GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(251 produits)
- Récepteur adrénergique(3.029 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(218 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(36 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(195 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(42 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(61 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
6012 produits trouvés pour "GPCR/G-Protéine"
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2-Iodomelatonin
CAS :2-Iodomelatonin, Ki 28 pM, is an MT1 agonist, >5x selective over MT2, used to map melatonin sites in brain/tissues.Formule :C13H15IN2O2Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :358.17Ref: TM-T10073
500mgÀ demander1mL*10mM (DMSO)34,00€10mg43,00€25mg79,00€50mg118,00€100mg178,00€200mg268,00€TIK-301
CAS :TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nMFormule :C14H17ClN2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :280.75ST3932
CAS :ST3932 is a ST1535 metabolite, is a adenosine A2A receptor antagonist(Kis of 8 nM and 33 nM for A2A and A1 receptors, respectively).Formule :C12H16N8ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :288.31PRX933 hydrochloride
CAS :PRX933 hydrochloride (GW876167 hydrochloride) is an agonist of 5-HT2C receptor and can be used in studies about hypertension acute treatment.Formule :C16H22ClN5O2Degré de pureté :99.51% - 99.89%Couleur et forme :SolidMasse moléculaire :351.84Ref: TM-T12565
1mg338,00€5mg538,00€1mL*10mM (DMSO)618,00€10mg858,00€25mg1.269,00€50mg1.720,00€100mg2.305,00€Iferanserin
CAS :Iferanserin (S-MPEC) is a selective antagonist of the 5-HT receptor (serotonin receptor) with an affinity for 5-HT2A receptors.Formule :C23H28N2OCouleur et forme :SolidMasse moléculaire :348.48Deramciclane
CAS :Deramciclane has high affinity for 5-HT2A and 5-HT2C receptors.Formule :C20H31NOCouleur et forme :SolidMasse moléculaire :301.47(±)-Tazifylline
CAS :(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.Formule :C23H32N6O3SDegré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :472.6Ref: TM-T10000
1mg140,00€5mg269,00€1mL*10mM (DMSO)350,00€10mg389,00€25mg610,00€50mg820,00€100mg1.063,00€Tedatioxetine hydrobromide
CAS :Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) is a serotonin-norepinephrine-dopamine reuptake inhibitor and 5-HT2A receptor antagonist.Formule :C18H22BrNSDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :364.34T-0509
CAS :T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle and selectively down-regulates rat cardiac beta 1-
Formule :C18H23NO5Degré de pureté :97.52% - 98.43%Couleur et forme :SolidMasse moléculaire :333.38p-MPPF dihydrochloride
CAS :p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.Formule :C25H29Cl2FN4O2Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :507.43Arvanil
CAS :Arvanil (N-Vanillylarachidonamide) is a synthetic capsaicin-amphetamine hybrid that acts as a ligand for VR1 and CB1, offering neuroprotective effects.Formule :C28H41NO3Degré de pureté :99.49%Couleur et forme :SolidMasse moléculaire :439.63LPA2 antagonist 1
CAS :LPA2 antagonist 1 is a potent LPA2 antagonist.Formule :C20H23Cl2N5O2S2Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :500.47Cyclazosin HCl
CAS :Cyclazosin HCl is an α-adrenergic receptor antagonist that can be used to study non-arteritic ischemic optic neuropathy.Formule :C23H28ClN5O4Degré de pureté :99.10%Couleur et forme :SolidMasse moléculaire :473.95L-694,247
CAS :L-694,247 is a 5-HT receptor agonist with affinity for 5-HT1D, 5-HT1A, 5-HT1B, 5-HT1C, and 5-HT1E receptors, and can be used to study neurological diseases.Formule :C20H21N5O3SDegré de pureté :98.36%Couleur et forme :White SolidMasse moléculaire :411.486-Chloromelatonin
CAS :6-Chloromelatonin: potent, stable melatonin agonist; binds MT2 receptors (pKi=9.77); could help research sleep disorders.Formule :C13H15ClN2O2Degré de pureté :97.26% - 99.25%Couleur et forme :SolidMasse moléculaire :266.72Ref: TM-T22530
1mg315,00€5mg745,00€10mg1.018,00€25mg1.431,00€50mg1.783,00€100mg2.250,00€500mg4.410,00€SKF83959
CAS :SKF83959: dopamine D1 partial agonist, Ki: D1(1.18 nM), D5(7.56 nM), D2(920 nM), D3(399 nM); improves cognitive function in depression, Alzheimer's.
Formule :C18H20ClNO2Degré de pureté :98.68%Couleur et forme :SolidMasse moléculaire :317.81CCX777
CAS :CCX777 is a partial agonist recruited to ACKR3 by β-arrestin-2 and is used in cancer research.Formule :C31H43N7O3SDegré de pureté :98.73%Couleur et forme :SolidMasse moléculaire :593.78Levobunolol hydrochloride
CAS :Levobunolol hydrochloride 是一种非选择性的 β-肾上腺素受体阻滞剂，可用于治疗青光眼和上斜肌肌障碍的研究。Formule :C17H26ClNO3Degré de pureté :98.49% - >99.99%Couleur et forme :SolidMasse moléculaire :327.85Org41841
CAS :Org41841 is an agonist of luteinising hormone/chorionic gonadotropin receptor and thyroid stimulating hormone receptor and can be used to study hyperthyroidism.Formule :C19H22N4O2S2Degré de pureté :99.46% - 99.92%Couleur et forme :SolidMasse moléculaire :402.53MRE3008F20
CAS :MRE3008F20 is an AA3R antagonist that inhibits Cl-IB-MECA-induced cAMP production and can be used to study glaucoma and asthma.Formule :C21H20N8O3Degré de pureté :97.29%Couleur et forme :SolidMasse moléculaire :432.44L748337
CAS :L748337 is a β3-adrenoceptor antagonist that inhibits β3-, β2-, and β1-adrenoceptors and inhibits the protective effects of CL316243.Formule :C26H31N3O5SDegré de pureté :99.67% - >99.99%Couleur et forme :SolidMasse moléculaire :497.61Pridefine
CAS :Pridefine: antidepressant, balances serotonin, dopamine, norepinephrine reuptake, weakly releases them.Formule :C19H21NDegré de pureté :99.15% - 99.66%Couleur et forme :SolidMasse moléculaire :263.38E-3620
CAS :E-3620 is a potent antagonist of the 5-HT3 receptor and can be used to study dyskinesia and gastrointestinal dysfunction.Formule :C20H27Cl2N3O2Degré de pureté :98.88% - 98.88%Couleur et forme :SolidMasse moléculaire :412.35PF 03654746 FA
PF 03654746 FA is a human histamine receptor H(3) antagonist that can be used to study cognitive impairment and Alzheimer's disease.Formule :C19H26F2N2O3Degré de pureté :99.44%Couleur et forme :SoildMasse moléculaire :368.42AVN-322
