
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.787 produits)
- Apoptose(6.265 produits)
- Cycle cellulaire/point de contrôle(4.800 produits)
- Chromatine/Épigénétique(2.446 produits)
- Signalisation du cytosquelette(1.530 produits)
- Altération de l'ADN/réparation de l'ADN(2.964 produits)
- Endocrinologie/Hormones(3.708 produits)
- Enzyme(3.669 produits)
- GPCR/G-Protéine(9.019 produits)
- Immunologie et Inflammation(3.883 produits)
- Virus de la grippe(301 produits)
- Signalisation JAK/STAT(414 produits)
- Signalisation MAPK(1.248 produits)
- Transporteur membranaire/Canal ionique(3.038 produits)
- Métabolisme(10.216 produits)
- Microbiologie/Virologie(7.607 produits)
- Neuroscience(10.383 produits)
- Autres inhibiteurs(36.019 produits)
- Oxydation-Réduction(42 produits)
- Signalisation PI3K/Akt/mTOR(1.442 produits)
- Protéases/Protéasome(1.726 produits)
- Cellules souche et Dérivés(823 produits)
- Tyrosine Kinase/Adaptateurs(2.039 produits)
- Ubiquitination(1.718 produits)
Affichez 16 plus de sous-catégories
66684 produits trouvés pour "Inhibiteurs"
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N-Methylbenzamide
CAS :N-Methylbenzamide is a potent phosphodiesterase 10A (PDE10A) inhibitor,with anti-cancer activity.Formule :C8H9NODegré de pureté :99.83%Couleur et forme :Physical Description Off-White Crystalline Solid (Ntp 1992)Masse moléculaire :135.16Indazole
CAS :Indazole, a heterocyclic compound, offers diverse biological activities.Formule :C7H6N2Degré de pureté :99.59% - 99.85%Couleur et forme :White Or Beige Crystalline PowderMasse moléculaire :118.14S-Dihydrodaidzein
CAS :S-Dihydrodaidzein ((3S)-7-hydroxy-3-(4-hydroxyphenyl)-2,3-dihydrochromen-4-one) is an enantiomer of dihydrodaidzein which is involved in equol biosynthesis in aFormule :C15H12O4Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :256.25Dasatinib
CAS :<p>Dasatinib (BMS-354825) is a tyrosine kinase inhibitor that inhibits Src and Bcr-Abl (Ki=16/30 pM) and is orally active and ATP-competitive.</p>Formule :C22H26ClN7O2SDegré de pureté :99.59% - 99.86%Couleur et forme :Pale-Yellow SolidMasse moléculaire :488.01L-Arabinopyranose
CAS :<p>L-Arabinopyranose (Pectinose) is an aldopentose, including an aldehyde (CHO) functional group.</p>Formule :C5H10O5Degré de pureté :99.86% - 99.91%Couleur et forme :White To Off White Crystalline PowderMasse moléculaire :150.13CSF1R-IN-1
CAS :CSF1R-IN-1 is a CSF1R inhibitor with IC50 of 0.5 nM.Formule :C25H20F3N5O2Degré de pureté :97.02% - 98.56%Couleur et forme :SolidMasse moléculaire :479.45Ref: TM-T10894
1mg94,00€5mg210,00€10mg325,00€25mg550,00€50mg787,00€100mg1.093,00€200mg1.454,00€1mL*10mM (DMSO)230,00€Retatrutide
CAS :Retatrutide (LY3437943) is a triple agonist of GCGR, GIPR and GLP-1R that can be used to study obesity.Formule :C221H342N46O68Degré de pureté :98.31%Couleur et forme :SolidMasse moléculaire :4732.09Pioglitazone hydrochloride
CAS :Pioglitazone hydrochloride (AD 4833) is the hydrochloride salt of an orally-active thiazolidinedione with antidiabetic properties and potential antineoplasticFormule :C19H20N2O3S·HClDegré de pureté :99.64% - >99.99%Couleur et forme :White Crystals Or Crystalline PowderMasse moléculaire :392.90Maprotiline hydrochloride
CAS :Maprotiline hydrochloride (Psymion) is a tetracyclic antidepressant akin to tricyclics with similar side effects.Formule :C20H24ClNDegré de pureté :99.68% - 99.84%Couleur et forme :White PowderMasse moléculaire :313.864Diclofenac
