GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.022 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(194 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5985 produits trouvés pour "GPCR/G-Protéine"
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Atenolol
CAS :Atenolol (Tenormin) is a selective β1 receptor antagonist.Formule :C14H22N2O3Degré de pureté :99.07% - 99.95%Couleur et forme :White Crystalline Powder SolidMasse moléculaire :266.34Tecastemizole
CAS :Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.Formule :C19H21FN4Degré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :324.4Ref: TM-T26253
1mg54,00€5mg118,00€1mL*10mM (DMSO)131,00€10mg168,00€25mg288,00€50mg414,00€100mg583,00€500mg1.161,00€AMK (hydrochloride)
CAS :AMK, a melatonin metabolite, scavenges oxygen, inhibits prostaglandin production, reduces lipid peroxidation, and affects Parkinson's in mouse studies.Formule :C12H17ClN2O3Couleur et forme :SolidMasse moléculaire :272.73Dapoxetine
CAS :Dapoxetine (Dapoxetina) is a selective serotonin reuptake inhibitor, for the treatment of premature ejaculation.Formule :C21H23NODegré de pureté :99.73%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :305.42PAMP-12(human, porcine) TFA
PAMP-12(human, porcine) TFA, a significant constituent of immunoreactive (ir)-PAMP, derives from the adrenomedullin precursor and functions as a potentCouleur et forme :Odour Solid(D-His(Bzl)6)-LHRH (1-7) (free acid)
CAS :(D-His(Bzl)6)-LHRH (1-7) free acid is a synthetic peptide derived from luteinizing hormone-releasing hormone (LHRH). It achieves enhanced stability and biological activity through the introduction of non-natural amino acid residues at specific positions within the LHRH molecule. This modification extends the drug's half-life in the body, reduces its rate of rapid metabolism and clearance, and subsequently increases its efficacy in inhibiting cell proliferation.Formule :C53H62N12O11Masse moléculaire :1043.1316,16-dimethyl Prostaglandin E1
CAS :16,16-dimethyl Prostaglandin E1 is a PGE1 (T1626) analog that induces bronchoconstriction and vascular smooth muscle contraction and inhibits indomethacin-Formule :C22H38O5Couleur et forme :SolidMasse moléculaire :382.541Neuropeptide W-23 (human) (TFA)
Neuropeptide W-23 (human) (NPW-23) TFA, representing the active form of Neuropeptide W, functions as an endogenous agonist for both NPBW1 (GPR7) and NPBW2 (GPR8Couleur et forme :Odour SolidAcetyl-(D-Arg2)-GRF (1-29) amide (human)
CAS :Acetyl-(D-Arg2)-GRF (1-29) amide (human) serves as an antagonist to growth hormone-releasing factor (GRF) and inhibits growth hormone (GH) secretion, withFormule :C154H255N47O43SMasse moléculaire :3485.03MRS8209
MRS8209 is an antagonist of the serotonin receptor (serotonin receptor), with a Ki value of 4.27 nM specifically for 5-HT2BR. It provides protective effects on pulmonary airway opening pressure (PAO) and is applicable in pulmonary fibrosis studies.Formule :C17H19IN6O2Couleur et forme :SolidMasse moléculaire :466.276LH-RH (4-10)
CAS :LH-RH (4-10), a heptapeptide from LHRH degradation, is made in macrophages and type II pneumocytes.Formule :C33H53N11O9Couleur et forme :SolidMasse moléculaire :747.84VIP(6-28)(human, rat, porcine, bovine)
CAS :VIP(6-28) blocks VIP-induced cAMP signaling in humans, rats, pigs, and cows.Formule :C126H207N37O34SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :2816.28Lamprey LH-RH I
CAS :Lamprey LH-RH I triggers ovulation and raises steroid levels in lamprey, inactive in other species.Formule :C58H79N15O15Couleur et forme :SolidMasse moléculaire :1226.34AP 811
CAS :AP 811: Selective NPR3 antagonist, Ki of 0.48 nM, >20,000x selective over NPR1, blocks ANP-induced pump stimulation.Formule :C46H66N12O8Couleur et forme :SolidMasse moléculaire :915.11[Lys8, Lys9]-Neurotensin (8-13)
CAS :[JMV438] is a Neurotensin analog, analgesic via NTS1/NTS2 activation, with K i of 0.33 nM (hNTS1) and 0.95 nM (hNTS2).Formule :C38H64N8O8Masse moléculaire :760.978A11
CAS :A11 (ANXA1-derived 11 amino acid–long peptide) serves as an inhibitor of the ANXA1-EphA2 interaction, reducing ANXA1 attachment to EphA2 while promoting the association of Cbl (an E3 ubiquitin ligase of EphA2) with EphA2. This peptide also effectively lowers EphA2 levels, greatly enhances EphA2 ubiquitination, and stimulates EphA2 internalization along with the colocalization of EphA2 and Cbl in nasopharyngeal carcinoma (NPC) cells. Moreover, A11 curtails NPC cell proliferation, migration, and invasion, and it suppresses angiogenesis.Formule :C53H88N14O19Couleur et forme :SolidMasse moléculaire :1225.35DD202-114
CAS :DD202-114 is an effective and selective agonist of GLP1R. It promotes the accumulation of cAMP, reduces blood glucose levels, and decreases food intake. Additionally, DD202-114 holds potential for research in type 2 diabetes mellitus (T2DM) and obesity studies.Formule :C33H35FN4O5Couleur et forme :SolidMasse moléculaire :586.65Biotinyl-neuropeptide W-23 (human)
CAS :Biotinyl-neuropeptide W-23 (human) is a biotinylated form of neuropeptide W-23 (human), which functions as an agonist for the NPBW1 (GPR7) and NPBW2 (GPR8)Formule :C129H197N37O30S2Couleur et forme :SolidMasse moléculaire :2810.3Contulakin G
CAS :Contulakin G: O-glycosylated neurotensin, weak neurotensin receptor agonist, strong antinociceptive.Formule :C88H140N20O37Masse moléculaire :2070.17PHI-27 (porcine)
CAS :PHI-27 (porcine) is a porcine-derived peptide consisting of 27 amino acids, utilized in the identification of peptide hormones and other bioactive peptides [1].Formule :C136H216N36O40Couleur et forme :SolidMasse moléculaire :2995.39(±)-Clopidogrel (hydrochloride)
CAS :Clopidogrel is an antithrombic compound whose active metabolite is a selective, irreversible antagonist of the platelet purinergic P2Y12 receptor (IC50 = 100 nMFormule :C16H17Cl2NO2SCouleur et forme :SolidMasse moléculaire :358.28MR 409
CAS :MR 409, a selective growth hormone-releasing hormone (GHRH) agonist, exhibits notable neuroprotective properties by augmenting endogenous neurogenesis inFormule :C153H252N44O43Couleur et forme :SolidMasse moléculaire :3395.9115(S)-Latanoprost