CAS :AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive impairment.Formule :C17H20ClN5O2SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :393.89Romifidine
CAS :Romifidine is used as a sedative in veterinary medicine mainly in large animals such as horses. It acts as an agonist at the α2 adrenergic receptor subtype.Formule :C9H9BrFN3Couleur et forme :SolidMasse moléculaire :258.09SLV-310
CAS :SLV-310 is a D2 receptor antagonist and 5-HT reuptake receptor inhibitor for the study of neurological disorders such as bipolar disorder and schizophrenia.Formule :C25H24FN3O2Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :417.48(Iso)-FK-480
CAS :(Iso)-FK-480 is a novel orally available cholecystokinin A (CCK-A) antagonist for investigational treatment of chronic pancreatitis.Formule :C26H19FN4O2Degré de pureté :98.36% - 99.41%Couleur et forme :SolidMasse moléculaire :438.45LY377604
CAS :LY377604 is a human β3-adrenergic receptor agonist (EC50: 2.4 nM) and β1/2-adrenergic receptor antagonist for the study of obesity.Formule :C31H32N4O4Degré de pureté :99.72% - >99.99%Couleur et forme :SolidMasse moléculaire :524.61ST1936
CAS :ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.Formule :C13H17ClN2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :236.74Ref: TM-T23396
1mg44,00€5mg111,00€1mL*10mM (DMSO)123,00€10mg178,00€25mg316,00€50mg470,00€100mg682,00€200mg954,00€SM-2470
CAS :SM-2470 is an α1-adrenoceptor antagonist with antihypertensive activity and hypocholesterolemic activity that inhibits cholesterol absorption.Formule :C23H30ClN5O3Degré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :459.97RXFP3/4 agonist 2
CAS :RXFP3/4 agonist 2 is a nonpeptide bis-RXFP3/4 agonist used in the study of diseases caused by metabolic abnormalities.Formule :C22H22N6O2Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :402.45Amgen-23
CAS :Amgen-23 is a selective and highly potent sphingosine kinase 1 (SPHK1) inhibitor that inhibits SPHK2 and can be used in anticancer research.Formule :C23H25Cl2N3O2SDegré de pureté :97.31%Couleur et forme :SolidMasse moléculaire :478.44AM404
CAS :AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer activities that blocks anandamide transport.Formule :C26H37NO2Couleur et forme :SolidMasse moléculaire :395.58RS 56812 hydrochloride
CAS :5-HT3 partial agonistFormule :C18H22ClN3O2Degré de pureté :98.62%Couleur et forme :SolidMasse moléculaire :347.84PF-184298
CAS :PF-184298 is a serotonin and norepinephrine monoamine reuptake inhibitor (SNRI) that inhibits dopamine reuptake.Formule :C15H20Cl2N2ODegré de pureté :98.67%Couleur et forme :SolidMasse moléculaire :315.24A-65186
CAS :A-65186 is a CCK antagonist used in the study of inflammation and gastrointestinal tract injury.Formule :C25H35N3O4Degré de pureté :98.85% - 99.94%Couleur et forme :SolidMasse moléculaire :441.56UNC9975
CAS :UNC9975 is a D(2) receptor agonist with antipsychotic activity used in the study of neurologic disorders such as schizophrenia.Formule :C23H28Cl2N4O2Degré de pureté :98.78% - 98.78%Couleur et forme :SolidMasse moléculaire :463.4ST 91
CAS :ST-91 is an agonist of α2-adrenoceptor with a mixed α-adrenergic receptor type/subtype selection profile.Formule :C13H20ClN3Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :253.77Ref: TM-T23397
5mg49,00€1mL*10mM (DMSO)50,00€10mg72,00€25mg142,00€50mg245,00€100mg354,00€200mg497,00€Clemastine
CAS :Clemastine (Meclastin) is an antagonist of the H1 receptor and exhibits anti-inflammatory effects.Formule :C21H26ClNODegré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :343.89PPTN hydrochloride
CAS :PPTN hydrochloride is a potent, high-affinity, competitive, highly selective P2Y14 receptor antagonist (KB: 434 pM), but no agonist or antagonist activity atFormule :C29H25ClF3NO2Degré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :511.96Quinupramine
CAS :Quinupramine: an oral antidepressant targeting the serotonin system; penetrates CNS; doesn’t affect β-adrenergic system.Formule :C21H24N2Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :304.43BMY-14802 hydrochloride
CAS :BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.Formule :C18H23ClF2N4ODegré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :384.85Amosulalol
CAS :Amosulalol is a combined alpha and beta adrenoceptor antagonist.Formule :C18H24N2O5SDegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :380.46Ref: TM-T30027
1mg175,00€2mg264,00€5mg404,00€1mL*10mM (DMSO)430,00€10mg592,00€25mg888,00€50mg1.243,00€100mg1.701,00€Benperidol
CAS :Benperidol (Anquil), a butanone derivative, has antipsychotic effects and blocks D2 receptors; useful in PET scans.Formule :C22H24FN3O2Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :381.44Ref: TM-T26360
1mg116,00€5mg276,00€1mL*10mM (DMSO)279,00€10mg410,00€25mg680,00€50mg938,00€100mg1.293,00€500mg2.593,00€Compound C108
CAS :Compound C108 is an inhibitor of GTPase-activating protein SH3 domain-binding protein 2 (G3BP2).
Formule :C15H14N2O3Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :270.28ASP-4058
CAS :ASP-4058: Safe, oral S1P1/S1P5 agonist; improves autoimmune encephalomyelitis in mice.Formule :C19H12F6N4O2Degré de pureté :99.92% - 99.96%Couleur et forme :SolidMasse moléculaire :442.31BAY 60-6583
CAS :BAY 60-6583 is a potent, high-affinity adenosine A2B receptor agonist (EC50 = 3 nM) with affinity for A2B receptors that exceeds that for A1, A2A, and A3Formule :C19H17N5O2SDegré de pureté :98.46% - 99.8%Couleur et forme :SolidMasse moléculaire :379.44Ref: TM-T14506
1mg39,00€2mg50,00€5mg84,00€1mL*10mM (DMSO)101,00€10mg116,00€25mg233,00€50mg376,00€100mg567,00€200mg797,00€SC 19220
CAS :SC 19220 is a prostaglandin E2 receptor EP1 antagonist that inhibits RANKL-induced osteoclastogenesis.Formule :C16H14ClN3O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :331.75Ref: TM-T23330
1mg47,00€5mg90,00€1mL*10mM (DMSO)99,00€10mg164,00€25mg322,00€50mg477,00€100mg668,00€200mg900,00€(Z)-Thiothixene
CAS :(Z)-Thiothixene (Thiothixene) is an antagonist of serotonergic receptor.
