GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(251 produits)
- Récepteur adrénergique(3.025 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(218 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(36 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(195 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
6011 produits trouvés pour "GPCR/G-Protéine"
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Rizatriptan sulfate
CAS :Rizatriptan sulfate is a selective serotonin 5-HTID receptor agonist derived from tryptamine.Formule :C15H21N5O4SCouleur et forme :SolidMasse moléculaire :367.42CGP 71683 (free base)
CAS :CGP 71683 (free base) is a potent and highly selective non-peptide antagonist of the NPY Y(5) receptor in the study of obesity.Formule :C26H29N5O2SCouleur et forme :SolidMasse moléculaire :475.61Taminadenant mesylate
CAS :Taminadenant (PBF-509/NIR-178) is an oral adenosine A2A receptor antagonist that activates T-cells to target tumor cells.Formule :C11H12BrN7O3SCouleur et forme :SolidMasse moléculaire :402.227SRI-37330 hydrochloride
CAS :SRI-37330 hydrochloride is an orally active thioredoxin-interacting protein (TXNIP) inhibitor. hydrochloride can be used to study type 2 diabetes.Formule :C16H20ClF3N4O2SCouleur et forme :SolidMasse moléculaire :424.87Selexipag
CAS :Selexipag (ACT-293987, NS-304) is a drug for PAH that dilates pulmonary vessels.Formule :C26H32N4O4SDegré de pureté :99.98% - >99.99%Couleur et forme :SolidMasse moléculaire :496.62Betahistine EP Impurity C
CAS :Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.Formule :C15H19N3Degré de pureté :99.93% - ≥95%Couleur et forme :SolidMasse moléculaire :241.33TFLLR-NH2 2TFA(197794-83-5(free base))
TFLLR-NH2 2TFA(197794-83-5(free base)) is an agonist of PAR1 (EC50 :1.9 μM).Formule :C35H55F6N9O10Degré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :875.87Escitalopram Oxalate
CAS :Escitalopram Oxalate ((S)-(+)Citalopram oxalate) is a selective serotonin (5-HT) reuptake inhibitor (SSRI) with Ki of 0.89 nM.Formule :C22H23FN2O5Degré de pureté :97.39% - 99.73%Couleur et forme :White SolidMasse moléculaire :414.43Ref: TM-T6493
10mg37,00€1mL*10mM (DMSO)42,00€25mg52,00€50mg63,00€100mg86,00€200mg118,00€500mg187,00€1g268,00€Pentagastrin
CAS :Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally, which can cause the secretion and synthesis ofFormule :C37H49N7O9SDegré de pureté :96.98% - 99.49%Couleur et forme :Fine Colorless Needle-Shaped Crystals From 2-Ethoxyethanol + Water SolidMasse moléculaire :767.89Praliciguat
CAS :Praliciguat (IW-1973) is an orally active sGC stimulator with a 197 nM EC50 in HEK-293 cells, enhances NO signaling, and is a vasodilator.Formule :C21H14F8N6O2Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :534.36Ref: TM-T16569
1mg142,00€2mg207,00€5mg349,00€1mL*10mM (DMSO)409,00€10mg537,00€25mg858,00€50mg1.161,00€100mg1.558,00€GSK2018682 HCl
CAS :GSK2018682 is a novel sphingosine-1-phosphate receptor 1 (s1p1) and 5 (s1p5) agonist.Formule :C22H22Cl2N4O4Couleur et forme :SolidMasse moléculaire :477.34Metoclopramide dihydrochloride
CAS :Metoclopramide dihydrochloride is a dopamine D2 antagonist that is used as an antiemetic.Formule :C14H24Cl3N3O2Couleur et forme :SolidMasse moléculaire :372.72Ursodeoxycholic acid sodium
CAS :Ursodeoxycholic acid sodium (Sodium Ursodeoxycholate) is a naturally occurring secondary bile acid with anti-inflammatory and cytoprotective activities.Formule :C24H40NaO4Degré de pureté :99.66% - 99.96%Couleur et forme :SolidMasse moléculaire :415.56BMY 7378 dihydrochloride
CAS :BMY 7378 dihydrochloride (BMY7378 HCl) , α1D-adrenergic receptor antagonist, is a weak partial agonist/antagonist of 5-HT1A receptor.Formule :C22H33Cl2N3O3Degré de pureté :97.32% - 99.08%Couleur et forme :SolidMasse moléculaire :458.42FK962
CAS :FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.Formule :C14H17FN2O2Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :264.3Ref: TM-T7829
2mg34,00€5mg52,00€1mL*10mM (DMSO)57,00€10mg82,00€25mg144,00€50mg200,00€100mg278,00€200mg389,00€BMS 182874 hydrochloride
CAS :BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.Formule :C17H20ClN3O3SDegré de pureté :97.01%Couleur et forme :SolidMasse moléculaire :381.88Ref: TM-T21790
1mg77,00€2mg92,00€5mg140,00€1mL*10mM (DMSO)146,00€10mg205,00€25mg343,00€50mg477,00€100mg665,00€200mg897,00€5-Benzyloxygramine
CAS :5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.Formule :C18H20N2ODegré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :280.36Landiolol hydrochloride
CAS :Landiolol hydrochloride (ONO-1101 hydrochloride) is an ultra-short-acting β1 selective adrenoceptor antagonist.Formule :C25H40ClN3O8Degré de pureté :99.91%Couleur et forme :White Crystalline PowderMasse moléculaire :546.05S1p receptor agonist 1
CAS :S1p receptor agonist 1 (S1p-receptor-agonist-1) is an S1P receptor agonist.Formule :C23H24FN3O3Degré de pureté :99.07% - 99.9%Couleur et forme :SolidMasse moléculaire :409.45WAY-100635 Monomaleate
CAS :WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.Formule :C25H34N4O2·C4H4O4Degré de pureté :98.44% - 99.46%Couleur et forme :SolidMasse moléculaire :538.64Ref: TM-T2631
2mg43,00€5mg63,00€1mL*10mM (DMSO)74,00€10mg89,00€25mg170,00€50mg315,00€100mg470,00€200mg680,00€500mg1.054,00€MCL0020
CAS :MCL0020 is a potent and selective melanocortin MC4 receptor antagonist, reverses stress-induced anorexia but has no effect on food intake in free-feeding rats.Formule :C34H39N7O4Degré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :609.72Indacaterol
CAS :Indacaterol (Onbrez; Arcapta) is a β2-Adrenergic Agonist. The mechanism of action of indacaterol is as an Adrenergic beta2-Agonist.Formule :C24H28N2O3Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :392.49Sonepiprazole mesylate
CAS :Sonepiprazole mesylate is a selective D4 antagonistFormule :C22H31N3O6S2Couleur et forme :SolidMasse moléculaire :497.63SAX-187
CAS :SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.Formule :C15H13ClN4O2S2Degré de pureté :97.82% - 98%Couleur et forme :SolidMasse moléculaire :380.87Ref: TM-T3183
1mg79,00€5mg152,00€1mL*10mM (DMSO)166,00€10mg245,00€25mg398,00€50mg532,00€100mg735,00€200mg973,00€Mequitazine
CAS :Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.Formule :C20H22N2SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :322.47[D-Phe12,Leu14]-Bombesin acetate