CAS :15(S)-Latanoprost, a latanoprost analog with inverted hydroxyl at C-15, has an IC50 of 24 nM and reduces IOP by 1 mmHg at 3 μg.Formule :C26H40O5Couleur et forme :SolidMasse moléculaire :432.59Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP (1-7)-GRF (8-27)
CAS :Acetyl-(D-Phe2,Lys15,Arg16,Leu27)-VIP(1-7)-GRF(8-27) is a selective antagonist [1] for the vasoactive intestinal peptide 1 (VIP 1) receptor.Formule :C150H246N44O38Couleur et forme :SolidMasse moléculaire :3273.83[Tyr1]-Somatostatin-14
CAS :[Tyr1]-Somatostatin-14 could binds to SSTR2.Formule :C82H108N18O20S2Masse moléculaire :1729.99Y4R agonist-1
CAS :Y4R Agonist-1 is a potent agonist of the Y4 receptor, exhibiting a K_i (inhibition constant) value of 0.048 nM.Formule :C51H80N18O11Masse moléculaire :1121.29N-Methyl-2-phenylpropan-1-amine hydrochloride
CAS :N-Methyl-2-phenylpropan-1-amine hydrochloride is an analogue of β-methylphenethylamine (BMPEA) and demonstrates neurotransmitter-releasing properties in experiments involving NET and DAT.Formule :C10H16ClNCouleur et forme :SolidMasse moléculaire :185.69[D-Phe2,6, Pro3]-LH-RH
CAS :[D-Phe2,6, Pro3]-LH-RH is a potent antagonist of luteinizing hormone-releasing hormone (LHRH).Formule :C59H80N14O13Couleur et forme :SolidMasse moléculaire :1193.35(Leu31,Pro34)-Peptide YY (human)
CAS :(Leu31,Pro34)-Peptide YY (human) is a derivative of Peptide YY, acting as a potent and selective Y1 receptor agonist with a dissociation constant (KD) of 1.0 nMFormule :C195H296N54O56Couleur et forme :SolidMasse moléculaire :4292.75CCK (27-33) (non-sulfated)
CAS :CCK (27-33), a non-sulfated peptide, inhibits [3H]naloxone binding (IC50=4uM) and guinea pig ileum contractions (IC50=17uM), reversed by naloxone.Formule :C45H57N9O10S2Couleur et forme :SolidMasse moléculaire :948.12Oxopurpureine
CAS :Oxopurpureine, classified as an oxoaporphine compound, functions to inhibit plant pathogens.Formule :C21H19NO6Couleur et forme :SolidMasse moléculaire :381.38BNP (1-21), Pro (Human)
CAS :BNP (1-21), Pro (Human) is a 21-amino acid peptide and a form of B-Type Natriuretic Peptide (BNP), a cardiac natriuretic hormone.Formule :C89H144N28O35Masse moléculaire :2166.26Cholecystokinin
CAS :Cholecystokinin, a peptide hormone, functions as a hunger suppressant by inhibiting food intake and promoting the digestion of fat and protein, and is employedCouleur et forme :SolidBrain Natriuretic Peptide-45, rat TFA
Brain Natriuretic Peptide-45, rat TFA (BNP-45, rat TFA) is an isoform of rat brain natriuretic peptide extracted from rat heart, exhibiting significantCouleur et forme :Odour Solid[D-Pro4,D-Trp7,9,10] Substance P (4-11)
CAS :[D-Pro4,D-Trp7,9,10] Substance P (4-11) serves as a potent antagonist of the tachykinin family of neuropeptides [1].Formule :C62H74N14O10SMasse moléculaire :1207.4Exendin-3
CAS :Exendin-3, a peptide from Gila monster venom, stimulates pancreatic secretion and belongs to the glucagon family.Formule :C184H282N50O61SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4202.57Antidepressant agent 10
CAS :Compound PDK0386, with CAS No. 87691-87-0, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0386 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formule :C11H13N3SMasse moléculaire :219.3064-Methylamphetamine hydrochloride
CAS :4-Methylamphetamine hydrochloride is a 5-HT1A receptor agonist that induces a decrease in body temperature in rats by binding to the 5-HT1A receptor. Additionally, it increases the extracellular levels of neurotransmitters norepinephrine (NE), dopamine (DA), and serotonin (5-HT) by affecting their transporters. 4-Methylamphetamine hydrochloride is applicable in the study of neurological disorders.Formule :C10H16ClNCouleur et forme :SolidMasse moléculaire :185.69Bosentan-d4
CAS :Bosentan-d4: deuterium version of Bosentan, competitive ET A/B antagonist, Ki: 4.7nM (ET A), 95nM (ET B) in human SMC.Formule :C27H25D4N5O6SCouleur et forme :SolidMasse moléculaire :555.64Prostaglandin B1
CAS :Prostaglandin B1 (PGB1), a metabolite of Prostaglandin E1, acts as a prostanoid receptor ligand [1] [2].Formule :C20H32O4Masse moléculaire :336.47Prolactin-Releasing Peptide (1-31), bovine
Prolactin-Releasing Peptide (1-31), bovine, is a fragment of prolactin-releasing peptide (PrRP).Formule :C44H80N14O15Masse moléculaire :1044.59276Thrombostatin cont-1
CAS :Thrombostatin cont-1, an analogue of the bradykinin metabolite thrombostatin, has been shown to reduce platelet activation in the canine carotid arteryFormule :C87H142N34O29S2Masse moléculaire :2192.4Endothelin 1 (swine, human) (TFA)
CAS :Synthetic human/swine Endothelin 1 (TFA) peptide; a potent vasoconstrictor acting on ET A and ET B receptors.Formule :C111H160F3N25O34S5Masse moléculaire :2605.93ent-8-iso Prostaglandin F2α
CAS :ent-8-iso Prostaglandin F2α is a potent vasoconstrictor of porcine retinal and cerebral microvessels with EC50 values of 30.6 and 53.5 nM, respectively.Formule :C20H34O5Couleur et forme :SolidMasse moléculaire :354.487Gastrin I (1-14), human TFA
Gastrin I (1-14), human TFA is 1-14 fragment of human gastrin I peptide.Formule :C81H101N16F3O29Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1819.75Anaritide
CAS :Anaritide, a synthetic form of atrial natriuretic peptide (ANP) composed of 25 amino acids, enhances the glomerular filtration rate by dilating afferent arterioles and constricting efferent arterioles. It is utilized for studying its effects on patients with acute tubular necrosis, with a focus on improving dialysis-free survival rates.Formule :C112H175N39O35S3Couleur et forme :SolidMasse moléculaire :2724.02LCKLSL
CAS :LCKLSL, an N-terminal hexapeptide, inhibits AnxA2 and tPA binding, reduces plasmin, and exhibits anti-angiogenic effects.Formule :C30H57N7O8SMasse moléculaire :675.89ANP (1-30), frog
CAS :ANP (1-30), frog, a peptide fragment sourced from atrial natriuretic peptide of frog origin, exhibits natriuretic, diuretic, and vasorelaxant properties.Formule :C131H217N49O41S4Couleur et forme :SolidMasse moléculaire :3262.69Uperolein
CAS :Uperolein, a physalaemin-like endecapeptide derived from the skin of Uperoleia rugosa and Uperoleia marmorata, exhibits spasmodic activity on theFormule :C57H79N13O16SMasse moléculaire :1234.38[D-His26]-Neuropeptide Y, human, rat