CAS :Diclofenac: a nonsteroidal compound inhibiting COX-1 and COX-2, reducing pro-inflammatory prostaglandins.Formule :C14H11Cl2NO2Degré de pureté :99.69% - 99.97%Couleur et forme :Crystals From Ether-Petroleum Ether SolidMasse moléculaire :296.15Sulfacarbamide
CAS :Sulfacarbamide (Sulfanilylurea) is a blood sugar-lowering agent.Formule :C7H9N3O3SDegré de pureté :95.6% - 99.72%Couleur et forme :SolidMasse moléculaire :215.23Robenacoxib
CAS :Robenacoxib (Onsior) is a non-steroidal compound with strong selectivity for cyclooxygenase-2 and anti-inflammatory activity.Formule :C16H13F4NO2Degré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :327.27Ref: TM-T26109
1mg69,00€2mg89,00€5mg149,00€10mg235,00€25mg455,00€50mg723,00€100mg938,00€500mg1.882,00€Nicotinic acid N-oxide
CAS :<p>Nicotinic acid N-oxide (Nicotinic acid 1-oxide) is a nicotinic acid derivative, used to treat hyperlipoidemia.</p>Formule :C6H5NO3Degré de pureté :99.93%Couleur et forme :Beige Fine Crystalline PowderMasse moléculaire :139.11Nilutamide
CAS :Nilutamide, a nonsteroidal anti-androgen, treats prostate cancer by blocking androgen receptors, not affecting other hormone receptors.Formule :C12H10F3N3O4Degré de pureté :98.67% - 99.78%Couleur et forme :Crystalline SolidMasse moléculaire :317.22Ravulizumab
CAS :Ravulizumab (ALXN1210) is a humanized antibody for blocking complement activation, treating PNH, aHUS, and myasthenia gravis.Degré de pureté :> 95%Couleur et forme :LiquidMasse moléculaire :145.80 kDaGiredestrant
CAS :Giredestrant (GDC-9545) is a potent oral anti-tumor ER antagonist competing with estradiol.Formule :C27H31F5N4ODegré de pureté :98.96% - 99.56%Couleur et forme :SolidMasse moléculaire :522.55Ref: TM-T11399
1mg111,00€5mg225,00€10mg354,00€25mg680,00€50mg1.074,00€100mg1.700,00€1mL*10mM (DMSO)259,00€Cav 2.2 blocker 1
CAS :Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.Formule :C25H29ClN2O2Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :424.96Ref: TM-T10690
1mg50,00€5mg111,00€10mg183,00€25mg340,00€50mg520,00€100mg780,00€200mg1.026,00€1mL*10mM (DMSO)117,00€Dimethyl sulfoxide
CAS :DMSO: polar solvent, aids drug penetration, cryopreservation, analgesic, anti-inflammatory.Formule :C2H6OSDegré de pureté :98%Couleur et forme :Clear LiquidMasse moléculaire :78.133Xentuzumab
CAS :Xentuzumab (BI836845) is a recombinant monoclonal antibody to humanised IGF ligand that inhibits AKT activation and can be used to study solid tumours.Degré de pureté :95.21% - >95.0% (SDS-PAGE); >95.0% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :143.7 kDaImidazole ketone erastin
CAS :View and buy Imidazole ketone erastin from TargetMol.Imidazole ketone erastin (IKE) is an inducer of ferroptosis. It has inhibition of the system Xc- cystine/glutamate transporter.Cited in 22 publications.Formule :C35H35ClN6O5Degré de pureté :98.48% - 99.87%Couleur et forme :SolidMasse moléculaire :655.14Ref: TM-T5523
1mg70,00€2mg96,00€5mg153,00€10mg195,00€25mg335,00€50mg512,00€100mg675,00€1mL*10mM (DMSO)170,00€BX430
CAS :BX430 is used for chronic pain and cardiovascular disease and it is a potent and selective noncompetitive allosteric human P2X4 receptor channels antagonistFormule :C15H15Br2N3ODegré de pureté :97.34%Couleur et forme :SolidMasse moléculaire :413.11Bax inhibitor peptide V5 acetate
