GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(251 produits)
- Récepteur adrénergique(3.027 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(218 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(36 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(195 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
6011 produits trouvés pour "GPCR/G-Protéine"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
UCM 608
CAS :UCM 608 (2-Phenylmelatonin) is an antagonist of melatonin-induced contractile responses at low concentrations and induces an increase in GDP-GTP exchange.Formule :C19H20N2O2Degré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :308.37Atipamezole
CAS :Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.Formule :C14H16N2Degré de pureté :99.88%Couleur et forme :Off-White To Light Yellow Crystal PowderMasse moléculaire :212.29Canagliflozin hemihydrate
CAS :Canagliflozin hemihydrate (TA 7284) treats type 2 diabetes by blocking SGLT2, leading to glucose excretion in urine.Formule :C48H52F2O11S2Degré de pureté :99.42% - 99.96%Couleur et forme :SolidMasse moléculaire :907.05Opipramol
CAS :Opipramol (Ensidon) is a compound with antidepressant activity, a sigma (σ) receptor agonist, and anxiolytic activity.Formule :C23H29N3ODegré de pureté :99.84% - 99.98%Couleur et forme :SolidMasse moléculaire :363.5Dexpramipexole
CAS :Dexpramipexole ((R)-Pramipexole) is a mitochondrial protective agent that maintains mitochondrial function and energy production.Formule :C10H17N3SDegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :211.33Rolofylline
CAS :Rolofylline (KW-3902) is an adenosine A1 receptor antagonist used to study acute congestive heart failure and renal dysfunction.Formule :C20H28N4O2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :356.46INCB 3284
CAS :INCB 3284, a potent human CCR2 antagonist with an IC50 of 3.7 nM, is researchable for acute liver failure and inhibits MCP-1/hCCR2 binding.Formule :C26H31F3N4O4Degré de pureté :97.81% - 99.42%Couleur et forme :SolidMasse moléculaire :520.54CB1/2 agonist 3
CAS :CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.Formule :C25H41NO2Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :387.6WIN 51,708
CAS :WIN 51,708 is an antagonist of neurokinin-1 receptor.Formule :C29H33N3ODegré de pureté :99%Couleur et forme :SolidMasse moléculaire :439.59AF-710B
CAS :AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.Formule :C20H27N3OSDegré de pureté :98.62% - 99.89%Couleur et forme :SolidMasse moléculaire :357.51Renzapride
CAS :Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.Formule :C16H22ClN3O2Degré de pureté :98.97% - 99.09%Couleur et forme :SolidMasse moléculaire :323.82Ref: TM-T38507
1mg93,00€2mg124,00€5mg200,00€10mg359,00€25mg692,00€50mg945,00€100mg1.279,00€200mg1.701,00€Atogepant
CAS :Atogepant (MK-8031) is an orally available, selective and potent calcitonin gene-related peptide receptor (CGRP) antagonist for the study of migraine.Formule :C29H23F6N5O3Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :603.52Ref: TM-T26682
1mg147,00€5mg250,00€10mg313,00€1mL*10mM (DMSO)334,00€25mg620,00€50mg1.108,00€100mg1.611,00€200mg2.178,00€Jatrorrhizine chloride
CAS :Jatrorrhizine chloride (Neprotine chloride) is an alkaloid isolated from Rhizoma coptidis with neuroprotective, antimicrobial, and antiplasmodial activities.Formule :C20H20ClNO4Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :373.8(S)-Mirtazapine
CAS :(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.Formule :C17H19N3Degré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :265.35Levocetirizine Dihydrochloride
CAS :Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.Formule :C21H27Cl3N2O3Degré de pureté :99.89%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :461.81Protein deglycase DJ-1 against-1
CAS :Protein deglycase DJ-1 against-1 penetrate the BBB and bind to DJ-1 protein,restoring neuronal cellular death in a neurotoxin MPTP-induced model of PD.Formule :C24H23N3O4Degré de pureté :97.23%Couleur et forme :SolidMasse moléculaire :417.46Pentoxyverine
CAS :Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.Formule :C20H31NO3Degré de pureté :97.11%Couleur et forme :SolidMasse moléculaire :333.47Fenoprofen
CAS :Fenoprofen (LILLY-5385) is a non-steroidal anti-inflammatory compound and a modifier enhancer of the melanocortin receptor, increasing ERK1/2 activation.Formule :C15H14O3Degré de pureté :98.4%Couleur et forme :SolidMasse moléculaire :242.27(S)-VU0637120
CAS :(S)-VU0637120 is a selective neuropeptide Y(4)R-mutant antagonist used in the study of metabolic disorders.Formule :C16H19N3O5S2Degré de pureté :99.74%Couleur et forme :SolidMasse moléculaire :397.47Trabodenoson
CAS :Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.Formule :C15H20N6O6Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :380.36Ref: TM-T34914
1mg40,00€1mL*10mM (DMSO)88,00€5mg89,00€10mg116,00€25mg187,00€50mg285,00€100mg411,00€200mg577,00€LP-533401 hydrochloride
CAS :LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.Formule :C27H23ClF4N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :562.94S-Methoprene
CAS :S-Methoprene (ZR2458), a juvenile hormone analog, acts as an insecticide influencing redox activity and male sex differentiation.
