GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.024 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.029 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(159 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(443 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(22 produits)
- Récepteur du glucagon(196 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(42 produits)
- Récepteur opioïde(326 produits)
- PAFR(14 produits)
- PKA(53 produits)
- Récepteur S1P(17 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5980 produits trouvés pour "GPCR/G-Protéine"
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Pneumadin, rat
CAS :Rat Pneumadin (PNM), a decapeptide, stimulates AVP release, exerting strong antidiuretic effects in animals with an active AVP system.Formule :C47H74N12O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1047.178PAR 4 (1-6) (TFA)
PAR 4 (1-6) TFA (GYPGQV TFA), a hexapeptide derived from protease-activated receptor 4 (PAR 4), serves as a specific agonist for PAR 4.Formule :C28H41N7O9·xC2HF3O2Couleur et forme :SolidUrocortin II, mouse
CAS :Mouse Urocortin II: Selective CRF2 agonist, Ki 0.66 nM for CRFR2, >100 nM for CRFR1, affects central neural circuits.Formule :C187H320N56O50Couleur et forme :SolidMasse moléculaire :4152.96Dolcanatide
CAS :Dolcanatide: oral GC-C agonist with laxative, pain-relief, and anti-inflammatory properties for IBD research.Formule :C65H104N18O26S4Couleur et forme :SolidMasse moléculaire :1681.89A 76154
CAS :A 76154 is an antagonist of leutenizing hormone releasing hormone (LHRH).Formule :C70H93FN12O12Couleur et forme :SolidMasse moléculaire :1313.584LHRH, Ala(6)-
CAS :LHRH, Ala(6)- is a synthetic luteinizing hormone-releasing hormone agonist agent.Formule :C56H77N17O13Couleur et forme :SolidMasse moléculaire :1196.32Lys-[Des-Arg9]Bradykinin TFA
CAS :Lys-[Des-Arg9]Bradykinin TFA: natural kinin, selective B1 agonist; Ki: 0.12 nM (human), 1.7 nM (mouse), 0.23 nM (rabbit); weak on B2 receptors.Formule :C54H75F6N13O15Couleur et forme :SolidMasse moléculaire :1260.24Bodilisant
CAS :Bodilisant: nanomolar-affinity hH3R ligand, derived from piperidine, with BODIPY fluorophore.Formule :C27H34BF2N3OCouleur et forme :SolidMasse moléculaire :465.4Denrakibart
Denrakibart is a humanized IgG2κ antibody targeting CCL17, with HumanIgG2kappa, Isotype Control serving as the corresponding isotype control.Couleur et forme :Odour LiquidParstatin(human) TFA
Parstatin(human) TFA, a cell-penetrating PAR-1 thrombin receptor agonist peptide, effectively inhibits angiogenesis, as indicated by studies [1] [2].Formule :C193H331F3N64O55S3Couleur et forme :SolidMasse moléculaire :4581.28SFNGGP-NH2
CAS :SFNGGP-NH2 is a biologically active peptide that interacts with Protease-Activated Receptor 3 (PAR-3), a high-affinity thrombin receptor.Formule :C25H36N8O8Couleur et forme :SolidMasse moléculaire :576.6L 366811
CAS :L 366811 is a potent oxytocin antagonist.Formule :C43H56N8O6Couleur et forme :SolidMasse moléculaire :780.95Ici 216140
CAS :ICI 216140: GRP/bombesin receptor 2 blocker, potent at 2 nM. Reduces amylase at 2 mg/kg and lowers bombesin-induced blood pressure at 1 mM in rats.Formule :C45H65N13O8Couleur et forme :SolidMasse moléculaire :916.08Lanerkitug
Lanerkitug is a humanized IgG1λ2 antibody that targets CCR8, with HumanIgG1lambda2, Isotype Control serving as its corresponding isotype control.Couleur et forme :Odour LiquidProtease-Activated Receptor-1, PAR-1 Agonist
CAS :Selective peptide agonist that mimics thrombin to activate PAR-1 receptor, enabling targeted receptor activation.Formule :C35H58N10O9Couleur et forme :SolidMasse moléculaire :762.91A-286501
CAS :A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.Formule :C11H14BrN5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :328.17HL2-m5