Formule :C23H29N3O2S2Degré de pureté :99.21%Couleur et forme :Yellow To Yellow With A Tan Cast PowderMasse moléculaire :443.63Olorinab
CAS :Olorinab (APD 371) (APD 371) is a highly potent, selective and fully efficacious cannabinoid receptor type 2 (CB2) agonist. With an EC50 of 6.2 nM for hCB2.Formule :C18H23N5O3Degré de pureté :97.67% - 98.47%Couleur et forme :SolidMasse moléculaire :357.4148740 RP
CAS :48740 RP (RP 55779) is an antagonist of platelet-activating factor.Formule :C12H11N3OSDegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :245.3Ref: TM-T10159
1mg338,00€5mg537,00€1mL*10mM (DMSO)537,00€10mg858,00€25mg1.269,00€50mg1.720,00€100mg2.305,00€JZP-361
CAS :JZP-361: selective MAGL inhibitor (IC50 = 46 nM); weaker on FAAH, hABHD6; anti-histamine; for asthma research.Formule :C22H20ClN5ODegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :405.88Fananserin
CAS :Fananserin: Oral 5-HT2A antagonist (Ki=0.37 nM, rat), blocks human D4 receptor (Ki=2.93 nM).Formule :C23H24FN3O2SDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :425.52Ref: TM-T15270
2mg39,00€5mg52,00€1mL*10mM (DMSO)58,00€10mg77,00€25mg110,00€50mg166,00€100mg236,00€200mg349,00€ADR-851 free base
CAS :ADR-851 free base is an antagonist of the HT3 receptor.Formule :C14H18ClN3O2Degré de pureté :97.88% - 98.39%Couleur et forme :SolidMasse moléculaire :295.77Sergliflozin etabonate
CAS :Sergliflozin etabonate (KGT-1251) is an inhibitor of SGLT2 and can be used in studies about type 2 diabetes and obesity.Formule :C23H28O9Degré de pureté :97.88%Couleur et forme :SolidMasse moléculaire :448.46Ref: TM-T28757
1mg93,00€1mL*10mM (DMSO)200,00€5mg203,00€10mg304,00€25mg492,00€50mg655,00€100mg893,00€CYM5181
CAS :CYM5181 is related to the body's immune system and can be used to study multiple sclerosis, transplant rejection, and adult respiratory distress syndrome.Formule :C17H17N3O3Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :311.34Pitolisant
CAS :Pitolisant is a potent and selective nonimidazole inverse agonist that acts on the recombinant human histamine H3 receptor with Ki of 0.16 nM.Formule :C17H26ClNODegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :295.85Ref: TM-T60636
5mg46,00€1mL*10mM (DMSO)49,00€10mg66,00€25mg114,00€50mg178,00€100mg295,00€500mg708,00€KSK94
CAS :KSK94 is an H3 receptor antagonist that inhibits sigma-2 receptors , with a Ki value of 75.2 nM, and can be used to study injurious pain.Formule :C25H26N4ODegré de pureté :99.60%Couleur et forme :SolidMasse moléculaire :398.5SLP9101555
SLP9101555 is a potent and selective sphingosine kinase 2 (SphK2) inhibitor with a Ki of 90 nM.SLP9101555 has a high affinity for SphK2, which is 200-fold
Formule :C16H22BrClN2Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :357.72Ref: TM-T63047
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€Immethridine dihydrobromide
CAS :Immethridine dihydrobromide is a histamine H3 receptor agonist.Formule :C9H11Br2N3Degré de pureté :97.61% - 98.14%Couleur et forme :SolidMasse moléculaire :321.01CV-6209
CAS :CV-6209 is a potent antagonist of the platelet-activating factor (PAF) receptor.Formule :C34H60ClN3O6Degré de pureté :>99.99% - >99.99%Couleur et forme :SolidMasse moléculaire :642.31KP136
CAS :KP136 is an orally effective antiallergic compound (IC50: 76.1 μg/mL for histamine release and 63 ug/mL for degranulation).Formule :C16H18N4O3Degré de pureté :98.3% - 98.61%Couleur et forme :SolidMasse moléculaire :314.34Runcaciguat
CAS :Runcaciguat, a soluble guanylate cyclase stimulator, aids in cardiovascular and renal research.Formule :C23H22Cl2F3NO3Degré de pureté :99.17%Couleur et forme :SolidMasse moléculaire :488.33Sinitrodil
CAS :Sinitrodil (ITF-296) is a guanylate cyclase stimulant that may be used in the treatment of myocardial ischemia and angina pectoris.Formule :C10H10N2O5Degré de pureté :97.03%Couleur et forme :SolidMasse moléculaire :238.2Ref: TM-T34648
1mg132,00€5mg315,00€1mL*10mM (DMSO)380,00€10mg477,00€25mg773,00€50mg1.063,00€100mg1.431,00€500mg2.872,00€L 674573
CAS :L 674573 is an inhibitor of leukotriene biosynthesis.Formule :C28H27NO3SDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :457.58LY 272015 hydrochloride
CAS :LY 272015 hydrochloride is a 5-HT2B receptor antagonist.Formule :C21H25ClN2O2Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :372.89OPC-51803
CAS :OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.Formule :C26H32ClN3O2Degré de pureté :98.93% - >99.99%Couleur et forme :SolidMasse moléculaire :454Cianopramine
CAS :Cianopramine (Ro 112465) is a selective 5-hydroxytryptamine uptake inhibitor and a tricyclic antidepressant used in the study of neurological disorders.Formule :C20H23N3Degré de pureté :99.92% - 99.92%Couleur et forme :SolidMasse moléculaire :305.42CYM50374
CAS :CYM50374 inhibits Sphingosine-1-phosphate receptor 4 (S1P4 ) with an IC50 of µM.Formule :C19H19NO3SDegré de pureté :98.35% - 98.96%Couleur et forme :SolidMasse moléculaire :341.42KSK68
CAS :KSK68 is a sigma-1 and histamine H3 receptor antagonist with analgesic activity, inhibits H3 receptors and can be used to study pain.Formule :C23H28N2O2Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :364.48NP10679
CAS :NP10679 is a N-methyl-D-aspartate (NMDA) receptor inhibitor of the GluN2B subunit that inhibits histamine H1, hERG channels, and CYPase.Formule :C23H26F3N3O3Degré de pureté :99.43%Couleur et forme :SolidMasse moléculaire :449.47Rafabegron
CAS :Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of diabetes and obesity.Formule :C21H23ClN2O4Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :402.87SDZ-62-434
CAS :SDZ-62-434 is a platelet-activating factor inhibitor with antitumor activity and may be used in the study of leukemia.Formule :C23H27Cl2N3Degré de pureté :98.38%Couleur et forme :SolidMasse moléculaire :416.39Nonabine
CAS :Nonabine is a compound with strong antiemetic properties that can be used to prevent nausea and vomiting associated with cancer chemotherapy.Formule :C25H33NO2Degré de pureté :99.82% - 99.94%Couleur et forme :SolidMasse moléculaire :379.54CP 96021
CAS :"CP 96021 is an antagonist of 5-HT1/2 receptors, with anti-inflammatory and anti-ulcer effects for treating GI tract and asthma."