[D-His26]-Neuropeptide Y, human, rat is a synthetic variant of neuropeptide Y (NPY). This compound acts as a Y1R agonist and may help prevent the development of anxiety, social disorders, and depressive symptoms. It has potential as an early intervention treatment for post-traumatic stress responses.Formule :C180H276N54O55SMasse moléculaire :4106.01808Pindolol
CAS :Pindolol is an effective, non-selective, and specific beta-receptor blocker that acts as a partial beta-adrenergic receptor agonist and a localized 5-HT1A receptor antagonist (Ki=33nM). Pindolol has intrinsic sympathetic activity (ISA) and is primarily used to treat high blood pressure and certain heart conditions. Exhaustion.Formule :C14H20N2O2Couleur et forme :Crystals From Ethanol SolidMasse moléculaire :248.32Neurokinin A TFA
CAS :Neurokinin A TFA (NKA TFA) is a neuropeptide within the neurokinin family, serving as the endogenous ligand and agonist for the NK-2 (Neurokinin 2) receptor.Formule :C52H81F3N14O16SDegré de pureté :98.704%Couleur et forme :SolidMasse moléculaire :1247.34Dabelotine, (S)-
CAS :Dabelotine, (S)- is the S-isomer of Dabelotine. Dabelotine is an adrenergic agonist used in the study of dementia.Formule :C15H22N2O2Couleur et forme :SolidMasse moléculaire :262.35Pegapamodutide
CAS :Pegapamodutide (LY-2944876) is a dual glucagon-GLP-1 receptor agonist utilized in research concerning type 2 diabetes and obesity [1].Couleur et forme :Solid(D-Phe5,Cys6,11,N-Me-D-Trp8)-Somatostatin-14 (5-12) amide
CAS :Somatostatin analog (Compound 4) with Kd: SSTR5-0.61nM, SSTR3-11.05nM, SSTR2-23.5nM, SSTR1-1.2µM, SSTR4->1µM.Formule :C50H67N11O10S2Masse moléculaire :1046.26[D-p-Cl-Phe6,Leu17]-VIP TFA
[D-p-Cl-Phe6,Leu17]-VIP TFA acts as a competitive and selective antagonist of the vasoactive intestinal peptide (VIP) receptor, exhibiting an IC50 of 125.8 nM.Formule :C150H240F3ClN44O44Couleur et forme :SolidMasse moléculaire :3456.22(Asp28)-Glucagon (1-29) (human, rat, porcine)
CAS :"(Asp28)-Glucagon (1-29) (human, rat, porcine)" is an analog of glucagon with an aspartic acid (Asp) substitution at position 28, notably enhancing its aqueousFormule :C153H224N42O50SCouleur et forme :SolidMasse moléculaire :3483.73Liraglutide acetate
CAS :Liraglutide acetate is the acetate salt form of Liraglutide, which is a glucagon-like peptide-1 (GLP-1) receptor agonist, utilized in the study of type 2 diabetes.Formule :C172H265N43O51·xC2H4O2Couleur et forme :SolidMasse moléculaire :3751.20 (free base)Methylsolfonyl 25(S)-Δ7-dafachronic acid
Methylsulfonyl 25(S)-Δ7-dafachronic acid (compound 3) is a selective ssDAF-12 agonist with an IC50 value of 0.41 μM. It exhibits low cytotoxicity in HepG2 cells, with an IC50 value greater than 200 μM. Methylsulfonyl 25(S)-Δ7-dafachronic acid is applicable in the study of parasitic diseases.Formule :C28H45NO4SMasse moléculaire :491.30693Aldioxa
CAS :Aldioxa is a Gastrointestinal Agent.Formule :C4H7AlN4O5Couleur et forme :SolidMasse moléculaire :218.10Urodilatin
CAS :Urodilatin, an analogue of ANF-(99-126), serves as a diuretic-natriuretic regulatory peptide with applications in the study of acute renal failure, congestiveCouleur et forme :Solid5-trans Latanoprost
CAS :Latanoprost, an F-series prostaglandin analog for ocular hypertension, has a 5-trans isomer used as an analytical standard.Formule :C26H40O5Couleur et forme :SolidMasse moléculaire :432.601Vensemaglutide
CAS :Vensemaglutide is a glucagon-like peptide-1 (GLP-1) receptor agonist, utilized in research related to diabetes or other metabolic disorders.Formule :C214H337N49O67Masse moléculaire :4668.25pCPA methyl ester hydrochloride
CAS :pCPA methyl ester HCl inhibits tryptophan hydroxylase, 5-HT synthesis, crosses blood-brain barrier, lowers central 5-HT.
Formule :C10H13Cl2NO2Degré de pureté :99.73% - 99.88%Couleur et forme :SolidMasse moléculaire :250.12Gastrin-Releasing Peptide, human
CAS :Gastrin-releasing peptide, released by vagal fibers, stimulates stomach G cells to secrete gastrin, affecting acid secretion and gut motility.Formule :C130H204N38O31S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2859.38Big endothelin-1 (rat 1-39)
CAS :Big endothelin-1 (rat 1-39), a 39-residue peptide, induces a diuretic and natriuretic response in conscious Sprague-Dawley rats and elevates blood pressure inCouleur et forme :SolidFezolamine
CAS :Fezolamine: a new, non-tricyclic, oral antidepressant, selectively inhibits norepinephrine uptake over serotonin or dopamine.Formule :C20H23N3Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :305.42TH023
TH023 is an inhibitor of the TLR4 signaling pathway, specifically targeting the formation of TLR4 homodimers. In HEK-Blue hTLR4 cells, TH023 suppresses the secretion of embryonic alkaline phosphatase with an IC50 of 0.354 μM and inhibits NO expression in RAW264.7 cells, with an IC50 of 1.61 μM. Additionally, TH023 inhibits the activation of NF-κB and reduces the nuclear translocation of NF-κB p65. The compound demonstrates anti-inflammatory effects in a mouse model of LPS-induced acute sepsis and improves lung injury in mice.Formule :C22H21ClF2N4OCouleur et forme :SolidMasse moléculaire :430.88T-kinin
CAS :T-kinin (Ile-Ser-bradykinin) is a bradykinin-containing peptide utilized in inflammation research [1] [2].Formule :C59H89N17O14Masse moléculaire :1260.44Wy 41747
CAS :Wy 41747 is a long-acting somatostatin analogue utilized in research of diabetes mellitus [1].Formule :C73H92N18O16S2Masse moléculaire :1541.75PNMT-IN-1
PNMT-IN-1 (inhibitor 4) is a selective second generation inhibitor [1] of phenylethanolamine N-methyltransferase (PNMT), exhibiting a Ki value of 1.2 nM and anCouleur et forme :Odour Solid[Lys8] Vasopressin Desglycinamide
CAS :[Lys8] Vasopressin Desglycinamide, a vasopressin analog, supports the maintenance of active and passive avoidance behavior and aids in the facilitation ofFormule :C44H63N11O12S2Couleur et forme :SolidMasse moléculaire :1002.17Alkyne-βAG-TOCA
Alkyne-βAG-TOCA is an octreotide derivative that targets somatostatin receptor subtype 2 (SST2). It is utilized in the synthesis and research of radioconjugates (RDC).Formule :C48H65N11O15S2Couleur et forme :SolidMasse moléculaire :1100.22P2Y12R ligand-1
P2Y12R ligand-1 (Compound 41) is a high-affinity P2Y12 receptor ligand with a Ki of 17.1 nM. The [18F]-labeled version of P2Y12R ligand-1 is suitable for research involving brain PET imaging.Couleur et forme :Odour SolidPG 106 acetate