Bax inhibitor peptide V5 acetate (Bax inhibitor peptide V5 acetate(579492-81-2 free base)) is a Bax-mediated apoptosis inhibitor, used for cancer treatment.Formule :C29H54N6O8SDegré de pureté :99.2%Couleur et forme :SolidMasse moléculaire :646.85Ref: TM-T10463L
1mg52,00€2mg66,00€5mg88,00€10mg130,00€25mg275,00€50mg454,00€100mg588,00€200mg768,00€1mL*10mM (DMSO)140,00€Pentoxifylline
CAS :Pentoxifylline (PTX) stimulates cytokines, inhibits phosphodiesterase, enhances blood flow, and increases cell flexibility.Formule :C13H18N4O3Degré de pureté :99.26% - 99.93%Couleur et forme :SolidMasse moléculaire :278.31Clomipramine hydrochloride
CAS :Clomipramine HCl (Anafranil) is a serotonin-inhibiting tricyclic antidepressant, well-absorbed and metabolized to desmethylclomipramine in the liver.Formule :C19H23ClN2·HClDegré de pureté :99.04% - 99.47%Couleur et forme :White To Slightly Yellow Crystalline PowderMasse moléculaire :351.31Chlorobenzothiazolinone
CAS :Chlorobenzothiazolinone blocks human chymase at 90 μM, assessed by fluorescence using a specific peptide substrate after 1 hr.Formule :C7H4ClNOSDegré de pureté :99.42% - 99.77%Couleur et forme :SolidMasse moléculaire :185.63Octopamine hydrochloride
CAS :Octopamine hydrochloride is akin to noradrenaline and acts as a neurohormone, neurotransmitter, and neuromodulator in invertebrates.Formule :C8H12ClNO2Degré de pureté :98.87% - 99.85%Couleur et forme :White Or Off-White SolidMasse moléculaire :189.64CCX140
CAS :CCX140 (CCX140-B) (CCX140-B) is an antagonist of CCR2.Formule :C20H13ClF3N5O3SDegré de pureté :99.66% - 99.95%Couleur et forme :SolidMasse moléculaire :495.86Repaglinide
CAS :Repaglinide, a benzoic acid derivative, stimulates insulin, treats type 2 diabetes, and may rarely cause acute liver injury.Formule :C27H36N2O4Degré de pureté :99.73% - >99.99%Couleur et forme :White To Off-White SolidMasse moléculaire :452.59Spesolimab
CAS :Spesolimab (BI 655130) is an antibody targeting IL-36 receptor, key in immunity, for systemic pustular psoriasis and dermatitis studies.Degré de pureté :> 95%Couleur et forme :LiquidMasse moléculaire :150 kDaPyrantel tartrate
CAS :Pyrantel tartrate (Banminth) is broad spectrum anthelmintic for livestock.Formule :C15H20N2O6SDegré de pureté :99.96%Couleur et forme :White CrystalsMasse moléculaire :356.39Methyl salicylate
CAS :Methyl salicylate (Gaultheria oil) is an organic ester. For acute joint and muscular pain, methyl salicylate is used as a rubefacient and analgesic.Formule :C8H8O3Degré de pureté :99.97%Couleur et forme :Colourless To Slightly Yellow LiquidMasse moléculaire :152.15Sabatolimab
CAS :Sabatolimab (MBG453) is a humanized IgG4 antibody that inhibits TIM-3 to modulate immunity and shows promise as an immunosuppressant.Degré de pureté :> 95% - > 95%Couleur et forme :LiquidMasse moléculaire :145 kDa (average)Turosteride
CAS :Turosteride is a small molecule steroidal 5α-reductase (5α-reductase) inhibitor.Turosteride has antitumor activity for the treatment of oncologic diseases andFormule :C27H45N3O3Degré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :459.66Imipenem monohydrate
CAS :Imipenem monohydrate (Imipenem) is a β lactam antibiotic. Imipenem monohydrate acts on the bacterial cell wall. Cost-effective and quality-assured.Formule :C12H19N3O5SDegré de pureté :98.77% - 99.94%Couleur et forme :Off-White Nonhygroscopic CrytalsMasse moléculaire :317.36Itopride hydrochloride
