GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.004 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(155 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(192 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(326 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(17 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
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5971 produits trouvés pour "GPCR/G-Protéine"
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Dabelotine, (R)-
CAS :Dabelotine, (R)- is the R-isomer of Dabelotine. Dabelotine is an adrenergic agonist used in the study of dementia.Formule :C15H22N2O2Couleur et forme :SolidMasse moléculaire :262.35RVD-Hpα
CAS :N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.Formule :C65H105N19O17Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1424.66Prostaglandin D2 methyl ester
CAS :PGD2: made in mast cells during allergic reactions, causes vasodilation and inhibits blood clots. PGD2 methyl ester is a similar, fat-soluble prodrug.Formule :C21H34O5Couleur et forme :SolidMasse moléculaire :366.498L-797,591
CAS :L-797,591 is a selective agonist of somatostatin receptor subtype 1.Formule :C38H49N5O2Couleur et forme :SolidMasse moléculaire :607.83Samelisant
CAS :Samelisant (SUVN-G3031), a selective H3 inverse agonist, Ki=8.7/9.8 nM in humans/rats, has anti-narcoleptic properties.Formule :C21H31N3O3Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :373.49Ref: TM-T9770
1mg105,00€2mg158,00€5mg260,00€10mg416,00€25mg687,00€50mg964,00€100mg1.288,00€500mg2.602,00€1mL*10mM (DMSO)268,00€VIP(Guinea pig)
CAS :Neuropeptide with many biological actionsFormule :C147H239N43O42S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3344.86LUF6096
CAS :LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically whileFormule :C22H21Cl2N3ODegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :414.33L-796,778
CAS :L-796,778 is an SST3 agonist and a selective ligand of SST3, which can increase the level of cAMP in the body.Formule :C29H40N6O7Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :584.66Ref: TM-T32511
1mg175,00€5mg404,00€10mg592,00€25mg888,00€50mg1.243,00€100mg1.701,00€500mg3.402,00€1mL*10mM (DMSO)522,00€Methylsolfonyl 25(S)-Δ7-dafachronic acid
Methylsulfonyl 25(S)-Δ7-dafachronic acid (compound 3) is a selective ssDAF-12 agonist with an IC50 value of 0.41 μM. It exhibits low cytotoxicity in HepG2 cells, with an IC50 value greater than 200 μM. Methylsulfonyl 25(S)-Δ7-dafachronic acid is applicable in the study of parasitic diseases.Formule :C28H45NO4SMasse moléculaire :491.30693Add 4743
CAS :Add 4743 is an analog of sitoglitazone, which is also a fat-forming agent.Formule :C18H23NO4SCouleur et forme :SolidMasse moléculaire :349.44[Des-Arg9]-Bradykinin
CAS :[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.Formule :C44H61N11O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :904.02Luseogliflozin hydrate
CAS :Luseogliflozin hydrate: SGLT2 inhibitor, IC50 2.26 nM, oral, for type 2 diabetes research.Formule :C23H32O7SCouleur et forme :SolidMasse moléculaire :452.56Vanicoside E
CAS :Vanicoside E is an antioxidant and antitumor agent. Vanicoside E inhibits L-Tyrosine and L-DOPA with IC 50 s of 45.23 μM and 189.96 μM, respectively [1] [2] .Formule :C53H52O22Couleur et forme :SolidMasse moléculaire :1040.97(+)-Oxypeucedanin methanolate
CAS :(+)-Oxypeucedanin methanolate (compound 9) is a natural compound that inhibits prostaglandin E2 production [1].Formule :C17H18O6Couleur et forme :SolidMasse moléculaire :318.32PG106 TFA
PG106 TFA is a potent hMC3 antagonist (IC50=210 nM), inactive at hMC4 (EC50=9900 nM) and hMC5 receptors.Formule :C53H70F3N13O11Couleur et forme :SolidMasse moléculaire :1122.2GHRF, porcine
CAS :GHRF, porcine, a growth hormone releasing factor (GHRF) peptide (porcine), binds to the growth hormone secretagogue receptor (GHSR), thereby inducing theFormule :C219H365N73O66SCouleur et forme :SolidMasse moléculaire :5108.76α-Helical CRF(9-41) TFA
