10mg87,00€25mg166,00€50mg266,00€100mg442,00€500mg973,00€Perphenazine dihydrochloride
CAS :Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.Formule :C21H28Cl3N3OSDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :476.89BMS CCR2 22
CAS :BMS CCR2 22 is a potent and selective antagonist of CCR2 with calcium flux IC50 of 18 nM, chemotaxis IC50 of 1 nM, and binding IC50 of 5.1 nM.Formule :C28H34F3N5O4SDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :593.66Ref: TM-T14688
1mg55,00€5mg110,00€1mL*10mM (DMSO)147,00€10mg173,00€25mg349,00€50mg532,00€100mg718,00€200mg964,00€Halopemide
CAS :Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).Formule :C21H22ClFN4O2Degré de pureté :96.57%Couleur et forme :SolidMasse moléculaire :416.88BMS-817399
CAS :BMS-817399: oral CCR1 antagonist with binding and chemotaxis inhibition IC50s, potential for rheumatoid arthritis research.Formule :C23H36ClN3O4Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :454Ref: TM-T26861
1mg152,00€5mg319,00€1mL*10mM (DMSO)356,00€10mg485,00€25mg770,00€50mg1.035,00€100mg1.395,00€CCR1 antagonist 6
CAS :CCR1 antagonist 6 is a CCR1 antagonist (IC50: 3 nM).Formule :C21H23ClN4O3SDegré de pureté :99.15% - 99.92%Couleur et forme :SolidMasse moléculaire :446.95SMO-IN-2
CAS :SMO-IN-2 is a SMO inhibitor with antiproliferative activity and anticancer activity and inhibits Hh signaling.SMO-IN-2 can be used in the study of cancer.Formule :C25H25F4N5O2Degré de pureté :98.64%Couleur et forme :SolidMasse moléculaire :503.49Thonzylamine hydrochloride
CAS :Thonzylamine hydrochloride (Resistab) is an anticholinergic and antihistamine used as an antipruritic.Formule :C16H23ClN4ODegré de pureté :99.67%Couleur et forme :White Crystalline PowderMasse moléculaire :322.83Piromelatine
CAS :Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity withFormule :C17H16N2O4Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :312.32Ref: TM-T34081
1mg60,00€5mg130,00€1mL*10mM (DMSO)142,00€10mg178,00€25mg334,00€50mg522,00€100mg713,00€GSK2239633A
CAS :GSK2239633A is an allosteric antagonist of CC-chemokine receptor 4 (CCR4) with a pIC50 of 7.96 for the binding of [125I]-TARC to human CCR4.Formule :C24H25ClN4O5S2Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :549.06Ref: TM-T11481
500mgÀ demander1mg35,00€5mg79,00€1mL*10mM (DMSO)87,00€10mg118,00€25mg245,00€50mg355,00€100mg515,00€CCR2 antagonist 5
CAS :JNJ-41443532: oral hCCR2 antagonist, IC50=37 nM, anti-chemotaxis, treats inflammation & diabetes.Formule :C22H25F3N4O3SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :482.52Linetastine
CAS :Linetastine (TMK-688) inhibits 5-LOX, blocks leukotrienes, counters histamine; researched for asthma, atherosclerosis, ulcers.Formule :C35H40N2O6Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :584.7Sonedenoson
CAS :Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2;-O-ribose methyltransferase.Formule :C18H20ClN5O5Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :421.84H-9 dihydrochloride
CAS :H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.Formule :C11H15Cl2N3O2SDegré de pureté :97.3%Couleur et forme :SolidMasse moléculaire :324.23AZD8542
CAS :AZD8542 is an antagonist of Smoothened (SMO) with potential as an oncology therapeutic.Formule :C25H24N4O2Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :412.485-HT1A modulator 1
CAS :5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).Formule :C21H25N3O2SDegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :383.51RLX-33
CAS :RLX-33 blocks RXFP3 and relaxin 3 effects, controls food intake in rats, and may help study metabolic syndrome.Formule :C24H19ClN4O4Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :462.89Imiloxan
CAS :Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder.Formule :C14H16N2O2Degré de pureté :98.13% - 99.8%Couleur et forme :SolidMasse moléculaire :244.29Ricasetron
CAS :Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.Formule :C19H27N3ODegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :313.44KSK68
CAS :KSK68 is a sigma-1 and histamine H3 receptor antagonist with analgesic activity, inhibits H3 receptors and can be used to study pain.Formule :C23H28N2O2Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :364.48KSK94
CAS :KSK94 is an H3 receptor antagonist that inhibits sigma-2 receptors , with a Ki value of 75.2 nM, and can be used to study injurious pain.Formule :C25H26N4ODegré de pureté :99.60%Couleur et forme :SolidMasse moléculaire :398.548740 RP
CAS :48740 RP (RP 55779) is an antagonist of platelet-activating factor.Formule :C12H11N3OSDegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :245.3Ref: TM-T10159
1mg338,00€5mg537,00€1mL*10mM (DMSO)537,00€10mg858,00€25mg1.269,00€50mg1.720,00€100mg2.305,00€ML 10302 hydrochloride
CAS :ML 10302 hydrochloride is a specific agonist 5-HT4 and binds 5-HT receptors with Kis of 1.07 nM and 782 nM for 5-HT4 and 5-HT3.Formule :C15H22Cl2N2O3Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :349.25