CAS :Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.Formule :C20H27ClN2O4Degré de pureté :99.59%Couleur et forme :White Or Pale Brownish CrystalMasse moléculaire :394.9Delgocitinib
CAS :Delgocitinib is a potent JAK inhibitor (IC50: 2.8-58 nM), treats inflammatory diseases, and is the first topical drug for atopic dermatitis.Formule :C16H18N6ODegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :310.35Ref: TM-T15096
1mg169,00€5mg311,00€10mg487,00€25mg929,00€50mg1.415,00€100mg2.062,00€200mg2.775,00€1mL*10mM (DMSO)349,00€Sulfamethizole
CAS :Sulfamethizole (Sulfamethizol) is a sulfathiazole antibacterial reagent.Formule :C9H10N4O2S2Degré de pureté :99.52%Couleur et forme :White To Pale Yellow Crystalline PowderMasse moléculaire :270.33Hydroxyhexamide
CAS :Hydroxyhexamide ((±)-Hydroxyhexamid) is a pharmacologically active metabolite of Acetohexamide, used as a hypoglycemic agent.Formule :C15H22N2O4SDegré de pureté :98.91%Couleur et forme :SolidMasse moléculaire :326.41AZ7550 hydrochloride
CAS :AZ7550 hydrochloride (AZ7550 hydrochloride ), an active metabolite of AZD9291, inhibits the activity of IGF1R (IC50: 1.6 μM).Formule :C27H32ClN7O2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :522.04Ibuprofen
CAS :Ibuprofen, an NSAID, reduces pain, inflammation, and fever by limiting prostaglandin production.Formule :C13H18O2Degré de pureté :99.7% - 99.81%Couleur et forme :Colorless Solid CrystallineMasse moléculaire :206.28Lycorine hydrochloride
CAS :Lycorine hydrochloride (Narcissine hydrochloride) is VE-cadherin inhibitor,and has IC50 of 1.2μM in Hey1B cell.It is an HCV inhibitor with strong activity.Formule :C16H18ClNO4Degré de pureté :99.45% - 99.49%Couleur et forme :Fine Crystal PowderMasse moléculaire :323.77β-Cyclodextrin
CAS :β-Cyclodextrin (NSC 269471) is a member of the class of compounds known as oligosaccharides.Formule :C42H70O35Degré de pureté :97.13% - 99.92%Couleur et forme :White Solid PowderMasse moléculaire :1134.98PMX 205 acetate(514814-49-4 free base)
PMX 205 acetate is an antagonist of complement C5a receptor (C5aR; CD88).Formule :C47H66N10O8Degré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :899.09Ref: TM-T12506L1
1mg111,00€5mg281,00€10mg369,00€25mg785,00€50mg1.254,00€100mg1.832,00€1mL*10mM (DMSO)394,00€Vocacapsaicin hydrochloride
CAS :<p>Vocacapsaicin hydrochloride (CA-008 hydrochloride) is a non-opioid TRPV1 agonist, a raw material for capsaicin, and is used for pain relief.</p>Formule :C26H42ClN3O4Degré de pureté :99.66% - 99.80%Couleur et forme :SolidMasse moléculaire :496.08Linezolid
CAS :Linezolid (PNU-100766), the first of the oxazolidinone class, is a synthetic antibiotic used for the therapy of infections resulted from multi-resistantFormule :C16H20FN3O4Degré de pureté :99.73% - 99.99%Couleur et forme :White SolidMasse moléculaire :337.35Ref: TM-T0391
10mg50,00€25mg85,00€50mg96,00€100mg145,00€200mg175,00€500mg283,00€1mL*10mM (DMSO)46,00€Prednisolone disodium phosphate
CAS :Prednisolone disodium phosphate, a synthetic glucocorticoid, has immunomodulating and anti-inflammatory properties.Formule :C21H27Na2O8PDegré de pureté :97.1% - 99.16%Couleur et forme :SolidMasse moléculaire :484.39C16 Sphingomyelin (d18:1/16:0)
CAS :C16 Sphingomyelin (d18:1/16:0) (N-Palmitoyl-D-sphingomyelin) is a phospholipid analog of phospholipid bilayers, which can be used to study biofilm activity.Formule :C39H79N2O6PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :703.03α-Lipoic Acid