Formule :C29H21FN4OSDegré de pureté :97.81% - 99.62%Couleur et forme :SoildMasse moléculaire :492.57Evodenoson
CAS :Evodenoson (ATL313), a potent A2aR agonist, treats eye diseases, tumors, and immune disorders; potential for glaucoma and blood cancer studies.Formule :C23H29N7O6Degré de pureté :99.75% - 99.83%Couleur et forme :SolidMasse moléculaire :499.52SLF1081851
CAS :SLF1081851 is a Spns2 inhibitor. SLF1081851 inhibits S1P release with IC50 of 1.93 μM.Formule :C21H33N3ODegré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :343.51Femoxetine hydrochloride
CAS :Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.Formule :C20H26ClNO2Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :347.887-Hydroxy-DPAT hydrobromide
CAS :7-Hydroxy-DPAT hydrobromide is a D3 dopamine receptor agonist that blocks dopamine reuptake, used in research on neurological diseases.Formule :C16H26BrNODegré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :328.29GW438014A
CAS :GW438014A 是一种有效且具有选择性的 NPY-Y5 受体拮抗剂。GW438014A 对食物摄入并减少肥胖啮齿动物的体重增加具有抑制作用。Formule :C23H23N3O4SDegré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :437.51Ricasetron
CAS :Ricasetron (Brl 46470) is a 5-HT3 receptor antagonist with pro-axonal lysing properties and is used in the study of anxiety disorders and anxiety disorders.Formule :C19H27N3ODegré de pureté :99.52%Couleur et forme :SolidMasse moléculaire :313.44Viloxazine
CAS :Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activityFormule :C13H19NO3Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :237.29Torbafylline
CAS :Torbafylline is a xanthine-based PDE inhibitor reducing protein breakdown via PDE4/cAMP/EPAC/PI3K/Akt in rats with burns, cancer, or sepsis.Formule :C16H26N4O4Degré de pureté :99.96% - 99.97%Couleur et forme :SoildMasse moléculaire :338.4Ref: TM-T67965
1mg81,00€5mg172,00€1mL*10mM (DMSO)178,00€10mg259,00€25mg424,00€50mg583,00€100mg800,00€FPL 55712
CAS :FPL 55712 is a leukotriene receptor and SRS-A antagonist that inhibits bronchoconstriction and can be used in studies of asthma and coronary artery thrombosis.Formule :C27H30O9Degré de pureté :98.15% - 99.8%Couleur et forme :SolidMasse moléculaire :498.52Soquinolol
CAS :Soquinolol (Soquinolol mucate) is a beta-adrenergic receptor antagonist with weak local anesthetic activity.Soquinolol has good enteral efficacy and a longFormule :C17H26N2O3Degré de pureté :97.48% - 98.63%Couleur et forme :SolidMasse moléculaire :306.4TASP0390325
CAS :TASP0390325, a potent and orally active V1B receptor antagonist, has antidepressant and anxiolytic activities in rodents.Formule :C25H30Cl2FN5O4Degré de pureté :98.62%Couleur et forme :SolidMasse moléculaire :554.44ISAM-140
CAS :ISAM-140 is a potent and highly selective antagonist of A2B adenosine receptor.Formule :C19H19N3O3Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :337.37Antihistamine-1
CAS :Antihistamine-1 是能够渗透血脑屏障的 H1-抗组胺药 (Ki=6.9 nM), 它也是 CYP2D6 和 hERG 通道的抑制剂，其 IC50 值分别为 5.4 和 0.8 μM。Formule :C23H24FN5Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :389.47Imiloxan
CAS :Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder.Formule :C14H16N2O2Degré de pureté :98.13% - 99.8%Couleur et forme :SolidMasse moléculaire :244.29RG 7152
CAS :RG 7152 is a leukotriene D4 antagonist with anti-asthmatic properties and can be used in the study of asthma.Formule :C20H19N5O2Degré de pureté :98.45%Couleur et forme :SolidMasse moléculaire :361.4Molindone
CAS :Molindone: antipsychotic for schizophrenia; blocks dopamine, often paired with serotonin; dosage affects error/response rates.Formule :C16H24N2O2Degré de pureté :99.46% - 99.67%Couleur et forme :Off-White SolidMasse moléculaire :276.37Fipamezole
CAS :Fipamezole is a potent alpha2 adrenergic receptor antagonist that may be useful for studying autonomic dysfunction in Parkinson's disease.Formule :C14H15FN2Degré de pureté :99.32% - 99.97%Couleur et forme :SolidMasse moléculaire :230.28BMS-470539 dihydrochloride
CAS :BMS-470539 dihydrochloride is a MC-1 R agonist with anti-inflammatory activity.Formule :C32H43Cl2N5O4Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :632.62Sitaxsentan
CAS :Sitaxsentan (TBC-11251), a selective ETA receptor antagonist, prevents vasoconstriction by blocking endothelin.Formule :C18H15ClN2O6S2Degré de pureté :97.99% - 98.71%Couleur et forme :SolidMasse moléculaire :454.9RO3244794
CAS :RO3244794 is a selective prostacyclin (IP) receptor antagonist that can be used to study liver injury.Formule :C25H19F2NO5Degré de pureté :99.36%Couleur et forme :SolidMasse moléculaire :451.42PNU-282987 free base
CAS :PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for nervous system research.