α-Helical CRF(9-41) TFA acts as a competitive antagonist for the CRF2 receptor, possessing a binding constant (K B) of approximately 100 nM.Formule :C168H275F3N46O55S2Couleur et forme :SolidMasse moléculaire :3940.42Corazonin
CAS :Corazonin, a neuropeptide in insects, regulates caste identity and behavior, mainly in workers/foragers.Formule :C62H83N17O19Couleur et forme :SolidMasse moléculaire :1370.42dCNP
dCNP binds to NPR-B/C receptors (NPR-B/C receptor), initiating the cGMP signaling pathway and regulating vascular function. It exhibits anti-hypoxic effects by downregulating hypoxia-related genes such as HIF1α and HIF2α. Additionally, dCNP inhibits tumor stroma induction, demonstrating antifibrotic properties. It also enhances immune response by upregulating CTL, NK cells, and conventional type 1 dendritic cells in tumors.Formule :C141H248N38O36S3Couleur et forme :SolidMasse moléculaire :3147.918-Chloro caffeine
CAS :8-Chloro caffeine binds to adenosine receptors with a Ki of 30 µM. It enhances UV-induced chromosomal aberrations in the Cl-I type Chinese hamster embryo lung cells. 8-Chloro caffeine is a derivative of the methylxanthine alkaloid caffeine.Formule :C8H9ClN4O2Couleur et forme :SolidMasse moléculaire :228.64SAR441255
SAR441255 is a potent unimolecular peptide that acts as a GLP-1/GIP/GCG receptor triagonist, demonstrating balanced activation across all three target receptorsCouleur et forme :Odour SolidSubstance P (alligator)
CAS :Substance P from alligator: a neuropeptide with structure Arg-Pro-Arg-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2.Formule :C63H98N20O13SCouleur et forme :SolidMasse moléculaire :1375.64Amylin, amide, human TFA
Amylin, a 37-amino acid human hormone, moderates glucose regulation by reducing glucagon, delaying digestion, and increasing satiety.Formule :C167H262F3N51O57S2Couleur et forme :SolidMasse moléculaire :4017.3Pramlintide
CAS :Pramlintide, a polypeptide analog of human amylin, is an antidiabetic agent with antineoplastic properties in colorectal cancer.Couleur et forme :SolidCCZ01048 TFA
CCZ01048 TFA, α-MSH analog, binds MC1R with 0.31 nM affinity, internalizes in melanoma cells, and is stable for melanoma PET imaging.Formule :C73H106F3N21O18Couleur et forme :SolidMasse moléculaire :1622.75(Phe2,Orn8)-Oxytocin acetate
(Phe2,Orn8)-Oxytocin acetate: V1 agonist with EC50 of 280 nM for rabbit epididymis contractility.Formule :C44H69N13O13S2Couleur et forme :SolidMasse moléculaire :1052.23CART(55-102)(rat) TFA
Rat CART(55-102) TFA suppresses appetite, links to leptin/neuropeptide Y, and may induce anxiety/stress.Formule :C228H368F3N65O67S7Couleur et forme :SolidMasse moléculaire :5373.2DOTA-JR11
CAS :DOTA-JR11 is a somatostatin receptor 2 (SSTR2) antagonist that can be radiolabeled with 68Ga.Formule :C74H98ClN19O21S2Couleur et forme :SolidMasse moléculaire :1689.27Neuropeptide SF(mouse,rat) TFA
Neuropeptide SF TFA is a potent agonist for NPFF1 (Ki=48.4 nM) and NPFF2 (Ki=12.1 nM) and enhances ASIC3 current.Formule :C42H66F3N13O12Couleur et forme :SolidMasse moléculaire :1002.05Relamorelin TFA
CAS :Relamorelin (RM-131) TFA: ghrelin analog, GHSR agonist, 0.42 nM affinity, boosts growth hormone, enhances gastric emptying, potential in motility disorders.Formule :C45H51F3N8O7SCouleur et forme :SolidMasse moléculaire :905PAMP-12 (unmodified) (TFA)
PAMP-12 (unmodified) TFA, an endogenous peptide and potent MRGPRX2 (MrgX2) agonist (EC50=20-50 nM), induces hypotension by inhibiting catecholamine secretionFormule :C79H119F3N24O17Couleur et forme :SolidMasse moléculaire :1733.94PG-931 TFA
PG-931 TFA, a potent MC4 receptor agonist (IC50 0.58 nM), excels in selectivity and helps reverse hemorrhagic shock in vivo.Formule :C61H86F3N15O13Couleur et forme :SolidMasse moléculaire :1294.42Atilmotin
