GPCR/G-Protéine
Les inhibiteurs des GPCR/protéines G sont des composés qui ciblent les récepteurs couplés aux protéines G (GPCR) et les protéines G associées, qui jouent un rôle crucial dans la transmission des signaux de l'extérieur vers l'intérieur des cellules. Ces inhibiteurs sont essentiels pour étudier les voies de signalisation médiées par les GPCR, impliquées dans de nombreux processus physiologiques, y compris la perception sensorielle, la réponse immunitaire et la neurotransmission. Les inhibiteurs des GPCR sont également importants dans le développement de médicaments, car de nombreux agents thérapeutiques ciblent ces récepteurs. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de GPCR/protéines G de haute qualité pour soutenir vos recherches en pharmacologie, biologie cellulaire et domaines connexes.
Sous-catégories appartenant à la catégorie "GPCR/G-Protéine"
- récepteur 5-HT(1.025 produits)
- Récepteur d'adénosine(249 produits)
- Récepteur adrénergique(3.017 produits)
- Récepteur de la bombésine(35 produits)
- Récepteur de la bradykinine(61 produits)
- CXCR(158 produits)
- CaSR(34 produits)
- Récepteur cannabinoïde(217 produits)
- Cholécystokinine(1 produits)
- Récepteur de la dopamine(445 produits)
- Récepteur de l'endothéline(86 produits)
- Récepteur GNRH(84 produits)
- GPCR19(33 produits)
- GRK(33 produits)
- GTPase(23 produits)
- Récepteur du glucagon(194 produits)
- Hérisson/Smoothened(49 produits)
- Récepteur de l'histamine(385 produits)
- Récepteur LPA(21 produits)
- Récepteur de la mélatonine(26 produits)
- Récepteur OX(41 produits)
- Récepteur opioïde(327 produits)
- PAFR(14 produits)
- PKA(60 produits)
- Récepteur S1P(18 produits)
- SGLT(31 produits)
- Récepteur Sigma(46 produits)
Affichez 19 plus de sous-catégories
5983 produits trouvés pour "GPCR/G-Protéine"
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Lu AA33810
CAS :Lu AA33810 is a selective neuropeptide Y5 (NPY5) receptor antagonist with an oral activity and BBB permeability, anti-anxiety and antidepressant-like effects.Formule :C19H25N3O2S3Degré de pureté :97.92% - 99.61%Couleur et forme :SolidMasse moléculaire :423.62Syk Inhibitor II hydrochloride
CAS :Syk signaling is key in lupus. Syk inhibitors reduce inflammation and sepsis severity in FcgRIIb-/- mice, lowering cytokines and organ damage.Formule :C14H16ClF3N6ODegré de pureté :99.05%Couleur et forme :SolidMasse moléculaire :376.77Gastrin I, rat
CAS :Gastrin I, rat is a peptide hormone that effectively stimulates gastric acid secretion.Formule :C94H128N22O31S2Couleur et forme :SolidMasse moléculaire :2126.3PT-129
PT-129 is a PROTAC degrader targeting the NTF2 domain of G3BP1/2, degrading stress granules in stressed cells, suppressing proliferation.Formule :C46H48N8O12SCouleur et forme :SolidMasse moléculaire :936.98Amylin (8-37), rat
CAS :Amylin (8-37), rat, an analog of IAPP, blocks insulin's effects on muscle glucose uptake and glycogen storage.Formule :C140H227N43O43Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3200.61LY 293284
CAS :LY 293284 is a potent, selective full agonist of 5-HT1A receptor with anxiogenic effects in animal studies.Formule :C19H26N2OCouleur et forme :SolidMasse moléculaire :298.42MLGFFQQPKPR-NH2
CAS :MLGFFQQPKPR-NH2 is a reversed Substance P peptide. Substance P is a neuropeptide [1] .Formule :C63H98N18O13SCouleur et forme :SolidMasse moléculaire :1347.63NF157
CAS :NF157, a selective P2Y11 antagonist with pKi 7.35, lowers MMP-3/MMP-13, aiding OA treatment; IC50s: P2Y11 463 nM, P2Y1 1811 μM, P2Y2 170 μM.Formule :C49H28F2N6Na6O23S6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1437.1Heterobivalent ligand-1
Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.Formule :C86H115FN16O21Couleur et forme :SolidMasse moléculaire :1727.93Cyclic SSTR agonist octreotide
Cyclic SSTR agonist octreotide is a Octreotide , serving as the cyclic Somatostatin Receptor SSTR agonist [1] .Formule :C53H71N11O14S2Couleur et forme :SolidMasse moléculaire :1150.33Melanostatin, frog TFA
Melanostatin, frog TFA is an α-MSH release inhibitor, a 36 amino acid peptide isolated from the frog brain.Degré de pureté :99.23%Couleur et forme :Odour Solid(R)-CJ 11974
CAS :(R)-CJ 11974: non-peptide NK1 receptor antagonist, may relieve pain and prevent chemo-induced vomiting.Formule :C31H38N2ODegré de pureté :97.15%Couleur et forme :SoildMasse moléculaire :454.65Chemerin-9 (149-157) TFA
Chemerin-9 (149-157) TFA is a peptide located at positions 149-157 of chemerin-9, acting as a ChemR23/CMKLR1 agonist.Formule :C56H67F3N10O15Degré de pureté :99.77%Couleur et forme :SolidMasse moléculaire :1177.18Chir 2279
CAS :CHIR 2279, a peptoid trimer, binds alpha 1-adrenoceptors, blocking epinephrine effects in dogs (pseudo pA2 6.86).Formule :C34H36N4O4Couleur et forme :SolidMasse moléculaire :564.67dCNP
dCNP binds to NPR-B/C receptors (NPR-B/C receptor), initiating the cGMP signaling pathway and regulating vascular function. It exhibits anti-hypoxic effects by downregulating hypoxia-related genes such as HIF1α and HIF2α. Additionally, dCNP inhibits tumor stroma induction, demonstrating antifibrotic properties. It also enhances immune response by upregulating CTL, NK cells, and conventional type 1 dendritic cells in tumors.Formule :C141H248N38O36S3Couleur et forme :SolidMasse moléculaire :3147.91BMS-753426
CAS :BMS-753426 is a potent and orally bioavailable antagonist of CCR2 .