PG 106 acetate: Selective hMC3 receptor antagonist, IC50=210 nM; inactive on hMC5 and hMC4, EC50=9900 nM.Formule :C53H73N13O11Degré de pureté :98.24%Couleur et forme :SolidMasse moléculaire :1068.23CHS-114
CHS-114 (SRF-114) is a fully human IgG1 antibody targeting the (CCR8) receptor. It shows potential for research in head and neck squamous cell carcinoma (HNSCC). The isotype control for CHS-114 can be referred to as HumanIgG1kappa, Isotype Control.Couleur et forme :Odour LiquidAnti-TSHR Antibody (M22)
Anti-TSHR Antibody (M22) is a humanized IgG1 monoclonal antibody targeting the thyroid-stimulating hormone receptor (TSHR). This antibody is capable of inhibiting the interaction between TSH and TSHR.Couleur et forme :Odour Liquid[Ala11,D-Leu15]-Orexin B acetate
[Ala11,D-Leu15]-Orexin B acetate is a selective agonist of orexin-2 receptor (OX2) with an EC50 of 0.13 nM, showing 400-fold selectivity over OX1 (52 nM).Formule :C122H210N44O37SDegré de pureté :98.18%Couleur et forme :SolidMasse moléculaire :2917.31Efranarelaxin alfa
CAS :Efranarelaxin alfa is an agonist of the relaxin receptor. It shows potential for research in cardiovascular diseases and tissue repair.Couleur et forme :LiquidNI-203
NI-203 is a monoclonal antibody inhibitor that targets amylin and shows potential for research in type 2 diabetes.Couleur et forme :Odour LiquidTriamterene
CAS :Triamterene is a barosensitive epithelial sodium channel (ENaC) blocker with a diuretic effect. It can also act as an inhibitor of the TGR5 receptor, reducing GLP-1 secretion and cAMP level increases induced by TGR5 activation in a dose-dependent manner.Formule :C12H11N7Degré de pureté :99.77%Couleur et forme :Yellow Yellow SolidMasse moléculaire :253.26Minaprine
CAS :Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.Formule :C17H22N4ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :298.38CCR6 antagonist 1
CAS :CCR6 antagonist 1 blocks CCL20/CCR6, aiding autoimmune and IBD research.
Formule :C17H12F3NO2Degré de pureté :99.83%Couleur et forme :SoildMasse moléculaire :319.28CUR61414 hydrochloride
CUR61414 hydrochloride: potent cell-permeable Hedgehog pathway inhibitor, IC50=100-200 nM, selectively targets Smo (Ki=44 nM), induces cancer cell apoptosis.Formule :C31H43ClN4O5Degré de pureté :94.05%Couleur et forme :SolidMasse moléculaire :587.15Cisapride hydrate
CAS :Cisapride acts directly as a selective agonist of serotonin 5-HT4 receptor with IC50 value of 0.483 μM. And It also acts indirectly as a parasympathomimetic.Formule :C23H31ClFN3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :483.96Oxatomide
CAS :Oxatomide: Dual H1/P2X7 antagonist, antihistamine, anti-allergic, treats immune diseases, IC50: 0.95 μM (P2X7), 0.43 μM (5-HT).Formule :C27H30N4ODegré de pureté :99.28% - 99.72%Couleur et forme :White PowderMasse moléculaire :426.55Ref: TM-T19839
1mg35,00€5mg75,00€1mL*10mM (DMSO)84,00€10mg114,00€25mg222,00€50mg356,00€100mg557,00€500mg1.153,00€Benzomalvin C
CAS :Benzomalvin C, isolated from Penicillium, inhibits NK1 receptor and IDO with IC50 of 130 μM, and has a unique epoxide group at C-19/C-20.Formule :C24H17N3O3Couleur et forme :SolidMasse moléculaire :395.418SKF-83566 hydrochloride
CAS :SKF-83566 hydrochloride is a D1-like dopamine receptor antagonist, inhibiting dopamine transporters and mitigating GBP-induced CPP.Formule :C17H19BrClNODegré de pureté :99.27%Couleur et forme :SoildMasse moléculaire :368.69(R)-Citalopram oxalate
CAS :(R)-Citalopram oxalate is a weak selective serotonin reuptake inhibitor (SSRI) that antagonises its S-isomer (escitalopram), anticonvulsant and antidepressant
Formule :C22H23FN2O5Degré de pureté :99.76%Couleur et forme :White SolidMasse moléculaire :414.43W140 HBr
CAS :[(3S)-3-amino-4-(3-hexylanilino)-4-oxobutyl]phosphonic acid;hydrobromide is a S1P1 antagonist with Ki of 2.84 μM.Formule :C16H28BrN2O4PDegré de pureté :99.85%Couleur et forme :SoildMasse moléculaire :423.28Ref: TM-T60204
1mg115,00€2mg172,00€5mg255,00€1mL*10mM (DMSO)284,00€10mg375,00€25mg562,00€50mg787,00€100mg1.074,00€Noladin ether
CAS :Noladin ether (2-AG ether) is a cannabinoid CB1 receptor agonist.Formule :C23H40O3Couleur et forme :SolidMasse moléculaire :364.56Seglitide acetate
CAS :Seglitide acetate (MK-678) is a selective agonist of sst2 somatostatin receptor.Formule :C46H60N8O9Degré de pureté :98.87%Couleur et forme :SolidMasse moléculaire :869.02NPC 567 acetate
NPC 567 acetate is a bradykinin B2 antagonist and can be used in studies about the treatment of allergic airway disease.Formule :C62H91N19O15Degré de pureté :97.72%Couleur et forme :SolidMasse moléculaire :1342.5γ-Glu-Abu TFA
Gamma-Glu-AbuTFA is the TFA salt form of Gamma-Glu-Abu. This compound acts as an agonist for the calcium sensing receptor (CaSR), activating CaSR in HEK-293 cells with an EC50 of 0.21 μM.Formule :C11H17F3N2O7Couleur et forme :SolidMasse moléculaire :346.26Calcitonin-13C6,15N4 TFA
Calcitonin-13CIC6,15NIC4(salmon) (Salmon calcitonin-13CIC6,15NIC4) TFA is a version of calcitonin(salmon) labeled with carbon-13 and nitrogen-15. This hormone regulates calcium and acts dualistically as an agonist to both amylin and calcitonin receptors, promoting bone formation while inhibiting bone resorption.Formule :C1401C5H240N4315NO48S2·5C2HF3O2Couleur et forme :SolidMasse moléculaire :4007.93Neurokinin A(4-10)
CAS :Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .Formule :C34H54N8O10SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :766.91GLP-1R Agonist DMB
CAS :GLP-1R Agonist DMB is an agonist of glucagon-like peptide 1 receptor (GLP-1R; KB = 26.3 nM for the recombinant human receptor).Formule :C13H15Cl2N3O2SDegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :348.25Des His1, Glu8 Exendin-4
Des His1, Glu8 Exendin-4 is a glucagon-like peptide-1 receptor (GLP1R) antagonist that regulates blood glucose and is used in the study of diabetes and obesity.Formule :C179H277N47O59SDegré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :4063.46Edg-2 receptor inhibitor 1
CAS :Edg-2 receptor inhibitor 1 (SAR-100842) is an Edg-2 receptor inhibitor extracted (IC50: <0.1 μM).Formule :C27H27NO5Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :445.51Ref: TM-T4521