CAS :HL2-m5 is an inhibitor of the sonic hedgehog/patched (Shh/PTCH1) interaction, with a Kd for Shh of 170 nM. It effectively inhibits the activation of the Hedgehog signaling pathway and the transcription of Gli-controlled genes, with an IC50 of 230 nM.Formule :C70H101N15O24S3Couleur et forme :SolidMasse moléculaire :1632.83CCR4 antagonist 3
CAS :Orally active CCR4 antagonist with piperidinyl-azetidine; IC50: 22 nM (calcium flux), 50 nM (CTX); antitumor effects.Formule :C24H27Cl2N7OCouleur et forme :SolidMasse moléculaire :500.43BPP-2
BPP-2 is a GHSR ligand containing the element F. By labeling BPP-2 with the isotope 18F, a PET probe targeting GHSR can be produced. The binding affinity (Ki) of 18F-BPP-2 for GHSR is 274 nM.Formule :C27H28FN5O2Masse moléculaire :473.2227PSB-22269
PSB-22269 is identified as a GPR17 antagonist with a Ki value of 8.91 nM. It exhibits significant inhibitory effects in cAMP and G protein activation assays. Molecular docking studies indicate that the binding site of PSB-22269 includes positively charged arginine residues and a hydrophobic pocket. PSB-22269 promotes myelin regeneration strategies, offering potential for multiple sclerosis research.Formule :C26H21NO6Couleur et forme :SolidMasse moléculaire :443.45R 50595
CAS :R 50595 is a selective non-competitive cisapride antagonist.Formule :C30H35Cl2F2N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :594.52FR190997
CAS :FR190997 is an agonist of bradykinin B2 receptor.Formule :C37H33Cl2N5O5Couleur et forme :SolidMasse moléculaire :698.5915(S)-15-methyl Prostaglandin F2α methyl ester
CAS :15(S)-15-methyl Prostaglandin F2α methyl ester can be used in related research in the field of life sciences.Formule :C22H38O5Couleur et forme :SolidMasse moléculaire :382.53GLP-1(7-37)
CAS :GLP-1 (7-37) is a truncated, bioactive form of GLP-1 that is the product of proglucagon processing in intestinal endocrine L cells.Formule :C151H228N40O47Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3355.67Anticancer agent 258
CAS :Anticanceragent 258 is an imidazo[1,2-B][1,2,4]triazole derivative that modulates nuclear receptor activity. It exhibits an EC50 of 63 nM for Nurr in N2A cells and an IC50 of 0.1 pM for Nur77 in HEK293 cells. Anticanceragent 258 is applicable in studies related to cancer, metabolic disorders, and neurological diseases.Formule :C17H12F2N4Couleur et forme :SolidMasse moléculaire :310.3RS 18286
CAS :RS 18286 is a LHRH antagonist.Formule :C74H101Cl2N17O14Couleur et forme :SolidMasse moléculaire :1523.6LY-53857 free base
CAS :LY-53857 free base is a bioactive chemical.Formule :C23H32N2O3Couleur et forme :SolidMasse moléculaire :384.51CCK Octapeptide, non-sulfated acetate
CCK Octapeptide, non-sulfated acetate is a synthetic desulfated peptide of cholecystokinin.Formule :C51H66N10O15S2Degré de pureté :98.9700%Couleur et forme :SolidMasse moléculaire :1123.26HAEGTFTSDVS
CAS :HAEGTFTSDVS is the first N-terminal 1-11 residues of GLP-1 peptide.Formule :C48H71N13O20Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1150.18Setmelanotide Acetate(920014-72-8 free base)
CAS :Setmelanotide Acetate(920014-72-8 free base) (RM-493 Acetate) is a selective agonist of melanocortin 4 receptor (MC4R)(human and rat MC4R with EC50s of 0.27 nMFormule :C51H72N18O11S2Degré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :1177.35Ref: TM-T12882L
1mg131,00€5mg286,00€10mg430,00€25mg710,00€50mg998,00€100mg1.349,00€1mL*10mM (DMSO)555,00€BIIE-0246
CAS :BIIE-0246 is a selective NPY2R antagonist, IC50=15 nM at the rat [125I]PYY3-36 site, reduces NPY-stimulated expression of p-AKT S473 and P-p44/42 MAPK.Formule :C49H57N11O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :896.05(S)-Osanetant