Formule :C25H33F3N6O2Couleur et forme :SolidMasse moléculaire :506.574GHRF, porcine
CAS :GHRF, porcine, a growth hormone releasing factor (GHRF) peptide (porcine), binds to the growth hormone secretagogue receptor (GHSR), thereby inducing theFormule :C219H365N73O66SCouleur et forme :SolidMasse moléculaire :5108.76Asenapine citrate
CAS :Asenapine citrate: atypical antipsychotic for schizophrenia, bipolar disorder; targets serotonin, adrenoceptors, dopamine, histamine (pKi: 8.2-10.5).Formule :C23H24ClNO8Couleur et forme :SolidMasse moléculaire :477.89Human growth hormone-releasing factor TFA
Human growth hormone-releasing factor TFA is a hypothalamic peptide that promotes GH secretion by targeting pituitary GHRHR.Formule :C217H359F3N72O68SCouleur et forme :SolidMasse moléculaire :5153.67Guanylin(human)
CAS :Peptide that activates gut guanylyl cyclase, secreted by GI mucosa, regulates water and electrolytes in gut and kidneys.Formule :C58H87N15O21S4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1458.65Prostaglandin H1
CAS :Prostaglandin H1 is the cyclooxygenase metabolite of DGLA, a CRTh2 agonist and a precursor of a family of 1 anti-inflammatory prostaglandins.Formule :C20H34O5Couleur et forme :SolidMasse moléculaire :354.487Dexchlorpheniramine free base
CAS :Dexchlorpheniramine Maleate, a histamine receptor antagonist, is used to treat urticaria, allergic rhinitis, allergic conjunctivitis and pruritus.Formule :C16H19ClN2Degré de pureté :98%Couleur et forme :Oily Liquid SolidMasse moléculaire :274.79Substance P(1-7) TFA
CAS :Substance P(1-7) TFA is a fragment of neuropeptide P (SP), with anti-harmful effects, used in neurological disease research.Formule :C43H66F3N13O12Degré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :1014.06Vazegepant
CAS :Vazegepant is an intranasal CGRP receptor antagonist utilized for conducting acute migraine research.Formule :C36H46N8O3Degré de pureté :98.61% - 99.98%Couleur et forme :SolidMasse moléculaire :638.80Ref: TM-T38734
1mg96,00€5mg227,00€10mg335,00€25mg567,00€50mgÀ demander100mgÀ demander1mL*10mM (DMSO)305,00€9-deoxy-9-methylene Prostaglandin E2
CAS :9-deoxy-9-methylene PGE2: stable PGE2 analog with similar effects, less side effects, equal potency in rats, gerbils, primates.Formule :C21H34O4Couleur et forme :SolidMasse moléculaire :350.499HPP-9
HPP-9, a Proteolysis-Targeting Chimera (PROTAC) derived from Hedgehog Pathway Inhibitor-1 (HPI-1) with a pIC50 value of 6.71, is designed to degrade BETFormule :C49H52N6O11Couleur et forme :SolidMasse moléculaire :900.97Cyclosomatostatin Acetate
Cyclosomatostatin Acetate is an effective antagonist of the somatostatin receptor.Cyclosomatostatin Acetate inhibits SSTR1 signaling and decreases cell
Formule :C46H61N7O8Degré de pureté :98.83%Couleur et forme :SolidMasse moléculaire :840.02Ref: TM-T21567L
1mg150,00€2mg251,00€5mg373,00€10mg568,00€25mg843,00€50mg1.130,00€100mg1.529,00€200mg2.062,00€EP4 receptor antagonist 3
CAS :EP4 receptor antagonist 3 from patent WO2010019796 A1 targets EP4 for research on pain, arthritis, and cancer.Formule :C26H21F3N2O3SCouleur et forme :SolidMasse moléculaire :498.52HAEGTFTSD
CAS :HAEGTFTSD is GLP-1's initial segment; GLP-1 (7-36) amide, tied to food intake, stems from preproglucagon in L-cells.Formule :C40H57N11O17Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :963.94Adatanserin hydrochloride
CAS :Adatanserin hydrochloride (WY50324 hydrochloride) is a 5-HT(1A)/5-HT(2) receptor ligand that is neuroprotective and may be used in the study of depression.Formule :C21H32ClN5ODegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :405.96Thromboxane B1
CAS :Thromboxane B1 (TXB1) is a lipid eicosanoid, part of the TXB family, involved in blood clotting.Formule :C20H36O6Couleur et forme :SolidMasse moléculaire :372.5GPR55 agonist 4
GPR55 agonist 4 (Compound 28), with an EC50 of 131 nM for hGPR55 and 1.41 nM for rGPR55, effectively induces β-arrestin recruitment to human GPR55 [1].Formule :C19H16FN5O2Couleur et forme :SolidMasse moléculaire :365.36PD 142893
CAS :PD 142893 is a functional endothelin-stimulated vasoconstriction antagonist.Formule :C50H65N7O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :924.09Prostaglandin D2 methyl ester
CAS :PGD2: made in mast cells during allergic reactions, causes vasodilation and inhibits blood clots. PGD2 methyl ester is a similar, fat-soluble prodrug.Formule :C21H34O5Couleur et forme :SolidMasse moléculaire :366.498Binospirone
CAS :Binospirone (MDL 73005EF) is a 5-HT1A receptor agonist with anxiolytic activity used in the study of movement disorders associated with neurologic dysfunction.Formule :C20H26N2O4Degré de pureté :97.57% - 98.96%Couleur et forme :SoildMasse moléculaire :358.43Ref: TM-T71138L
1mg109,00€5mg261,00€10mg374,00€25mg583,00€50mg803,00€100mg1.063,00€200mg1.459,00€1mL*10mM (DMSO)33,00€tcY-NH2
CAS :Selective PAR4 antagonist peptide. Inhibits endostatin release and platelet aggregation induced by thrombin.Formule :C40H49N7O7Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :739.87Galanin (1-13)-Neuropeptide Y (25-36) amide
CAS :Galanin (1-13)-Neuropeptide Y (25-36) amide exhibits high-affinity binding to galanin receptors, similar to that of galanin itself [1].Formule :C136H209N41O34Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2962.37PACAP-related Peptide (rat) (trifluoroacetate salt)
PRP, a 29-amino acid peptide in the secretin/glucagon family, is found in rat brain regions and reproductive tissues.Couleur et forme :SolidRC-3095
CAS :RC-3095, a selective GRPR antagonist, has been shown to have anti-inflammatory properties in different models of inflammation.Formule :C56H79N15O9Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1106.32Tetrapeptide-1
CAS :Tetrapeptide-1 is a bioactive peptide renowned for its antioxidant properties and has been cited as an ingredient in cosmetics [1].Formule :C20H36N4O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :428.52Isobutyryl-L-carnitine
CAS :Isobutyryl-L-carnitine is a member of the class of compounds known as acylcarnitines. Isobutyryl-L-carnitine is a product of the acyl-CoA dehydrogenases.Formule :C11H21NO4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :231.29PACAP-38 (31-38), human, mouse, rat acetate