1mg97,00€2mg170,00€5mg274,00€1mL*10mM (DMSO)288,00€10mg426,00€25mg663,00€50mg947,00€100mg1.264,00€R 396
CAS :R 396 (Acleu-asp-gln-trp-phe-glynh2) is a linear hexapeptide and is also an NK-2 tachykinin receptor antagonist.Formule :C39H51N9O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :805.88BMS 193885
CAS :BMS 193885 is a selective and competitive neuropeptide Y(1) receptor antagonist with affinity of 3.3 nM.Formule :C36H48N4O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :680.79L-796,778
CAS :L-796,778 is an SST3 agonist and a selective ligand of SST3, which can increase the level of cAMP in the body.Formule :C29H40N6O7Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :584.66Ref: TM-T32511
1mg175,00€5mg404,00€1mL*10mM (DMSO)522,00€10mg592,00€25mg888,00€50mg1.243,00€100mg1.701,00€500mg3.402,00€p-MPPF
CAS :p-MPPF is a 5-HT antagonist that can be used to study neurological diseases.Formule :C25H27FN4O2Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :434.51Mazdutide acetate(2259884-03-0 free base)
Mazdutide acetate is a potent (GLP-1R and GCGR agonist that stimulates insulin secretion from mouse pancreatic islets , which can be used to study obesity.Degré de pureté :98.41%Couleur et forme :Odour SolidAtrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate
CAS :Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate is an NPR-A agonist and ANP hormone. Carperitide increases cGMP levels and reduces the heart's workload.Formule :C129H207N45O41S3Degré de pureté :99.78%Couleur et forme :SoildMasse moléculaire :3140.5Dalcotidine
CAS :Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, may lower relapse.Formule :C18H29N3O2Degré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :319.44Ref: TM-T31195
1mg63,00€5mg140,00€1mL*10mM (DMSO)140,00€10mg200,00€25mg324,00€50mg470,00€100mg662,00€200mg893,00€QWF acetate
QWF acetate is a Substance P antagonist peptide that specifically inhibits the binding to its receptor, NK1, and inhibits the activation of MRGPRX2.
Formule :C40H47N5O10Degré de pureté :96.65%Couleur et forme :SolidMasse moléculaire :757.84N-Nitroso Atenolol
CAS :N-Nitroso Atenolol is a derivative of Atenolol. At concentrations ranging from 0.1 to 1 mM, it induces DNA fragmentation in rat hepatocytes.Formule :C14H21N3O4Couleur et forme :SolidMasse moléculaire :295.33(±)-9-Nor-9α-hydroxy Hexahydrocannabinol
CAS :(±)-9-Nor-9α-hydroxy Hexahydrocannabinol is a cannabinoid-structured compound that exhibits potent cannabinoid-like activity in both dogs and mice.Formule :C20H30O3Couleur et forme :SolidMasse moléculaire :318.45CB2 receptor agonist 9
CAS :CB2 receptor agonist 9 (Compound 33) is an orally active agonist of cannabinoid receptor 2 (CB2 receptor) with an EC50 of 16.2 nM. It inhibits the expression of TNF-α, IL-1β, and IL-6, demonstrating anti-inflammatory activity in a DSS-induced acute colitis model in mice.Formule :C16H23N3O2SCouleur et forme :SolidMasse moléculaire :321.44SBI-810
CAS :SBI-810 is a functional selective β-arrestin-biased allosteric modulator of the neurotensin receptor 1 (NTSR1). In the presence of the endogenous ligand neurotensin (NT), SBI-810 regulates NTSR1 signaling through a G protein-specific mechanism. It fully antagonizes NT-induced Gq activation and partially antagonizes NT-induced Gi1 activation, allowing NTSR1 to activate GoA and G12.Formule :C27H34N4O2Couleur et forme :SolidMasse moléculaire :446.594-hydroxy DiPT hydrochloride
CAS :4-hydroxy DiPT (hydrochloride) is a 5-HT2A agonist that can induce head twitch response (HTR) in mice, indicating its hallucinogenic potential. This compound holds promise for research into hallucinogens.Formule :C16H25ClN2OCouleur et forme :SolidMasse moléculaire :296.84Δ8-THC methyl ether
CAS :Δ8-THC methyl ether (compound 3) demonstrates a strong docking score of -10.167 kcal/mol for the CB2 receptor. Additionally, Δ8-THC methyl ether exhibits antinociceptive activity in mice.Formule :C22H32O2Couleur et forme :SolidMasse moléculaire :328.494-Iodoamphetamine hydrochloride
CAS :4-Iodoamphetamine (p-Iodoamphetamine) hydrochloride is a halogenated phenethylamine characterized by the presence of an iodine atom at the para position of the phenyl group. It selectively induces serotonin release and inhibits reuptake in rat brain synaptosomes.Formule :C9H13ClINCouleur et forme :SolidMasse moléculaire :297.56δ8-THC acetate
CAS :Delta8-THC acetate (Delta8-tetrahydrocannabinol) is a psychoactive cannabinoid that binds to the cannabinoid receptor 1 (CB1 receptor) and exhibits anti-nausea, appetite-stimulating, and anti-inflammatory effects. It may also offer neuroprotective benefits and has potential applications in research on anxiety and depression.Formule :C23H32O3Couleur et forme :SolidMasse moléculaire :356.5Methamnetamine hydrochloride
CAS :Methamnetamine (PAL-1046) hydrochloride is a psychoactive substance derived from phenethylamine, known to cause excessive serotonin release.Formule :C14H18ClNCouleur et forme :SolidMasse moléculaire :235.75PAF C-18
CAS :PAF C-18 is a natural phospholipid molecule belonging to the platelet-activating factor (PAF) family,, involved in hemostasis and thrombosis by binding to PAFR.Formule :C28H58NO7PDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :551.74BAY-6672
CAS :BAY-6672 is, a selective,oral, highly potent human prostaglandin F (FP) receptor antagonist, exerts antifibrotic effects by inhibiting PGF₂α activity.Formule :C26H27BrClN3O3Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :544.87AD353
AD353 is a selective sigma-1 receptor ligand. It demonstrates high efficacy in models of capsaicin-induced allodynia and PGE2-induced mechanical hyperalgesia. Additionally, AD353 exhibits favorable pharmacokinetic properties.Formule :C23H30N2O2Couleur et forme :SolidMasse moléculaire :366.5PF-4363467
CAS :PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.Formule :C22H30N2O3SCouleur et forme :SolidMasse moléculaire :402.55Casopitant
CAS :Casopitant (GW679769) is an orally active neurokinin-1 (NK1) receptor antagonist, researched for its potential use in managing chemotherapy-induced nausea and vomiting (CINV) and postoperative nausea and vomiting (PONV).Formule :C30H35F7N4O2Couleur et forme :SolidMasse moléculaire :616.616-Fluoro-N,N-diethyltryptamine