CAS :<p>α-Lipoic Acid, a sulfur-containing octanoic acid derivative, is biosynthesized from linoleic acid and used in dietary supplements.</p>Formule :C8H14O2S2Degré de pureté :98.39% - 99.73%Couleur et forme :Forms Yellowish Flakes Light Yellow To Yellow PowderMasse moléculaire :206.33Anatibant 2HCl
CAS :<p>Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.</p>Formule :C34H36Cl2N6O5S·2ClHDegré de pureté :99.17% - 99.58%Couleur et forme :SoildMasse moléculaire :784.58Nisoldipine
CAS :Nisoldipine (BAY-k 5552) is a dihydropyridine calcium channel antagonist that acts as a potent arterial vasodilator and antihypertensive agent.Formule :C20H24N2O6Degré de pureté :98.79% - 99.57%Couleur et forme :SolidMasse moléculaire :388.41Fluorofenidone
CAS :<p>Fluorofenidone (AKF-PD) slows kidney fibrosis by inhibiting NADPH oxidase/ECM via PI3K/Akt, akin to AMR69 but less toxic with a longer half-life.</p>Formule :C12H10FNODegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :203.21Betamethasone dipropionate
CAS :<p>Betamethasone Dipropionate, a synthetic glucocorticoid, modulates gene expression to manage inflammation and autoimmune activity.</p>Formule :C28H37FO7Degré de pureté :98.13% - 99.59%Couleur et forme :PowderMasse moléculaire :504.59Diclofenac diethylamine
CAS :Diclofenac Diethylamine, a non-selective COX inhibitor, is utilized as a nonsteroidal anti-inflammatory drug (NSAID).Formule :C18H22Cl2N2O2Degré de pureté :99.81% - 99.87%Couleur et forme :SolidMasse moléculaire :369.29MIM1
CAS :MIM1 (Inhibitor of Mcl-1) is an myeloid cell factor 1 (Mcl-1) inhibitor.Formule :C17H21N3O3SDegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :347.43Ref: TM-T12041
1mg37,00€2mg52,00€5mg79,00€10mg119,00€25mgÀ demander50mgÀ demander1mL*10mM (DMSO)87,00€3-Methylsalicylic acid
CAS :3-Methylsalicylic acid (o-Cresotic acid) is a long-acting salicylate derivative with antilipidemic properties,which reduces plasma free fatty acid levels.Formule :C8H8O3Degré de pureté :97.36%Couleur et forme :SolidMasse moléculaire :152.15Axitinib
CAS :Axitinib (AG-013736) is a multi-targeted tyrosine kinase inhibitor that inhibits VEGFR1/2/3 and PDGFRβ. Axitinib has antitumor activity. Cost-effective and quality-assured.Formule :C22H18N4OSDegré de pureté :98.9% - 99.74%Couleur et forme :Off-White SolidMasse moléculaire :386.472-(2-Hydroxyethyl)pyridine
CAS :2-Pyridineethanol is used as an industrial chemistry intermediate.Formule :C7H9NODegré de pureté :99.90%Couleur et forme :Yellow-Brown Liquid LiquidMasse moléculaire :123.15SC-26196
CAS :SC-26196 is an orally active inhibitor of Delta6 desaturase (D6D) with IC50 of 0.2 μM in a rat liver microsomal assay, with antiinflammatory properties.Formule :C27H29N5Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :423.55DTNB
CAS :DTNB, or Ellman's Reagent, quantifies thiol groups and measures low-mass thiols like glutathione in pure and biological samples.Formule :C14H8N2O8S2Degré de pureté :97.11% - 99.51%Couleur et forme :Yellow SolidMasse moléculaire :396.35Clarithromycin
CAS :Clarithromycin (A-56268), a macrolide antibiotic, inhibits Cytochrome P450 3A4 and P-Glycoprotein.Formule :C38H69NO13Degré de pureté :98.77% - 99.89%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :747.95Pidotimod