CAS :Atilmotin is a gastrointestinal agent for treating motility disorders.Formule :C86H135N20O19Couleur et forme :SolidMasse moléculaire :1753.146MM 419447
CAS :MM 419447, a linaclotide metabolite, is a guanylate cyclase-C agonist showing potential in IBS-C research.Formule :C50H70N14O19S6Couleur et forme :SolidMasse moléculaire :1363.55(D-Phe12,Nle21,38,α-Me-Leu37)-CRF (12-41) (human, rat)
CAS :(D-Phe12,Nle21,38,α-Me-Leu37)-CRF (12-41) (human, rat) is a corticotropin-releasing factor (CRF) antagonist known to counteract the inhibitory effects of IL-1aFormule :C159H267N49O43Couleur et forme :SolidMasse moléculaire :3553.12[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)
CAS :'[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)' is a selective NK2R agonist with prokinetic activity for smooth muscle studies.Formule :C39H64N8O10Couleur et forme :SolidMasse moléculaire :804.97Neuropeptide Y (2-36) (porcine)
CAS :Porcine Neuropeptide Y (2-36) is 97.14% similar to rat/human, an agonist for Y5, Y2, Y1 receptors, used in obesity research.Formule :C181H278N54O55Couleur et forme :SolidMasse moléculaire :4090.47Prepro-ANF (56-92), human
CAS :Human prepro-ANF (56-92) activates renal guanylate cyclase and boosts its activity.Formule :C173H270N44O57Couleur et forme :SolidMasse moléculaire :3878.26Protease-Activated Receptor-1, PAR-1 Agonist TFA
PAR-1 Agonist TFA: Selective peptide, mimics thrombin, activates PAR-1 receptor.Couleur et forme :Liquid(Trp7,β-Ala8)-Neurokinin A (4-10)
CAS :(Trp7,β-Ala8)-Neurokinin A (4-10) is a potent neurokinin-3 (NK3) antagonist [1] .Formule :C41H57N9O10SCouleur et forme :SolidMasse moléculaire :868.01Cyclosomatostatin TFA
Cyclosomatostatin TFA blocks SST receptor, reduces CRC cell growth, ALDH+ size, and sphere-formation.Formule :C46H58F3N7O8Couleur et forme :SolidMasse moléculaire :893.99Sauvagine TFA
Sauvagine TFA: frog-derived, 40-amino-acid CRF agonist; stimulates ACTH release, affects diuresis, cardiovascular system, endocrine glands.Formule :C204H347F3N56O65S1Couleur et forme :SolidMasse moléculaire :4713.33L-797,591 hydrochloride
L-797,591 HCl activates SSTR1, boosts p-ERK5 with AG1478, and enhances p38 phosphorylation, reversible by AG1478.Formule :C38H50ClN5O2Degré de pureté :98.65% - >99.99%Couleur et forme :SoildMasse moléculaire :644.30Galanin-Like Peptide (rat)
CAS :Galanin-Like Peptide (rat), a neuropeptide comprising 60 amino acids, plays a crucial role in regulating feeding, body weight, and energy metabolism [1].Formule :C288H461N87O83SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :6502.34Jmv 176
CAS :Jmv 176 is a CCK agonist when first given and becomes a cholecystokinin antagonist after 3-4 hours.Formule :C53H70N8O15SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1091.24GI-560192
CAS :GI-560192 (RL-0070933), a potent smo modulator, EC50: 0.02µM; affects smoothened in cilia via hedgehog signaling.Formule :C20H16N2O2Degré de pureté :99.53%Couleur et forme :SoildMasse moléculaire :316.35Ref: TM-T64351
1mg85,00€5mg170,00€10mg250,00€25mg371,00€50mg522,00€100mg712,00€200mg954,00€1mL*10mM (DMSO)170,00€PSB-1114 triethylamine
PSB-1114 triethylamine is a potent, enzymatically stable, P2Y2 receptor agonist with a 134 nM EC50, exhibiting greater than 50-fold selectivity over P2Y4 (EC50Formule :C10H15F2N3O13P3S·xC6H15NDegré de pureté :98%Couleur et forme :SolidBradykinin (1-7)
CAS :Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.Formule :C35H52N10O9Degré de pureté :98%Couleur et forme :White Lyophilized PowderMasse moléculaire :756.85α-CGRP (mouse, rat) TFA
α-CGRP (mouse, rat) TFA, a neuropeptide belonging to the calcitonin gene-related peptide (CGRP) family, is predominantly located at neuromuscular junctions andFormule :C162H262N50O52S2·C2HF3O2Degré de pureté :98%Couleur et forme :SolidLinaclotide acetate
CAS :Linaclotide acetate, an oral guanylate cyclase C agonist with 14 amino acids, treats constipation-predominant IBS and chronic constipation.