Formule :C14H17ClN2ODegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :264.75ReN-1869
CAS :ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity for the study of neurological diseasesFormule :C24H27NO2Degré de pureté :99.83% - 99.98%Couleur et forme :SolidMasse moléculaire :361.48Egis-11150
CAS :Egis-11150 is a potent inhibitor of adrenergic alpha1, alpha2c, 5-HT2a, 5HT7 receptors.Formule :C19H21ClFN5O2Degré de pureté :97.49% - >99.99%Couleur et forme :SolidMasse moléculaire :405.85RLX-33
CAS :RLX-33 blocks RXFP3 and relaxin 3 effects, controls food intake in rats, and may help study metabolic syndrome.Formule :C24H19ClN4O4Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :462.89Lorglumide sodium salt
CAS :Lorglumide sodium salt (CR-1409 sodium salt) is an antagonist of cholecystokinin receptors (CCK).Formule :C22H31Cl2N2NaO4Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :481.39ML-354
CAS :ML354 is a selective antagonist of PAR4 with an IC 50 of 140 nM [1].Formule :C16H14N2O3Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :282.29Milenperone
CAS :Milenperone (R 34009) is a novel anti-invasive compound for the control of behavioral disorders in patients with epilepsy and alcoholism.Formule :C22H23ClFN3O2Degré de pureté :98.09% - 99.84%Couleur et forme :SolidMasse moléculaire :415.89Impromidine hydrochloride
CAS :Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.Formule :C14H26Cl3N7SDegré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :430.83Midaglizole hydrochloride
CAS :Midaglizole hydrochloride (DG5128) is an α2-adrenoceptor antagonist with 7.4x more affinity than α1-adrenoceptors (pKi=6.28).Formule :C16H19Cl2N3Degré de pureté :99.39% - 99.82%Couleur et forme :SolidMasse moléculaire :324.25Ref: TM-T11015
1mg54,00€5mg119,00€1mL*10mM (DMSO)152,00€10mg188,00€25mg306,00€50mg416,00€100mg532,00€200mg705,00€NF-56-EJ40
CAS :NF-56-EJ40 is an effective and highly selective antagonist of human SUCNR1 with an IC50 of 25 nM and a Ki of 33 nM.Formule :C27H29N3O3Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :443.54Elinogrel
CAS :Elinogrel (PRT060128) is a competitive and reversible antagonist of platelet P2Y12 with IC50 of 20 nM and exhibits potent antiplatelet effects.Formule :C20H15ClFN5O5S2Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :523.95Ref: TM-T11177
1mg34,00€5mg66,00€1mL*10mM (DMSO)77,00€10mg92,00€25mg161,00€50mg224,00€100mg313,00€200mg447,00€5-HT1A modulator 1
CAS :5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).Formule :C21H25N3O2SDegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :383.51RS 42358-197
CAS :RS 42358-197 (RS 25259-007) is a competitive 5-HT3 receptor antagonist.Formule :C19H23ClN2ODegré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :330.85Ref: TM-T20739
1mg158,00€1mL*10mM (DMSO)349,00€5mg351,00€10mg527,00€25mg783,00€50mg1.054,00€100mg1.414,00€200mg1.908,00€FK-453
CAS :FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.Formule :C23H25N3O2Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :375.46NE-100 hydrochloride
CAS :NE-100 hydrochloride (NE-100 HCl) is a potent and selective antagonist of σ1 (IC50 = 4.16 nM) with antipsychotic activity.Formule :C23H34ClNO2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :391.98Ref: TM-T20797
1mg43,00€2mg54,00€5mg87,00€10mg130,00€25mg210,00€50mg313,00€100mg465,00€200mg662,00€500mg982,00€AZD8542
CAS :AZD8542 is an antagonist of Smoothened (SMO) with potential as an oncology therapeutic.Formule :C25H24N4O2Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :412.48Camonagrel
CAS :Camonagrel is a compound that has inhibitory effects on Prostaglandin E2.Formule :C15H16N2O3Degré de pureté :98.71% - 99.25%Couleur et forme :SolidMasse moléculaire :272.3Sonedenoson
CAS :Sonedenoson (MRE0094) is an adenosine A(2A) receptor agonist and potential inhibitor potentially targeting SARS-CoV-2 coronavirus 2;-O-ribose methyltransferase.Formule :C18H20ClN5O5Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :421.84Isbogrel
CAS :Isbogrel (CV4151) is a TXA2 synthase inhibitor for researching arrhythmias, ischemic attacks, and thrombosis.Formule :C18H19NO2Degré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :281.35Linetastine
CAS :Linetastine (TMK-688) inhibits 5-LOX, blocks leukotrienes, counters histamine; researched for asthma, atherosclerosis, ulcers.Formule :C35H40N2O6Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :584.7GS-9667
CAS :GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia viaFormule :C21H24FN5O4SDegré de pureté :99.77% - 99.96%Couleur et forme :SolidMasse moléculaire :461.51Lecozotan HCl
CAS :Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.
