
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.782 produits)
- Apoptose(6.263 produits)
- Cycle cellulaire/point de contrôle(4.792 produits)
- Chromatine/Épigénétique(2.441 produits)
- Signalisation du cytosquelette(1.528 produits)
- Altération de l'ADN/réparation de l'ADN(2.965 produits)
- Endocrinologie/Hormones(3.707 produits)
- Enzyme(3.667 produits)
- GPCR/G-Protéine(9.009 produits)
- Immunologie et Inflammation(3.875 produits)
- Virus de la grippe(301 produits)
- Signalisation JAK/STAT(414 produits)
- Signalisation MAPK(1.248 produits)
- Transporteur membranaire/Canal ionique(3.033 produits)
- Métabolisme(10.209 produits)
- Microbiologie/Virologie(7.592 produits)
- Neuroscience(10.381 produits)
- Autres inhibiteurs(36.040 produits)
- Oxydation-Réduction(42 produits)
- Signalisation PI3K/Akt/mTOR(1.442 produits)
- Protéases/Protéasome(1.724 produits)
- Cellules souche et Dérivés(826 produits)
- Tyrosine Kinase/Adaptateurs(2.035 produits)
- Ubiquitination(1.717 produits)
Affichez 16 plus de sous-catégories
66683 produits trouvés pour "Inhibiteurs"
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mPEG-DSPE sodium
CAS :mPEG-DSPE sodium (DSPE-mPEG2000 sodium) is a PROTAC linker belonging to PEG and is involved in the synthesis of PROTAC molecules.Formule :C45H87NNaO11PCouleur et forme :SolidMasse moléculaire :2808.74Donanemab
CAS :Donanemab (LY3002813), a humanized IgG1 antibody, targets N-terminal Aβ for potential early Alzheimer's research.Degré de pureté :95%Couleur et forme :LiquidTPC2-A1-P
CAS :TPC2-A1-P is a TPC2 agonist that can differentially activate two-pore channel 2 (TPC2) and mimic the activation of TPC2 with NAADP and PIP (2).Formule :C20H21BrF3NO3Degré de pureté :98.49%Couleur et forme :SolidMasse moléculaire :460.29Ref: TM-T36806
1mg97,00€5mg236,00€10mg394,00€25mg750,00€50mg1.216,00€100mg1.853,00€1mL*10mM (DMSO)240,00€Panomifene TFA
Panomifene TFA(GYKl13504 TFA) is a antagonist of ERs with anticancer activity that can be used to study breast cancer and musculoskeletal diseases.Formule :C27H25F6NO4Degré de pureté :99.74%Couleur et forme :SoildMasse moléculaire :541.4815-Methyl Palmitic Acid
CAS :15-methyl Palmitic Acid is a methylated fatty acid that is widely found in animal lipids and may be involved in the regulation of fat metabolism.Formule :C17H34O2Degré de pureté :99.82%Couleur et forme :SolidMasse moléculaire :270.45Nardeterol HCl
<p>Nardeterol HCl is a β-adrenergic receptor partial agonist used in the study of the central nervous system.CAS 번호13460-73-83-4</p>Formule :C20H25ClFN3O2Degré de pureté :97.72% - 98.65%Couleur et forme :SoildMasse moléculaire :393.88Pranazepide
CAS :Pranazepide (FK 480) is a small molecule cholecystokinin receptor antagonist used to study digestive disorders and pancreatitis.Formule :C26H19FN4O2Degré de pureté :97.43% - 99.53%Couleur et forme :SolidMasse moléculaire :438.45AKOS037652256
CAS :AKOS037652256 modulates TRPML, treating TRPML-linked diseases like lysosomal disorders, muscular dystrophy, neurodegeneration, and oxidative stress.Formule :C24H26ClFN4O4S2Degré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :553.07Phosphonic acid, [(2R,3S)-3-methyloxiranyl]-, calcium salt
CAS :Phosphonic acid, [(2R,3S)-3-methyloxiranyl]-, calcium salt (9CI) (phosphonomycin calcium) is an antibiotic, used for the treatment of urinary tract infectionsFormule :C3H5O4P·CaDegré de pureté :99.56% - 99.68%Couleur et forme :SolidMasse moléculaire :176.12Eplerenone
CAS :<p>Eplerenone (CGP 30083) is an aldosterone receptor antagonist and potassium-sparing diuretic used in the therapy of hypertension.</p>Formule :C24H30O6Degré de pureté :99.75% - ≥98%Couleur et forme :White SolidMasse moléculaire :414.49Emibetuzumab