CAS :(S)-Osanetant, an S-enantiomer, is a selective NK3 antagonist with potential for treating schizophrenia and has anxiolytic and antidepressant effects.Formule :C35H41Cl2N3O2Couleur et forme :SolidMasse moléculaire :606.62Kassinin
CAS :Kassinin is a peptide derived from the Kassina frog. It belongs to tachykinin family of neuropeptides.Formule :C59H95N15O18SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1334.54GHRF, porcine
CAS :GHRF, porcine, a growth hormone releasing factor (GHRF) peptide (porcine), binds to the growth hormone secretagogue receptor (GHSR), thereby inducing theFormule :C219H365N73O66SCouleur et forme :SolidMasse moléculaire :5108.76Kisspeptin 13
CAS :<p>Kisspeptin 13 activates GPR54 & GnRH receptors, boosts memory, and aids in Alzheimer's research.</p>Formule :C78H107N21O18Couleur et forme :SolidMasse moléculaire :1626.81FLLRN
CAS :<p>FLLRN is a biologically active peptide serving as a PAR1-specific antagonist.</p>Formule :C31H51N9O7Couleur et forme :SolidMasse moléculaire :661.79Sarafotoxin S6c
CAS :Highly selective ETB endothelin receptor agonist (Ki values are 0.29 and 28000 nM at ETB and ETA receptors respectively).Formule :C103H147N27O37S5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2516Bradykinin (1-7)
CAS :Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.Formule :C35H52N10O9Degré de pureté :98%Couleur et forme :White Lyophilized PowderMasse moléculaire :756.85Methionyl-Lysyl-Bradykinin
CAS :Methionyl-Lysyl-Bradykinin (Met-Lys-Bradykinin), a Bradykinin analogue, is a kinin [1] [2] .Formule :C61H94N18O13SCouleur et forme :SolidMasse moléculaire :1319.58Bim 21009
CAS :Bim 21009 is an inhibitor of gonadorelin.Formule :C74H92ClN17O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1463.08YFLLRNP
CAS :YFLLRNP is a biologically active peptide functioning as a partial agonist of PAR-1, selectively activating the G12/13 signaling pathway.Formule :C45H67N11O10Couleur et forme :SolidMasse moléculaire :922.08[8-L-arginine] deaminovasopressin
CAS :[8-L-arginine] deaminovasopressin (dAVP) is a vasopressin analog [1] .Formule :C46H64N14O13S2Couleur et forme :SolidMasse moléculaire :1085.22Tau conotoxin CnVA
CAS :Tau conotoxin CnVA, a small peptide found in the venom of Conus consors (cone snail), is a member of the T1 cone snail peptide superfamily. It demonstrates high selectivity for the somatostatin sst3 receptor with a Ki value of 1.5 µM. Tau conotoxin CnVA is unique as the only known toxin interacting with this subfamily of G protein-coupled receptors (GPCR). This compound is useful for research related to diseases associated with the sst3 receptor, such as pancreatic cancer or pituitary adenomas.Formule :C72H116N24O17S4Couleur et forme :SolidMasse moléculaire :1718.1SC-53116
CAS :SC-53116 HCl can increase the production of serotonin in central nervous system tissues and is a psychoactive agent.Formule :C16H22ClN3O2Couleur et forme :SolidMasse moléculaire :323.82Lobeline sulfate
CAS :Lobeline sulfate, an alkaloid like nicotine, aids in smoking cessation, insomnia, and respiratory issues. Less potent on nicotinic receptors.Formule :C22H29NO6SDegré de pureté :98%Couleur et forme :White PowderMasse moléculaire :435.54GB-110 hydrochloride
GB-110 HCl: potent, nonpeptidic oral PAR2 agonist; triggers Ca2+ release in HT29 cells; EC50 0.28 μM.Formule :C33H49ClN6O5Couleur et forme :SolidMasse moléculaire :645.23HTL22562
CAS :HTL22562 is a calcitonin gene-related peptide (CGRP) receptor antagonist for acute treatment of migraine.Formule :C40H49N11O5Couleur et forme :SolidMasse moléculaire :763.904(±)5(6)-EET
CAS :5(6)-EET is a fully racemic version of the enantiomeric forms biosynthesized from arachidonic acid by cytochrome P450 enzymes.Formule :C20H32O3Couleur et forme :SolidMasse moléculaire :320.473Substance P (1-9)