Formule :C19H34O3Degré de pureté :97.05% - 98.55%Couleur et forme :SolidMasse moléculaire :310.47Medetomidine
CAS :Medetomidine (MPV785 free base) is a selective α2-adrenoceptor agonist, with sedative and analgesic and vasoconstrictive hypoxic , in small animal anesthesia.Formule :C13H16N2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :200.28Ref: TM-T21492
2mg38,00€5mg57,00€1mL*10mM (DMSO)62,00€10mg77,00€25mg128,00€50mg193,00€100mg290,00€200mg447,00€Nebentan potassium
CAS :Nebentan potassium (YM598) is an ETA receptor antagonist that inhibits pulmonary arterial hypertension and is used in the study of neurologic diseases.Formule :C24H20KN5O5SDegré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :529.61Ref: TM-T36008
1mg52,00€2mg77,00€5mg111,00€1mL*10mM (DMSO)133,00€10mg177,00€25mg313,00€50mg502,00€100mg680,00€200mg888,00€WAY-100635 maleate
CAS :WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).Formule :C25H34N4O2·xC4H4O4Degré de pureté :99.96%Couleur et forme :White SolidMasse moléculaire :538.645Ref: TM-T3453
2mg43,00€5mg63,00€1mL*10mM (DMSO)74,00€10mg89,00€25mg150,00€50mg215,00€100mg316,00€500mg765,00€Poly-D-lysine hydrobromide (MW 30000-70000)
CAS :Poly-D-lysine hydrobromide (MW 30000-70000) (Poly-D-lysine HBr) is a peptide CaSR agonist that removes proteinase K-resistant PrP from SN56 neuroblastoma cells.Formule :(C6H14N2O2)x·xHBrCouleur et forme :SolidMasse moléculaire :227.102Ozanimod hydrochloride
CAS :Ozanimod (RPC-1063) HCl is a selective S1P1/S1P5 modulator with high affinity, used in relapsing MS research.Formule :C23H25ClN4O3Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :440.92Ref: TM-T62552
1mg47,00€5mg92,00€1mL*10mM (DMSO)101,00€10mg137,00€25mg268,00€50mg432,00€100mg620,00€200mg875,00€BMS-986278
CAS :BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb values of 6.9 nM and 4.0 nM for human and mouse LPA1,Formule :C22H31N5O5Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :445.51Citalopram
CAS :Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.Formule :C20H21FN2ODegré de pureté :99.78% - 99.89%Couleur et forme :SolidMasse moléculaire :324.39GAT211
CAS :GAT211 (AZ-4) is a cannabinoid 1 receptor (CB1R) positive allosteric modulator (PAM) for the study of epilepsy.Formule :C22H18N2O2Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :342.39Ref: TM-T27405
1mg34,00€5mg66,00€1mL*10mM (DMSO)73,00€10mg90,00€25mg148,00€50mg210,00€100mg310,00€500mg750,00€SB 243213
CAS :SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.Formule :C22H19F3N4O2Degré de pureté :98.78% - 99.86%Couleur et forme :SolidMasse moléculaire :428.41(R)-Mirtazapine
CAS :(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.Formule :C17H19N3Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :265.35Latrepirdine dihydrochloride
CAS :Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.Formule :C21H25N3·2HClDegré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :392.37Trazpiroben
CAS :Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.Formule :C31H39N3O4Degré de pureté :99.41% - >99.99%Couleur et forme :SolidMasse moléculaire :517.66Benzylthiouracil
CAS :Benzylthiouracil (6-Benzyl-2-thiouracil) induces ANCA-associated glomerulonephritis in Graves' disease patients and is used to study hyperthyroidism.Formule :C11H10N2OSDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :218.28Syk Inhibitor II
CAS :Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).Formule :C14H15F3N6ODegré de pureté :97.63%Couleur et forme :SolidMasse moléculaire :340.3(S)-Pramipexole-(N-Propyl-2,2,3,3,3-d5) Dihydrochloride
CAS :(S)-Pramipexole-(N-Propyl-2,2,3,3,3-d5) Dihydrochloride is a deuterated compound of (S)-Pramipexole Dihydrochloride. (S)-Pramipexole Dihydrochloride has a CAS number of 104632-25-9. Pramipexole dihydrochloride could be used to treat Parkinson disease.Formule :C10H14D5Cl2N3SCouleur et forme :SolidMasse moléculaire :289.28Hydroxyzine-d8 DiHCl
CAS :Hydroxyzine-d8 DiHCl is a deuterated compound of Hydroxyzine DiHCl. Hydroxyzine DiHCl has a CAS number of 2192-20-3.Formule :C21H21D8Cl3N2O2Couleur et forme :SolidMasse moléculaire :455.88Ropinirole
CAS :Ropinirole, D2-like agonist, no D1 affinity, Ki 29 nM for D2, treats Parkinson's.Formule :C16H24N2ODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :260.38SR59230A hydrochloride
CAS :SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue thermogenesis.Formule :C21H28ClNO2Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :361.91L-745870
CAS :L-745870 is a D4 receptor antagonist that also inhibits D2 receptors, 5-HT2 receptors, and α-adrenergic receptors.Formule :C18H19ClN4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :326.82R 59-022
CAS :R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.Formule :C27H26FN3OSDegré de pureté :98.55%Couleur et forme :SolidMasse moléculaire :459.58Ref: TM-T16709
1mg35,00€5mg74,00€1mL*10mM (DMSO)75,00€10mg119,00€25mg269,00€50mg447,00€100mg733,00€200mg973,00€Travoprost
CAS :Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.Formule :C26H35F3O6Degré de pureté :97.39% - 99.58%Couleur et forme :Colorless OilMasse moléculaire :500.55Ref: TM-T5841
1mg46,00€5mg88,00€1mL*10mM (DMSO)96,00€10mg120,00€25mg175,00€50mg255,00€100mg371,00€200mg507,00€PACAP (1-38), human, ovine, rat