Formule :C61H83N15O23S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1586.79Heterobivalent ligand-1
Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.Formule :C86H115FN16O21Couleur et forme :SolidMasse moléculaire :1727.93Adrenomedullin (16-31), human
CAS :Adrenomedullin (16-31), human is amino acid residues 16-31 fragment of human adrenomedullin (hADM).Formule :C82H129N25O21S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1865.19Chir 2279
CAS :CHIR 2279, a peptoid trimer, binds alpha 1-adrenoceptors, blocking epinephrine effects in dogs (pseudo pA2 6.86).Formule :C34H36N4O4Couleur et forme :SolidMasse moléculaire :564.67YM 218
CAS :YM 218 is a novel, potent, selective antagonist of nonpeptide vasopressin V1A receptor.Formule :C35H38F2N4O4Couleur et forme :SolidMasse moléculaire :616.7Pneumadin, rat
CAS :Rat Pneumadin (PNM), a decapeptide, stimulates AVP release, exerting strong antidiuretic effects in animals with an active AVP system.Formule :C47H74N12O15Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1047.178NN1213
NN1213 (Peptide 21) is a long-acting human amylin peptide analogue that functions as a selective amylin receptor agonist. It has an EC50 of 0.177 nM for hAMY3R and 0.262 nM for rAMY3R. In both rat and dog models, NN1213 significantly reduces appetite and is utilized in anti-obesity research.Couleur et forme :Odour SolidOno 3708
CAS :Ono-3708 is a potent antagonist of the thromboxane A2/prostaglandin endoperoxide receptor in vitro and in vivo.Formule :C23H37NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :391.54RWJ 676070
CAS :RWJ 676070 is an antagonist of vasopressin V1A/V2 receptor.Formule :C30H26ClFN2O5Couleur et forme :SolidMasse moléculaire :548.9917-phenoxy trinor Prostaglandin F2α ethyl amide
CAS :Prostaglandin F2α (PGF2α), acting through the FP receptor, causes smooth muscle contraction and exhibits potent luteolytic activity.Formule :C25H37NO5Couleur et forme :SolidMasse moléculaire :431.573ZM 253270
CAS :ZM 253270 is an nonpeptide neurokinin A antagonist.Formule :C22H26ClN7O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :471.95Emoghrelin
CAS :Emoghrelin, extracted from Heshouwu (Polygonum multiflorum), promotes the secretion of growth hormone by activating the ghrelin receptor [1].Formule :C24H22O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :518.42FR190997
CAS :FR190997 is an agonist of bradykinin B2 receptor.Formule :C37H33Cl2N5O5Couleur et forme :SolidMasse moléculaire :698.59γ-Glu-Abu TFA
Gamma-Glu-AbuTFA is the TFA salt form of Gamma-Glu-Abu. This compound acts as an agonist for the calcium sensing receptor (CaSR), activating CaSR in HEK-293 cells with an EC50 of 0.21 μM.Formule :C11H17F3N2O7Couleur et forme :SolidMasse moléculaire :346.26TGR5 agonist 1
Compound 18 (TGR5 agonist 1) is a potent agonist of TGR5, exhibiting an EC50 value of 0.31 µM [1].Formule :C28H48NNaO6SCouleur et forme :SolidMasse moléculaire :549.74Synephrine hemitartrate
CAS :Synephrine hemitartrate, an alkaloid from Citrus aurantium, is a sympathomimetic for weight loss, with α and β-adrenergic action.Formule :C9H13NO2C4H6O6Couleur et forme :SolidMasse moléculaire :242.26GLP-1R Antagonist 1
CAS :GLP-1R Antagonist 1 is an orally active, CNS penetrant and non-competitive glucagon-like peptide 1 receptor (GLP-1R) antagonist (IC50: 650 nM).Formule :C16H11ClF6N4O2Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :440.73Carbocyclic Thromboxane A2
CAS :Carbocyclic Thromboxane A2 can be used in related research in the field of life sciences. Its product number is T36548 and CAS number is 74034-56-3.Formule :C22H36O3Couleur et forme :SolidMasse moléculaire :348.527ACTH (22-39)
CAS :ACTH (22-39) is an adrenocorticotropic hormone (ACTH) fragment and it is the 22-39 sequence of ACTH.Formule :C90H125N19O32Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1985.06Alverine hydrochloride