PACAP-38 (31-38) acetate stimulates PAC1 receptor and boosts NPY and catecholamine in sympathetic neurons.Formule :C49H87N17O13Degré de pureté :99.92%Couleur et forme :SolidMasse moléculaire :1122.32Lanepitant 2HCl
CAS :Lanepitant 2HCl is a non-peptide neurokinin-1 receptor antagonist that can be used to study painful neuropathy-like disorders such as migraine.Formule :C33H47Cl2N5O3Degré de pureté :98.67%Couleur et forme :SolidMasse moléculaire :632.66PSMA/GRPR ligand 1
PSMA/GRPR ligand 1 (compound 3) is a bispecific ligand with dual targeting capabilities for tumors that express PSMA(+) and GRPR(+).Couleur et forme :Odour SolidSigma-1 receptor antagonist 5
Sigma-1 receptor antagonist 5 (compound 12), a 4-pyridylpiperidine derivative, exhibits analgesic properties through its antagonistic action on sigma receptorsFormule :C26H27N3ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :397.51Invopressin
CAS :Invopressin (Compound 42), a vasopressin V1A receptor partial agonist (EC50: 1.0 nM), is utilized in research related to cirrhosis conditions such as bacterialFormule :C110H161N31O27S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2413.78LHRH
CAS :Luteinizing hormone-releasing hormone (LHRH) is a neuropeptide produced in the hypothalamus that plays a pivotal role in regulating reproduction and hasFormule :C55H74N16O14Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1183.27α-CGRP (mouse, rat) TFA
α-CGRP (mouse, rat) TFA, a neuropeptide belonging to the calcitonin gene-related peptide (CGRP) family, is predominantly located at neuromuscular junctions andFormule :C162H262N50O52S2·C2HF3O2Degré de pureté :98%Couleur et forme :SolidOxmetidine FA
Oxmetidine FA is an orally available specific histamine H2 receptor antagonist with antiulcerogenic properties.Formule :C20H23N5O5SDegré de pureté :97.34%Couleur et forme :SoildMasse moléculaire :445.49PSB-1114 triethylamine
PSB-1114 triethylamine is a potent, enzymatically stable, P2Y2 receptor agonist with a 134 nM EC50, exhibiting greater than 50-fold selectivity over P2Y4 (EC50Formule :C10H15F2N3O13P3S·xC6H15NDegré de pureté :98%Couleur et forme :SolidCB2R agonist 3
CB2R agonist 3, a potent activator of cannabinoid receptor 2 (CB2R), exhibits an EC50 value of 0.37μM, indicative of its significant role in the immune system [Degré de pureté :98%Couleur et forme :Odour Solid4-Hydroxy MPT
CAS :4-Hydroxy MPT (4-OH-MPT) is a serotonin-active compound that acts as an agonist for 5-HT2A and 5-HT2B receptors, with EC50 values of 3.82 nM and 3.4 nM, respectively.Formule :C14H20N2OCouleur et forme :SolidMasse moléculaire :232.32Prostaglandin K1
CAS :Prostaglandin K1 (compound 46) is a structurally modified prostanoid analog with an EC50 and Ki of 2800 nM for the EP1 receptor.Formule :C20H32O5Couleur et forme :SolidMasse moléculaire :352.47FGH31
FGH31 (Compound 24), a dopamine D4 agonist, exhibits potent and selective GRK2-dependency with a K i of 1.6 nM and partially activates β-arrestin [1].Formule :C33H36N4O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :520.66BAY-6672
CAS :BAY-6672 is, a selective,oral, highly potent human prostaglandin F (FP) receptor antagonist, exerts antifibrotic effects by inhibiting PGF₂α activity.Formule :C26H27BrClN3O3Degré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :544.87SSTR4 agonist-1
CAS :SSTR4agonist-1 (Compound 47) is a selective agonist of the somatostatin receptor 4 (SSTR4), with an EC50 of 4.7 nM. It has a half-life of over 130 minutes in human liver microsomes.Formule :C16H23N3O2Couleur et forme :SolidMasse moléculaire :289.37LY 344864 racemate
CAS :LY 344864 racemate is a 5-HT1F receptor agonist.Formule :C21H22FN3ODegré de pureté :99.75%Couleur et forme :SoildMasse moléculaire :351.42Casopitant
CAS :Casopitant (GW679769) is an orally active neurokinin-1 (NK1) receptor antagonist, researched for its potential use in managing chemotherapy-induced nausea and vomiting (CINV) and postoperative nausea and vomiting (PONV).Formule :C30H35F7N4O2Couleur et forme :SolidMasse moléculaire :616.61Org 13011
CAS :Org 13011 has CNS activity and induces conditioned taste aversion by mediating 5-HT 1A receptors.Formule :C18H25F3N4ODegré de pureté :98.02%Couleur et forme :SoildMasse moléculaire :370.41Ref: TM-T28258L
1mg109,00€5mg261,00€10mg374,00€25mg583,00€50mg803,00€100mg1.063,00€200mg1.431,00€1mL*10mM (DMSO)266,00€MEN 11270
CAS :B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.Formule :C60H90N20O11SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1299.56Misoprostol acid
CAS :Misoprostol acid is an active metabolite of Misoprostol,can be used for non-steroidal anti-inflammatory drug-induced (NSAID) gastric ulcers.Formule :C21H36O5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :368.51Labradimil
CAS :Labradimil, a bradykinin B2 agonist, boosts brain drug delivery and tumor survival rates.Formule :C49H75N15O12SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1098.29Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate
CAS :Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate is an NPR-A agonist and ANP hormone. Carperitide increases cGMP levels and reduces the heart's workload.Formule :C129H207N45O41S3Degré de pureté :99.78%Couleur et forme :SoildMasse moléculaire :3140.519(S)-HETE
CAS :19-HETE, a CYP450 arachidonic acid metabolite from kidneys, consists of 70% (S) and 30% (R) isomers and dilates renal vessels.Formule :C20H32O3Couleur et forme :SolidMasse moléculaire :320.473MDL 29913
CAS :NK2 tachykinin receptor selective antagonist.Formule :C40H56N8O6Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :745Latanoprost lactone diol
CAS :Latanoprost lactone diol, a key intermediate for synthesizing Latanoprost (a prostaglandin F2α analogue), lowers IOP by activating FP receptors.Formule :C18H24O4Degré de pureté :98%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :304.38UCM 549
CAS :UCM 549 is a bioactive chemical.Formule :C19H21NO2Couleur et forme :SolidMasse moléculaire :295.38SphK1&2-IN-1
CAS :SphK1&2-IN-1 is a sphingosine kinase inhibitor with anti-inflammatory, antitumor and hemostatic effects.