CAS :PACAP (1-38), human, ovine, rat (Pituitary Adenylate Cyclase Activating Polypeptide 38) is a neuropeptide with 38 amino acid residues.Formule :C203H331N63O53SDegré de pureté :96.93% - 98.16%Couleur et forme :SolidMasse moléculaire :4534.26Cyproheptadine hydrochloride
CAS :Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.Formule :C21H21N·HClDegré de pureté :99.88% - 99.97%Couleur et forme :SolidMasse moléculaire :323.86Mibavademab
CAS :Mibavademab is a humanized anti-leptin receptor (LEPR) mAb under investigation for treating congenital leptin deficiency.Degré de pureté :95%Couleur et forme :LiquidMasse moléculaire :~150 kDaArazasetron HCl
CAS :Arazasetron is an antiemetic which acts as a 5-HT3 receptor antagonist, pKi = 9.27.Formule :C17H20ClN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :349.81DL-Phenylephrine HCl
CAS :DL-Phenylephrine HCl is a selective agonist of the alpha1-adrenergic receptor.Formule :C9H14ClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :203.67Keto Ziprasidone
CAS :Ziprasidone, an antipsychotic agent, functions as a dual antagonist of 5-HT (serotonin) and dopamine receptors.Formule :C21H19ClN4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :426.92GPR183-IN-1
CAS :GPR183-IN-1 (compound 15) is an effective orally active inhibitor of GPR183. It inhibits Ca2+ mobilization with an IC50 value of 39.97 nM. GPR183-IN-1 holds potential for research in cancer, autoimmune diseases, pain, and osteoporosis.Formule :C16H19BrN2O2Couleur et forme :SolidMasse moléculaire :351.24Fremanezumab
CAS :Fremanezumab (TEV-48125) is a humanised monoclonal antibody targeting CGRP, capable of neutralising human, mouse and rat CGRP, migraine.Degré de pureté :95% - 97.6% (SDS-PAGE); 95.9% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :145.49 kDaEscitalopram
CAS :Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.Formule :C20H21FN2ODegré de pureté :99.82%Couleur et forme :White Or White Crystalline PowderMasse moléculaire :324.39N-Methyl amisulpride
CAS :N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.Formule :C18H29N3O4SCouleur et forme :SolidMasse moléculaire :383.51P2Y14R antagonist 1
CAS :P2Y14R antagonist 1 (compound I-17) is a selective oral that inhibits inflammatory response in acute gouty arthritis the NLRP3/GSDMD y and cellular pyroptosis.Formule :C15H12BrN3O2Degré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :346.18Eptinezumab
CAS :Eptinezumab is a humanised monoclonal antibody targeting CGRP (calcitonin gene-related peptide), which prevents CGRP binding to its receptor, migraine.
Degré de pureté :95% - 95%Couleur et forme :LiquidTriflupromazine
CAS :Triflupromazine is a dopamine receptor D1/D2 antagonist and LHDA inhibitor that suppresses dopamine activity in (CNS)mental disorders, sedation, and antiemesis.Formule :C18H19F3N2SCouleur et forme :SolidMasse moléculaire :352.42Buflomedil
CAS :Buflomedil is a vasoactive compound. Buflomedil has been used for peripheral arterial diseases.Formule :C17H25NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :307.38Meticillin
CAS :Methicillin: Narrow-spectrum beta-lactam, penicillin-type antibiotic for certain gram-positive bacterial infections.Formule :C17H20N2O6SCouleur et forme :SolidMasse moléculaire :380.42Carlumab
CAS :Carlumab is a high-affinity human monoclonal antibody that targets CCL2, suppressing the recruitment of monocytes/macrophages in the tumour microenvironment.Degré de pureté :95%Couleur et forme :LiquidMasse moléculaire :144.87 kDaGLP-1 Receptor modulator 1
CAS :GLP-1 Receptormodulator 1 (Compound 7) is an effective positive allosteric modulator of the GLP-1 receptor. It is utilized in the research of obesity and type 2 diabetes.Formule :C18H21NOSMasse moléculaire :299.43Metoxibutropate
CAS :Metoxibutropate is a biochemical.Formule :C20H24O3Couleur et forme :SolidMasse moléculaire :312.4Olopatadine
CAS :Olopatadine is an antihistamine and anti-allergy medication for itchy eyes, also possibly treats red skin syndrome.Formule :C21H23NO3Degré de pureté :98%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :337.41Methaphenilene hydrochloride
CAS :Methaphenilene hydrochloride is an H1 receptor antagonist with antihistaminic and anticholinergic activity, in allergic inflammation and autonomic research.Formule :C15H21ClN2SDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :296.86Risperidone Mesylate
CAS :Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.Formule :C24H31FN4O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :506.5917-phenyl trinor Prostaglandin F2α isopropyl ester
CAS :17-phenyl trinor PGF2α N-ethyl amide is an F-series prostaglandin analog which has been approved for use as an ocular hypotensive drug, sold under the AllerganFormule :C26H38O5Couleur et forme :SolidMasse moléculaire :430.58Blontuvetmab
CAS :Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].Degré de pureté :95% - 95%Couleur et forme :LiquidRocatinlimab
CAS :Rocatinlimab (AMG 451) (KHK4083) is a fully human, non-fucosylated IgG1 anti-OX40 monoclonal antibody indicated for atopic dermatitis (AD) research [1].Couleur et forme :LiquidPF-610355
CAS :PF-610355 is a long-acting and potent β2-adrenergic receptor agonist (EC50: 0.26 nM).PF-610355 can be used to study asthma and COPD.