Formule :C28H30ClN5O3Degré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :520.02Repinotan
CAS :Repinotan (BAY x 3702 free base) is a 5-HT1A receptor agonist used in acute ischemic stroke studies.Formule :C21H24N2O4SDegré de pureté :99%Couleur et forme :SolidMasse moléculaire :400.49SF-22
CAS :SF-22 is a Y2R antagonist with potential anti-inflammatory activity that can be used to study diseases associated with neurological disorders.Formule :C28H26N2O3SDegré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :470.58Cilansetron
CAS :Cilansetron is an effective and selective 5-HT3 receptor antagonist that can be used for related diseases caused by colitis.Formule :C20H21N3ODegré de pureté :99.82% - 99.98%Couleur et forme :SolidMasse moléculaire :319.4N 0861
CAS :N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.Formule :C13H17N5Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :243.31Ref: TM-T70722
1mg164,00€2mg234,00€5mg389,00€10mg532,00€25mg820,00€50mg1.063,00€100mg1.423,00€200mg1.945,00€Piromelatine
CAS :Piromelatine is an agonist of melatonin MT1/MT2 receptors, 5-HT1A and 5-HT1D, and an antagonist of 5-HT2B.Piromelatine has antinociceptive activity withFormule :C17H16N2O4Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :312.32Ref: TM-T34081
1mg60,00€5mg130,00€1mL*10mM (DMSO)142,00€10mg178,00€25mg334,00€50mg522,00€100mg713,00€Tildacerfont
CAS :Tildacerfont inhibits CRF1, lowers ACTH/adrenal androgens, and aids in congenital adrenal hyperplasia research.Formule :C20H26ClN5OSDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :419.97SMO-IN-2
CAS :SMO-IN-2 is a SMO inhibitor with antiproliferative activity and anticancer activity and inhibits Hh signaling.SMO-IN-2 can be used in the study of cancer.Formule :C25H25F4N5O2Degré de pureté :98.64%Couleur et forme :SolidMasse moléculaire :503.49Spizofurone
CAS :Spizofurone (Espizofurona) has anti-ulcer activity, protective effect on the gastric mucosa of rats and can increase alkaline secretion.Formule :C12H10O3Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :202.21Dimethindene
CAS :Dimethindene (Dimetindeno) is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects.Formule :C20H24N2Degré de pureté :98.3% - 98.99%Couleur et forme :SolidMasse moléculaire :292.42CCR1 antagonist 6
CAS :CCR1 antagonist 6 is a CCR1 antagonist (IC50: 3 nM).Formule :C21H23ClN4O3SDegré de pureté :99.15% - 99.92%Couleur et forme :SolidMasse moléculaire :446.95Adoprazine
CAS :Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.Formule :C24H24FN3O2Degré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :405.46Ref: TM-T10249
1mg60,00€5mg130,00€1mL*10mM (DMSO)142,00€10mg205,00€25mg363,00€50mg580,00€100mg782,00€BMS-817399
CAS :BMS-817399: oral CCR1 antagonist with binding and chemotaxis inhibition IC50s, potential for rheumatoid arthritis research.Formule :C23H36ClN3O4Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :454Ref: TM-T26861
1mg152,00€5mg319,00€1mL*10mM (DMSO)356,00€10mg485,00€25mg770,00€50mg1.035,00€100mg1.395,00€Landipirdine
CAS :Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders such as dementia.Formule :C18H19FN2O3SDegré de pureté :97.61% - 99.99%Couleur et forme :SolidMasse moléculaire :362.42Eclazolast
CAS :Eclazolast (RHC 2871), a lipophilic anti-allergic, inhibits mast cell mediator release by affecting Fc(epsilon)RI-related processes, dose-dependently.Formule :C12H12ClNO4Degré de pureté :98.29% - 98.61%Couleur et forme :SolidMasse moléculaire :269.68Ref: TM-T25360
1mg112,00€1mL*10mM (DMSO)249,00€5mg261,00€10mg396,00€25mg655,00€50mg888,00€100mg1.251,00€500mg2.493,00€LY-2624803
CAS :LY-2624803 is a 5-HT2A receptor antagonist and histamine receptor inverse agonist that can be used to improve slow wave sleep.Formule :C22H25N3O3Degré de pureté :99.78% - 99.97%Couleur et forme :SolidMasse moléculaire :379.45Regrelor disodium
CAS :Regrelor disodium (INS 50589) is a p2y12 receptor antagonist that prevents thrombosis, effectively inhibits vascular smooth muscle cell contraction, inhibitsFormule :C22H23N6Na2O8PDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :576.41GR 46611
CAS :GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in studies about the treatment of epilepsy.Formule :C23H27N3O2Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :377.48VA-K-14 hydrochloride
CAS :VA-K-14 hydrochloride（VAK14 HCl） is a selective thyrotropin receptor (TSHR) antagonist (IC50= 12.3 μM) that inhibits TSHR stimulation by serum and monoclonalFormule :C18H16ClN3SDegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :341.86Aplindore Fumarate
CAS :Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia research.Formule :C22H22N2O7Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :426.42Perphenazine dihydrochloride
CAS :Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.Formule :C21H28Cl3N3OSDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :476.89L-161982
CAS :L-161982 is a selective EP4 receptor antagonist that inhibits PGE2-induced ERK phosphorylation and cell proliferation in HCA-7 cells.Cost-effective and quality-assured.Formule :C32H29F3N4O4S2Degré de pureté :99.58% - 99.6%Couleur et forme :SolidMasse moléculaire :654.72Ref: TM-T15681
1mg66,00€5mg122,00€1mL*10mM (DMSO)170,00€10mg200,00€25mg424,00€50mg608,00€100mg848,00€200mg1.144,00€GBR 12783 dihydrochloride
CAS :GBR 12783 dihydrochloride inhibits dopamine uptake in rats/mice; IC50s: 1.8/1.2 nM. Enhances memory, boosts hippocampal acetylcholine.Formule :C28H34Cl2N2ODegré de pureté :98.08%Couleur et forme :SolidMasse moléculaire :485.49rel-(1R,2R)-Vesamicol Hydrochloride
CAS :rel-(1R,2R)-Vesamicol Hydrochloride is a acetylcholine transport inhibitor.Formule :C17H26ClNODegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :295.85CyPPA
CAS :CyPPA enhances SK channels, reducing firing rate and extending apamin-sensitive afterhyperpolarization.Formule :C16H23N5Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :285.39Ref: TM-T20968
2mg42,00€5mg62,00€1mL*10mM (DMSO)66,00€10mg87,00€25mg166,00€50mg266,00€100mg442,00€500mg973,00€Crinecerfont
CAS :Crinecerfont (SSR-125543) is a CRF1 antagonist, useful in congenital adrenal hyperplasia research.Formule :C27H28ClFN2OSDegré de pureté :97.79% - 98.55%Couleur et forme :SolidMasse moléculaire :483.04Medifoxamine
CAS :Medifoxamine (LG 152) is a selective non-monoamine oxidase inhibitor that exhibits antidepressant activity through inhibition of 5 HT reuptake.MedifoxamineFormule :C16H19NO2Degré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :257.33Ref: TM-T24444
1mg94,00€5mg222,00€1mL*10mM (DMSO)245,00€10mg334,00€25mg602,00€50mg845,00€100mg1.099,00€Teniloxazine
CAS :Teniloxazine is an orally available antidepressant compound with anti-hypoxic properties.Formule :C16H19NO2SDegré de pureté :99.29%Couleur et forme :SolidMasse moléculaire :289.39LTB4-IN-1
CAS :LTB4-IN-1 (Anti-inflammatory agent 2) with IC50 of 70 nM is an inhibitor of leukotriene synthesis (LTB4).Formule :C26H30N2O4SDegré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :466.59Ref: TM-T10917
1mg261,00€5mg515,00€1mL*10mM (DMSO)653,00€10mg874,00€25mg1.288,00€50mg1.755,00€100mg2.358,00€Selodenoson
CAS :Selodenoson (RG-14202) is a selective adenosine A1 receptor agonist used to slow the heart rate in patients with atrial fibrillation and to treat arrhythmias.Formule :C17H24N6O4Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :376.41Litoxetine
CAS :Litoxetine: a selective 5-HT inhibitor & 5-HT3 antagonist, used as an antidepressant with antiemetic effects, Ki=85 nM.Formule :C16H19NODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :241.33Ref: TM-T67956
1mg92,00€1mL*10mM (DMSO)178,00€5mg207,00€10mg309,00€25mg527,00€50mg755,00€100mg1.044,00€500mg2.088,00€Taprizosin
CAS :Taprizosin（UK-338003） is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of benign prostatic hyperplasia.Formule :C25H26N6O4SDegré de pureté :98.10% - 99.11%Couleur et forme :SolidMasse moléculaire :506.58Nexopamil
CAS :Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.