Formule :C14H14N2O3SDegré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :290.34Linzagolix choline
CAS :Linzagolix choline is a GnRH antagonist. It can be used to study pain associated with uterine fibroids and endometriosis.Formule :C27H28F3N3O8SDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :611.59Lanepitant
CAS :Lanepitant (LY303870) is a non-peptide neurokinin-1 (NK-1) antagonist with analgesic activity for the prevention of migraine.Formule :C33H45N5O3Degré de pureté :97.71%Couleur et forme :SolidMasse moléculaire :559.74Ethylpropyltryptamine
CAS :Ethylpropyltryptamine (EPT) is an orally active novel psychoactive substance. It is predicted to act as a partial agonist of the 5-HT2A receptor.Formule :C15H22N2Couleur et forme :SolidMasse moléculaire :230.35Bradykinin (1-7)
CAS :Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.Formule :C35H52N10O9Degré de pureté :98%Couleur et forme :White Lyophilized PowderMasse moléculaire :756.85L-796,778
CAS :L-796,778 is an SST3 agonist and a selective ligand of SST3, which can increase the level of cAMP in the body.Formule :C29H40N6O7Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :584.66Ref: TM-T32511
1mg175,00€5mg404,00€10mg592,00€25mg888,00€50mg1.243,00€100mg1.701,00€500mg3.402,00€1mL*10mM (DMSO)522,00€(S)-Osanetant
CAS :(S)-Osanetant, an S-enantiomer, is a selective NK3 antagonist with potential for treating schizophrenia and has anxiolytic and antidepressant effects.Formule :C35H41Cl2N3O2Couleur et forme :SolidMasse moléculaire :606.62Spiroglumide
CAS :Spiroglumide, a CCKB-gastrin antagonist that inhibits dose-dependent pentagastrin-induced acid hypersecretion with an ID50 of 20.1 (8.67-46.4) mg / kg, could beFormule :C21H26Cl2N2O4Degré de pureté :98.23%Couleur et forme :SoildMasse moléculaire :441.35MM 07
CAS :Biased agonist for apelin/G protein pathway, enhances eNOS and cell growth, reduces apoptosis, improves heart function, and dilates vessels.Formule :C67H106N22O14S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1539.9Benzomalvin B
CAS :Benzomalvin B, a metabolite from Penicillium, blocks 24% NK1 receptor binding at 100 μg/ml.Formule :C24H17N3O2Couleur et forme :SolidMasse moléculaire :379.419Cetirizine Impurity C
CAS :Cetirizine Impurity C - a metabolite of hydroxyzine, is a long-acting, oral H1-antihistamine.Formule :C21H25ClN2O3Couleur et forme :SolidMasse moléculaire :388.89VVZ-149
VVZ-149 is an antagonist of both serotonin receptor 2A (5HT2A) and glycine transporter type 2 (GlyT2), with potential anti-nociceptive activity.Couleur et forme :SolidA2A/A3 AR antagonist-1
A2A/A3 AR antagonist-1 is a dual fluorescent AR ligand with K i of 90 nM (hA2A) & 31.8 nM (hA3).Formule :C56H71N15O12S2Couleur et forme :SolidMasse moléculaire :1210.39Neuropeptide Y (13-36), amide, human
CAS :Neuropeptide Y (13-36), amide, human is a neuropeptide Y receptor agonist.Formule :C134H207N41O36SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3000.4ALEPH hydrochloride
CAS :ALEPH (hydrochloride) acts as a partial agonist of h5-HT2A and h5-HT2B receptors, with EC50 values of 10.3 nM and 19.2 nM, respectively. It can induce head twitch responses in mice, with an ED50 of 0.80 mg/kg.Formule :C12H20ClNO2SCouleur et forme :SolidMasse moléculaire :277.81GLP-1(7-37)
CAS :GLP-1 (7-37) is a truncated, bioactive form of GLP-1 that is the product of proglucagon processing in intestinal endocrine L cells.Formule :C151H228N40O47Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3355.67Blue FPG-A trisodium
CAS :Blue FPG-A trisodium is a P2X1 & P2Y1 receptor antagonist, IC50: 35.5 μM & 2.6 μM, related to RB2.Formule :C29H17ClN7Na3O11S3Couleur et forme :SolidMasse moléculaire :840.1A3AR modulator 1
MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.Formule :C23H25IN4Couleur et forme :SolidMasse moléculaire :484.38[Des-His1,Glu9]-Glucagon amide
CAS :Glucagon blocker with pA2 of 7.2; no agonist effect. Boosts insulin; prevents glucagon-driven hyperglycemia in rabbits and diabetic rats.Formule :C148H221N41O47SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3358.68R 396
CAS :R 396 (Acleu-asp-gln-trp-phe-glynh2) is a linear hexapeptide and is also an NK-2 tachykinin receptor antagonist.Formule :C39H51N9O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :805.88Mini Gastrin I, human
CAS :Mini Gastrin I, human, is a truncated form of the human gastrin peptide, encompassing amino acids 5-17 of the original sequence.Formule :C74H99N15O26SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1646.73MrgprX2 antagonist-4
CAS :MrgprX2 antagonist-4, from patent US20210128561A1, inhibits MrgprX2 receptor; useful for skin inflammation studies.Formule :C16H19N3OCouleur et forme :SolidMasse moléculaire :269.348Spantide I
CAS :Spantide antagonizes both bombesin & substance P. It is also tachykinin receptor antagonist.Formule :C75H108N20O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1497.79Calcitonin Gene Related Peptide (CGRP) II, rat
CAS :CGRP II is a potent vasodilator that boosts pancreatic enzyme levels by activating β-cell receptors.Formule :C163H267N51O50S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3805.31Survodutide TFA
Survodutide TFA (BI 456906 TFA) is a GCGR/GLP-1R dual agonist, a peptide compound used in obesity research.Formule :C192H289N47O61·xC2HF3OC2Degré de pureté :99.29% - 99.96%Couleur et forme :SolidMasse moléculaire :4231.62 (free base)4-Hydroxy MET
CAS :4-Hydroxy MET (4-HO-MET) is a tryptamine-based new psychoactive substance (NPS), structurally similar to the endogenous neurotransmitter serotonin. It has hallucinogenic properties that affect mood, movement, and cognitive functions.Formule :C13H18N2OCouleur et forme :SolidMasse moléculaire :218.3Luseogliflozin
CAS :Luseogliflozin inhibits SGLT2 for glucose uptake with 1.10 nM potency.Formule :C23H30O6SCouleur et forme :SolidMasse moléculaire :434.55Eloralintide sodium
Eloralintide sodium (LY-3841136 sodium) is an AMYR (amylin receptor) agonist applicable for studying type 2 diabetes and obesity.Formule :C201H319N49O65S2·xNaDegré de pureté :98.66%Couleur et forme :SolidMasse moléculaire :4526.1 (free base)17-phenoxy trinor Prostaglandin F2α ethyl amide
CAS :Prostaglandin F2α (PGF2α), acting through the FP receptor, causes smooth muscle contraction and exhibits potent luteolytic activity.Formule :C25H37NO5Couleur et forme :SolidMasse moléculaire :431.573Galanin (1-16), mouse, porcine, rat TFA