CAS :Substance P (1-9), a nonapeptide, slows its own inactivation and stimulates neurons.Formule :C52H77N15O12Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1104.26Hemokinin 1, human TFA
Hemokinin-1 is a human TFA and selective NK1 agonist; also activates NK2 & NK3 and induces opioid-independent analgesia.Formule :C56H85F3N14O16SCouleur et forme :SolidMasse moléculaire :1299.42Vicasinabin
CAS :Vicasinabin: potent CB2 agonist; researches chronic pain, atherosclerosis, bone mass, neuroinflammation.Formule :C15H22N10OCouleur et forme :SolidMasse moléculaire :358.41P4pal10 TFA
P4pal10 TFA, the TFA salt form of P4pal10, serves as an antagonist of the protease-activated receptor 4 (PAR4). This compound inhibits platelet aggregation and thrombin generation induced by tissue factor (TF), exhibiting anticoagulant and antithrombotic activities. Additionally, P4pal10 TFA alleviates carrageenan-induced edema and neutrophil infiltration, and ameliorates damage in rat myocardial ischemia/reperfusion (I/R) models.Couleur et forme :Odour Solid[Pro34]Neuropeptide Y, porcine
CAS :[Pro34]Neuropeptide Y, porcine functions as a selective agonist for the NPY (Y1) receptor and induces vasoconstriction in the guinea pig's caval vein [1].Formule :C190H286N54O56Couleur et forme :SolidMasse moléculaire :4222.63α-Bulnesene
CAS :α-Bulnesene, a novel PAF (platelet-activating factor) receptor antagonist, exhibits an IC50 of 17.62 μM. It can be isolated from patchouli. α-Bulnesene inhibits both PAF and arachidonic acid-induced aggregation of rabbit platelets.Formule :C15H24Couleur et forme :SolidMasse moléculaire :204.35Lys-γ3-MSH(human)
CAS :Pro-opiomelanocortin (POMC) derived peptide that stimulates lipolysisFormule :C128H193N45O39SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3018.25CCR4 antagonist 3 hydrochloride
CAS :Orally active CCR4 antagonist 3 hydrochloride with potent selectivity, IC50s: 22/50 nM; has antitumor properties.Formule :C24H27Cl2N7O·xHClCouleur et forme :SolidNeuropeptide Y 13-36 (porcine)
CAS :Neuropeptide Y 13-36 (porcine) is a selective neuropeptide Y2 receptor agonist.Formule :C135H209N41O36Couleur et forme :SolidMasse moléculaire :2982.408GLP-1R agonist 16
CAS :Compound 115a, a GLP-1R agonist, effectively activates the GLP-1 receptor with an EC50 of 0.15 nM [1].Formule :C50H58FN10O6PCouleur et forme :SolidMasse moléculaire :945.038-iso Prostaglandin E2
CAS :"8-iso PGE2: Isoprostane from arachidonic acid, potent rat renal vasoconstrictor, reduces GFR and renal flow by 80%, no BP effect."Formule :C20H32O5Couleur et forme :SolidMasse moléculaire :352.47Thioperamide maleate
CAS :Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31Formule :C19H28N4O4SDegré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :408.52Cinnamtannin A2
CAS :<p>Cinnamtannin A2, a tetrameric procyanidin, boosts GLP-1, insulin, CRH expression, and has antioxidant, anti-diabetic, nephroprotective properties.</p>Formule :C60H50O24Couleur et forme :SolidMasse moléculaire :1155.02GLP-1 receptor agonist 8
CAS :GLP-1 receptor agonist 8, potent for diabetes and obesity research, may also study NAFLD.Formule :C34H36ClFN6O4Couleur et forme :SolidMasse moléculaire :647.14{Val1}-Exendin-3/4
{Val1}- exendin-3/4 is the first n-terminal 1-28 residue of exendin-4 peptide.Formule :NADegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3241.7DETQ
CAS :DETQ enhances human D1 dopamine receptor signaling, EC50=5.8 nM, less effective in rats/mice, inactive on D5.Formule :C22H25Cl2NO3Couleur et forme :SolidMasse moléculaire :422.34Abediterol napadisylate
CAS :Abediterol napadisylate is a novel long-acting β2-agonist in persistent asthma that is efficacy, safe, and tolerable.Formule :C60H68F4N4O14S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1209.32[Des-His1,Glu9]-Glucagon amide