[D-Phe12,Leu14]-Bombesin acetate inhibits bombesin-stimulated secretion.Formule :C77H118N22O20Degré de pureté :98.41% - 99.14%Couleur et forme :SolidMasse moléculaire :1671.9Ranitidine
CAS :Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors).Formule :C13H22N4O3SDegré de pureté :99.52%Couleur et forme :Solid SolidMasse moléculaire :314.40Orexin B, rat, mouse Acetate
Orexin B, rat, mouse Acetate (Rat orexin B) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.Formule :C128H219N45O36SDegré de pureté :94.61%Couleur et forme :SolidMasse moléculaire :2996.45S1RA hydrochloride
CAS :S1RA hydrochloride (E-52862 hydrochloride) is an effective and specific sigma-1 receptor(σ1R, Ki: 17 nM) antagonist, and has good selectivity against σ2R (Ki >Formule :C20H24ClN3O2Degré de pureté :98% - 99.84%Couleur et forme :SolidMasse moléculaire :373.87Ref: TM-T4229
1mg35,00€5mg75,00€1mL*10mM (DMSO)84,00€10mg105,00€25mg205,00€50mg334,00€100mg492,00€500mg973,00€Ciproxifan maleate
CAS :Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinityFormule :C20H22N2O6Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :386.4Ref: TM-T2004
1mg40,00€2mg52,00€5mg75,00€1mL*10mM (DMSO)82,00€10mg101,00€25mg205,00€50mg380,00€100mg565,00€Epinastine hydrochloride
CAS :Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.Formule :C16H15N3·HClDegré de pureté :99.26% - 99.62%Couleur et forme :White SolidMasse moléculaire :285.77BWX 46 Acetate
BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.Formule :C118H190N36O30S2Degré de pureté :96.86%Couleur et forme :SolidMasse moléculaire :2657.12Raclopride
CAS :Raclopride is a selective antagonist of dopamine D2/D3 receptor.Formule :C15H20Cl2N2O3Degré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :347.24Neurotensin(8-13) 3TFA(60482-95-3(free base))
CAS :Neurotensin(8-13) 3TFA is Neurotensin (NT) fragment. Neurotensin(8-13) 3TFA results in a decrease in cell-surface NT1 receptors (NTR1) density.Formule :C40H65F3N12O10Degré de pureté :98.31%Couleur et forme :SolidMasse moléculaire :931.03Ref: TM-T7617L
1mg35,00€5mg73,00€10mg107,00€1mL*10mM (DMSO)132,00€25mg207,00€50mg313,00€100mg447,00€200mg620,00€SCH 58261
CAS :SCH 58261 is a potent and selective A2a adenosine receptor antagonist.The Ki =2.3 nM for rat A2a and 2 nM is for bovine A2a.Formule :C18H15N7ODegré de pureté :99.07% - 99.75%Couleur et forme :SolidMasse moléculaire :345.36Ref: TM-T6979
1mg38,00€2mg49,00€5mg80,00€1mL*10mM (DMSO)81,00€10mg118,00€25mg213,00€50mg344,00€100mg550,00€Piboserod
CAS :Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.Formule :C22H31N3O2Degré de pureté :97.21% - 99.49%Couleur et forme :SolidMasse moléculaire :369.5Ref: TM-T2278
1mg38,00€2mg50,00€5mg84,00€10mg118,00€1mL*10mM (DMSO)120,00€25mg220,00€50mg403,00€100mg582,00€500mg1.198,00€L-745870 trihydrochloride
CAS :L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.Formule :C18H22Cl4N4Degré de pureté :97.52%Couleur et forme :SolidMasse moléculaire :436.214i
CAS :4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.Formule :C16H12ClN3ODegré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :297.74CGP71683 hydrochloride
CAS :CGP71683 hydrochloride: NPY5 receptor antagonist, Ki=1.3 nM; inactive at Y1 (Ki >4000 nM) and Y2 (Ki=200 nM).Formule :C26H30ClN5O2SDegré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :512.07Neurokinin A(4-10) TFA(97559-35-8 free base)
Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].Formule :C36H55F3N8O12SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :880.93Bevantolol hydrochloride
CAS :Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.Formule :C20H28ClNO4Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :381.9Pimozide
CAS :Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.Formule :C28H29F2N3ODegré de pureté :99.63% - >99.99%Couleur et forme :SolidMasse moléculaire :461.55RS 504393
CAS :RS 504393 is a highly selective CCR2 chemokine receptor antagonist (IC50s: 89 nM and > 100 μM for human recombinant CCR2 and CCR1).Formule :C25H27N3O3Degré de pureté :98.64% - 99.62%Couleur et forme :SolidMasse moléculaire :417.5Idazoxan hydrochloride
CAS :Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.Formule :C11H12N2O2·HClDegré de pureté :99.42% - 99.84%Couleur et forme :SolidMasse moléculaire :240.69Ref: TM-T0115
2mg34,00€5mg49,00€1mL*10mM (DMSO)52,00€10mg73,00€25mg126,00€50mg177,00€100mg266,00€200mg394,00€Dimaprit dihydrochloride
CAS :Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.Formule :C6H15N3S·2HClDegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :234.19HPI 1
CAS :HPI 1 suppresses Hh pathway: IC50 = 1.5 μM (Shh, SAG), 4 μM (Gli2), 6 μM (Gli1) in Shh-LIGHT2 cells.Formule :C27H29NO6Degré de pureté :97.6%Couleur et forme :SolidMasse moléculaire :463.52Ref: TM-T22089
1mg44,00€2mg57,00€5mg96,00€1mL*10mM (DMSO)102,00€10mg128,00€25mg207,00€50mg308,00€100mg447,00€500mg973,00€N-Desmethylclozapine
CAS :N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.Formule :C17H17ClN4Degré de pureté :97.25% - 99.83%Couleur et forme :Yellow Crystalline SolidMasse moléculaire :312.8Ref: TM-T5158
2mg34,00€5mg48,00€1mL*10mM (DMSO)58,00€10mg79,00€25mg152,00€50mg235,00€100mg344,00€200mg490,00€ZK 756326
CAS :ZK 756326: Selective CCR8 agonist, IC50 1.8 μM (human), 2.6 μM (mouse), no CCR4/5, CXCR3/4 action, 28-fold selectivity vs 26 GPCRs, anti-HIV fusion.Formule :C21H28N2O3Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :356.46OXOMEMAZINE
CAS :Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.Formule :C18H22N2O2SDegré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :330.44AZD2098
CAS :AZD2098 is a potent CC-chemokine receptor 4 (CCR4) inhibitor used for asthma research.Formule :C11H9Cl2N3O3SDegré de pureté :99.80% - >99.99%Couleur et forme :SolidMasse moléculaire :334.18Ref: TM-T4300
1mg34,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg105,00€25mg217,00€50mg334,00€100mg502,00€500mg1.063,00€Clemizole
CAS :Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.Formule :C19H20ClN3Degré de pureté :98% - 99.65%Couleur et forme :SolidMasse moléculaire :325.84Ref: TM-T1822
1mg42,00€5mg82,00€1mL*10mM (DMSO)93,00€10mg101,00€25mg152,00€50mg256,00€100mg460,00€500mg973,00€AC-55541
CAS :AC-55541 (AOB2796), a PAR2 agonist, activates PAR2 in cellular proliferation assays, phosphatidylinositol hydrolysis assays, and Ca(2+) mobilization assays.