Galanin (1-16) agonizes hippocampal receptors; Kd 3 nM. Active on locus coeruleus neurons in mice, pigs, rats.Formule :C80H117F3N20O23Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1783.9Bertilimumab
CAS :Bertilimumab (CAT 213; iCo-008), a human monoclonal antibody that targets eotaxin-1 (CCL11), shows promise in the research of allergic disorders [1].Couleur et forme :LiquidBesipirdine hydrochloride
CAS :Besipirdine hydrochloride is a non-receptor-dependent cholinomimetic compound with cardiovascular activity that inhibits the uptake of biogenic amines.Formule :C16H18ClN3Degré de pureté :98.45%Couleur et forme :SoildMasse moléculaire :287.79MI 1544
CAS :MI 1544 is a LHRH antagonist.Formule :C71H94ClN17O13Couleur et forme :SolidMasse moléculaire :1429.09CI-988 hemihydrate
CI-988 hemihydrate (PD134308) is a potent and selective orally active CCK2R (cholecystokinin 2 receptor) antagonist, with an IC50 of 1.7 nM for mouse cortical CCK2. It is over 1600 times more selective for CCK2 than for CCK1 receptors. CI-988 hemihydrate exhibits anxiolytic and antitumor properties.Formule :C35H42N4O6H2OMasse moléculaire :632.321PAF C-18
CAS :PAF C-18 is a natural phospholipid molecule belonging to the platelet-activating factor (PAF) family,, involved in hemostasis and thrombosis by binding to PAFR.Formule :C28H58NO7PDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :551.745-HT2A receptor agonist-6
CAS :5-HT2A receptor agonist-6 (compound 47) is a selective agonist of the 5-HT2A receptor with a pEC50 value of 6.58.Formule :C18H19N3O3Couleur et forme :SolidMasse moléculaire :325.36CAY10509
CAS :CAY10509 is a PGF2α analogue and acts as an FP receptor inhibitor with an IC50 of 30 nM. It shows potential for use in studying the physiological regulatory mechanisms related to prostaglandins.Formule :C23H35FO5SCouleur et forme :SolidMasse moléculaire :442.58Ramelteon metabolite M-II
CAS :Ramelteon M-II binds MT1/MT2 with IC50s: 208/1470 pM; it's the main metabolite and a melatonin receptor agonist.Formule :C16H21NO3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :275.34exo-Tetrahydrocannabivarin
CAS :exo-Tetrahydrocannabivarin (Compound 12) is an analog of Δ9,11-THC. It weakly binds to cannabinoid receptors (CB) with an IC50 of 1.4 μM. In mice, exo-Tetrahydrocannabivarin exhibits activity related to both motor function and analgesia.Formule :C19H26O2Couleur et forme :SolidMasse moléculaire :286.41Neuropeptide Y 13-36 (porcine)
CAS :Neuropeptide Y 13-36 (porcine) is a selective neuropeptide Y2 receptor agonist.Formule :C135H209N41O36Couleur et forme :SolidMasse moléculaire :2982.408MLS1082
CAS :MLS1082 is a D1-like dopamine receptor (D1R) orthosteric modulatothat stimulates G-protein signaling upon dopamine activation for neurodegenerative disorders.Formule :C24H23N3O2Degré de pureté :99.53%Couleur et forme :SolidMasse moléculaire :385.46FFN246
CAS :FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation andFormule :C15H13FN2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :256.27Emoghrelin
CAS :Emoghrelin, extracted from Heshouwu (Polygonum multiflorum), promotes the secretion of growth hormone by activating the ghrelin receptor [1].Formule :C24H22O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :518.42BIBP3226
CAS :BIBP3226 is a potent and selective antagonist for the Neuropeptide Y receptor Y1 and the neuropeptide FF receptor.Formule :C27H31N5O3Couleur et forme :SolidMasse moléculaire :473.57(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
CAS :(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].Formule :C52H76N14O11S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1137.38Albiglutide fragment TFA
Albiglutide fragment (GLP-1 (7-36) analog) TFA represents a biologically active segment of Albiglutide, resistant to DPP-4 degradation due to its structure as aFormule :C148H224N40O45·xC2HF3O2Couleur et forme :SolidTCMCB07
CAS :TCMCB07, a cyclic nonapeptide, serves as an orally active, brain-penetrant antagonist of the melanocortin receptor 4 (MC4R), with significant implications inFormule :C63H87N15O11Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1230.461-39-Corticotropin (human)(TFA)
ACTH (1-39) human (TFA) is a melanocortin agonist that boosts adrenal CS production and affects the CNS and immune system.Formule :C207H308N56O58S·C2HF3O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4655.16PSB 0777 ammonium hydrate
PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM forFormule :C18H20N5O7S2·NH4·75H2ODegré de pureté :98%Couleur et forme :SolidMasse moléculaire :532.09Levocarnitine propionate hydrochloride
CAS :Levocarnitine propionate hydrochloride (ST-261) is used for the treatment of the deterioration of renal function, congestive heart failure, and other diseases.Formule :C10H20ClNO4Degré de pureté :90% - 99.77%Couleur et forme :SolidMasse moléculaire :253.72[D-Pro2] Spantide I TFA
[D-Pro2] Spantide I TFA is an analog of Spantide I, a selective antagonist of the NK1 receptor [1].Formule :C75H108N20O13·xC2HF3O2Degré de pureté :98%Couleur et forme :SolidHemokinin 1 (mouse)
CAS :Hemokinin 1 (mouse) is a selective excitogen 1 receptor agonist with a Ki value of 0.175 nM for the human NK1 receptor and 560 nM for the human NK2 receptor.Formule :C61H100N22O15SDegré de pureté :98%Couleur et forme :White PowderMasse moléculaire :1413.65Ala5-Galanin (2-11)
CAS :Ala5-Galanin (2-11) is a specific agonist for the galanin receptor 2 (GAL2R) with an affinity constant (Ki) of 258 nM [1].Formule :C54H81N13O13Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1120.3Bradykinin (1-6)
CAS :Bradykinin (1-6) is a stable, CPY-cleaved metabolite that triggers pain, induces muscle contractions, and activates NO synthetase.Formule :C30H45N9O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :659.73Sigma-1 receptor antagonist 4
Sigma-1 receptor antagonist 4 (Compound 32) is a potent σ1R antagonist that significantly enhances morphine's analgesic effects and reverses morphine-inducedFormule :C22H26N2OCouleur et forme :SolidMasse moléculaire :334.45Nebentan
CAS :Nebentan (YM598) is an oral, selective ETA antagonist; Ki: 0.697 nM (ETA), 569 nM (ETB); may slow cor pulmonale, myocardial infarction.