CAS :Emibetuzumab: potent humanized MET antibody, antitumor, inhibits HGF/MET pathways, for advanced prostate cancer research.Degré de pureté :SDS-PAGE:96.2%;SEC-HPLC:98.8%Couleur et forme :LiquidMasse moléculaire :143.74 kDaHydrocortisone Valerate
CAS :Hydrocortisone Valerate (Westcort) has anti-inflammatory, antipruritic and vasoconstrictive properties.Formule :C26H38O6Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :446.58Sulfacetamide sodium
CAS :<p>Sulfacetamide sodium (Sulamyd sodium) is an anti-infective agent. It is used topically to treat orally for urinary tract infections and skin infections.</p>Formule :C8H9N2NaO3SDegré de pureté :99.90% - 99.96%Couleur et forme :White Crystalline PowderMasse moléculaire :236.22Olutasidenib
CAS :Olutasidenib (FT-2102), an IDH1 inhibitor (IC50: 21.2/114 nM), is studied for treating AML/MDS and can cross the blood-brain barrier.Formule :C18H15ClN4O2Degré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :354.79Ref: TM-T16384
1mg62,00€5mg169,00€10mg264,00€25mg487,00€50mg710,00€100mg998,00€200mg1.320,00€1mL*10mM (DMSO)178,00€Piperacillin sodium
CAS :(CL227193) )binds to and inactivates penicillin-binding proteins (PBPs), enzymes located on the inner membrane of the bacterial cell wall, resulting in theFormule :C23H26N5NaO7SDegré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :539.54Oxidopamine hydrobromide
CAS :Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.Formule :C8H12BrNO3Degré de pureté :98.22% - 99.88%Couleur et forme :Beige To Brown Fine Crystalline PowderMasse moléculaire :250.09Darifenacin hydrobromide
CAS :Darifenacin hydrobromide (UK-88525) is a selective muscarinic receptor antagonist used to treat urinary incontinence and overactive bladder syndrome.Formule :C28H31BrN2O2Degré de pureté :99.75% - >99.99%Couleur et forme :SolidMasse moléculaire :505.45Sulfamethazine
CAS :Sulfamethazine (Sulfadimidine) is a sulfanilamide anti-infective agent. It has a spectrum of antimicrobial action similar to other sulfonamides.Formule :C12H14N4O2SDegré de pureté :99.88%Couleur et forme :White White Crystalline PowderMasse moléculaire :278.33Cav 2.2 blocker 1
CAS :Cav 2.2 blocker 1 is an N-type calcium channel (Cav 2.2; IC50: 1 nM) blocker for the treatment of pain.Formule :C25H29ClN2O2Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :424.96Ref: TM-T10690
1mg50,00€5mg111,00€10mg183,00€25mg340,00€50mg520,00€100mg780,00€200mg1.026,00€1mL*10mM (DMSO)117,00€Sulindac
CAS :Sulindac (Sulindac sulfoxide) is a sulfinylindene derivative prodrug with potential antineoplastic activity.Formule :C20H17FO3SDegré de pureté :99.09% - 99.15%Couleur et forme :Yellow SolidMasse moléculaire :356.41Dropropizine
CAS :<p>Dropropizine (UCB-1967), a racemic non-opiate antitussive agent, is served as a cough suppressant.</p>Formule :C13H20N2O2Degré de pureté :99.38%Couleur et forme :White Or Almost White PowderMasse moléculaire :236.31Glucosamine
CAS :<p>Glucosamine (Chitosamine) is used as a dietary supplement. Glucosamine has pharmacological effects on osteoarthritis cartilage. High-Quality, Low-Cost!</p>Formule :C6H13NO5Degré de pureté :99.8% - 99.8%Couleur et forme :CoaMasse moléculaire :179.17Dienestrol
CAS :Dienestrol (Restrol) is a synthetic and nonsteroidal estrogen, which is an estrogen receptor agonist.Formule :C18H18O2Degré de pureté :96.73% - 98%Couleur et forme :Minute Needles From Dilute Alc SolidMasse moléculaire :266.33AS-1763