Formule :C34H39N3O6SDegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :617.76Tulobuterol
CAS :Tulobuterol is mainly used for the prevention and treatment of bronchial asthma, asthmatic bronchitis and chronic bronchitis. Research shows that it could inhibit rhinovirus infection in primary cultures of human tracheal epithelial cells.Formule :C12H18ClNOCouleur et forme :Crystalline SolidMasse moléculaire :227.73Mirtazapine D3
CAS :Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .Formule :C17H19N3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :268.37Mianserin-d3
CAS :Mianserin-d3 is a deuterated compound of Mianserin. Mianserin has a CAS number of 24219-97-4. Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, antianxiety, antiemetic, hypotrophic, hypnotic and antihistamine effects, and can be used as a combination of norepinephrine and specific serotonin to treat depression.Formule :C18H17D3N2Couleur et forme :SolidMasse moléculaire :267.38Brexpiprazole-d8
CAS :Brexpiprazole D8 is a deuterium-modified partial agonist of 5-HT1A and dopamine receptors, with Ki values of 0.12 nM and 0.3 nM respectively.Formule :C25H27N3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :441.62Dapagliflozin-d5
CAS :Dapagliflozin D5 (BMS-512148 D5) is deuterated Dapagliflozin. Dapagliflozin is a competitive SGLT2 inhibitor.Formule :C21H25ClO6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :413.9Amitriptyline-d6 Hydrochloride
CAS :Amitriptyline-d6 Hydrochloride is a deuterated compound of Amitriptyline Hydrochloride. Amitriptyline Hydrochloride has a CAS number of 549-18-8. Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.Formule :C20H18D6ClNCouleur et forme :SolidMasse moléculaire :319.90Cinnarizine D8
CAS :Cinnarizine D8 is a deuterium-labeled Cinnarizine which is an antihistamine and a calcium channel blocker.Formule :C26H28N2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :376.57315-keto Prostaglandin F2α
CAS :15-keto Prostaglandin F2α is a metabolite of Prostaglandin F2α that lowers intraocular pressure in rabbits.Formule :C20H32O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :352.47Dopamine D4 receptor ligand 2
CAS :Compound 17, a dopamine D4 receptor ligand, exhibits high potency and selectivity with IC 50 values of 0.057 nM for D4, and >1000, 220, and 270 nM for D2, 5-HT1A, and α1 receptors, respectively [1].Formule :C20H24ClN3O2Couleur et forme :SolidMasse moléculaire :373.88AR244555
CAS :AR244555 is a bioactive chemical.Formule :C23H23ClF2N2OCouleur et forme :SolidMasse moléculaire :416.89Atenolol Hydrochloride
CAS :Atenolol Hydrochloride is a selective antagonist of ß1 receptor.Formule :C14H23ClN2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :302.80PSB-KK1445
CAS :PSB-KK1445 is a potent and selective agonist of GPR18, exhibiting EC50 values of 45.4 nM for humans and 124 nM for mice. The selectivity of PSB-KK1445 for GPR18 over the CB receptor subtypes GPR55 and GPR183 exceeds 200-fold.Formule :C24H23FN6O2Masse moléculaire :446.486-hydroxy Buspirone
CAS :6-Hydroxy Buspirone, an active metabolite of the anxiolytic compound buspirone, is produced via the cytochrome P450 (CYP) isoform CYP3A4.Formule :C21H31N5O3Couleur et forme :SolidMasse moléculaire :401.507-Desmethyl-3-hydroxyagomelatine
CAS :7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.Formule :C14H15NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :245.277-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene
CAS :7-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene is a liver receptor homolog-1 (LRH-1) antagonist (IC50: 3.1 μM).Formule :C42H44N2O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :704.87Ridazolol HCl
CAS :Ridazolol HCl (CAS 413) is a novel β-adrenoceptor (β-AR) blocker with α-adrenerolytic activity.Formule :C15H19Cl3N4O3Degré de pureté :99.48%Couleur et forme :SoildMasse moléculaire :409.75-Methyltryptamine hydrochloride
CAS :5-Methyltryptamine hydrochloride is a high-affinity 5-HT1C receptor ligand and a partial agonist of 5-HT. 5-Methyltryptamine hydrochloride protects mice subjected to burn, tourniquet and endotoxin shock.Formule :C11H15ClN2Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :210.703Dehydroabiethylamine
CAS :Dehydroabiethylamine (NSC-2955) boosts liver CYP2B, blocks PDKs & cholesterol transport, and has anti-tumor effects.Formule :C20H31NDegré de pureté :98.79%Couleur et forme :Pale Yellow Viscous Liquid /Technical Grade/ Viscous Colorless To Amber LiquidMasse moléculaire :285.47Vanoxerine
CAS :Vanoxerine is an antagonist of dopamine transporter (Ki: 16.9nM).Formule :C28H32F2N2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :450.56MK-447
CAS :MK-447 is a nonsteroidal antiinflammatory agent.Formule :C11H16INODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :305.16Penbutolol sulfate
CAS :Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.Formule :C18H29NO2H2O4SDegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :340.47Roxatidine acetate
CAS :Roxatidine acetate: anti-ulcer, blocks histamine, reduces acid. Safer at lower doses.Formule :C19H28N2O4Degré de pureté :98%Couleur et forme :White Or Off-White PowderMasse moléculaire :348.44Itopride free base
CAS :Itopride HCl combats dyspepsia and GERD, inhibiting AChE and blocking D2 receptors.