CAS :Glucagon blocker with pA2 of 7.2; no agonist effect. Boosts insulin; prevents glucagon-driven hyperglycemia in rabbits and diabetic rats.Formule :C148H221N41O47SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3358.68ONO-0300302
CAS :ONO-0300302: LPA1 antagonist, treats Benign Prostatic Hyperplasia, IC50 = 0.16 nM, reduces IUP in rats and dogs for 12h.Formule :C29H35NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :477.59[D-Trp34]-Neuropeptide Y
CAS :Potent NPY Y5 receptor agonist (pEC50 = 7.82); highly selective; induces hyperphagia, body weight gain; orally active.Formule :C196H289N55O56Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4311.77[Ala17]-MCH acetate
[Ala17]-MCH acetate is a selective ligand for MCHR1 with a Ki of 0.16 nM and Kd of 0.37 nM(Eu3+ chelate-labeled).Formule :C99H159N29O28S4Degré de pureté :98.92%Couleur et forme :SolidMasse moléculaire :2331.76AGN 191976
CAS :AGN 191976 is a novel thromboxane A2-mimetic.Formule :C21H32O6Couleur et forme :SolidMasse moléculaire :380.481Oxyntomodulin
CAS :GLP-1 analog modulates appetite, boosts metabolism, and curbs gastric acid. Increases cAMP, mildly stimulates glucagon receptor.Formule :C192H295N59O60SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4421.86σ1R-IN-1
σ1R-IN-1 ((R,R)-1a) is an effective σ-1R inhibitor with an IC50 of 110 nM. It shows promising potential for use in research related to neuropsychiatric disorders.Formule :C15H22N2Couleur et forme :SolidMasse moléculaire :230.35Tezusomant
CAS :Tezusomant is an antagonist of the growth hormone receptor (growth hormone receptor). It is being investigated for potential use in conditions like acromegaly, which are caused by excessive secretion of growth hormone.Formule :C120H171N23O32SCouleur et forme :SolidMasse moléculaire :2479.84MM 07
CAS :Biased agonist for apelin/G protein pathway, enhances eNOS and cell growth, reduces apoptosis, improves heart function, and dilates vessels.Formule :C67H106N22O14S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1539.9Adenosine 3'-monophosphate (sodium salt hydrate)
Adenosine 3'-monophosphate (sodium salt hydrate) (3'-AMP) is a nucleotide and cAMP-generating agonist that elevates cAMP levels in NG108-15 cells.Formule :C10H15N5NaO8PCouleur et forme :SolidMasse moléculaire :387.22B-Raf IN 14
CAS :B-Raf IN 14 is a BRAF inhibitor.Formule :C15H14BrN5O3SDegré de pureté :98.38%Couleur et forme :SolidMasse moléculaire :424.27Maridebart
CAS :Maridebart is a humanized IgG1-kappa monoclonal antibody that targets the GIPR (gastric inhibitory polypeptide receptor) [1].Couleur et forme :LiquidJKC363 TFA
JKC363 TFA is an MC4 receptor antagonist with 90x more affinity than MC3 (IC50: 0.5 nM vs 44.9 nM), blocks α-MSH's effect on TRH, and is anti-hyperalgesic.Formule :C71H93F3N19O18S2Couleur et forme :SolidMasse moléculaire :1620.73U 67827E
CAS :U 67827E is a long-lasting cholecystokinin agonist. It acts by decreases food intake.Formule :C53H68N10O17SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1149.24AA 497 HCl
CAS :AA 497, a beta-2 agonist, suppresses Ca spikes.Formule :C14H22ClNO3Couleur et forme :SolidMasse moléculaire :287.78Vapiprost
CAS :Vapiprost is an antagonist of the thromboxane receptor and a prostaglandin receptor.Formule :C30H39NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :477.64sGnRH-A
CAS :sGnRH-A, a salmon GnRH analog, boosts growth hormone and induces ovulation for artificial insemination.Formule :C64H83N17O12Couleur et forme :SolidMasse moléculaire :1282.45(p-Iodo-Phe7)-ACTH (4-10)
CAS :(p-Iodo-Phe7)-ACTH (4-10), an ACTH derivative and MC receptor antagonist, inhibits α-MSH-induced grooming in rats.Formule :C44H58IN13O10SCouleur et forme :SolidMasse moléculaire :1087.98α-MSH TFA