Formule :C25H20BrN5O3Degré de pureté :98% - 99.33%Couleur et forme :SolidMasse moléculaire :518.36Litorin acetate(55749-97-8 Free base)
Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.Formule :C53H72N14O13SDegré de pureté :98.61%Couleur et forme :SolidMasse moléculaire :1145.29LY334370
CAS :LY334370 is a selective 5-HT1F receptor agonist with a Ki of 1.6 nMFormule :C21H22FN3ODegré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :351.42Ozagrel hydrochloride
CAS :Ozagrel hydrochloride (OKY-046 HCl) is a selective thromboxane A(2) synthetase inhibitor used for the improvement of postoperative cerebrovascular contractionFormule :C13H12N2O2·HClDegré de pureté :99.80%Couleur et forme :White Or Off White Crystalline PowderMasse moléculaire :264.71CCG215022
CAS :CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 μM and 3.9±1 μM for GRK2, 5 and 1, respectively.Formule :C26H22FN7O3Degré de pureté :97.63% - 99.69%Couleur et forme :SolidMasse moléculaire :499.5Ref: TM-T3498
1mg56,00€5mg114,00€1mL*10mM (DMSO)127,00€10mg178,00€25mg394,00€50mg655,00€100mg1.035,00€Clemizole hydrochloride
CAS :Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.Formule :C19H21Cl2N3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :362.3PF-4136309
CAS :PF-4136309 (INCB8761) is a specific, effective, and orally bioavailable CCR2 antagonist.Formule :C29H31F3N6O3Degré de pureté :98.85% - 99.47%Couleur et forme :SolidMasse moléculaire :568.59PGS-IN-1
CAS :PGS-IN-1 (KME-4) is a potent inhibitor of prostaglandin synthetase (PGS, IC50: 0.28 μM) and 5-lipoxygenase (IC50: 1.05 μM).Formule :C19H26O3Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :302.41BMS-813160
CAS :BMS-813160 is the first dual CCR2/CCR5 antagonist to enter Clinical development for cardiovascular.Formule :C25H40N8O2Degré de pureté :99.66% - 99.79%Couleur et forme :SolidMasse moléculaire :484.64Ref: TM-T4584
1mg63,00€5mg137,00€1mL*10mM (DMSO)145,00€10mg187,00€25mg341,00€50mg567,00€100mg810,00€500mg1.644,00€BX471
CAS :BX471 (BX 471) is a potent, selective non-peptide CCR1 antagonist.Formule :C21H24ClFN4O3Degré de pureté :98% - 99.98%Couleur et forme :SolidMasse moléculaire :434.89Ref: TM-T2375
1mg35,00€5mg86,00€1mL*10mM (DMSO)95,00€10mg117,00€25mg200,00€50mg313,00€100mg489,00€200mg740,00€Glasdegib
CAS :Glasdegib (PF-04449913) (PF-04449913) is a potent, and orally bioavailable Smoothened (Smo) inhibitor with IC50 of 5 nM. Phase 2.Formule :C21H22N6ODegré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :374.44Maraviroc
CAS :Maraviroc: a CCR5 antagonist blocking HIV-1 entry; IC50s—MIP-1α: 3.3nM, MIP-1β: 7.2nM, RANTES: 5.2nM.Formule :C29H41F2N5ODegré de pureté :97.13% - 99.59%Couleur et forme :Brown SolidMasse moléculaire :513.67Ref: TM-T6016
5mg49,00€1mL*10mM (DMSO)56,00€10mg90,00€25mg152,00€50mg259,00€100mg465,00€200mg600,00€500mg945,00€Cenicriviroc
CAS :Cenicriviroc (TAK-652), oral CCR2/CCR5 blocker, inhibits HIV-1/HIV-2, with strong anti-infective/anti-inflammatory effects.Formule :C41H52N4O4SDegré de pureté :97.87%Couleur et forme :SolidMasse moléculaire :696.94Ref: TM-TQ0297
1mg63,00€2mg90,00€5mg133,00€1mL*10mM (DMSO)200,00€10mg212,00€25mg423,00€50mg550,00€100mg715,00€200mg964,00€SAG
CAS :SAG (Smoothened Agonist) is a Smo receptor agonist (EC50=3 nM) that is cell-permeable and selective.
Formule :C28H28ClN3OSDegré de pureté :97.37% - 98.88%Couleur et forme :SolidMasse moléculaire :490.06Ciliobrevin A
CAS :Ciliobrevin A (HPI-4) is an inhibitor of hedgehog signaling pathway with an IC50 <10 μM.Formule :C17H9Cl2N3O2Degré de pureté :98.54% - 99.57%Couleur et forme :SolidMasse moléculaire :358.18Ref: TM-T3156
2mg39,00€5mg56,00€1mL*10mM (DMSO)65,00€10mg80,00€25mg165,00€50mg224,00€100mg314,00€200mg467,00€SANT-1
CAS :SANT-1 directly binds to Smoothened (Smo) receptor (Kd: 1.2 nM) and inhibits Smo agonist effects (IC50: 20 nM).Formule :C23H27N5Degré de pureté :99.93% - >99.99%Couleur et forme :SolidMasse moléculaire :373.49Vercirnon
CAS :Vercirnon (Traficet-EN) is a selective and potent antagonist of CCR9 (IC50: 10 nM). It is also used in the research of inflammatory bowel diseases.Formule :C22H21ClN2O4SDegré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :444.93Ref: TM-T17225
1mg100,00€5mg245,00€1mL*10mM (DMSO)344,00€10mg385,00€25mg645,00€50mg888,00€100mg1.234,00€500mg2.457,00€SAG hydrochloride (912545-86-9(free base))
CAS :SAG hydrochloride (912545-86-9(free base)) (Smoothened Agonist HCl) acts as an SMO agonist.Formule :C28H29Cl2N3OSDegré de pureté :99.19% - 99.97%Couleur et forme :SolidMasse moléculaire :526.52Ref: TM-T4211
1mg49,00€2mg65,00€5mg90,00€1mL*10mM (DMSO)105,00€10mg114,00€25mg222,00€50mg334,00€100mg502,00€200mg717,00€R243
CAS :R243 is CCR8 signaling and chemotaxis inhibitor.Formule :C21H27NO4Degré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :357.44Ref: TM-T24700
1mg40,00€2mg52,00€5mg80,00€1mL*10mM (DMSO)90,00€10mg117,00€25mg207,00€50mg333,00€100mg495,00€Sonidegib
CAS :Sonidegib (Erismodegib), a Smoothened (Smo) antagonist, inhibits Hedgehog (Hh) signaling with IC50 of 1.3 nM (mouse) and 2.5 nM (human), respectively.Formule :C26H26F3N3O3Degré de pureté :98% - 99.97%Couleur et forme :SolidMasse moléculaire :485.5Salmeterol Xinafoate
CAS :Salmeterol Xinafoate (GR 33343X xinafoate) is a long-acting β2-adrenergic receptor agonist with anti-inflammatory effects, used in the treatment of asthma.Formule :C36H45NO7Degré de pureté :98% - 98.24%Couleur et forme :White SolidMasse moléculaire :603.75MRT-81
CAS :MRT-81 blocks Smo receptors in Shh-light2 cells at 41 nM IC50, showing strong hedgehog pathway inhibition, useful in cancer research.Formule :C31H29N3O5SDegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :555.64Ref: TM-T9532
1mg46,00€5mg92,00€1mL*10mM (DMSO)110,00€10mg138,00€25mg241,00€50mg349,00€100mg479,00€200mg657,00€Geissoschizine methyl ether