CAS :Pidotimod is a synthetic dipeptide with immunomodulatory properties.Formule :C9H12N2O4SDegré de pureté :97.56% - 99.74%Couleur et forme :Almost White To White Crystalline PowderMasse moléculaire :244.27ART558
CAS :ART558 is a potent, selective, low molecular weight, allosteric DNA polymerase activity of Polθ inhibitor (IC50=7.9 nM).Formule :C21H21F3N4O2Degré de pureté :99.18% - 99.67%Couleur et forme :SolidMasse moléculaire :418.41Bupivacaine hydrochloride
CAS :Bupivacaine hydrochloride (Vivacaine) is a long-lasting, amide local anesthetic that blocks sodium channels, inhibiting nerve impulses and sensation.Formule :C18H28N2O·HClDegré de pureté :99.89% - 99.9%Couleur et forme :SolidMasse moléculaire :324.89Mitotane
CAS :<p>Mitotane (NCI-C04933) is a derivative of the insecticide dichlorodiphenyldichloroethane that specifically inhibits cells of the adrenal cortex.</p>Formule :C14H10Cl4Degré de pureté :99.89% - ≥95%Couleur et forme :Less Powder (Ntp 1992) Physical Description Colorless Powder (Ntp 1992)Masse moléculaire :320.04Oxaquin TEA
<p>Oxaquin TEA (MCB-3837 TEA), a precursor compound to MCB3681, is a DNA topoisomerase inhibitor that can be used to study Clostridium difficile infections and</p>Formule :C37H48F2N5O11PDegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :807.77Ethambutol dihydrochloride
CAS :Ethambutol dihydrochloride (CL40881) is a bacteriostatic antimycobacterial agent, which obstructs the formation of cell wall by inhibiting arabinosylFormule :C10H26Cl2N2O2Degré de pureté :98% - 99.95%Couleur et forme :Crystals White PowderMasse moléculaire :277.24Decitabine
CAS :Decitabine (Deoxycytidine) is a deoxycytidine analog, a DNA methyltransferase inhibitor with oral activity.Formule :C8H12N4O4Degré de pureté :98.06% - 99.87%Couleur et forme :Physical Description Fine White Crystalline Powder Used As A DrugMasse moléculaire :228.21Tepotinib
CAS :Tepotinib (EMD-1214063) is a selective, orally, and ATP-competitive c-MET tyrosine kinase inhibitor. Tepotinib has antitumor effect. Cost-effective and quality-assured.Formule :C29H28N6O2Degré de pureté :98% - 99.91%Couleur et forme :SolidMasse moléculaire :492.57Ref: TM-T6121
1mg39,00€2mg52,00€5mg85,00€10mg120,00€25mg225,00€50mg375,00€100mg532,00€200mg768,00€1mL*10mM (DMSO)92,00€Zatolmilast
CAS :Zatolmilast (BPN14770) is an allosteric inhibitor of selective phosphodiesterase 4D (PDE4D; IC50s: 7.8 nM and 7.4 nM for PDE4D7 and PDE4D3).Formule :C21H15ClF3NO2Degré de pureté :98.20%Couleur et forme :SolidMasse moléculaire :405.8Ref: TM-T10590
1mg70,00€5mg135,00€10mg245,00€25mg409,00€50mg562,00€100mg780,00€200mg1.026,00€1mL*10mM (DMSO)149,00€GABAA receptor agent 1
CAS :<p>GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.</p>Formule :C13H8ClN3O2Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :273.67BOS-172722
CAS :BOS-172722 is an inhibitor of monopolar spindle 1 (MPS1) checkpoint(IC50 of 2 nM).Formule :C24H30N8ODegré de pureté :99.37%Couleur et forme :SolidMasse moléculaire :446.55Torsemide
CAS :<p>Torsemide (AC-4464), a sulfonylurea loop diuretic, has a long action duration, high plasma protein binding, and a long half-life.</p>Formule :C16H20N4O3SDegré de pureté :99.81%Couleur et forme :Crystalline SolidMasse moléculaire :348.42Monensin sodium salt
CAS :Monensin sodium is an antiprotozoal agent produced by Streptomyces cinnamonensis.Monensin sodium salt (Monensin A sodium salt) causes a marked enlargement ofFormule :C36H61NaO11Degré de pureté :90% - 98.9%Couleur et forme :Almost White SolidMasse moléculaire :692.85Rimantadine hydrochloride