CAS :AS-1763 is an orally available and selective BTK inhibitor with an IC50 of 0.85 nM.Formule :C33H31FN6O3Degré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :578.64BCI
CAS :BCI ((E)-BCI) is an allosteric inhibitor of dual-specificity phosphatase (DUSP; EC50s: 13.3 and 8.0 μM for DUSP6 and DUSP1 in cells) and does not inhibit DUSP5.Formule :C22H23NODegré de pureté :99.33% - 99.66%Couleur et forme :SolidMasse moléculaire :317.42GSK-3 inhibitor 4
CAS :Orally active GSK-3 inhibitor 4 targets GSK-3α/β, CDK2/5 (IC50: 0.45-0.68 μM) and may aid in Alzheimer's research by lowering Tau protein.Formule :C22H15F2N5ODegré de pureté :99.82%Couleur et forme :SoildMasse moléculaire :403.38Ref: TM-T77341
1mg333,00€5mg922,00€10mg1.140,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg3.734,00€LY 2389575 hydrochloride
CAS :LY2389575 hydrochloride is a selective mGlu3 NAM with 190 nM IC50, increases Mrc1, and aids Alzheimer's research.Formule :C15H16BrCl3N4Degré de pureté :99.9%Couleur et forme :SolidMasse moléculaire :438.58Acridine Orange hydrochloride
CAS :Acridine Orange is a cell-permeable fluorescent dye, binding to nucleic acids, used for staining and fluorescence cytochemistry; may mutate microorganisms.Formule :C17H20ClN3Degré de pureté :98.27% - 99.3%Couleur et forme :Orange PowderMasse moléculaire :301.81Pemetrexed disodium
CAS :<p>Pemetrexed disodium treats lung cancer/mesothelioma; may cause moderate serum enzyme elevation, rarely acute liver injury.</p>Formule :C20H19N5Na2O6Degré de pureté :99.29% - 99.49%Couleur et forme :Crystalline SolidMasse moléculaire :471.37Felbinac
CAS :Felbinac (Dapson), a topical medicine, is an active metabolite of fenbufen. Felbinac is belonging to the family of NSAIDs of the arylpropionic acid class.Formule :C14H12O2Degré de pureté :99.47%Couleur et forme :Beige Beige PowderMasse moléculaire :212.24Dimetridazole
CAS :Dimetridazole (1, 2-Dimethyl-5-nitroimidazole) is a agent that combats protozoan infections. Dimetridazole is a nitroimidazole class drug.Formule :C5H7N3O2Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :141.13Gut restricted-7
CAS :Gut restricted-7 (GR-7) (GR-7) is a covalent and orally active pan-bile salt hydrolase (BSH) inhibitor.Formule :C25H40FNaO6SDegré de pureté :98.81% - 99.27%Couleur et forme :SolidMasse moléculaire :510.64KRAS G12C inhibitor 19
CAS :KRAS G12C inhibitor 19 is a potent KRAS G12C inhibitor that shows anti-tumor activity in cellular assays, and the family inhibits tumor growth.Formule :C25H19ClF2N4O3SDegré de pureté :97.46%Couleur et forme :SolidMasse moléculaire :528.96APX-115 free base
CAS :APX-115 free base (Ewha-18278 free base) (Ewha-18278 free base) is a potent, orally active pan NADPH oxidase (Nox) inhibitor (Kis: 1.08 μM, 0.57 μM, and 0.63 μMFormule :C17H17N3ODegré de pureté :98.39%Couleur et forme :SolidMasse moléculaire :279.34Ref: TM-T10353
1mg49,00€5mg97,00€10mg160,00€25mg329,00€50mg533,00€100mg822,00€200mg1.130,00€1mL*10mM (DMSO)123,00€SHIP2-IN-1
CAS :SHIP2-IN-1 is a potent SHIP2 inhibitor(IC50 : 2 µM),and used in the research of Alzheimer’s disease.Formule :C17H13Cl2FN4ODegré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :379.22Ref: TM-T12901
1mg81,00€5mg170,00€10mg259,00€25mg429,00€50mg605,00€100mg815,00€200mg1.093,00€1mL*10mM (DMSO)180,00€Sanguinarine chloride
CAS :<p>Sanguinarine chloride (Pseudochelerythrine chloride), a benzophenanthridine alkaloid, stimulates apoptosis by activating the production of reactive oxygen</p>Formule :C20H14ClNO4Degré de pureté :98% - 99.41%Couleur et forme :SolidMasse moléculaire :367.78Clonidine hydrochloride