CAS :6-Fluoro-N,N-diethyltryptamine (6-F-DET) exhibits affinity for the 5-HT2A receptor.Formule :C14H19FN2Couleur et forme :SolidMasse moléculaire :234.3117-TFM-PGF1α
CAS :17-TFM-PGF1α (Compound 8) is a saturated prostaglandin analog. It exhibits a high affinity and receptor selectivity for the human prostaglandin F receptor (hFP receptor), with an EC50 of 85 nM.Formule :C24H35F3O5Couleur et forme :SolidMasse moléculaire :460.53Eloralintide
CAS :Eloralintide (LY 3841136) is an AMYR agonist, anticipated for research in type 2 diabetes and obesity.Formule :C201H319N49O65S2Couleur et forme :SolidMasse moléculaire :4526.1CAY10509
CAS :CAY10509 is a PGF2α analogue and acts as an FP receptor inhibitor with an IC50 of 30 nM. It shows potential for use in studying the physiological regulatory mechanisms related to prostaglandins.Formule :C23H35FO5SCouleur et forme :SolidMasse moléculaire :442.585-MeO-MET
CAS :5-MeO-MET (5-Methoxy-N-methyl-N-ethyltryptamine) is a compound belonging to the 5-methoxytryptamine class. It acts as an agonist for 5-HT1A and 5-HT2A receptors. In mice, 5-MeO-MET inhibits locomotion and has sedative effects.Formule :C14H20N2OCouleur et forme :SolidMasse moléculaire :232.3225N-NBOMe hydrochloride
CAS :25N-NBOMe hydrochloride is a derivative of 2C-N and acts as an agonist for the 5-HT2A and 5-HT2C receptors, with Ki values of 0.144 nM and 1.06 nM, respectively. It has minimal effect on the release of preloaded neurotransmitters from recombinant dopamine, serotonin, and norepinephrine transporters.Formule :C18H23ClN2O5Couleur et forme :SolidMasse moléculaire :382.84Δ8-THC-C8
CAS :Δ8-THC-C8 is a semi-synthetic cannabinoid. It acts as an agonist for the cannabinoid receptor 1 (CB1) with an EC50 value of 13.8 nM.Formule :C24H36O2Couleur et forme :SolidMasse moléculaire :356.544-Bromo-2,5-DMMA
CAS :4-Bromo-2,5-DMMA (Compound 2) demonstrates affinity for the 5-HT2 binding site and has an ED50 of 0.82 mg/kg in rat discrimination experiments.Formule :C12H18BrNO2Couleur et forme :SolidMasse moléculaire :288.18hA3AR agonist 2
hA3AR agonist 2 is a potent activator of A3AR, with a Ki value of 3.5 nM.Formule :C11H14ClN5O2SCouleur et forme :SolidMasse moléculaire :315.78APP-FUBINACA
CAS :APP-FUBINACA is a cannabinoid receptor agonist, classified as a phenylalanine amide-based indazole-3-carboxamide derivative. It exhibits neurostimulatory effects.Formule :C24H21FN4O2Couleur et forme :SolidMasse moléculaire :416.45Latanoprost tris(triethylsilyl) ether
CAS :Latanoprosttris(triethylsilyl) ether is a precursor in the synthesis of Latanoprost, which serves as an agonist for the prostaglandin F2α (PGF2α) receptor, also known as the FP receptor.Formule :C44H82O5Si3Couleur et forme :SolidMasse moléculaire :775.38Pafenolol
CAS :Pafenolol is a P-glycoprotein modulator with a Ki value of 5.5 µM. pafenolol is an orally available and selective beta-adrenergic receptor antagonist.Formule :C18H31N3O3Degré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :337.46Arotinolol hydrochloride
CAS :Arotinolol HCl is a non-selective α/β-blocker, anti-hypertensive, anti-obesity, and improves aortic stiffness.Formule :C15H22ClN3O2S3Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :408FFN246
CAS :FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation andFormule :C15H13FN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :256.27Emoghrelin
CAS :Emoghrelin, extracted from Heshouwu (Polygonum multiflorum), promotes the secretion of growth hormone by activating the ghrelin receptor [1].Formule :C24H22O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :518.42α-CGRP (mouse, rat) TFA
α-CGRP (mouse, rat) TFA, a neuropeptide belonging to the calcitonin gene-related peptide (CGRP) family, is predominantly located at neuromuscular junctions andFormule :C162H262N50O52S2·C2HF3O2Degré de pureté :98%Couleur et forme :SolidPSB-1114 triethylamine
PSB-1114 triethylamine is a potent, enzymatically stable, P2Y2 receptor agonist with a 134 nM EC50, exhibiting greater than 50-fold selectivity over P2Y4 (EC50Formule :C10H15F2N3O13P3S·xC6H15NDegré de pureté :98%Couleur et forme :Solid(Leu31,Pro34)-Peptide YY (human) (TFA)
"(Leu31,Pro34)-Peptide YY (human) (TFA) is the trifluoroacetic acid (TFA) form of (Leu31,Pro34)-Peptide YY (human), a derivative of Peptide YY that acts as aFormule :C195H296N54O56·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4292.75 (free base)Mibenratide TFA
Mibenratide TFA, a small cyclic peptide, functions as an adrenergic β1 receptor antagonist and has potential applications in heart failure research [1].Degré de pureté :98%Couleur et forme :Odour SolidMuscarinic toxin 3
CAS :Muscarinic toxin 3 (MT3), a potent non-competitive antagonist of mAChR and adrenoceptors, exhibits pIC50 values of 6.71 for M1, 8.79 for M4, 8.86 for α1A, 7.57Formule :C319H489N89O97S8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :7379.35AB21 oxalate
AB21 oxalate, a potent and selective S1R antagonist, exhibits binding affinities (Kis) of 13 nM and 102 nM for S1R and S2R, respectively.Formule :C25H30N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :438.525-HT6 agonist 1
Compound 19, a 5-HT6 agonist with an affinity (K i : 5 nM), exhibits antidepressant-like effects and enhances cognitive function while also inhibiting plateletFormule :C17H22Cl2N6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :413.37human GALP (3-32)
Human GALP (3-32) (Galanin-like peptide (3-32)) serves as a high-affinity agonist for galanin receptors GalR1 (IC50 = 33 nM) and GalR2 (IC50 = 15 nM), asFormule :C137H213N43O38SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3102.49Sigma-1 receptor antagonist 5
Sigma-1 receptor antagonist 5 (compound 12), a 4-pyridylpiperidine derivative, exhibits analgesic properties through its antagonistic action on sigma receptorsFormule :C26H27N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :397.51CB2R agonist 2
CB2R agonist 2 (cis-17-para) is a CB2R agonist [1].Degré de pureté :98%Couleur et forme :Odour SolidPhoenixin-14
CAS :Phoenixin-14 (PNX-14), an active endogenous isoform, induces an anxiolytic effect by activating the AHA GnRH system in mice and protects against ischemia/
Formule :C75H110N18O20Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1583.78Uroguanylin (human)