Formule :C20H26N2O4Couleur et forme :WhiteMasse moléculaire :358.43Pardoprunox
CAS :Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.Formule :C12H15N3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :233.27Caerulein, desulfated
CAS :Caerulein, desulfated (FI-6934, desulfated) is a desulfated compound formed after caerulein hydrolysis, a neuropeptide with lower smooth muscle activity.Formule :C58H73N13O18SDegré de pureté :99.46%Couleur et forme :SolidMasse moléculaire :1272.34Tivumecirnon
CAS :Tivumecirnon (FLX475) is a selective and oral CCR4 antagonist inhibits the infiltration and migration of Treg into the tumour microenvironment, antitumourFormule :C24H27Cl2F3N6ODegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :543.41Ref: TM-T69834
1mg171,00€5mg418,00€1mL*10mM (DMSO)500,00€10mg666,00€25mg1.334,00€50mg2.071,00€100mg2.879,00€Bethanidine sulfate
CAS :Bethanidine sulfate and its ortho-chloro derivative (BW 392C60) are potent adrenergic neuron blockers exhibiting sympathomimetic effects similar to those of bromobenzamine and guanethidine in various animal models, particularly in cats. These compounds inhibit the release of norepinephrine during neural stimulation and enhance the responsiveness of smooth muscle to epinephrine and norepinephrine. Notably, bethanidine sulfate increases the pressor response to tyramine, although this effect diminishes with higher doses. Unlike guanethidine, bethanidine sulfate does not deplete pressor amines in the iris of cats following administration. Additionally, it temporarily suppresses autonomic cholinergic mechanisms and can cause transient neuromuscular paralysis at large doses, contrasting its long-term adrenergic neuron blocking effects.Formule :C20H32N6O4SCouleur et forme :SolidMasse moléculaire :452.57S 25585
CAS :S 25585 is a neuropeptide Y (NPY) Y5 receptor antagonist.Formule :C22H23F3N4O6SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :528.5R-138727
CAS :R-138727 is a novel P2Y12 receptor inhibitor.Formule :C18H20FNO3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :349.42Isoproterenol sulfate anhydrous
CAS :Isoproterenol sulfate anhydrous is a useful alkaloid. It is used for biological research.Formule :C22H36N2O10SDegré de pureté :98%Couleur et forme :CoaMasse moléculaire :520.59Ticlopidine
CAS :Ticlopidine (PCR 5332) is an antiplatelet drug in the thienopyridine family which is an adenosine diphosphate (ADP) receptor inhibitor.Formule :C14H14ClNSDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :263.79Amthamine
CAS :Compound AMTHAMINE DIHYDROBROMIDE is a useful organic compound for research related to life sciences.Formule :C6H11N3SCouleur et forme :SoildMasse moléculaire :157.24Ketanserinol
CAS :Ketanserinol is a metabolite of the antihypertensive drug ketanserin, which blocks 5-HT2 receptors to treat protamine-induced pulmonary hypertension.Formule :C22H24FN3O3Couleur et forme :SolidMasse moléculaire :397.44Proxyfan Oxalate
CAS :Proxyfan Oxalate is a potent antagonist of the histamine H3 receptor (histamine H3 receptor), with Ki values of 2.9 nM for rats and 2.7 nM for humans. Its inhibitory effect on H3 receptors is over 1000 times stronger than its effect on other histamine receptors.Formule :C15H18N2O5Couleur et forme :SolidMasse moléculaire :306.31Ciproxifan
CAS :Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).Formule :C16H18N2O2Degré de pureté :98.00%Couleur et forme :SolidMasse moléculaire :270.33Amidephrine hydrochloride
CAS :Amidephrine hydrochloride is a biochemical.Formule :C10H17ClN2O3SCouleur et forme :SolidMasse moléculaire :280.77Amidephrine
CAS :Amidephrine is an adrenergic agent.Formule :C10H16N2O3SCouleur et forme :SolidMasse moléculaire :244.31Litorin
CAS :Litorin suppresses appetite and stimulates smooth muscle, gastrin, gastric acid, and pancreatic secretion.Formule :C51H68N14O11SCouleur et forme :White PowderMasse moléculaire :1085.24SB 271046 hydrochloride
CAS :SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is > 200-fold selective over 55 other receptors, enzymes and ion channels.Formule :C20H22ClN3O3S2·HClDegré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :488.45Norreticuline
CAS :Norreticuline is a potential adrenoceptor-α/β agonist and CYP2D6 and D2 receptor inhibitor for the study of neurodegenerative diseases.Formule :C18H21NO4Couleur et forme :SolidMasse moléculaire :315.36(RS)-ICI-118551 Hydrochloride
CAS :ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3Formule :C17H27NO2·HClDegré de pureté :98.02%Couleur et forme :SolidMasse moléculaire :313.86Diclofensine
CAS :Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.Formule :C17H17Cl2NODegré de pureté :97.01% - 98.13%Couleur et forme :SolidMasse moléculaire :322.23Hydroxy ziprasidone
CAS :Hydroxy ziprasidone is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a 5-HT and dopamine receptor antagonist.Formule :C21H21ClN4O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :428.94MCI-225 dehydratase
CAS :MCI-225 dehydratase is an oral, selective inhibitor of noradrenaline reuptake, and functions as a 5-HT3 antagonist, exhibiting antidepressant effects in vivo .Formule :C17H18ClFN4SCouleur et forme :SolidMasse moléculaire :364.87Paroxetine hydrochloride hemihydrate
CAS :Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).Formule :C38H44Cl2F2N2O7Degré de pureté :99.949%Couleur et forme :SolidMasse moléculaire :749.67LY 344864
CAS :LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.Formule :C21H22FN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :351.42Guacetisal
CAS :Guacetisal, from acetylsalicylic acid and guaiacol, may treat chronic bronchitis.Formule :C16H14O5Degré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :286.28Ref: TM-T15447
2mg43,00€5mg60,00€1mL*10mM (DMSO)73,00€10mg99,00€25mg177,00€50mg225,00€100mg316,00€200mg442,00€Lodoxamide tromethamine