CAS :Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.Formule :C9H10Cl3N3Degré de pureté :99.16% - 99.86%Couleur et forme :SolidMasse moléculaire :266.55Belimumab
CAS :Belimumab, a human IgG1λ monoclonal antibody, blocks BAFF, treating lupus and related fatigue.Degré de pureté :SDS-PAGE:98.4%;SEC-HPLC:98.4%Couleur et forme :LiquidMasse moléculaire :144.07 kDaTerazosin hydrochloride
CAS :<p>Terazosin HCl (Hytrin) treats BPH and hypertension by blocking alpha1, affecting bladder and vessel muscles.</p>Formule :C19H26ClN5O4Degré de pureté :99.69% - 99.91%Couleur et forme :SolidMasse moléculaire :423.89Emodin
CAS :Emodin (Frangula emodin) is a selective 11β-HSD1 inhibitor,IC50 of 186 and 86 nM against 11β-HSD1 in humans and mice. High-Quality, Low-Cost!Formule :C15H10O5Degré de pureté :98.37% - 99.53%Couleur et forme :Physical Description Orange Needles Or Powder (Ntp 1992)Masse moléculaire :270.24Dimethylsulfamoyl chloride
CAS :Dimethylsulfamoyl chloride (DMSC) is an organosulfur compoundused in organic synthesis and laboratory reagents.Formule :C2H6ClNO2SDegré de pureté :99.31%Couleur et forme :Less Liquid Colorless LiquidMasse moléculaire :143.59NaV1.7 inhibitor-1
CAS :NaV1.7 inhibitor-1, an efficacious inhibitor of voltage-gated sodium channel (NaV) 1.7 (IC50 of 0.6 nM for hNaV1.7).Formule :C23H30FNO4SDegré de pureté :99.89%Couleur et forme :SolidMasse moléculaire :435.55Ref: TM-T12181
1mg104,00€5mg255,00€10mg406,00€25mg700,00€50mg938,00€100mg1.378,00€1mL*10mM (DMSO)280,00€Decarboxy Moxifloxacin
CAS :Decarboxylated moxifloxacin is a moxifloxacin derivative, an oral antibiotic for sinusitis, bronchitis, and pneumonia.Formule :C20H24FN3O2Degré de pureté :99.65%Couleur et forme :SolidMasse moléculaire :357.42Mefloquine hydrochloride
CAS :Mefloquine hydrochloride (Mefloquin hydrochloride) is a quinoline derivative used for the prevention and therapy of P. falciparum malaria.Formule :C17H17ClF6N2ODegré de pureté :99% - 99.99%Couleur et forme :Off-White To Yellow SolidMasse moléculaire :414.77Ketanserin
CAS :Ketanserin: quinazoline derivative, 5-HT2 receptor antagonist, may lower blood pressure and inhibit blood clots.Formule :C22H22FN3O3Degré de pureté :99.19% - 99.73%Couleur et forme :SolidMasse moléculaire :395.43Atorvastatin lactone
CAS :Atorvastatin lactone is a prodrug form of atorvastatin. Which is an orally active 3-hydroxy-3-methylglutaryl coenzyme A (HMG-CoA) reductase inhibitor.Formule :C33H33FN2O4Degré de pureté :98.05% - 98.16%Couleur et forme :SolidMasse moléculaire :540.62(E/Z)-BCI
CAS :(E/Z)-BCI (NSC-150117), a dual-specificity phosphatase 6 (DUSP6) inhibitor with anti-inflammatory properties, reduces LPS-induced inflammatory mediators and ROSFormule :C22H23NODegré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :317.42Ref: TM-T11139
1mg80,00€5mg155,00€10mg283,00€25mg452,00€50mg638,00€100mg848,00€200mg1.121,00€1mL*10mM (DMSO)170,00€PF429242 dihydrochloride
CAS :<p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>Formule :C25H37Cl2N3O2Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :482.49Naluzotan hydrochloride
CAS :<p>Naluzotan hydrochloride, a hERG K+ blocker (IC50: 3800 nM) and potent 5-HT1A agonist (IC50: ~20 nM, Ki: ~5.1 nM), is used in anxiety and depression studies.</p>Formule :C23H39ClN4O3SDegré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :487.1Adropin (34-76) (human, mouse, rat)
CAS :Adropin (34-76) (human, mouse, rat) is a peptide that attenuates liver fibrosis and insulin resistance. Cost-effective and quality-assured.Formule :C190H293N55O68S2Degré de pureté :94.23% - 99.95%Couleur et forme :SolidMasse moléculaire :4499.82GNE-781