Formule :C24H21N5O5SCouleur et forme :SolidMasse moléculaire :491.52L-797,591
CAS :L-797,591 is a selective agonist of somatostatin receptor subtype 1.Formule :C38H49N5O2Couleur et forme :SolidMasse moléculaire :607.83Xenopus orexin B
CAS :Xenopus orexin B, a neuropeptide identified as an endogenous ligand for an orphan G-protein-coupled receptor, acts as a potent agonist of OX2R [1].Formule :C130H219N45O40S2Couleur et forme :SolidMasse moléculaire :3116.54NESS 0327
CAS :NESS 0327 is a high selectivity antagonist of the cannabinoid CB1 receptor. NESS 0327 is more than 60,000-fold selective for the CB1 receptor.Formule :C24H23Cl3N4ODegré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :489.82[D-Trp8]-γ-MSH
CAS :[D-Trp8]-γ-MSH is a selective melanocortin 3 (MC3) receptor agonist (IC50 values are 6.7, 340 and 600 nM for human MC3, MC5 and MC4 receptors respectively).Formule :C74H99N21O16SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1570.79Corynanthine
CAS :Corynanthe is a plant alkaloid. Corynanthe also has an alpha-2-adrenergic blocking activity.Formule :C21H26N2O3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :354.44Guanylin TFA (mouse,rat)
Guanylin (mouse, rat) TFA is a peptide composed of 15 amino acids and acts as an activator of intestinal guanylate cyclase. This compound is utilized in research related to diarrhea.Formule :C60H90N16O22S4·xC2HF3O2Couleur et forme :SolidMasse moléculaire :1515.71 (free base)Cholecystokinin (26-33) free acid
CAS :Cholecystokinin (26-33) free acid is part of CCK and induces mild taste aversion conditioning in rats.Formule :C49H61N9O14S2Degré de pureté :99.14%Couleur et forme :SoildMasse moléculaire :1064.19LCKLSL acetate
LCKLSL acetate is a potent AnxA2 inhibitor, blocking tPA binding and plasmin production, with anti-angiogenic effects.Formule :C32H61N7O10SDegré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :735.93MrgprX2 antagonist-3
CAS :MrgprX2 antagonist-3 (compound E117) is a MrgprX2 antagonist applicable for investigating cutaneous inflammation.Formule :C16H20FN3O2SDegré de pureté :98.06%Couleur et forme :SolidMasse moléculaire :337.41Ref: TM-T40271
1mg54,00€5mg114,00€10mg180,00€25mg362,00€50mg572,00€100mg914,00€1mL*10mM (DMSO)127,00€PAR 4 (1-6)
CAS :PAR 4 (1-6) can be used for relevant research in the life sciences. Its product number is T36293 and CAS number is 225779-44-2.Formule :C28H41N7O9Couleur et forme :SolidMasse moléculaire :619.676Preclamol hydrochloride
CAS :Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.Formule :C14H22ClNOCouleur et forme :SolidMasse moléculaire :255.78β-CGRP (mouse)
β-CGRP (mouse), a calcitonin gene-related peptide, induces vasodilation and is applicable in research areas including cardiovascular, pro-inflammatory, migraine, and metabolic studies.Formule :C165H265N49O55S2Couleur et forme :SolidMasse moléculaire :3879.29PROTAC(H-PGDS)-8
CAS :PROTAC(H-PGDS)-8 is a PROTAC degrader targeting Hematopoietic prostaglandin D synthase (H-PGDS), exhibiting an IC50 of 0.14 μM [1].Formule :C41H40N8O7Couleur et forme :SolidMasse moléculaire :756.81Adenosine receptor agonist 1
Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.Formule :C12H14ClN5O2SeCouleur et forme :SolidMasse moléculaire :374.68CRF, bovine
CAS :CRF, bovine is a potent agonist of CRF receptor, and displaces [125I-Tyr]ovine CRF with a Ki of 3.52 nM.Formule :C206H340N60O63SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4697.34Adrenomedullin (1-50), rat
CAS :Rat adrenomedullin (1-50) is a 50-AA peptide; induces arterial vasodilation by activating CGRP1 receptors.Formule :C248H381N77O75S5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :5729.5Ecnoglutide
CAS :Ecnoglutide (XW003) is a glucagon-like peptide 1 (GLP-1) receptor agonist [1] .Formule :C194H304N48O61Couleur et forme :SolidMasse moléculaire :4284.76LSN3160440
CAS :LSN3160440 is a GLP-1R allosteric modulator and PPI stabilizer aiding inactive GLP-1 attachment.Formule :C27H27Cl2N3OCouleur et forme :SolidMasse moléculaire :480.43Tetrahydro-β-carboline
CAS :Compound Fr12161, with CAS No. 16502-01-5, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound Fr12161 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formule :C11H12N2Degré de pureté :96.31%Couleur et forme :Tan SolidMasse moléculaire :172.2264cAC 253 acetate
cAC 253 acetate (TP2135 Free base) is an amylin antagonist. cAC 253 acetate inhibits 125I-adrenomedullin binding, with an IC50 of 25 nM.
Formule :C128H206N42O42S2Degré de pureté :98.16% - 99.99%Couleur et forme :SoildMasse moléculaire :3069.39Xanthine amine congener trihydrochloride
CAS :Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.Formule :C21H29ClN6O4Degré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :464.95α-Helical CRF(9-41) TFA
α-Helical CRF(9-41) TFA acts as a competitive antagonist for the CRF2 receptor, possessing a binding constant (K B) of approximately 100 nM.Formule :C168H275F3N46O55S2Couleur et forme :SolidMasse moléculaire :3940.42[D-Phe12,Leu14]-Bombesin
CAS :Bombesin receptor blocker; stops binding in rat brain (IC50=2 μM), hinders amylase release (IC50=4 μM), reduces appetite suppression in vivo.Formule :C77H113F3N22O20Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1724.9Cortistatin-14 acetate
Cortistatin-14 acetate, a neuropeptide have structural similarity to somatostatin-14, binds and exerts its function via the somatostatin receptors (sst1-sst5).