Formule :C24H40N2O3Degré de pureté :97.87% - >99.99%Couleur et forme :SolidMasse moléculaire :404.59Antalarmin hydrochloride
CAS :Antalarmin hydrochloride, a CRF1 antagonist, offers anti-inflammatory benefits and prevents stress ulcers in IBS.Formule :C24H35ClN4Degré de pureté :99.84% - 99.85%Couleur et forme :SolidMasse moléculaire :415.02Masupirdine free base
CAS :Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used to study neurological disorders like Alzheimer's disease.Formule :C21H24BrN3O3SDegré de pureté :98.36% - 99.65%Couleur et forme :SolidMasse moléculaire :478.4Milveterol HCl
CAS :Milveterol HCl is a long-acting β(2) -adrenergic receptor agonist for the potential treatment of chronic obstructive pulmonary disease (COPD).Formule :C25H30ClN3O4Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :471.982'-MeCCPA
CAS :2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.Formule :C16H22ClN5O4Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :383.835-HT2 antagonist 1
CAS :5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.Formule :C22H29FN4O2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :400.49Ref: TM-T12597
1mg642,00€5mg1.288,00€1mL*10mM (DMSO)1.521,00€10mg1.738,00€25mg2.583,00€50mg3.484,00€100mg4.708,00€CB1 agonist 1
CAS :CB1 agonist 1 is a potent CB1 agonist with a pIC50 value of 5.7 for CB1 receptors.CB1 agonist 1 can be used to study brain disorders, pain, and inflammation.Formule :C24H24N2O5SDegré de pureté :98.56%Couleur et forme :SolidMasse moléculaire :452.52MK-0686
CAS :MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.Formule :C22H19ClF4N2O4Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :486.84Safotibant
CAS :Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edemaFormule :C25H34N4O5SDegré de pureté :99.62% - 99.67%Couleur et forme :SolidMasse moléculaire :502.63DA-6886
CAS :DA-6886 is a 5-HT4 agonist, relaxes rat oesophagus, with 1000x selectivity over hERG channels, pIC50: 4.3.Formule :C19H28Cl2N6O2Degré de pureté :99.91% - 99.99%Couleur et forme :SolidMasse moléculaire :443.37APNEA
CAS :APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.Formule :C18H22N6O4Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :386.41TC LPA5 4
CAS :TC LPA5 4 is a LPA5 receptor antagonist.Formule :C23H23ClN2O3Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :410.89Ref: TM-T23438
1mg49,00€5mg98,00€1mL*10mM (DMSO)107,00€10mg157,00€25mg324,00€50mg485,00€100mg713,00€200mg982,00€LAS38096
CAS :LAS38096 is an A2B adenosine receptor antagonist (Ki : 17 nM) that is potent, selective and efficient .Formule :C17H12N6ODegré de pureté :99.18% - 99.95%Couleur et forme :SolidMasse moléculaire :316.32JP1302
CAS :JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, renal issues.Formule :C24H24N4Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :368.47PSB-16133 sodium
CAS :PSB-16133 sodium is a selective P2Y purine receptor variant antagonist with an IC of 233 nM.Formule :C28H21N2NaO5S2Degré de pureté :98.03% - 98.93%Couleur et forme :SolidMasse moléculaire :552.60KI-7
CAS :KI-7 is an adenosine A2B receptor positive allosteric modulator.Formule :C23H18N2O2Degré de pureté :98.33%Couleur et forme :SolidMasse moléculaire :354.4Ref: TM-T9238
2mg35,00€5mg55,00€1mL*10mM (DMSO)62,00€10mg95,00€25mg172,00€50mg264,00€100mg399,00€200mg560,00€Ticalopride
CAS :Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.Formule :C14H20ClN3O3Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :313.78SB 218795
CAS :SB 218795 is an effective and selective antagonist of NK3 with a Ki 13 nM for hNK3 which is about 90-fold and 7000-fold selectivity over hNK2 and hNK1.Formule :C25H20N2O3Degré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :396.44Ref: TM-T23316
1mg49,00€2mg63,00€5mg90,00€1mL*10mM (DMSO)109,00€10mg160,00€25mg313,00€50mg505,00€100mg713,00€500mg1.504,00€Efletirizine
CAS :Efletirizine (UCB-28754), a histamine blocker and 5-LO inhibitor, aids in topical allergy treatment.Formule :C21H24F2N2O3Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :390.42AM-1235
CAS :AM-1235 is a potent and selective cannabinoid receptor CB1 agonist.Formule :C24H21FN2O3Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :404.43CCG 203769
CAS :CCG 203769 (Thiadiazolidinone (TDZD) deriv. 6) is a selective inhibitor of RGS4 with an IC50 of 17 nM for the RGS4-Gαo protein-protein interaction.Formule :C8H14N2O2SDegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :202.27Ref: TM-T10705
1mg84,00€5mg177,00€1mL*10mM (DMSO)195,00€10mg250,00€25mg444,00€50mg622,00€100mg893,00€500mg1.783,00€A-437203
CAS :A-437203 (Lu201640), selective D3 antagonist with Ki: D2-71nM, D3-1.6nM, D4-6220nM; based on 1H-pyrimidin-2-one scaffold.Formule :C20H27F3N6OSDegré de pureté :98.80%Couleur et forme :SolidMasse moléculaire :456.53Ref: TM-T10213
1mg94,00€5mg188,00€1mL*10mM (DMSO)215,00€10mg264,00€25mg411,00€50mg532,00€100mg740,00€200mg982,00€Lensiprazine
CAS :Lensiprazine (SLV314) is a potent dopamine D(2) receptor antagonist that acts as a serotonin reuptake inhibitor , and can be used to study bipolar disorder andFormule :C24H27FN4O2Degré de pureté :97.86%Couleur et forme :SolidMasse moléculaire :422.5PF-00217830
CAS :PF-00217830: agonist at serotonin 1A & dopamine D2, antagonist at serotonin 2A, potential schizophrenia study drug.Formule :C26H30N4O2Degré de pureté :98.72%Couleur et forme :SolidMasse moléculaire :430.54Octimibate
CAS :Octimibate: non-prostaglandin antiplatelet, treats cardiovascular disease, aids atherosclerosis/thrombosis research.Formule :C29H30N2O3Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :454.56Ticolubant
CAS :Ticolubant: Oral LTB4 antagonist, Ki=0.78 nM; blocks Ca2+ migration, IC50=6.6 nM; anti-inflammatory in mice.Formule :C23H19Cl2NO3SDegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :460.37Masilukast
CAS :Masilukast(MCC-847) is an oral leukotriene D4 (LTD4) receptor antagonist for the study of diseases associated with inflammation.Formule :C31H32F3N3O5SDegré de pureté :99.23% - 99.62%Couleur et forme :SolidMasse moléculaire :615.66Pirodomast
CAS :Pirodomast is a thromboxane A (TXA2) synthase inhibitor.Formule :C18H17N3O2Degré de pureté :99.14%Couleur et forme :SolidMasse moléculaire :307.35E6801
CAS :E6801: selective 5-HT6 agonist for research in dementia, Parkinson's, depression, obesity, epilepsy, anxiety, etc.Formule :C17H18ClN5O2S2Degré de pureté :96.32% - 97.24%Couleur et forme :SolidMasse moléculaire :423.94CL 316243
CAS :CL316243 is a highly potent selective agonist of β3-adrenoceptor.Cost-effective and quality-assured.Formule :C20H18ClNNa2O7Degré de pureté :98.00% - 99.68%Couleur et forme :SolidMasse moléculaire :465.79Adenosine antagonist-1
CAS :Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.