CAS :GNE-781: potent CBP inhibitor (IC50: 0.94 nM), also targets BRET/BRD4(1) (IC50: 6.2/5100 nM).Formule :C27H33F2N7O2Degré de pureté :99.25% - 99.64%Couleur et forme :SolidMasse moléculaire :525.59Ref: TM-T15405
1mg138,00€5mg298,00€10mg485,00€25mg808,00€50mg1.093,00€100mg1.483,00€1mL*10mM (DMSO)343,00€Tea polyphenol
CAS :Tea polyphenol, also called green tea extract, are a mixture of chemical compounds, such as flavanoids and tannins, found naturally in tea.Formule :C17H19N3ODegré de pureté :98%Couleur et forme :Yelloish Green Free Flowing PowderMasse moléculaire :281.36Hexyl gallate
CAS :Hexyl gallate (Gallic acid hexyl ester), an alkyl ester derivative of gallic acid, exhibits potent antimalarial activity against Plasmodium falciparum (IC50: 0.Formule :C13H18O5Degré de pureté :99.78%Couleur et forme :SolidMasse moléculaire :254.28Dibenzosuberol
CAS :Dibenzosuberol is used as a Pharmaceutical intermediate.Formule :C15H14ODegré de pureté :98.73%Couleur et forme :White Fluffy PowderMasse moléculaire :210.27CL-82198
CAS :CL-82198, a selective MMP-13 inhibitor, serves as a pharmacological intervention to halt the progression of osteoarthritis (OA).Formule :C17H22N2O3Degré de pureté :95.91%Couleur et forme :SolidMasse moléculaire :302.37Ref: TM-T14978
5mg47,00€10mg73,00€25mg153,00€50mg243,00€100mg378,00€200mg552,00€500mg868,00€1mL*10mM (DMSO)50,00€Cy3 NHS ester
CAS :Cy3 NHS ester is a fluorescent dye used to label amino groups in proteins, peptides, antibodies, and oligonucleotides.Cost-effective and quality-assured.Formule :C34H40ClN3O4Degré de pureté :97.35% - 97.55%Couleur et forme :SolidMasse moléculaire :590.15CU-T12-9
CAS :CU-T12-9 is a potent TLR1/2 agonist(EC50 of 52.9 nM in HEK-Blue hTLR2 SEAP assay).Formule :C17H13F3N4O2Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :362.31Ref: TM-T15017
1mg52,00€5mg111,00€10mg169,00€25mg283,00€50mg432,00€100mg615,00€1mL*10mM (DMSO)124,00€(3S,4R,5S)-1,3,4,5,6-Pentahydroxyhexan-2-one
CAS :(3S,4R,5S)-1,3,4,5,6-Pentahydroxyhexan-2-one (L(-)-Sorbopyranose) is a ketose belonging to the group of sugars known as monosaccharides.Formule :C6H12O6Degré de pureté :99.97%Couleur et forme :Rhombohedral Crystals From Ethanol White To Off-White Crystalline PowderMasse moléculaire :180.16Pizotifen Malate
CAS :Pizotifen Malate (BC-105 malate), a highly selective 5-HT receptor blocking agent, is a drug based on benzocycloheptane.Formule :C19H21NS·C4H6O5Degré de pureté :99.96% - >99.99%Couleur et forme :SolidMasse moléculaire :429.53Elexacaftor
CAS :Elexacaftor (VX-445) is a cystic fibrosis transmembrane conductance regulator (CFTR) corrector.Cost-effective and quality-assured.Formule :C26H34F3N7O4SDegré de pureté :98.87% - 99.87%Couleur et forme :SolidMasse moléculaire :597.65Ref: TM-T14935
1mg87,00€2mg137,00€5mg243,00€10mg393,00€25mg772,00€50mg1.074,00€100mg1.444,00€1mL*10mM (DMSO)320,00€Levosulpiride
CAS :Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.Formule :C15H23N3O4SDegré de pureté :98.20% - 99.88%Couleur et forme :White Crystalline PowderMasse moléculaire :341.43Vincamine
CAS :Vincamine, from Vinca minor, is an alkaloid used as a vasodilator and antihypertensive for brain circulation issues.Formule :C21H26N2O3Degré de pureté :98.96%Couleur et forme :White To Almost White Fine Crystalline PowderMasse moléculaire :354.44dAURK-4 hydrochloride
dAURK-4 hydrochloride, a derivative of Alisertib, functions as a potent and selective degrader of AURKA (Aurora A), exhibiting anticancer properties [1].Formule :C52H53Cl2FN8O12Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :1071.93Cinnarizine