CAS :α-Melanocyte-stimulating hormone (α-MSH) is a 13-amino acid peptide hormone produced by post-translational processing of proopiomelanocortin (POMC) in theFormule :C79H110F3N21O21SCouleur et forme :SolidMasse moléculaire :1778.9313,14-dihydro Prostaglandin F2α
CAS :13,14-dihydro Prostaglandin F2α (13,14-dihydro PGF2α) is the analog of PGF2α which has no unsaturation in the lower side chain.Formule :C20H36O5Couleur et forme :SolidMasse moléculaire :356.503PF-9184
CAS :PF-9184 inhibits human mPGES-1 selectively, with an IC50 of 16.5 nM, and reduces IL-1β-stimulated PGE2 production in vitro.Formule :C21H14Cl2N2O4SDegré de pureté :97.43%Couleur et forme :SolidMasse moléculaire :461.32Mosliciguat
CAS :Mosliciguat is a guanylate cyclase activator.Formule :C41H36ClF3N2O5Couleur et forme :SolidMasse moléculaire :729.19Cafelkibart
Cafelkibart is a chimeric IgG1κ monoclonal antibody targeting CCR8, with HumanIgG1kappa, Isotype Control serving as its corresponding isotype control.Couleur et forme :Odour LiquidACTH (3-24) (human, bovine, mouse, ovine, porcine, rabbit, rat)
CAS :ACTH (3-24) is the fragment 3-24 of ACTH, used in disease research including cancer and immune disorders.Formule :C124H196N38O27SCouleur et forme :SolidMasse moléculaire :2683.19L-796,778 acetate
L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for sst1, sst2, sst4 and sst5, IC50 is >1000nM.Formule :C31H44N6O9Degré de pureté :98%Couleur et forme :SoildMasse moléculaire :644.72Exendin-4 (3-39)
CAS :<p>Exendin-4 (3-39) is a truncated peptide missing first 2 amino acids of Exendin-4, a potent GLP-1r agonist used in diabetes and HPA axis research.</p>Formule :C176H272N46O58SCouleur et forme :SolidMasse moléculaire :3992.44CKLF1-C27 TFA
CKLF1-C27 peptide activates ERK1/2 via CCR4, competes with CKLF1, promotes HUVEC growth, and has psoriasis research potential.Formule :C153H244F3N39O39Couleur et forme :SolidMasse moléculaire :3310.8LY83583
CAS :<p>LY83583 is a soluble guanylate cyclase competitive inhibitor with IC50 of 2 µM.</p>Formule :C15H10N2O2Degré de pureté :99.54% - 99.80%Couleur et forme :SolidMasse moléculaire :250.25Norisoboldine hydrochloride
CAS :<p>Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.</p>Formule :C18H20ClNO4Couleur et forme :SolidMasse moléculaire :349.81Ala-parafluoroPhe-Arg-Cha-Cit-Tyr-NH2
CAS :Ala-parafluoroPhe-Arg-Cha-Cit-Tyr-NH2 is a biologically active peptide functioning as a selective agonist for Protease Activated Receptor 1 (PAR-1), a subtypeFormule :C42H63FN12O8Couleur et forme :SolidMasse moléculaire :883.02NPS ALX Compound 4a hydrochloride(1:1)
NPS ALX Compound 4a hydrochloride(1:1) is a potent and selective 5-hydroxytryptamine6 (5-HT6) receptor antagonist, with an IC50 of 7.2 nM and a Ki of 0.2 nM.Formule :C25H26ClN3O2SDegré de pureté :99.84%Couleur et forme :SoildMasse moléculaire :468.01Ref: TM-T12262L1
1mg40,00€5mg88,00€10mg119,00€25mg198,00€50mg288,00€100mg393,00€200mg520,00€1mL*10mM (DMSO)97,00€PAR-2 (1-6) (human)
CAS :PAR-2 (1-6) (human) (SLIGKV), a peptide ligand, is a PAR-2 agonist [1] .Formule :C28H53N7O8Couleur et forme :SolidMasse moléculaire :615.76GLP-1R agonist 19
CAS :GLP-1R agonist 19 (M3190) is a potent, selective GLP-1 receptor agonist that demonstrates excellent plasma and liver microsomal stability, along with low hERG toxicity [1].Formule :C94H136FN21O25Couleur et forme :SolidMasse moléculaire :1979.21SphK1&2-IN-1
CAS :<p>SphK1&2-IN-1 is a sphingosine kinase inhibitor with anti-inflammatory, antitumor and hemostatic effects.</p>Formule :C14H14N2O3SDegré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :290.34Cagrilintide
CAS :<p>Cagrilintide: a long-acting amylin analogue, potential obesity treatment, reduces appetite and weight.</p>Formule :C194H312N54O59S2Couleur et forme :SolidMasse moléculaire :4409.01
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