Formule :C83H118N20O20S2Degré de pureté :98.24% - 99.63%Couleur et forme :SoildMasse moléculaire :1780.08Peptide C105Y TFA
Peptide C105Y TFA is a cell-penetrating peptide synthesized based on the amino acid sequence of residues 359-374 of α1-antitrypsin. It enhances the gene expression of DNA nanoparticles.Formule :C97H148N20O23S·xC2HF3O2BQ-123 TFA
BQ-123 TFA: Potent ETA antagonist, IC50 = 7.3 nM, Ki = 25 nM, inhibits ET-1 cell proliferation, lowers rat BP.Formule :C33H43F3N6O9Couleur et forme :SolidMasse moléculaire :724.72Scyliorhinin II
CAS :Scyliorhinin II, a cyclic Tachykinin peptide, is a potent NK3 receptor agonist.Formule :C77H119N21O26S3Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1851.09Thioperamide maleate
CAS :Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31Formule :C19H28N4O4SDegré de pureté :98.48%Couleur et forme :SolidMasse moléculaire :408.52PF-03382792
CAS :PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.Formule :C23H32FN3O4Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :433.52Substance P (4-11)
CAS :Substance P (4-11), a C-terminal fragment of Substance P, acts as a highly selective agonist for NK1 receptors, demonstrating specificity in its interaction.Formule :C46H67N11O10SCouleur et forme :SolidMasse moléculaire :966.16Utreglutide
CAS :Utreglutide is a potent glucagon-like peptide 1 (GLP-1) receptor agonit [1] .Formule :C191H298N46O58Couleur et forme :SolidMasse moléculaire :4166.67Selepressin acetate
Selepressin acetate is a useful organic compound for research related to life sciences and the catalog number is T73654.Formule :C48H77N13O13S2Couleur et forme :SolidMasse moléculaire :1108.33Peptide YY (PYY) (3-36), porcine TFA
Peptide YY (PYY) (3-36), porcine TFA, functions as a gut hormone that serves as a Y2 receptor agonist, effectively reducing appetite [1].Formule :C176H272N52O54·C2HF3O2Couleur et forme :SolidMasse moléculaire :4094.44Dotanoc
CAS :Dotanoc is a ligand to make gallium Ga 68-DOTANOC, which is a gallium Ga 68-radiolabeled analog of somatostatin.Formule :C69H94N14O17S2Couleur et forme :SolidMasse moléculaire :1455.71[Ala2] Endothelin-3, human
CAS :[Ala2] Endothelin-3, a linear ET-3 analog with Ala replacing Cys, stimulates endothelial cell migration.Formule :C120H166N26O32S4Couleur et forme :SolidMasse moléculaire :2613.02CCK (26-30) (sulfated)
CAS :CCK (26-30) is a digestive and satiety-related peptide fragment inhibiting [125I]CCK-33 binding by 10% at 0.1 mM.Formule :C33H41N7O12S2Couleur et forme :SolidMasse moléculaire :791.85(D-Ser4,D-Ser(tBu)6,Azagly10)-LHRH
CAS :Analog of LHRH, stimulates LH and FSH release, controls reproduction.Formule :C59H84N18O14Couleur et forme :SolidMasse moléculaire :1269.41S1PR1 modulator 1
CAS :S1PR1 modulator 1 is a selective inhibitor of S1PR1 with a pIC50 of 7.6.Formule :C23H24N2O3SDegré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :408.51(S, R)-LSN 3318839
CAS :(S,R)-LSN 3318839 enhances GLP-1R, shows strong blood sugar lowering in animals, works with sitagliptin.Formule :C26H23Cl2N3O2Degré de pureté :99.41%Couleur et forme :SoildMasse moléculaire :480.39TRV045
CAS :TRV045 is a selective agonist of the sphingosine-1-phosphate (S1P) subtype 1 receptor and does not impact lymphocyte trafficking. It possesses antiepileptic properties.Formule :C18H18N4O3Couleur et forme :SolidMasse moléculaire :338.36Sarafotoxin S6b
CAS :non-selective endothelin receptor agonistFormule :C110H163N27O34S5Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :2567.96Kisspeptin 13
CAS :Kisspeptin 13 activates GPR54 & GnRH receptors, boosts memory, and aids in Alzheimer's research.Formule :C78H107N21O18Couleur et forme :SolidMasse moléculaire :1626.81Orexin B, human
CAS :Orexin B, human agonizes Orexin receptors (OX1 Ki=420 nM, OX2 Ki=36 nM), promotes feeding in rats, and is a neuropeptide.Formule :C123H212N44O35SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :2899.34Alsactide
CAS :Alsactide, an adrenocorticotropic hormone (ACTH) agonist and a heptadecapeptide analogue, is utilized in the study of the central nervous system [1].Formule :C99H155N29O21SCouleur et forme :SolidMasse moléculaire :2119.53Amylin (8-37), human
CAS :Human-derived Amylin (8-37) is a vasodilator in rat arteries and forms aggregates linked to type II diabetes.Formule :C138H216N42O45Couleur et forme :SolidMasse moléculaire :3183.495[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)
CAS :'[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)' is a selective NK2R agonist with prokinetic activity for smooth muscle studies.Formule :C39H64N8O10Couleur et forme :SolidMasse moléculaire :804.97GLP-1R agonist 14
CAS :GLP-1R agonist 14, also known as Compound 14, is a potent agonist of the GLP-1 receptor, demonstrating an EC50 range of 0-20 nM against human GLP-1 [1].Formule :C45H42F2N10O5Couleur et forme :SolidMasse moléculaire :840.88PAR650097
PAR650097 is a humanized monoclonal antibody targeting PAR2, used in migraine research.Degré de pureté :96.67% (SEC-HPLC) - 98.83% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :144.1 kDaAngiopeptin TFA
CAS :Angiopeptin TFA: somatostatin analogue, sst2/sst5 partial agonist (IC50: 0.26/6.92 nM), suppresses GH & IGF-1, for atherosclerosis research.Formule :C58H73F6N11O14S2Couleur et forme :SolidMasse moléculaire :1326.39Prepro-ANF (56-92), human
CAS :Human prepro-ANF (56-92) activates renal guanylate cyclase and boosts its activity.Formule :C173H270N44O57Couleur et forme :SolidMasse moléculaire :3878.26Protease-Activated Receptor-1, PAR-1 Agonist TFA
PAR-1 Agonist TFA: Selective peptide, mimics thrombin, activates PAR-1 receptor.Couleur et forme :LiquidAdrenomedullin (AM) (22-52), human TFA