CAS :Uroguanylin (human) serves as a natural ligand for the Guanylyl Cyclase C (GCC) receptor in metastatic colorectal cancer tumors and exhibits anti-tumor effectsFormule :C64H102N18O26S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1667.86LHRH
CAS :Luteinizing hormone-releasing hormone (LHRH) is a neuropeptide produced in the hypothalamus that plays a pivotal role in regulating reproduction and hasFormule :C55H74N16O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1183.27CB2R agonist 3
CB2R agonist 3, a potent activator of cannabinoid receptor 2 (CB2R), exhibits an EC50 value of 0.37μM, indicative of its significant role in the immune system [Degré de pureté :98%Couleur et forme :Odour SolidFGH31
FGH31 (Compound 24), a dopamine D4 agonist, exhibits potent and selective GRK2-dependency with a K i of 1.6 nM and partially activates β-arrestin [1].Formule :C33H36N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :520.66MRS7925
MRS7925 (Compound 43) serves as a potent antagonist of the 5-HT2B receptor, with an inhibition constant (Ki) of 17 nM, and is utilized in the study of fibrosisFormule :C20H26IN5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :511.36[D-Pro2] Spantide I TFA
[D-Pro2] Spantide I TFA is an analog of Spantide I, a selective antagonist of the NK1 receptor [1].Formule :C75H108N20O13·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidTetrapeptide-1
CAS :Tetrapeptide-1 is a bioactive peptide renowned for its antioxidant properties and has been cited as an ingredient in cosmetics [1].Formule :C20H36N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :428.52PSB 0777 ammonium hydrate
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM forFormule :C18H20N5O7S2·NH4·75H2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :532.09D3R ligand 1
D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor (Ki=66 nM), incorporating a THPB template.Formule :C27H37NO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :455.59NF546 hydrate
NF546 (hydrate), a selective non-nucleotide P2Y11 agonist, exhibits a pEC50 value of 6.27 and induces interleukin-8 secretion from human monocyte-derivedFormule :C47H44N6Na4O17P4·5H2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1424.01Guanylin (mouse, rat)
CAS :Guanylin (mouse, rat), a peptide consisting of 15 amino acids, acts as an activator of intestinal guanylate cyclase and is utilized in diarrhea research [1].Formule :C60H90N16O22S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1515.71A3AR agonist 2
Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM.Formule :C34H34N6O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :622.67Stressin I TFA
Stressin I (Cyclo(31-34)[DPhe12, Nle21, 38, Glu31, Lys34]Ac-hCRF(4-41)) TFA, with a K i of 1.7 nM, is a potent and selective agonist of the CRF1 receptor.Degré de pureté :98%Couleur et forme :Odour SolidVal9-Oxytocin
CAS :Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete antagonist of the vasopressin (V1a) receptor.Formule :C46H72N12O12S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1049.27Ala5-Galanin (2-11)
CAS :Ala5-Galanin (2-11) is a specific agonist for the galanin receptor 2 (GAL2R) with an affinity constant (Ki) of 258 nM [1].Formule :C54H81N13O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1120.3AD186
AD186, a potent and selective S1R agonist, exhibits dissociation constants (Kis) of 2.7 nM for S1R and 27 nM for S2R.Formule :C22H28N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :320.47Galanin-Like Peptide (porcine)
CAS :Galanin-Like Peptide (porcine) is a 60 amino acid neuropeptide originally isolated from the porcine hypothalamus.Formule :C281H443N81O78Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :6204.02hNTS1R agonist-1
Compound 10, an hNTS1R agonist-1, acts as a full agonist with a strong affinity for hNTS1R (K i: 6.9 nM), showing the ability to cross the blood-brain barrier (Formule :C37H62N10O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :790.95N,N′-Diferuloylputrescine
CAS :N,N′-Diferuloylputrescine acts as a pigment inhibitor, showing a 57% reduction in pigmentation.Formule :C24H28N2O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :440.49Vilanterol
CAS :Vilanterol is a selective long-acting beta2-adrenergic agonist (LABA) used in the treatment of COPD and asthma.Formule :C24H33Cl2NO5Degré de pureté :97.47% - 99.46%Couleur et forme :SolidMasse moléculaire :486.43Ref: TM-T2645
1mg39,00€5mg84,00€1mL*10mM (DMSO)90,00€10mg114,00€25mg173,00€50mg227,00€100mg339,00€200mg504,00€Nadolol
CAS :Nadolol is a non-selective beta-adrenergic antagonist with antihypertensive and antiarrhythmic activities.Formule :C17H27NO4Degré de pureté :99.87% - 99.92%Couleur et forme :White To Off-White Crystalline Powder SolidMasse moléculaire :309.40Esprolol
CAS :Esprolol (ACC-9369 free base) is a novel beta-adrenergic antagonist used to study exertional angina.Formule :C17H27NO4Degré de pureté :71.58% - 99.16%Couleur et forme :SoildMasse moléculaire :309.4Ref: TM-T27286L
1mg80,00€2mg105,00€5mg172,00€10mg253,00€25mg414,00€50mg583,00€100mg783,00€200mg1.054,00€PACAP (6-27) (human, chicken, mouse, ovine, porcine, rat) (trifluoroacetate salt)
PACAP (6-27) is an antagonist for PACAP receptors with varying IC50s; blocks cAMP in neuroblastoma and breast cancer cells.Couleur et forme :LiquidPACAP-related Peptide (human) (trifluoroacetate salt)
Endogenous 29-amino acid PRP belongs to secretin/glucagon family, found in pancreas, adrenal glands, and some VIP tumors; secreted by CHO-K1 cells.Couleur et forme :LiquidPACAP-related Peptide (rat) (trifluoroacetate salt)
PRP, a 29-amino acid peptide in the secretin/glucagon family, is found in rat brain regions and reproductive tissues.Couleur et forme :SolidCorticotropin-releasing factor (human) acetate
Corticotropin-releasing factor (human) acetate stimulates to synthesize and secret adrenocorticotropin in the anterior pituitary.Degré de pureté :98.30%Couleur et forme :LiquidPACAP-38 (31-38), human, mouse, rat acetate
PACAP-38 (31-38) acetate stimulates PAC1 receptor and boosts NPY and catecholamine in sympathetic neurons.Formule :C49H87N17O13Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :1122.32Nα-Methylhistamine FA