CAS :Geissoschizine methyl ether: an alkaloid from Uncaria hook, key in Yokukansan, impacts mood and social behavior enhancing serotonin activity.Formule :C22H26N2O3Degré de pureté :99.24% - 99.68%Couleur et forme :SolidMasse moléculaire :366.45Ref: TM-TN1032
1mg130,00€2mg187,00€5mg319,00€1mL*10mM (DMSO)326,00€10mg485,00€25mg770,00€50mg1.035,00€100mg1.395,00€VUF10460
CAS :VUF10460 is a non-imidazole histamine H4 receptor agonist.Formule :C15H19N5Degré de pureté :99.44% - 99.57%Couleur et forme :SolidMasse moléculaire :269.34Ansofaxine hydrochloride
CAS :Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).Formule :C24H32ClNO3Degré de pureté :99.57% - 99.77%Couleur et forme :SolidMasse moléculaire :417.97Treprostinil
CAS :Treprostinil (Orenitram) is a potent DP1, IP and EP2 agonist (EC50: 0.6/1.9/6.2 nM).Formule :C23H34O5Degré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :390.51Ref: TM-T5150
1mg34,00€1mL*10mM (DMSO)60,00€5mg71,00€10mg108,00€25mg221,00€50mg355,00€100mg533,00€200mg755,00€BA 1 acetate(183241-31-8 free base)
BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.Formule :C59H80N14O13Degré de pureté :95.3%Couleur et forme :SolidMasse moléculaire :1193.35Nelotanserin
CAS :Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).Formule :C18H15BrF2N4O2Degré de pureté :98.42% - 99.88%Couleur et forme :SolidMasse moléculaire :437.24Ref: TM-T7350
1mg38,00€2mg50,00€1mL*10mM (DMSO)80,00€5mg84,00€10mg113,00€25mg178,00€50mg333,00€100mg495,00€500mg1.071,00€Lecirelin acetate(61012-19-9 free base)
Lecirelin acetate is a synthetic GnRH (gonadotropin releasing hormone) analogue which shows a great efficacy in the treatment of bovine ovarian follicular cystsFormule :C61H88N16O14Degré de pureté :98.1%Couleur et forme :SolidMasse moléculaire :1269.45Phenylbiguanide
CAS :Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)Formule :C8H11N5Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :177.21Lys-[Des-Arg9]Bradykinin acetate
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 andFormule :C52H77N13O13Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :1092.27I-191
CAS :I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.Formule :C23H26FN5O2Degré de pureté :99.8%Couleur et forme :SolidMasse moléculaire :423.48Gastrin I (human) acetate
Gastrin I (human) acetate (Gastrin-17 acetate) is the endogenous peptide produced in the stomach, and increases gastric acid secretion via cholecystokinin 2 (Formule :C99H128N20O33SDegré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :2158.25AR-M 1896 Acetate
AR-M 1896 Acetate is the selective agonist of GalR2.Formule :C56H85N13O16Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :1196.35Ref: TM-T21646L
1mg305,00€5mg605,00€10mg827,00€25mg1.215,00€1mL*10mM (DMSO)1.251,00€50mg1.603,00€100mg2.142,00€AM966
CAS :AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.Formule :C27H23ClN2O5Degré de pureté :98.06% - 99.79%Couleur et forme :SolidMasse moléculaire :490.93Lurasidone hydrochloride
CAS :Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.Formule :C28H36N4O2S·HClDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :529.14Ref: TM-T1735
5mg39,00€1mL*10mM (DMSO)54,00€10mg59,00€25mg75,00€50mg90,00€100mg137,00€200mg213,00€500mg447,00€Eledoisin Related Peptide 2TFA
Eledoisin Related Peptide 2TFA (Eledoisin Related Peptide 2TFA (2990-43-4(free base))) is a tachykinin receptor ligand.Formule :C38H60F6N8O10SDegré de pureté :99%Couleur et forme :SolidMasse moléculaire :934.99Sitaxsentan sodium
CAS :Sitaxsentan sodium (TBC11251 sodium salt) is a highly selective antagonist of endothelin A receptors.Formule :C18H14ClN2O6S2·NaDegré de pureté :98.39% - 99.01%Couleur et forme :SolidMasse moléculaire :476.89GBR 12935 dihydrochloride
CAS :GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.Formule :C28H36Cl2N2ODegré de pureté :99.09% - ≥95%Couleur et forme :SolidMasse moléculaire :487.5LIXIVAPTAN
CAS :Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)Formule :C27H21ClFN3O2Degré de pureté :98.36%Couleur et forme :SolidMasse moléculaire :473.93Ref: TM-T7303
2mg34,00€5mg66,00€1mL*10mM (DMSO)70,00€10mg99,00€25mg205,00€50mg334,00€100mg522,00€200mg743,00€Pergolide
CAS :Pergolide is a long-acting and orally active dopamine receptor D1/D2 agonist and ergoline derivative, used in the study of Parkinson's diseaseFormule :C19H26N2SDegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :314.49Ref: TM-T21340
2mg37,00€5mg54,00€1mL*10mM (DMSO)60,00€10mg77,00€25mg110,00€50mg164,00€100mg237,00€200mg350,00€FSLLRY-NH2 TFA(245329-02-6 free base)
FSLLRY-NH2 TFA inhibits PAR2, reverses taxol-induced pain, and reduces itch in mice; blocks ERK and collagen in fibroblasts.Formule :C41H61F3N10O10Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :910.99Brexpiprazole
CAS :Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.Formule :C25H27N3O2SDegré de pureté :99.06% - 99.96%Couleur et forme :SolidMasse moléculaire :433.57Ref: TM-T2306
1mL*10mM (DMSO)À demander5mg50,00€10mg63,00€25mg75,00€50mg88,00€100mg94,00€200mg140,00€500mg259,00€NIBR-0213
CAS :NIBR-0213 is a potent and selective competitive S1P1 antagonist.Cost-effective and quality-assured.Formule :C27H29ClN2O3Degré de pureté :98.36% - 99.34%Couleur et forme :SolidMasse moléculaire :464.98Urapidil
CAS :Urapidil (Ebrantil), a sympatholytic antihypertensive drug, acts as a 5-HT1A receptor agonist and as an α1-adrenoceptor antagonist.Formule :C20H29N5O3Degré de pureté :99.85% - >99.99%Couleur et forme :SolidMasse moléculaire :387.48Norepinephrine bitartrate salt
CAS :Norepinephrine bitartrate salt is an adrenergic neurotransmitter.Formule :C12H17NO9Degré de pureté :97.32% - 99.97%Couleur et forme :SolidMasse moléculaire :319.27LRGILS-NH2 acetate