CAS :Alverine hydrochloride is a parasympatholytic.Formule :C20H28ClNCouleur et forme :SolidMasse moléculaire :317.9Corticotropin-releasing factor (human) acetate
Corticotropin-releasing factor (human) acetate stimulates to synthesize and secret adrenocorticotropin in the anterior pituitary.Degré de pureté :98.30%Couleur et forme :LiquidFezolamine
CAS :Fezolamine: a new, non-tricyclic, oral antidepressant, selectively inhibits norepinephrine uptake over serotonin or dopamine.Formule :C20H23N3Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :305.42LTB4-IN-2
LTB4-IN-2 (Compound 6x) is a selective inhibitor of Leukotriene B4 (LTB4), acting by specifically targeting the 5-Lipoxygenase-activating protein (FLAP) with anFormule :C24H17N5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :439.568-iso Prostaglandin E2 isopropyl ester
CAS :8-iso PGE2 isopropyl ester: lipophilic, hydrolyzes to acid in vivo, used as prodrug, less active than parent acid.Formule :C23H38O5Couleur et forme :SolidMasse moléculaire :394.54Brain Natriuretic Peptide-45, mouse
CAS :Mouse BNP-45, a heart-derived peptide, lowers blood pressure and increases sodium excretion.TH023
TH023 is an inhibitor of the TLR4 signaling pathway, specifically targeting the formation of TLR4 homodimers. In HEK-Blue hTLR4 cells, TH023 suppresses the secretion of embryonic alkaline phosphatase with an IC50 of 0.354 μM and inhibits NO expression in RAW264.7 cells, with an IC50 of 1.61 μM. Additionally, TH023 inhibits the activation of NF-κB and reduces the nuclear translocation of NF-κB p65. The compound demonstrates anti-inflammatory effects in a mouse model of LPS-induced acute sepsis and improves lung injury in mice.Formule :C22H21ClF2N4OCouleur et forme :SolidMasse moléculaire :430.88Apelin-12 acetate
Apelin-12 acetate possesses a high affinity to orphan receptor APJ receptor.Formule :C66H107N21O16SDegré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :1482.75Ref: TM-T39823L
1mg128,00€5mg172,00€10mg269,00€25mg429,00€50mg610,00€100mg820,00€1mL*10mM (DMSO)430,00€LRGILS-NH2
CAS :LRGILS-NH2, reverse sequence of SLIGRL-NH2, is a control peptide for PAR2, affecting gut transit.Formule :C29H56N10O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :656.82L-770644 dihydrochloride
CAS :L-770644 dihydrochloride is a potent and selective agonist of the human beta3 adrenergic receptor.Formule :C30H38ClN7O4SCouleur et forme :SolidMasse moléculaire :628.19c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm
CAS :c(Bua-Cpa-Thi-Val-Asn-Cys)-Pro-Agm: potent, selective V2R agonist; EC50: 0.25 nM (hV2R), 0.05 nM (rV2R).Formule :C47H69ClN12O9S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1045.71Exendin-3/4 (59-86)
Exendin-3/4 (59-86) is a Exendin-4 peptide derivative.Formule :NADegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3055.49Ro 25-1553
CAS :Ro 25-1553 is a 31-amino acid analog of vasoactive intestinal peptide (VIP) that functions as an agonist for the VIP2 receptor (VPAC2 receptor). In guinea pig models, Ro 25-1553 exhibits bronchodilator effects on tracheal smooth muscle contraction induced by neural stimuli or Carbachol.Formule :C160H258N46O46Couleur et forme :SolidMasse moléculaire :3562.04(Hyp³)-Bradykinin acetate
(Hyp³)-Bradykinin acetate is an agonist of bradykinin B2 receptor and stimulates inositol phosphate production in cultured human fibroblasts.Formule :C52H77N15O14Degré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :1136.26Clotizolam
CAS :Clotizolam is a thienotriazolodiazepine derivative with PAF antagonistic properties, exhibiting sedative, anxiolytic, anticonvulsant, and muscle relaxant effects.Formule :C15H10Cl2N4SCouleur et forme :SolidMasse moléculaire :349.24Wy 41747