CAS :Rimantadine hydrochloride (Meradane) is an RNA synthesis inhibitor that is used as an antiviral agent in the prophylaxis and treatment of influenza.Formule :C12H21N·HClDegré de pureté :99.47% - 99.85%Couleur et forme :White Crystalline SolidMasse moléculaire :215.76Thioctamide
CAS :Thioctamide is 6,8-dithiooctanoic amide; carboxyl changes to amide linking to proteins/amines.Formule :C8H15NOS2Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :205.34Rotenolone
CAS :<p>Rotenolone (12alpha-HYDROXYROTENONE) is a metabolite of Rotenone which is a natural compound derived from plants of the genera Derris and Lonchocarpus.</p>Formule :C23H22O7Degré de pureté :99.27%Couleur et forme :SolidMasse moléculaire :410.42Oxantel Pamoate
CAS :<p>Oxantel Pamoate (Oxantel embonate) is used as an Antinematodal agent.</p>Formule :C36H32N2O7Degré de pureté :99% - 99.89%Couleur et forme :SolidMasse moléculaire :604.65(E/Z)-BCI
CAS :(E/Z)-BCI (NSC-150117), a dual-specificity phosphatase 6 (DUSP6) inhibitor with anti-inflammatory properties, reduces LPS-induced inflammatory mediators and ROSFormule :C22H23NODegré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :317.42Ref: TM-T11139
1mg80,00€5mg155,00€10mg283,00€25mg452,00€50mg638,00€100mg848,00€200mg1.121,00€1mL*10mM (DMSO)170,00€Tazobactam
CAS :<p>Tazobactam (YTR-830H) is an antibacterial penicillin derivative which inhibits the action of bacterial beta-lactamases.</p>Formule :C10H12N4O5SDegré de pureté :99.53%Couleur et forme :White To Off-White Solid PowderMasse moléculaire :300.29Bronopol
CAS :Bronopol (BNPD): Low-toxicity antimicrobial, highly effective against Gram-negative bacteria.Formule :C3H6BrNO4Degré de pureté :98.96% - 99.85%Couleur et forme :White Crystalline PowderMasse moléculaire :199.992-Chlorophenothiazine
CAS :2-Chlorophenothiazine is used as the intermediate of Chlorpromazine hydrochloride.Formule :C12H8ClNSDegré de pureté :98.18%Couleur et forme :Gray PowderMasse moléculaire :233.72Ziprasidone hydrochloride monohydrate
CAS :Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychoticFormule :C21H21ClN4OS·HCl·H2ODegré de pureté :98% - 99.83%Couleur et forme :Off-White PowderMasse moléculaire :467.12Amatuximab
CAS :Amatuximab is a chimeric humanized IgG1/k antibody targeting MSLN with antitumor effects for solid tumors.Degré de pureté :SDS-PAGE:95.2%;SEC-HPLC:98.4%Couleur et forme :LiquidMasse moléculaire :144.31 kDaEntecavir
CAS :Entecavir (SQ34676), a guanosine analogue, treats chronic HBV; may cause hepatitis B flares, not clear liver injury.Formule :C12H15N5O3Degré de pureté :99.14% - >99.99%Couleur et forme :White To Off-White/Yellow Crystalline PowderMasse moléculaire :277.28Ref: TM-T0085L
2mg35,00€5mg50,00€10mg87,00€25mg116,00€50mg166,00€100mg230,00€200mg344,00€1mL*10mM (DMSO)50,00€Aminoguanidine hydrochloride
CAS :Aminoguanidine hydrochloride (Hydrazinecarboximidamide) is a diamine oxidase and NO synthase inhibitor, used in the treatment of diabetic nephropathy.Formule :CH6N4·HClDegré de pureté :99.80%Couleur et forme :White To Off-White SolidMasse moléculaire :110.55Oxaliplatin
CAS :Oxaliplatin (L-OHP) is a DNA alkylating agent, an inhibitor of DNA synthesis.Formule :C8H14N2O4PtDegré de pureté :97% - 99.93%Couleur et forme :SolidMasse moléculaire :397.29Trimipramine maleate