LRGILS-NH2 acetate is a PAR-2-inactive reversed peptide.Formule :C29H56N10O7Degré de pureté :96.65%Couleur et forme :SolidMasse moléculaire :656.82Hemopressin (human, mouse) acetate
Hemopressin: Nonapeptide, α1-hemoglobin derivative, CB1 inverse agonist, isolated from rats, oral, reduces inflammatory pain.Formule :C52H83N13O14Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :1114.29Brimonidine Tartrate
CAS :Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM).Formule :C15H16BrN5O6Degré de pureté :99.95%Couleur et forme :Off-White Crystalline SolidMasse moléculaire :442.22Ki16425
CAS :Ki16425 (Debio 0719) is a competitive, potent and reversible antagonist to LPA1, LPA2 and LPA3 with Ki of 0.34 μM, 6.5 μM and 0.93 μM, respectively.Formule :C23H23ClN2O5SDegré de pureté :97.6% - 97.78%Couleur et forme :SolidMasse moléculaire :474.96Perospirone hydrochloride
CAS :Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.Formule :C23H31ClN4O2SDegré de pureté :99.37%Couleur et forme :White SolidMasse moléculaire :463Serotonin
CAS :Serotonin (5-hydroxytryptamine) is a monoamine neurotransmitter in the CNS and an endogenous 5-HT receptor agonist. High-Quality, Low-Cost!Formule :C10H12N2ODegré de pureté :97.47% - 99.92%Couleur et forme :SolidMasse moléculaire :176.22Melatonin
CAS :Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.Formule :C13H16N2O2Degré de pureté :98% - 99.89%Couleur et forme :Pale Yellow Leaflets From Benzene SolidMasse moléculaire :232.28Verucerfont
CAS :Verucerfont (NBI77860) is an antagonist of corticotropin-releasing factor receptor 1 (CRF1) .Formule :C22H26N6O2Degré de pureté :99.90%Couleur et forme :SolidMasse moléculaire :406.48Ref: TM-T7361
1mg60,00€2mg87,00€5mg130,00€1mL*10mM (DMSO)142,00€10mg205,00€25mg376,00€50mg573,00€100mg803,00€tcY-NH2 TFA(327177-34-4 free base)
tcY-NH2 TFA is a selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.Formule :C42H50F3N7O9Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :853.9PD-168077 maleate
CAS :PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)Formule :C24H26N4O5Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :450.49Ref: TM-T5047
2mg34,00€5mg50,00€1mL*10mM (DMSO)55,00€10mg75,00€25mg142,00€50mg231,00€100mg344,00€200mg490,00€8-Cyclopentyl-1,3-dimethylxanthine
CAS :8-Cyclopentyl-1,3-dimethylxanthine (CPT) is a potent antagonist of adenosine A1 receptor.Formule :C12H16N4O2Degré de pureté :98.58% - 99.9%Couleur et forme :SolidMasse moléculaire :248.283-AQC
CAS :3-AQC is a competitive antagonist of 5-HT3.Formule :C20H21N5O4Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :395.41CHEMBL241987
CAS :CHEMBL241987 targets the Adenosine receptor A3 (human)Formule :C16H11N3ODegré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :261.28Avexitide
CAS :Avexitide (Exendin-3 (9-39) amide) (Exendin (9-39)) is a specific and competitive antagonist of glucagon-like peptide-1 (GLP-1) receptor.Formule :C149H234N40O47SDegré de pureté :98% - 99.65%Couleur et forme :SolidMasse moléculaire :3369.76Methyldopa hydrate
CAS :Methyldopa hydrate (MK-351 hydrate) is a DOPA decarboxylase inhibitor and indirect α2-adrenergic receptor agonist used to treat hypertension.Formule :C10H13NO4H2ODegré de pureté :99.67%Couleur et forme :White SolidMasse moléculaire :238.24Tiprenolol
CAS :Tiprenolol is a beta adrenergic receptor antagonist.[1]Formule :C13H21NO2SDegré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :255.38Ref: TM-T50081
1mg52,00€1mL*10mM (DMSO)89,00€5mg98,00€10mg146,00€25mg235,00€50mg319,00€100mg447,00€200mg587,00€BAR 501 impurity
CAS :BAR 501 impurity 在 BAR501 制剂中发现的一种杂质，可作为 G 蛋白偶联胆汁酸激活受体 (GP-BAR1) 的激动剂。 BAR501 杂质 (10 µM) 在 GP-BAR1 报告基因检测中诱导荧光素酶活性增加 150%。Formule :C26H46O3Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :406.64Conopressin S acetate(111317-90-9 free base)
Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1bFormule :C43H77N17O12S2Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :1088.32AVN-101
CAS :AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.Formule :C21H25ClN2Degré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :340.89Ref: TM-T26690
1mg34,00€5mg75,00€1mL*10mM (DMSO)92,00€10mg114,00€25mg205,00€50mg334,00€100mg557,00€200mg790,00€Canagliflozin
CAS :Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor. Canagliflozin is used to treat type II diabetes mellitus. Cost-effective and quality-assured.Formule :C24H25FO5SDegré de pureté :98.01% - >99.99%Couleur et forme :SolidMasse moléculaire :444.52Ref: TM-T1782
2mg34,00€5mg48,00€1mL*10mM (DMSO)50,00€10mg63,00€25mg82,00€50mg90,00€100mg116,00€500mg260,00€Veralipride
CAS :Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.Formule :C17H25N3O5SDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :383.46Betahistine dihydrochloride
CAS :Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator.Formule :C8H14Cl2N2Degré de pureté :99.22% - 99.88%Couleur et forme :White To Light Yellow Crystalline PowderMasse moléculaire :209.12Mosapride
CAS :Mosapride (AS-4370) is a selective 5HT4 agonistFormule :C21H25ClFN3O3Degré de pureté :99.56%Couleur et forme :White To Off-White Crystalline SolidMasse moléculaire :421.89KH7
CAS :KH7 is a soluble inhibitor of adenylyl cyclase (sAC)-specific.Formule :C17H15BrN4O2SDegré de pureté :98.43%Couleur et forme :SolidMasse moléculaire :419.3ONO-7300243
CAS :ONO-7300243 is an antagonist of lysophosphatidic acid receptor 1 (LPA1; IC50 : 0.16 μM).Formule :C28H31NO5Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :461.55Thrombin Receptor Activator for Peptide
Thrombin Receptor Activator (TRAP) or Coagulation Factor II (1-5), used in CHD research.Formule :C32H51F3N8O9Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :748.79NAN-190 hydrobromide
CAS :NAN-190 hydrobromide is an antagonist of serotonin receptor 5-HT.