CAS :Wy 41747 is a long-acting somatostatin analogue utilized in research of diabetes mellitus [1].Formule :C73H92N18O16S2Masse moléculaire :1541.75Desmethyl Mirtazapine (hydrochloride)
CAS :Desmethyl mirtazapine is a metabolite of the antidepressant mirtazapine.1It is formed from mirtazapine by the cytochrome P450 (CYP) isoform CYP3A4.Formule :C16H18ClN3Couleur et forme :SolidMasse moléculaire :287.79Berobenatide
CAS :Berobenatide is a glucagon-like peptide-1 (GLP-1) receptor agonist.Couleur et forme :SolidFFN246
CAS :FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation andFormule :C15H13FN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :256.27Cholecystokinin Octapeptide, desulfated
CAS :Cholecystokinin Octapeptide, desulfated (CCK Octapeptide, non-sulfated) is an octapeptide composed of 8 amino acids from cholecystokinin-8.Formule :C49H62N10O13S2Degré de pureté :97.12%Couleur et forme :SolidMasse moléculaire :1063.21GLP-1R agonist 15
CAS :GLP-1R agonist 15 (Compound 101) is a GLP-1 receptor agonist [1] .Formule :C46H47FN8O7SCouleur et forme :SolidMasse moléculaire :874.98Apigenin 6,8-di-C-α-L-arabinopyranoside
CAS :Apigenin 6,8-di-C-alpha-L-arabinopyranoside is a useful organic compound for research related to life sciences.Formule :C25H26O13Couleur et forme :SolidMasse moléculaire :534.47BM213 acetate
BM213 acetate is a selective C5aR1 agonist with antitumor activity that induces C5aR1-mediated calcium mobilization and pERK1/2 signaling.
Formule :C45H74N12O12Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :975.14D-Epinephrine
CAS :D-Epinephrine: a hormone and drug, boosts heart rate, muscle blood flow, pupil size, and sugar levels in stress responses.
Formule :C9H13NO3Couleur et forme :SolidMasse moléculaire :183.2[Tyr3]Octreotate
CAS :[Tyr3]Octreotate is a long peptide compound containing 8 amino acids and is a functional DOTA chelating agent with covalent bonds.Formule :C49H64N10O12S2Degré de pureté :98.21%Couleur et forme :SoildMasse moléculaire :1049.22Cortistatin-14
CAS :Cortistatin-14, a neuropeptide structurally similar to growth inhibitor-14, is used to study sepsis-induced cognitive impairment.Formule :C81H114N20O18S2Degré de pureté :98.06% - 98.23%Couleur et forme :SolidMasse moléculaire :1720.03α-helical CRF 9-41 acetate
α-helical CRF 9-41 acetate is a competitive antagonist of CRF2 (KB = 100 nM) and a partial agonist of CRF1 (EC50 = 140 nM).
Degré de pureté :96.60%Couleur et forme :SolidMasse moléculaire :#N/ARef: TM-TP2048L
1mg208,00€5mg500,00€10mg672,00€25mg1.017,00€50mg1.359,00€100mg1.853,00€200mg2.498,00€MLS1082
CAS :MLS1082 is a D1-like dopamine receptor (D1R) orthosteric modulatothat stimulates G-protein signaling upon dopamine activation for neurodegenerative disorders.Formule :C24H23N3O2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :385.46Leukotriene B5
CAS :LTB5, an eicosapentaenoic acid metabolite via 5-LO, has varied bioactivities and enhances bullfrog lung strip contraction.Formule :C20H30O4Couleur et forme :SolidMasse moléculaire :334.4561-(4-Fluorobenzyl)-1H-indazole-3-carboxylic acid
CAS :1-(4-Fluorobenzyl)-1H-indazole-3-carboxylic acid (Compound 31) is a metabolite of AB-FUBINACA. It acts as an MRGPRX4 antagonist with an IC50 greater than 2.5 μM.Formule :C15H11FN2O2Couleur et forme :SolidMasse moléculaire :270.26AC-264613
CAS :AC-264613 is an agonist of the GPCR protease-activated receptor 2 (PAR2). AC-264613 suppresses interferon regulatory factor 5.Formule :C19H18BrN3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :400.28sGC activator 2
sGC activator 2 (Compound 16a) acts as an activator of soluble guanylate cyclase (sGC), enhancing the production of cGMP and exhibiting vasoprotective and anti-inflammatory properties.Formule :C21H21FN8O3Couleur et forme :SolidMasse moléculaire :452.44
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