Nα-Methylhistamine FA is a histamine H3 receptor agonistFormule :C7H13N3O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :171.2Tirzepatide
CAS :Tirzepatide (LY-3298176) is a dual glucose-dependent polypeptide (GIP) (EC50=0.042 nM) and glucagon-like peptide-1 (GLP-1) (EC50=0.086 nM) receptor agonist.Formule :C225H348N48O68Degré de pureté :99.52% - 99.99%Couleur et forme :SolidMasse moléculaire :4813.45Meclinertant
CAS :Meclinertant: selective NTS1 antagonist, blocks Ca2+ mobilization, with anxiolytic and anti-addictive properties.Formule :C32H31ClN4O5Degré de pureté :97.51% - 99.44%Couleur et forme :SolidMasse moléculaire :587.07Tiaspirone hydrochloride
CAS :Tiaspirone hydrochloride (BMY-13859 hydrochloride) exhibits antipsychotic activity and influences the electrophysiological activity of dopaminergic neurons.Formule :C24H33ClN4O2SDegré de pureté :99.87%Couleur et forme :SoildMasse moléculaire :477.06Tamsolusin Hydrochloride
CAS :Tamsolusin Hydrochloride (YM 12617) is a highly selective alpha-1A adrenergic receptor antagonist used in the treatment of benign prostatic hypertrophy.Formule :C20H29ClN2O5SDegré de pureté :99.92%Couleur et forme :SoildMasse moléculaire :444.97Vazegepant
CAS :Vazegepant is an intranasal CGRP receptor antagonist utilized for conducting acute migraine research.Formule :C36H46N8O3Degré de pureté :98.61% - 99.98%Couleur et forme :SolidMasse moléculaire :638.80Ref: TM-T38734
1mg90,00€5mg215,00€1mL*10mM (DMSO)289,00€10mg318,00€25mg537,00€50mg767,00€100mg1.054,00€Lysosphingomyelin (d18:1)
CAS :Sphingomyelins are phosphorylcholine, sphingosine, and fatty acid. Lysosphingomyelin, missing the fatty acid, activates diverse cellular pathways.Formule :C23H49N2O5PCouleur et forme :SolidMasse moléculaire :464.628GRK2 Inhibitor
CAS :GRK2 Inhibitor is an inhibitor of β-Adrenergic Receptor Kinase 1 (β ARK1).Formule :C12H9NO6Couleur et forme :SolidMasse moléculaire :263.2Docosahexaenoic acid ethyl ester
CAS :Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.Formule :C24H36O2Degré de pureté :98.35%Couleur et forme :SolidMasse moléculaire :356.54Sulfisoxazole (Standard)
CAS :Sulfisoxazole (Standard) is the standard substance of Sulfisoxazole, and it is applicable for quantitative analysis, quality control, and related research in biochemical experiments. Sulfisoxazole (Sulfafurazole) is a short-acting sulfonamide antibacterial with activity against a wide range of gram-negative and gram-positive organisms.Sulfisoxazole inhibits breast cancer exosome release by targeting endothelin receptor A.Formule :C11H13N3O3SCouleur et forme :White To Cream PowderMasse moléculaire :267.30SUN B8155
CAS :SUN B8155 is a CT receptor agonist that induces cAMP formation in cells expressing recombinant human CT receptor.Formule :C14H15N3O3Degré de pureté :99.38% - 99.99%Couleur et forme :SolidMasse moléculaire :273.29Cudarolimab
CAS :Cudarolimab (IBI-101) is a fully human anti-OX40 antibody with potential immune checkpoint inhibitory and anti-tumor activity for the study of cancer.Degré de pureté :97.5% (SDS-PAGE); 98.2% (SEC-HPLC) - 97.5% (SDS-PAGE); 98.2% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :145.67 kDaFenoterol-d6 Hydrobromide
CAS :Fenoterol-d6 Hydrobromide is a deuterated compound of Fenoterol Hydrobromide. Fenoterol Hydrobromide has a CAS number of 1944-12-3. Fenoterol hydrobromide, the hydrobromide salt of fenoterol, is a β2 adrenoreceptor agonist with bronchodilator activity.Formule :C17H16D6BrNO4Masse moléculaire :390.301-Methyl-4-imidazoleacetic Acid (hydrochloride)
CAS :MIMA, a stable histamine byproduct from N-methylhistamine oxidation, indicates systemic mastocytosis via urinary levels.Formule :C6H9ClN2O2Couleur et forme :SolidMasse moléculaire :176.601Eplivanserin (mixture)
CAS :Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist,Formule :C19H21FN2O2Couleur et forme :SolidMasse moléculaire :328.387Quetiapine-d8 Fumarate
CAS :Quetiapine-d8 Fumarate is a deuterated compound of Quetiapine Fumarate. Quetiapine Fumarate has a CAS number of 111974-72-2. Quetiapine Fumarate, an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar II depression, bipolar I depression.Formule :C25H21D8N3O6SCouleur et forme :SolidMasse moléculaire :507.63Furprofen
CAS :Furprofen, an NSAID, inhibits PGE synthesis, offers analgesic effects, and is orally taken for pain relief.Formule :C14H12O4Degré de pureté :98.62% - 99.25%Couleur et forme :SolidMasse moléculaire :244.24Hydroxyzine dihydrochloride-d4
CAS :Hydroxyzine dihydrochloride-d4 is a deuterated compound of Hydroxyzine dihydrochloride.Formule :C21H25D4Cl3N2O2Couleur et forme :SolidMasse moléculaire :451.85Lanreotide
CAS :Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.Formule :C54H69N11O10S2Couleur et forme :SolidMasse moléculaire :1096.32SAR247799
CAS :SAR247799 is a selective and G-protein-biased S1P1 agonist that activates downstream G-protein signaling pathways more preferentially on endothelial cells.Formule :C21H16ClN3O5Couleur et forme :SolidMasse moléculaire :425.82(Rac)-Rotigotine hydrochloride
CAS :(Rac)-Rotigotine hydrochloride is a racemate of Rotigotine. Rotigotine is a full agonist of dopamine receptor, a partial the 5-HT1A receptor agonist.Formule :C19H26ClNOSCouleur et forme :SolidMasse moléculaire :351.93UCSF924
CAS :UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).Formule :C20H22N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :322.4rac-Propranolol-d7
CAS :Rac-Propranolol-d7 is the deuterated form of Rac-Propranolol. Propranolol is a β-adrenergic receptor antagonist that inhibits β1AR.Formule :C16H14D7NO2Couleur et forme :SolidMasse moléculaire :266.39Pramipexole dihydrochloride
CAS :Pramipexole dihydrochloride could be used to treat Parkinson disease.Formule :C10H18ClN3SDegré de pureté :98%Couleur et forme :White Crystalline PowderMasse moléculaire :247.79Granisetron
CAS :Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.
Formule :C18H24N4OCouleur et forme :SolidMasse moléculaire :312.41SBI-810 hydrochloride
CAS :SBI-810 hydrochloride is a β-arrestin-2 (βarr2)-biased allosteric modulator of NTSR1 (neurotensin receptor 1), exerting analgesic effects.Formule :C27H35ClN4O2Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :483.05
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