Formule :C23H28BrN3O3Degré de pureté :95.20%Couleur et forme :SolidMasse moléculaire :474.39HAEGTFT acetate(926018-95-3 free base)
HAEGTFT acetate is the first N-terminal 1-7 residues of GLP-1 peptide.Formule :C35H51N9O14Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :821.84Linzagolix
CAS :Linzagolix is a small-molecule, non-peptide, orally active gonadotropin-releasing hormone antagonist (GnRH antagonist) which is under development by KisseiFormule :C22H15F3N2O7SDegré de pureté :99.33%Couleur et forme :SolidMasse moléculaire :508.42ACH-000143
CAS :ACH-000143 是一种可口服的褪黑素受体激动剂，对 MT1 和 MT2 的EC50值分别为0.06 和0.32 nM。Formule :C13H16ClN3O3Degré de pureté :98.15%Couleur et forme :SolidMasse moléculaire :297.74Ref: TM-T9193
1mg50,00€5mg110,00€1mL*10mM (DMSO)122,00€10mg172,00€25mg304,00€50mg424,00€100mg583,00€200mg785,00€Ablukast
CAS :Ablukast (Ro 23-3544) is a leuktriene receptor antagonist. Ablukast acts as an anti-asthmatic.Formule :C28H34O8Degré de pureté :98.58%Couleur et forme :SolidMasse moléculaire :498.56GW842166X
CAS :GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.Formule :C18H17Cl2F3N4O2Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :449.25SCH-23390 hydrochloride
CAS :SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Formule :C17H19Cl2NODegré de pureté :98% - 99.83%Couleur et forme :SolidMasse moléculaire :324.24Ref: TM-T4369
1mg39,00€2mg50,00€5mg78,00€1mL*10mM (DMSO)78,00€10mg97,00€25mg195,00€50mg369,00€100mg550,00€Clozapine N-Oxide
CAS :View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.Formule :C18H19ClN4ODegré de pureté :98.65% - 99.94%Couleur et forme :SolidMasse moléculaire :342.82OXA (17-33) acetate
OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).Formule :C79H125N23O22Degré de pureté :98.52%Couleur et forme :SolidMasse moléculaire :1748.98MK-0557
CAS :MK-0557 is a selective and orally available antagonist of the neuropeptide Y5 receptor (Ki: 1.6 nM).Formule :C22H19FN4O3Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :406.41Ref: TM-TQ0286
1mg34,00€5mg67,00€1mL*10mM (DMSO)75,00€10mg92,00€25mg166,00€50mg264,00€100mg371,00€200mg517,00€2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base)
2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) is a potent and selective protease-activated receptor 2 (PAR2) agonist.Formule :C38H64F3N11O10Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :891.98Ditolylguanidine
CAS :Ditolylguanidine (Di-o-tolylguanidine) is an agonist of sigma receptor (σ1/σ2 receptor).Formule :C15H17N3Degré de pureté :98.42%Couleur et forme :White To Pinkish Solid PowderMasse moléculaire :239.32Midodrine
CAS :Midodrine ((±)-Midodrin), an adrenergic alpha-1 agonist, belongs to the class of medications known as vasopressors.Formule :C12H18N2O4Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :254.28CGS 21680 Hydrochloride
CAS :CGS 21680 Hydrochloride (CGS 21680 HCl)(IC50=22 nM), an adenosine receptor agonist, exhibits 140-fold potency in A2 receptor over A1 receptor.Formule :C23H29N7O6·HClDegré de pureté :96.74% - 99.53%Couleur et forme :SolidMasse moléculaire :535.98Ref: TM-T6441
1mg38,00€2mg50,00€5mg81,00€1mL*10mM (DMSO)95,00€10mg109,00€25mg215,00€50mg389,00€100mg575,00€Hydroxyzine dihydrochloride
CAS :Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.Formule :C21H27ClN2O2·2HClDegré de pureté :99.46% - 99.79%Couleur et forme :Oil PowderMasse moléculaire :447.83Dapagliflozin ((2S)-1,2-propanediol, hydrate)
CAS :Dapagliflozin ((2S)-1,2-propanediol, hydrate) (BMS-512148 (2S)-1,2-propanediol, hydrate) is a selective, orally active inhibitor of the renal sodium-glucose co-Formule :C24H35ClO9Degré de pureté :99.88% - 99.94%Couleur et forme :SolidMasse moléculaire :502.98Pridopidine
CAS :Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's R6/2 mice.Formule :C15H23NO2SDegré de pureté :95.2% - 99.89%Couleur et forme :SolidMasse moléculaire :281.41lumateperone Tosylate
CAS :lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Formule :C31H36FN3O4SDegré de pureté :95.83% - 99.95%Couleur et forme :SolidMasse moléculaire :565.7Peptide YY (PYY) (3-36), human
CAS :Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) is a gut hormone peptide. Peptide YY (PYY) (3-36), human acts as a Y2 receptor agonist to reduce appetite.Formule :C176H272N52O54Degré de pureté :97.76%Couleur et forme :SolidMasse moléculaire :3980.42Doxazosin
CAS :Doxazosin (UK 33274) is a long-lasting inhibitor of α1-adrenoceptors that is widely used to treat benign prostatic hyperplasia and lower urinary tract symptoms.Formule :C23H25N5O5Degré de pureté :99.47% - 99.87%Couleur et forme :SolidMasse moléculaire :451.48ZM241385
CAS :ZM-241385 is a high-affinity antagonist ligand selective for the adenosine A2A receptor.
Formule :C16H15N7O2Degré de pureté :97.02% - 99.69%Couleur et forme :SolidMasse moléculaire :337.34Vilazodone Hydrochloride
CAS :Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of theFormule :C26H27N5O2·HClDegré de pureté :99.56% - >99.99%Couleur et forme :SolidMasse moléculaire :477.99S 38093 HCl
CAS :S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.Formule :C17H25ClN2O2Degré de pureté :97.91%Couleur et forme :SolidMasse moléculaire :324.85Ref: TM-T4087
1mg37,00€5mg71,00€1mL*10mM (DMSO)71,00€10mg92,00€25mg164,00€50mg225,00€100mg323,00€200mg437,00€Cetirizine Impurity B dihydrochloride
CAS :Cetirizine Impurity B dihydrochloride is a Cetirizine antihistamine byproduct with anti-allergic properties.Formule :C19H23Cl3N2O2Degré de pureté :97.33%Couleur et forme :SolidMasse moléculaire :417.76Reboxetine mesylate
CAS :Reboxetine mesylate (FCE20124 mesylate) is a norepinephrine reuptake inhibitor (Ki: 8.2 nM).Formule :C19H23NO3·CH4O3SDegré de pureté :99.18% - 99.87%Couleur et forme :Tan Or Off-White Cyrstalline SolidMasse moléculaire :409.5Derenofylline
CAS :Derenofylline is a selective and potent adenosine A(1) antagonist in vitro (Ki=1 nM)Formule :C18H20N4ODegré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :308.38NNC-0640
CAS :NNC-0640 is a negative allosteric modulator of Human Glucagon Receptor with an IC50 of 69.2 nM.Formule :C29H31N7O4SDegré de pureté :97.04%Couleur et forme :SolidMasse moléculaire :573.67Ref: TM-T7364
1mg46,00€2mg62,00€5mg90,00€1mL*10mM (DMSO)90,00€10mg160,00€25mg281,00€50mg430,00€100mg620,00€Diquafosol tetrasodium
CAS :Diquafosol Tetrasodium is a P2Y2 receptor agonist that stimulates the secretion of mucins from ocular tissues Diquafosol tetrasodium (INS365) improves tear filmFormule :C18H22N4Na4O23P4Degré de pureté :98.25% - 99.97%Couleur et forme :SolidMasse moléculaire :878.23Antalarmin
CAS :Antalarmin is a CRHR1 antagonist that blocks adrenocorticotropin-releasing hormone-induced hypertension, blocks CRF activation.Formule :C24H34N4Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :378.55Ref: TM-T70433
1mg81,00€5mg170,00€1mL*10mM (DMSO)173,00€10mg241,00€25mg408,00€50mg552,00€100mg745,00€Xaliproden hydrochloride
CAS :Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.Formule :C24H23ClF3NDegré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :417.89Ref: TM-T9272
1mg38,00€5mg80,00€1mL*10mM (DMSO)92,00€10mg114,00€25mg222,00€50mg356,00€100mg512,00€200mg735,00€CAY10526