CAS :Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergicFormule :C19H28ClN5O12Degré de pureté :98.8%Couleur et forme :SolidMasse moléculaire :553.91MK-5046
CAS :MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).Formule :C20H18F6N4ODegré de pureté :98.56%Couleur et forme :SolidMasse moléculaire :444.37Dolasetron Mesylate
CAS :Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea followingFormule :C20H24N2O6SDegré de pureté :99.05%Couleur et forme :White PowderMasse moléculaire :420.48RP101442
CAS :RP101442: Ozanimod metabolite, selective S1PR1 agonist, EC50: 2.6 nM (S1PR1), 171 nM (S1PR5).Formule :C23H22N4O3Couleur et forme :SolidMasse moléculaire :402.45RXFP3/4 agonist 2
CAS :RXFP3/4 agonist 2 is a nonpeptide bis-RXFP3/4 agonist used in the study of diseases caused by metabolic abnormalities.Formule :C22H22N6O2Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :402.45FR-194921
CAS :FR-194921: potent oral adenosine A1 antagonist, improves cognition, reduces anxiety, similar efficacy in humans, rats, mice.Formule :C23H23N5OCouleur et forme :SolidMasse moléculaire :385.46GSK-239512
CAS :GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.Formule :C23H27N3O2Degré de pureté :99.62% - 99.74%Couleur et forme :SolidMasse moléculaire :377.48L 11204
CAS :L 11204 is an antifertility in vivo. It is an inhibitor of prostaglandin synthesis.Formule :C18H17N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :291.35T-0509
CAS :T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle and selectively down-regulates rat cardiac beta 1-
Formule :C18H23NO5Degré de pureté :97.52% - 98.43%Couleur et forme :SolidMasse moléculaire :333.38ST3932
CAS :ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).Formule :C12H16N8ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :288.31Odapipam
CAS :Odapipam is a selective and high affinity antagonist of benzazepine dopamine D1 receptor (Kd of 0.18 nM).Formule :C19H20ClNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :329.82TD-5471 hydrochloride
CAS :TD-5471 hydrochloride is a selective and potent long-acting human β2-adrenergic receptor agonist for the treatment of chronic obstructive pulmonary disease (Formule :C32H32ClN3O4Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :558.07PRX933 hydrochloride
CAS :PRX933 hydrochloride (GW876167 hydrochloride) is an agonist of 5-HT2C receptor and can be used in studies about hypertension acute treatment.Formule :C16H22ClN5O2Degré de pureté :99.51% - 99.89%Couleur et forme :SolidMasse moléculaire :351.84Ref: TM-T12565
1mg338,00€5mg538,00€1mL*10mM (DMSO)618,00€10mg858,00€25mg1.269,00€50mg1.720,00€100mg2.305,00€Bremazocine
CAS :Bremazocineis a potent opiate kappa-agonist and centrally acting analgesic.Formule :C20H29NO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :315.45(±)-Tazifylline
CAS :(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.Formule :C23H32N6O3SDegré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :472.6Ref: TM-T10000
1mg140,00€5mg269,00€1mL*10mM (DMSO)350,00€10mg389,00€25mg610,00€50mg820,00€100mg1.063,00€Way 100289
CAS :Way 100289 is a selective 5-HT3 receptor antagonist.Formule :C20H27N3O3Couleur et forme :SolidMasse moléculaire :357.45FR 64822
CAS :FR64822, a non-opioid pain reliever, is effective in rodent tests with an ED50 of 1.8 mg/kg orally.Formule :C11H14N4OCouleur et forme :SolidMasse moléculaire :218.26TC-2153
CAS :TC-2153 inhibits STEP, boosts BDNF, lowers MAOA/5-HT1A mRNA, and blocks 5-HT2A signaling with low toxicity.Formule :C7H5ClF3NS5Couleur et forme :SolidMasse moléculaire :355.89SK1-IN-1
CAS :SK1-IN-1 is a SPHK1 inhibitor (IC50: 58 nM), with potential anticancer activity, and can be used to study cancer and neurodegenerative diseases.Formule :C22H30N4O3Degré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :398.5Naminterol
CAS :Naminterol is a phenethanolamine derivative is an agonist of β2 adrenoceptor with bronchodilatory properties, and used for treatment of asthma.Formule :C19H26N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :330.42Pronethalol hydrochloride
CAS :β-adrenergic antagonistFormule :C15H20ClNODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :265.78L-803087
CAS :L-803087: potent sst4 receptor agonist, 0.7 nM Ki, 280x selectivity, boosts AMPA responses & seizures in mice.Formule :C25H29F2N5O3Degré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :485.53Ref: TM-T11800
1mg50,00€5mg112,00€1mL*10mM (DMSO)126,00€10mg175,00€25mg366,00€50mg585,00€100mg928,00€200mg1.234,00€SGS518 oxalate
CAS :SGS518 oxalate is a 5-HT6 antagonist.Formule :C23H24F2N2O7SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :510.51Licogliflozin
CAS :Licogliflozin (LIK066) is an inhibitor of sodium-glucose cotransporter (SGLT1 and SGLT2).Formule :C23H28O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :416.46L-692429
CAS :L-692429 (MK-0751) is a GHS agonist with high affinity for G protein-coupled receptors and can be used to study acromegaly and obesity.Formule :C29H31N7O2Degré de pureté :98.64% - 99.90%Couleur et forme :SolidMasse moléculaire :509.614Ref: TM-T11798
1mg147,00€5mg356,00€1mL*10mM (DMSO)400,00€10mg530,00€25mg848,00€50mg1.153,00€100mg1.549,00€Amibegron
CAS :Amibegron: oral β3 adrenergic agonist, CNS-penetrating, with antidepressant and anxiolytic properties.Formule :C22H26ClNO4Couleur et forme :SolidMasse moléculaire :403.9Benafentrine dimaleate
CAS :Benafentrine dimaleate is a platelet activating factor receptor (PAFR) antagonists and phosphodiesterase (PDE) 3/4 inhibitors.Formule :C31H35N3O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :625.63Metitepine
CAS :Metitepine is a serotonin receptor antagonist in the CNS used as an antipsychotic.Formule :C20H24N2S2Couleur et forme :SolidMasse moléculaire :356.55YM 114