CAS :Trimipramine maleate, a tricyclic antidepressant, blocks serotonin and norepinephrine reuptake, boosting their levels and duration.Formule :C24H30N2O4Degré de pureté :99.47%Couleur et forme :SolidMasse moléculaire :410.51VU0650786
CAS :VU0650786: selective mGlu3 NAM, CNS-penetrant, IC50 392 nM, shows antidepressant/anxiolytic effects in rodents.Formule :C18H15ClFN5O2Degré de pureté :99.09%Couleur et forme :SolidMasse moléculaire :387.8Ref: TM-T13318
1mg96,00€5mg235,00€10mg329,00€25mg560,00€50mg800,00€100mg1.103,00€1mL*10mM (DMSO)259,00€4-(Aminomethyl)benzoic acid
CAS :4-(Aminomethyl)benzoic acid (PAMBA), an antifibrinolytic, is an unnatural amino acid derivative.Formule :C8H9NO2Degré de pureté :99.55% - 99.64%Couleur et forme :White To Light Yellow Crystal PowderMasse moléculaire :151.16Calcein
CAS :Calcein is a fluorescent dye for detecting lipid vesicle leaks and calcium titration with EDTA.Formule :C30H26N2O13Degré de pureté :≥98%Couleur et forme :Orange PowderMasse moléculaire :622.53Kinetin
CAS :Kinetin (N6-Furfuryladenine), a type of cytokinin, has plant growth regulation effects.Formule :C10H9N5ODegré de pureté :99.55% - 99.83%Couleur et forme :Platelets From Absolute Ethanol SolidMasse moléculaire :215.21Ethopabate
CAS :Ethopabate (Ethyl pabate) is an inhibitor of folate metabolism, used as a coccidiostat in poultry.Formule :C12H15NO4Degré de pureté :98.44%Couleur et forme :White PowderMasse moléculaire :237.25Garetosmab
CAS :Garetosmab (REGN 2477), a human IgG4 monoclonal antibody, inhibits activin A for potential cancer treatment and FOP study.Degré de pureté :> 95% - > 95%Couleur et forme :LiquidMasse moléculaire :145.52 kDaUC-514321
CAS :UC-514321 directly targets STAT3/5 and represses TET1 expression.Formule :C26H35NO5Degré de pureté :98.50%Couleur et forme :SolidMasse moléculaire :441.56Ref: TM-T13950
1mg74,00€5mg160,00€10mg250,00€25mg502,00€50mg753,00€100mg1.130,00€200mg1.549,00€1mL*10mM (DMSO)170,00€Arimoclomol maleate
CAS :Arimoclomol maleate (BRX-220) (BRX-220) is a heat shock protein (HSP) co-inducer.Formule :C18H24ClN3O7Degré de pureté :99.44% - 99.98%Couleur et forme :SolidMasse moléculaire :429.85Ilginatinib maleate
CAS :<p>Ilginatinib maleate (NS-018 maleate) is a highly active and orally bioavailable inhibitor of JAK2.</p>Formule :C25H24FN7O4Degré de pureté :99.74% - 99.82%Couleur et forme :SolidMasse moléculaire :505.5NS1652
CAS :<p>NS1652 is an anion conductance inhibitor. NS1652 blocks chloride channel has an IC50 of 1.6 μM in human and mouse red blood cells.</p>Formule :C15H11F3N2O3Degré de pureté :99.62%Couleur et forme :SolidMasse moléculaire :324.25SCD1 inhibitor-4
CAS :<p>SCD1 inhibitor-4 is stearoylCoA desaturase-1 (SCD1) inhibitor. SCD1 inhibitor-4 can be used for the research of diabetes.</p>Formule :C17H16F3N5ODegré de pureté :99.71%Couleur et forme :SolidMasse moléculaire :363.34Lenvatinib
CAS :Lenvatinib (E7080) is a multi-target receptor tyrosine kinase inhibitor that inhibits VEGFR1-3, FGFR1-4, KIT, PDGFR, and RET, and has oral activity.Formule :C21H19ClN4O4Degré de pureté :98.46% - 99.96%Couleur et forme :SolidMasse moléculaire :426.85Azobenzene
CAS :Azobenzene, an aryl azo compound with a N=N bond between two phenyl rings, represents a broad molecule class.Formule :C12H10N2Degré de pureté :98.45%Couleur et forme :Orange-Red Leaflets Physical Description Orange-Red Crystals Or Dark Brown Chunky Solid (Ntp 1992)Masse moléculaire :182.22