CAS :CAY10526 (BTH) is a selective mPGES-1 inhibitor that acts as an inhibitor of the NF-κB signaling pathway.Formule :C12H7BrO3SDegré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :311.15Cerlapirdine
CAS :Cerlapirdine (PF-05212365), a 5-HT6 receptor antagonist, is in trials for Alzheimer's and schizophrenia cognition issues.Formule :C22H23N3O3SDegré de pureté :98.77%Couleur et forme :SolidMasse moléculaire :409.5Ref: TM-T30798
1mg81,00€5mg170,00€1mL*10mM (DMSO)198,00€10mg274,00€25mg543,00€50mg780,00€100mg1.074,00€Elinzanetant
CAS :Elinzanetant is a dual antagonist of neurokinin (NK) receptors 1 and 3 and modulates reproductive hormone secretion.Formule :C33H35F7N4O3Degré de pureté :98% - 99.13%Couleur et forme :SolidMasse moléculaire :668.64Ref: TM-T38144
1mg92,00€2mg118,00€5mg192,00€1mL*10mM (DMSO)284,00€10mg313,00€25mg528,00€50mg740,00€100g4.977,00€M871 acetate
M871 acetate is a selective galanin GAL2 receptor antagonist (Ki values are 13.1 and 420 nM at GAL2 and GAL1 receptors, respectively).It blocks pronociceptiveFormule :C110H167N27O30Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :2347.67Eltoprazine hydrochloride
CAS :Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,Formule :C12H17ClN2O2Degré de pureté :99.35%Couleur et forme :SolidMasse moléculaire :256.73Guanfacine hydrochloride
CAS :Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.Formule :C9H10Cl3N3ODegré de pureté :99.89% - 99.91%Couleur et forme :SolidMasse moléculaire :282.55Galanin Receptor Ligand M35 TFA
Galanin Receptor Ligand M35 TFA is a high-affinity ligand and antagonist of galanin receptor (Kd=0.1 nM).Formule :C109H154N27F3O28Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :2347.62TY-52156
CAS :TY-52156 is an effective and selective S1P3 receptor antagonist (Ki: 110 nM).Formule :C18H19Cl2N3ODegré de pureté :99.91% - 99.91%Couleur et forme :SolidMasse moléculaire :364.27Ref: TM-T17183
2mg38,00€5mg57,00€1mL*10mM (DMSO)63,00€10mg93,00€25mg158,00€50mg281,00€100mg484,00€200mg647,00€BD-1047 dihydrobromide
CAS :BD-1047 dihydrobromide (BD1047.2HBr) , a selective functional antagonist of sigma receptors, has antipsychotic activity in animal models predictive of efficacyFormule :C13H22Br2Cl2N2Degré de pureté :98.13% - 99.39%Couleur et forme :SolidMasse moléculaire :437.04Ref: TM-T1740
1mg37,00€2mg48,00€5mg73,00€1mL*10mM (DMSO)74,00€10mg95,00€25mg168,00€50mg290,00€100mg490,00€Amperozide
CAS :Amperozide (FG 5606), an atypical antipsychotic, antagonizes 5-HT2A and modulates dopamine activity for schizophrenia treatment.Formule :C23H29F2N3ODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :401.49Ref: TM-T23733
1mg87,00€5mg178,00€10mg295,00€1mL*10mM (DMSO)321,00€25mg497,00€50mg708,00€100mg964,00€500mg1.918,00€Nemifitide acetate(173240-15-8 free base)
Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.Formule :C35H47FN10O8Degré de pureté :97.97%Couleur et forme :SolidMasse moléculaire :754.85Carazolol
CAS :Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.Formule :C18H22N2O2Degré de pureté :99% - 99.53%Couleur et forme :Yellowish SolidMasse moléculaire :298.38L-732138
CAS :L-732138 is a potent and competitive antagonist of neurokinin-1 (NK-1) receptor(IC50 : 2.3 nM)Formule :C22H18F6N2O3Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :472.38Ref: TM-T8235
1mL*10mM (DMSO)À demander5mg50,00€10mg80,00€25mg135,00€50mg192,00€100mg286,00€200mg416,00€Indophagolin
CAS :Indophagolin: autophagy inhibitor, IC50 140 nM; blocks P2X4, P2X1, P2X3 receptors, IC50s 2.71, 2.40, 3.49 μM.Formule :C19H15BrClF3N2O3SDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :523.75Phenelzine
CAS :Phenelzine is a MAOI antidepressant, boosting brain catecholamines, effective for endogenous depression.Formule :C8H12N2Degré de pureté :98%Couleur et forme :LiquidMasse moléculaire :136.19Ref: TM-T9540
5mgÀ demander10mgÀ demander25mgÀ demander50mgÀ demander100mgÀ demander200mgÀ demander500mgÀ demanderDesmopressin acetate (16679-58-6 free base)
CAS :Desmopressin (16679-58-6), a synthetic vasopressin analog, treats nocturia, enuresis, and diabetes insipidus by reducing urine production.Formule :C48H68N14O14S2Degré de pureté :98.84% - >99.99%Couleur et forme :SolidMasse moléculaire :1129.26Zatebradine
CAS :Zatebradine is a potent hyperpolarization-activated cyclic nucleotide-gated (HCN) channels inhibitor(IC50 of 1.96 μM).Formule :C26H36N2O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :456.57Azaphen dihydrochloride monohydrate
CAS :Azaphen dihydrochloride monohydrate is a 5-hydroxytryptamine reabsorption inhibitor with antidepressant activity and can be used to study neurological diseases.Formule :C16H23Cl2N5O2Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :388.29RS-67333
CAS :RS-67333 is a partial agonist of 5-HT4R with neuroprotective effects.Formule :C19H29ClN2O2Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :352.9Bay 55-9837 acetate
Bay 55-9837 acetate is a potent and highly selective VPAC2 agonist(Kd = 0.65 nM) and can be used in type 2 diabetes studies.Degré de pureté :98.27%Couleur et forme :LiquidMasse moléculaire :N/APancreatic Polypeptide, rat acetate
Pancreatic Polypeptide, rat acetate is an agonist of NPY receptor, with high affinity at NPYR4.Degré de pureté :97.53%Couleur et forme :SolidMasse moléculaire :N/ARef: TM-TP1044L
1mg215,00€5mg510,00€10mg692,00€25mg1.009,00€50mg1.378,00€100mg1.863,00€200mg2.520,00€Neuropeptide Y (29-64), amide, human acetate
Neuropeptide Y (29-64), amide, human acetate is involved in Alzheimer's disease (AD) and protects rat cortical neurons against β-Amyloid toxicity.Degré de pureté :98.42%Couleur et forme :LiquidMasse moléculaire :N/APancreatic Polypeptide (human) acetate
Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist.Degré de pureté :97.26%Couleur et forme :LiquidMasse moléculaire :N/AHuman growth hormone-releasing factor acetate
Human growth hormone-releasing factor acetate is a hypothalamic polypeptide and stimulates GH production and release by binding to the GHRH Receptor (GHRHR) onDegré de pureté :99.26%Couleur et forme :LiquidMasse moléculaire :N/AK 41498 aceate
K41498 acetate, a potent CRF2 antagonist (Ki: 0.66/0.62 nM for CRF2α/β) with 425 nM for CRF1; blocks aSvg-30 effect on cAMP in cells.Degré de pureté :96.4%Couleur et forme :LiquidMasse moléculaire :N/AVercirnon sodium
CAS :Vercirnon (GSK1605786A) sodium: oral CCR9 antagonist, inhibits Ca2+ mobilization/chemotaxis, IC50 = 2.6-5.4 nM, selective for CCR9 vs. CCR1-12/CX3CR1-7.Formule :C22H21ClN2NaO4SCouleur et forme :SolidMasse moléculaire :467.92BRL-15572 dihydrochloride
CAS :BRL-15572 dihydrochloride: 5-HT1D antagonist, pKi 7.9, also binds 5-HT1A/2B, 60x selective over 5-HT1B.Formule :C25H27ClN2O·2HClDegré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :479.87Neuropeptide S (Rat) acetate
Neuropeptide S (Rat) acetate is an endogenous ligand of a previously orphan G-protein-coupled receptor now named NPS receptor.Formule :C97H164N34O29Degré de pureté :95.36%Couleur et forme :SolidMasse moléculaire :2270.59Ref: TM-TP1982L
1mg93,00€2mg117,00€5mg182,00€10mg269,00€25mg429,00€50mg610,00€100mg820,00€200mg1.099,00€(+)-PD 128907 hydrochloride
CAS :(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .
Formule :C14H20ClNO3Degré de pureté :97.76%Couleur et forme :SolidMasse moléculaire :285.77Histrelin acetate
CAS :Histrelin acetate is a nonapeptide analog of gonadotropin-releasing hormone (GnRH) with added potency.Formule :C68H90N18O14Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :1383.55RFRP3(human) acetate(311309-27-0 free base)
RFRP-3(human) acetate inhibits gonadotropin, blocks Ca2+ mobilization, acts on NPFF1 receptors, and has an IC50 of 0.7 nM against cAMP production.Formule :C47H76N14O12Degré de pureté :97.09%Couleur et forme :SolidMasse moléculaire :1029.19TG4-155
CAS :TG4-155: brain-penetrant EP2 inhibitor, KB 2.4 nM; >1000x weaker at EP4, KB 11.4 μM; selective over other receptors/channels.Formule :C23H26N2O4Degré de pureté :97.2%Couleur et forme :SolidMasse moléculaire :394.46Ref: TM-T5482
2mg35,00€5mg52,00€1mL*10mM (DMSO)57,00€10mg94,00€25mg178,00€50mg313,00€100mg464,00€200mg660,00€Alprenolol benzoate
CAS :Alprenolol benzoate is the benzoate salt of Alprenolol -- a beta blocker.Formule :C22H29NO4Couleur et forme :SolidMasse moléculaire :371.48SB-200646
CAS :SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptorFormule :C15H14N4ODegré de pureté :99.61%Couleur et forme :SolidMasse moléculaire :266.3ML221
CAS :ML221 is a potent apelin /APJ functional antagonist, inhibiting apelin-13-mediated activation of APJ, with IC50s of 0.70 μM in the cAMP assay, and 1.75 μM inFormule :C17H11N3O6SDegré de pureté :97.74%Couleur et forme :SolidMasse moléculaire :385.35Ref: TM-T4390
2mg34,00€5mg50,00€1mL*10mM (DMSO)52,00€10mg80,00€25mg137,00€50mg215,00€100mg349,00€200mg512,00€Obestatin (rat) acetate
Obestatin (rat) acetate is an endogenous ligand of G-protein coupled receptor 39 (GPR39).Formule :C114H174N34O31Degré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :2516.81Ref: TM-TP2279L
1mg77,00€2mg97,00€5mg156,00€10mg225,00€25mg375,00€50mg535,00€100mg730,00€200mg938,00€FAUC-365
CAS :FAUC-365 is a D3 dopamine receptor agonist.Formule :C23H25Cl2N3OSDegré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :462.44Ref: TM-T21667
1mg50,00€5mg105,00€1mL*10mM (DMSO)116,00€10mg160,00€25mg305,00€50mg485,00€100mg700,00€500mg1.459,00€Vipadenant
CAS :Vipadenant (CEB-4520)(BIIB-014) is an adenosine A2a antagonist with Ki of 1.3 nM; less potent for A1(Ki=69 nM).Formule :C16H15N7ODegré de pureté :97.25% - 97.36%Couleur et forme :SolidMasse moléculaire :321.34Ref: TM-T2373
2mg35,00€5mg51,00€10mg80,00€25mg131,00€50mg210,00€1mL*10mM (DMSO)215,00€100mg313,00€200mg445,00€γ-Mangostin
CAS :Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.Formule :C23H24O6Degré de pureté :98.55% - 99.08%Couleur et forme :SolidMasse moléculaire :396.43Lurasidone
CAS :Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Formule :C28H36N4O2SDegré de pureté :99.78% - 99.91%Couleur et forme :SolidMasse moléculaire :492.68Substance P (7-11)
CAS :Substance P (7-11) (Substance P 7-11(TFA)) is a C-terminal fragment of Substance P .Formule :C31H44N6O5SDegré de pureté :98.39%Couleur et forme :SolidMasse moléculaire :612.78Aplindore
CAS :Aplindore is a dopamine receptor agonist used in the therapeutic treatment of Parkinson's Disease.Formule :C18H18N2O3Couleur et forme :SolidMasse moléculaire :310.35Talnetant hydrochloride
CAS :Talnetant (SB 223412) hydrochloride, an NK3 antagonist, selectively binds hNK-3 at 1.4 nM, much less to hNK-2, none to hNK-1 at 100 μM.Formule :C25H23ClN2O2Couleur et forme :SolidMasse moléculaire :418.92Decynium 22
CAS :Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitorFormule :C23H23IN2Degré de pureté :99.92%Couleur et forme :Dark Red CrystalsMasse moléculaire :454.35Diclofensine hydrochloride
CAS :Diclofensine hydrochloride (Ro 8-4650 hydrochloride) 是一种高效单胺再摄取抑制剂，在大鼠脑突触体中能够阻断多巴胺 (IC50=0.74 nM)、去甲肾上腺素 (IC50=2.3 nM) 和 5-羟色胺 (IC50=3.7 nM)。Formule :C17H18Cl3NODegré de pureté :98.86% - 99.93%Couleur et forme :SolidMasse moléculaire :358.69ML-191
CAS :ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2.Formule :C24H25N3O3Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :403.47Quipazine
CAS :Quipazine: 5-HT agonist, Ki 1.4 nM at 5-HT3R, anti-SARS-CoV-2 (EC50 31.64 μM), for neurological research.Formule :C13H15N3Couleur et forme :SolidMasse moléculaire :213.28
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