CAS :YM 114 is an anatagonist of 5-HT(3) receptor.Formule :C16H18ClN3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :303.79ChemR23-IN-2
CAS :ChemR23-IN-2 is a potent, orally active inhibitor of ChemR23 (IC50: 3.2 nM).Formule :C29H26N4O5Couleur et forme :SolidMasse moléculaire :510.54mCPBG
CAS :mCPBG is a potent high affinity agonist of 5-HT3 receptor.Formule :C8H10ClN5Couleur et forme :SolidMasse moléculaire :211.65Iprindole
CAS :Iprindole, a tricyclic indole antidepressant, is a dual weak inhibitor of noradrenaline and 5-HT uptake [1].Formule :C19H28N2Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :284.44Ref: TM-T37015
2mg34,00€5mg50,00€10mg75,00€1mL*10mM (DMSO)79,00€25mg145,00€50mg253,00€100mg432,00€200mg618,00€2-(E-2-decenoylamino)ethyl 2-(cyclohexylethyl) sulfide
CAS :2-Decenoylaminoethyl cyclohexylethyl sulfide prevents stress ulcers, stabilizes phospholipase A2 and prostaglandin E2.Formule :C20H37NOSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :339.58PRX-08066 Maleic acid
CAS :PRX-08066 Maleic acid is the salt form of PRX-08066.PRX-08066 is a 5-HT receptor 2B antagonist that induces selective vasodilation of the pulmonary artery.Formule :C23H21ClFN5O4SDegré de pureté :97.59%Couleur et forme :SolidMasse moléculaire :517.96Ref: TM-T6959
1mg79,00€5mg168,00€10mg220,00€1mL*10mM (DMSO)380,00€25mg398,00€50mg587,00€100mg835,00€200mg1.134,00€Sipagladenant
CAS :Sipagladenant: oral inverse agonist for A2A adenosine receptor, may aid frontal lobe dysfunction research.Formule :C20H19N3O4SCouleur et forme :SolidMasse moléculaire :397.45Tei 6472
CAS :Tei 6472 is a more hydrophilic form of TEI-1338 which is a novel, selective lipoxygenase inhibitor.Formule :C32H39N3O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :545.67Sch 33303
CAS :Sch 33303 is an antiallergy agents.Formule :C19H16N2O3Couleur et forme :SolidMasse moléculaire :320.34(+/-)-PPCC oxalate
CAS :Sigma receptor ligand with high sigma-1 affinity; binds sigma-2 as well (Ki = 1.5 & 50.8 nM). Selective over dopaminergic, muscarinic receptors, DAT, SERT.Formule :C50H60N2O10Couleur et forme :SolidMasse moléculaire :849.034CB2 modulator 1
CAS :CB2 modulator 1 is a potent CB2 modulator. It can be used for the research for immune disorders, osteoporosis, inflammation, renal ischemia.Formule :C18H19F3N4O2Degré de pureté :99.6%Couleur et forme :SolidMasse moléculaire :380.36Butopamine
CAS :Butopamine differs from dobutamine in location of only one hydroxyl group, but is no longer a catecholamine.Formule :C18H23NO3Couleur et forme :SolidMasse moléculaire :301.38Adenosine receptor A1 antagonist 5
CAS :1,3-Dipropyl-8-phenylxanthine is an adenosine antagonist, oxypurine, insecticide, and reduces high blood pressure.Formule :C17H20N4O2Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :312.37Niperotidine
CAS :Niperotidine is an antagonist of histamine H2-receptor.Formule :C20H26N4O5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :434.51Orexin receptor antagonist 2
CAS :Compound 30, potent orexin antagonist with pKis of 7.69/9.78, potential for insomnia research.Formule :C25H31N5O2Couleur et forme :SolidMasse moléculaire :433.55Ko-3290
CAS :Ko-3290 is a cardioselective antagonist of β-adrenoceptors known for its antilipolytic effects in animals.Formule :C19H25N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :343.42(Iso)-FK-480
CAS :(Iso)-FK-480 is a novel orally available cholecystokinin A (CCK-A) antagonist for investigational treatment of chronic pancreatitis.Formule :C26H19FN4O2Degré de pureté :98.36% - 99.41%Couleur et forme :SolidMasse moléculaire :438.45Amitriptylinoxide
CAS :Amitriptylinoxide is an antidepressant.Formule :C20H23NODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :293.4GCGR antagonist 2
CAS :Orally active GCGR antagonist 2, a furan-2-carbohydrazide, binds hGluR at 2.3 nM. Blocks glucagon, inhibits rat receptor at 0.43 nM.Formule :C28H26N4O2Couleur et forme :SolidMasse moléculaire :450.53SLM6031434 (free base)
CAS :SLM6031434 (free base) is an inhibitor of sphingosine kinase type 2 (SphK2). It consists of pedant 1-guanidino-2-phenyloxadiazolylpyrrolidine group.Formule :C22H30F3N5O2Couleur et forme :SolidMasse moléculaire :453.5LEQ-506
CAS :LEQ506, an oral Smoothened antagonist, may inhibit cancer growth by blocking the Hedgehog signaling pathway.Formule :C27H29N5OCouleur et forme :SolidMasse moléculaire :439.55CID1172084
CAS :CID1172084, a novel high-potent GPR55 agonist, interacts with cannabinoid receptors.Formule :C23H18FN5O2S2Couleur et forme :SolidMasse moléculaire :479.55PF-4522654
CAS :PF-4522654 is a potent and selective 5-HT2C receptor agonist.Formule :C16H18F2N4Couleur et forme :SolidMasse moléculaire :304.34PD 118717
CAS :PD 118717: a piperazinyl benzopyranone dopamine agonist with potential antipsychotic properties and no neurological side effects in tests.Formule :C20H22N4O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :366.41CGS 12066B dimaleate
CAS :5-HT1B full agonistFormule :C25H25F3N4O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :566.48ZM 169369
CAS :ICI 169369, a 5-HT2/5-HT1C antagonist, can evoke endothelium-dependent relaxation in rabbit aorta.Formule :C19H20N2SCouleur et forme :SolidMasse moléculaire :308.44WAY208466 dihydrochloride
CAS :WAY208466 dihydrochloride is a 5-HT6 receptor agonist (EC50=7.3 nM) with antidepressant and anxiolytic activity.Formule :C17H20Cl2FN3O2SDegré de pureté :98.43% - 99.56%Couleur et forme :SolidMasse moléculaire :420.33Cetrorelix Acetate
CAS :Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.Formule :C70H92ClN17O14·xC2H4O2Degré de pureté :97.96%Couleur et forme :SolidMasse moléculaire :1491.11LP44 hydrochloride
CAS :LP44 hydrochloride is a 5-HT7 agonist with analgesic effects on formalin-induced orofacial pain in mice and can be used to study neuroinflammation.Formule :C27H38ClN3OSDegré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :488.13SLM6031434 HCl