Adrenomedullin (AM) human (22-52) is a truncated NH2 TFA-modified adrenal medullary receptor antagonist.Formule :C161H253N46F3O50Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3690.062-Furoyl-LIGRLO-amide
CAS :2-Furoyl-LIGRLO-amide TFA is a peptide that acts as a proteinase-activated receptor-2 (PAR2) agonist, and contains a furoyl group addition at its N-terminal.Formule :C36H63N11O8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :777.95Cagrilintide acetate
.Cagrilintide is a long-acting amylin analog,treat diabetes and obesity by reducing appetite through activation of the AMY3R and calcitonin receptor.Formule :C196H316N54O61S2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :4469.06α-CGRP, rat
CAS :Endogenous neuropeptide, potent vasodilatorFormule :C162H262N50O52S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :3806.25[D-Trp34]-Neuropeptide Y
CAS :Potent NPY Y5 receptor agonist (pEC50 = 7.82); highly selective; induces hyperphagia, body weight gain; orally active.Formule :C196H289N55O56Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4311.77[Arg-15,20,21,Leu17]-PACAP-Gly-Lys-Arg-NH2
CAS :[Arg-15,-20,-21, Leu17]-PACAP-Gly-Lys-Arg-NH2 (BM-PACAP) is a synthetic analogue of PACAP 1-27 that exhibits a relaxant effect [1].Formule :C157H253N53O42Couleur et forme :SolidMasse moléculaire :3555.02(Phe2,Orn8)-Oxytocin
CAS :(Phe2,Orn8)-Oxytocin: Selective V1 agonist, induces rabbit epididymis contractility, EC50=280 nM.Formule :C42H65N13O11S2Couleur et forme :SolidMasse moléculaire :992.18Orexin B, rat, mouse TFA
Orexin B, rat/mouse TFA, activates OX1-R & OX2-R receptors, influencing food intake, energy, and sleep regulation.Formule :C128H216F3N45O36SCouleur et forme :SolidMasse moléculaire :3050.42Adrenotensin (human)
CAS :Adrenotensin: human 153-185 fragment of Adrenomedullin precursor, a 52-amino acid peptide in CGRP hormone family.Formule :C143H224N42O43Couleur et forme :SolidMasse moléculaire :3219.56Kisspeptin-10, rat TFA
Kisspeptin-10, a rat TFA, constricts blood vessels, inhibits vessel growth, and counters Methotrexate reproductive toxicity.Formule :C65H84F3N17O17Couleur et forme :SolidMasse moléculaire :1432.46Naratriptan D3 Hydrochloride
CAS :Naratriptan D3 Hydrochloride is the deuterium labeled Naratriptan, is a selective agonist of 5-HT1 receptor subtype.Formule :C17H26ClN3O2SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :374.94[D-Phe12]-Bombesin
CAS :Bombesin receptor antagonist
Formule :C74H112N22O18SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1629.88Angiopeptin
CAS :Angiopeptin is a synthetic octapeptide analog of somatostatin; suppresses accelerated transplant atherosclerosis in rabbit heart arteries.Formule :C54H71N11O10S2Couleur et forme :SolidMasse moléculaire :1098.34Exendin-3
CAS :Exendin-3, a peptide from Gila monster venom, stimulates pancreatic secretion and belongs to the glucagon family.Formule :C184H282N50O61SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4202.57Antisauvagine-30
CAS :CRF2 receptor antagonist; Kd 1.4 nM (mCRF2β), 153.6 nM (rCRF1). Blocks sauvagine-induced cAMP in cells & stress-related responses in mice.Formule :C161H274N48O46SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :3650.29Apelin-36(human)
CAS :Endogenous APJ agonist, EC50=20nM, regulates cardiovascular function, fluid balance, and feeding; blocks certain HIV strains.Formule :C184H297N69O43SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :4195.87Meluadrine tartrate
CAS :Meluadrine tartrate is an endogenous metabolite.Formule :C16H24ClNO8Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :393.82Biotin-NeurokininA
Biotin-NeurokininA: biotinylated peptide, NK-2 receptor agonist, key in human airway and gut function.Formule :C60H94N16O16S2Couleur et forme :SolidMasse moléculaire :1359.61Protease-Activated Receptor-1 antagonist 2
CAS :Orally active PAR-1 antagonist with 7 nM IC50; potential for CVD research.Formule :C24H23F2N3O2Couleur et forme :SolidMasse moléculaire :423.46Zebrafish Kisspeptin-1
CAS :Zebrafish Kisspeptin-1 is the core sequence of the neuropeptide kisspeptin-1, which plays a crucial role in regulating the release of gonadotropin-releasing hormone (GnRH) and modulating the reproductive system.Formule :C58H84N16O15Couleur et forme :SolidMasse moléculaire :1245.39BAM(8-22)
CAS :Potent MRGPRX1 agonist peptide; first found in bovine adrenal glands. Non-opioid, lacking met-enkephalin motif. EC50: 8-150 nM.Formule :C91H127N25O23SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :1971.22Haloperidol D4
CAS :Haloperidol D4 is deuterium-labeled haloperidol.Formule :C21H23ClFNO2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :379.89(Ala13)-Apelin-13 TFA
'(Ala13)-Apelin-13 TFA acts as a potent antagonist of the apelin receptors (APJ) and impedes gastric motility via the vagal cholinergic pathway [1].'Formule :C63H107N23O16S·xC2HF3O2Couleur et forme :SolidMasse moléculaire :1474.73 (free acid)P2Y14R antagonist 3
P2Y14R antagonist 3 (compound A) is an orally active P2Y14R antagonist with an IC50 of 23.60 nM and a Kd of 7.26 μM. It mitigates lung injury in mice induced by Lipopolysaccharides (LPS) and can be utilized in the study of inflammatory diseases.Formule :C26H25N5O5Couleur et forme :SolidMasse moléculaire :487.51Exendin-4 (3-39)
CAS :Exendin-4 (3-39) is a truncated peptide missing first 2 amino acids of Exendin-4, a potent GLP-1r agonist used in diabetes and HPA axis research.
Formule :C176H272N46O58SCouleur et forme :SolidMasse moléculaire :3992.44[cPP1-7,NPY19-23,Ala31,Aib32,Gln34]-hPancreatic Polypeptide
CAS :Potent, selective NPY Y5 receptor agonist; IC50: 0.24 nM (Y5), >500 nM (Y2), 530 nM (Y1), 51 nM (Y4); Ki: 0.1-0.15 nM (Y5); increases food intake in vivo.Formule :C183H281N57O54S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :4207.67
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