Formule :C18H13N7SDegré de pureté :99.28% - 99.95%Couleur et forme :SolidMasse moléculaire :359.41CB1R antagonist 1
CAS :CB1R antagonist 1 is a potent CB1R antagonist that can be used to study diseases related to the nervous system.Formule :C18H23F3N2O3SDegré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :404.45AZ-1355
CAS :AZ-1355 is a novel dibenzoxepine derivative with lipid-lowering properties.Formule :C17H17NO4Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :299.32Ref: TM-T13563
1mg78,00€1mL*10mM (DMSO)156,00€5mg170,00€10mg224,00€25mg338,00€50mg460,00€100mg600,00€200mg820,00€RS 67333 hydrochloride
CAS :RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.Formule :C19H30Cl2N2O2Degré de pureté :98.78%Couleur et forme :SolidMasse moléculaire :389.36Itasetron
CAS :Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer treatments.Formule :C16H20N4O2Degré de pureté :98.58% - 99.68%Couleur et forme :SolidMasse moléculaire :300.36MLS1547
CAS :MLS1547 is a potent D2 receptor G protein-biased agonist (Ki=1.2 μM, EC50=0.37 μM in Ca2+ assay).Formule :C19H19ClN4ODegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :354.83L-693,403 maleate
CAS :L-693,403 maleate has analgesic activity.Formule :C24H27NO4Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :393.48Ref: TM-T22899
1mg315,00€5mg745,00€10mg1.018,00€25mg1.431,00€50mg1.783,00€100mg2.250,00€500mg4.410,00€Terbogrel
CAS :Terbogrel is an antiplatelet drug, blocking thromboxane A2 receptor/synthase. Helps prevent clots.Formule :C23H27N5O2Degré de pureté :98.95%Couleur et forme :SolidMasse moléculaire :405.49PD 168568 dihydrochloride
CAS :PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).Formule :C22H29Cl2N3ODegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :422.39Ref: TM-T12383
5mg46,00€10mg55,00€1mL*10mM (DMSO)57,00€25mg111,00€50mg166,00€100mg235,00€200mg329,00€Ancriviroc
CAS :Ancriviroc (SCH-351125) is an orally bioavailable small molecule chemokine receptor CCR5 antagonist.Cost-effective and quality-assured.Formule :C28H37BrN4O3Degré de pureté :99.76% - 99.82%Couleur et forme :SolidMasse moléculaire :557.533YIL 781
CAS :YIL 781 is a selective ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM), showing a weak affinity for kinesin receptors (K = 6 μM).Formule :C24H28FN3O2Degré de pureté :98.8%Couleur et forme :SolidMasse moléculaire :409.5BL-1020 Mesylate
CAS :BL-1020 Mesylate (CYP-1020 Mesylate) is a GABA A receptor agonist and D2 antagonist used in studies of neurodegeneration.Formule :C28H45ClN4O11S4Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :777.39LX-2931
CAS :LX-2931(LX-3305) is a sphingosine-1-phosphate cleavage enzyme (S1P) inhibitor for the treatment of rheumatoid arthritis.Formule :C9H15N3O5Degré de pureté :98.85% - 99.83%Couleur et forme :SolidMasse moléculaire :245.23Ecastolol
CAS :Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.Formule :C26H33N3O6Degré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :483.56Ref: TM-T11148
1mg349,00€5mg697,00€1mL*10mM (DMSO)880,00€10mg888,00€25mg1.395,00€50mg1.783,00€100mg2.530,00€N-[(4-Aminophenyl)methyl]adenosine
CAS :N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).Formule :C17H20N6O4Degré de pureté :98.75%Couleur et forme :SolidMasse moléculaire :372.38Ref: TM-T16166
1mg52,00€5mg111,00€1mL*10mM (DMSO)141,00€10mg166,00€25mg318,00€50mg504,00€100mg803,00€Ensaculin
CAS :Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.Formule :C26H32N2O5Degré de pureté :99.56% - 99.81%Couleur et forme :SolidMasse moléculaire :452.54L 651896
CAS :L 651896 is an inhibitor of 5-lipoxygenase.Formule :C18H18O3Degré de pureté :96.06% - 99.85%Couleur et forme :SolidMasse moléculaire :282.33ABT-080
CAS :ABT-080 (VML 530), a leukotriene synthesis inhibitor, is used potentially for treatment of asthma.
Formule :C37H31N2NaO4Degré de pureté :98.42%Couleur et forme :SolidMasse moléculaire :590.64Tedatioxetine
CAS :Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.Formule :C18H21NSDegré de pureté :99.76% - >99.99%Couleur et forme :SolidMasse moléculaire :283.43Proxyfan
CAS :Proxyfan is a high-affinity protean antagonist/agonist of H3 receptors from full agonist to full inverse agonist, depending on given tissue or brain region.Formule :C13H16N2ODegré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :216.28D18024
CAS :D18024 is a phthalazinonderivat with anti-allergic and anti-histamine effect.Formule :C29H31ClFN3ODegré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :492.03Ref: TM-T10945
1mg349,00€5mg697,00€1mL*10mM (DMSO)880,00€10mg888,00€25mg1.395,00€50mg1.783,00€100mg2.530,00€
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