CAS :SLM6031434 HCl (SLM-6031434 HCl) is a SphK2 inhibitor that reduces LPS-induced TNF伪 and IL-1尾 production.Formule :C22H31ClF3N5O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :489.96WB 4101 hydrochloride
CAS :α1A-adrenergic antagonistFormule :C19H24ClNO5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :381.85SM-2470
CAS :SM-2470 is an α1-adrenoceptor antagonist with antihypertensive activity and hypocholesterolemic activity that inhibits cholesterol absorption.Formule :C23H30ClN5O3Degré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :459.97Methdilazine Hydrochloride
CAS :Methdilazine Hydrochloride (Bristaline) is a histamine H1 receptor antagonist for dermatologic conditions and relief of itching by allergies or rhinitis.Formule :C18H21ClN2SCouleur et forme :Light-Tan Crystalline Powder 4 8-6 (Ntp 1992)Masse moléculaire :332.89Napitane
CAS :napitane (A 75200) is a novel catecholamine uptake inhibitor with inhibitory effects on α-adrenergic receptors and potential antidepressant activity for the
Formule :C22H25NO2Degré de pureté :99.77% - 99.89%Couleur et forme :SolidMasse moléculaire :335.44Amthamine dihydrobromide
CAS :H2 agonistFormule :C6H13Br2N3SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :319.06Pargolol hydrochloride
CAS :Pargolol hydrochloride is an antagonist of β adrenergic receptor.Formule :C16H24ClNO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :313.82AS1069562
CAS :AS1069562 inhibits 5-HT/NE reuptake, boosts IGF-1, FGF2 mRNA in dorsal root ganglia, spinal cord.Formule :C20H23NO5SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :389.46Losmiprofen
CAS :Losmiprofen is a nonsteroidal compound of antiinflammatory.Formule :C17H15ClO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :318.75ML230
CAS :ML230 is a selective ATP-binding cassette (ABC) transporter ABCG2 inhibitor.Formule :C25H21N5O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :439.47SMM-189
CAS :SMM-189 is a potent and selective CB2 inverse agonist.Formule :C19H12Cl2O3Couleur et forme :SolidMasse moléculaire :359.2AMX12006
CAS :AMX12006, a potent and selective EP4 antagonist, exhibits cytotoxic and antitumor activity, demonstrating oral activity with an IC50 of 4.3 nM [1].Formule :C26H22F3N3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :481.47Cafaminol
CAS :Cafaminol (methylcoffanolamine) is a vasoconstrictor and anticatarrhal of the methylxanthine family related to caffeine which is used as a nasal decongestant.Formule :C11H17N5O3Couleur et forme :SolidMasse moléculaire :267.28Levobunolol hydrochloride
CAS :Levobunolol hydrochloride 是一种非选择性的 β-肾上腺素受体阻滞剂，可用于治疗青光眼和上斜肌肌障碍的研究。Formule :C17H26ClNO3Degré de pureté :98.49% - >99.99%Couleur et forme :SolidMasse moléculaire :327.85Ricinelaidic Acid
CAS :Ricinelaidic acid blocks LTB4 receptors; hampers human neutrophil responses; reduces rat bronchoconstriction by 46% at 1 mg/kg i.v.Formule :C18H34O3Couleur et forme :SolidMasse moléculaire :298.46DAT 582
CAS :DAT 582 is a novel serotonin3 receptor antagonist. It is also an effective and long-lasting antiemetic agentFormule :C22H28ClN5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :413.95PF2562
CAS :PF2562: Dopamine D1 ligand, agonist/partial agonist. Binds D1 receptor (Ki: 113 nM), active in cAMP assay (EC50: 568 nM).Formule :C19H17N5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :331.37Lidanserin
CAS :Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.Formule :C26H31FN2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :454.53Albuterol adipate
CAS :Albuterol adipate, a β2-AR agonist salt, treats asthma/COPD, with high selectivity for pulmonary over cardiac receptors.Formule :C32H52N2O10Couleur et forme :SolidMasse moléculaire :624.77S 14063
CAS :S 14063 is a potent 5-HT1A receptor antagonist devoid of beta-adrenoceptor blocking properties.Formule :C22H29Cl2N3O2SCouleur et forme :SolidMasse moléculaire :470.45BW 245C
CAS :BW 245C is a DP1 agonist with an inhibitory effect on the aggregation response of collagen and can be used to study diseases such as stroke.Formule :C19H32N2O5Degré de pureté :≥99%Couleur et forme :SolidMasse moléculaire :368.47Glemanserin
CAS :Glemanserin (MDL11939) is a specific 5-HT2A antagonist with Ki values of 0.54 nM, 2.5 nM and 2.89 nM for rabbit, human and rat 5-HT2A.Formule :C20H25NODegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :295.42Ref: TM-T22964
1mg38,00€5mg84,00€1mL*10mM (DMSO)84,00€10mg119,00€25mg259,00€50mg409,00€100mg605,00€500mg1.288,00€Daglutril
CAS :Daglutril is a NEP/ECE inhibitor for treating hypertension, heart failure, and pulmonary issues, blocking big endothelin-1 conversion.Formule :C31H38N2O6Couleur et forme :SolidMasse moléculaire :534.64Cyclazosin HCl
CAS :Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.Formule :C23H28ClN5O4Degré de pureté :99.10%Couleur et forme :SolidMasse moléculaire :473.95SB 272183
CAS :SB 272183 is a highly potent dual 5-HT1A and 5-HT1B antagonists as potential antidepressant drug.Formule :C29H28ClN5ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :498.02VPC 23019
CAS :VPC 23019 is a competitive antagonist at the S1P1 and S1P3 receptors (pKi= 7.86 and 5.93, respectively).Formule :C17H29N2O5PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :372.4Acetylaszonalenin
CAS :Acetylaszonalenin, from A. flavipes, is an NK1 receptor antagonist with a Ki of 170 μM, blocking substance P.Formule :C25H25N3O3Couleur et forme :SolidMasse moléculaire :415.48Ambucetamide
CAS :Ambucetamide is an antispasmodic, it may inhibit or diminish the spontaneous rhythmical activity of the human myometrium.Formule :C17H28N2O2Couleur et forme :SolidMasse moléculaire :292.42
![7-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT10189.webp&w=3840&q=75)