CAS :Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause Parkinson-like symptoms.Formule :C26H28N2Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :368.51Rifaximin
CAS :Rifaximin: an oral semi-synthetic antibiotic from rifamycin SV; targets bacterial RNA polymerase to halt growth.Formule :C43H51N3O11Degré de pureté :99.18% - 99.40%Couleur et forme :Red-Orange Crystalline PowderMasse moléculaire :785.88Ethidium bromide
CAS :<p>Ethidium bromide: trypanocidal, potential antiviral, binds to nucleic acids, inhibits acetylcholine receptors, fluorescent; used in biochemistry.</p>Formule :C21H20BrN3Degré de pureté :99.14% - >99.99%Couleur et forme :Dark Red Crystals From Alcohol Red-To-Brown CrystalsMasse moléculaire :394.32Oxybuprocaine hydrochloride
CAS :Oxybuprocaine hydrochloride (Oxybuprocaine HCl), a local anesthetic, is used especially in otolaryngology and ophthalmology.Formule :C17H29ClN2O3Degré de pureté :>99.99%Couleur et forme :White Crystalline PowderMasse moléculaire :344.88MLi-2
CAS :MLi-2: Novel, potent CNS-active LRRK2 inhibitor; IC50s: 0.76nM in vitro, 1.4nM cellular, 3.4nM binding.Formule :C21H25N5O2Degré de pureté :98.96%Couleur et forme :SolidMasse moléculaire :379.46Ref: TM-T16115
1mg58,00€2mg88,00€5mg133,00€10mg188,00€25mg432,00€50mg652,00€100mg929,00€1mL*10mM (DMSO)142,00€Anetumab
CAS :Anetumab: a human anti-mesothelin IgG1 for synthesizing Anetumab ravtansine, potentially treating metastatic pleural mesothelioma.Degré de pureté :SDS-PAGE:95.2%;SEC-HPLC:98.4%Couleur et forme :LiquidMasse moléculaire :143.77 kDaSLU-PP-1072
CAS :SLU-PP-1072: inverse agonist for ERRα/γ, disrupts PCa metabolism, induces apoptosis, studies prostate cancer.Formule :C18H12N2O3SDegré de pureté :97.66%Couleur et forme :SoildMasse moléculaire :336.36Miconazole nitrate
CAS :Miconazole nitrate, an antifungal, targets fungal cell membranes rich in ergosterol, distinct from mammalian cells.Formule :C18H15Cl4N3O4Degré de pureté :99.51%Couleur et forme :White Crystal PowderMasse moléculaire :479.15Proglumide
CAS :Proglumide (Binoside), an anti-ulcer drug, is a CCKA/CCKB antagonist that lowers gastric secretion and gastrointestinal motility.Formule :C18H26N2O4Degré de pureté :99.4% - 99.45%Couleur et forme :White Crystalline PowderMasse moléculaire :334.41REV 5901A
CAS :REV 5901A (REV 5901 HCl) is a leukotriene receptor antagonist and 5-LOX inhibitor with antimicrobial activity that attenuates the growth of colon cancer in miceFormule :C22H26ClNO2Degré de pureté :98.04%Couleur et forme :SoildMasse moléculaire :371.90Abexinostat
CAS :Abexinostat (PCI-24781) is a pan-HDAC inhibitor, strongest on HDAC1; less so on HDACs 2, 3, 6, 10. Very select for HDAC8. In Phase 1/2 trials.Formule :C21H23N3O5Degré de pureté :98.19% - 98.43%Couleur et forme :SolidMasse moléculaire :397.42Tolazoline hydrochloride
CAS :Tolazoline hydrochloride (NSC35110 (hydrochloride)) is a non-selective competitive α-adrenergic receptor antagonist used in treatment of persistent pulmonaryFormule :C10H13ClN2Degré de pureté :99.67%Couleur et forme :Pale Yellow Crystalline SolidMasse moléculaire :196.68Topilutamide
CAS :Topilutamide (Fluridil) is a topical nonsteroidal antiandrogen.Formule :C13H11F6N3O5Degré de pureté :98.77% - 99.24%Couleur et forme :SolidMasse moléculaire :403.23Ref: TM-T13184
1mg56,00€5mg119,00€10mg188,00€25mg393,00€50mg615,00€100mg877,00€200mg1.198,00€1mL*10mM (DMSO)131,00€Endoxifen (E-isomer)
CAS :Endoxifen E-isomer (E-Endoxifen) is the E-isomer of (Z)-Endoxifen. Endoxifen E-isomer has antiestrogenic effects.Formule :C25H27NO2Degré de pureté :98.57%Couleur et forme :SolidMasse moléculaire :373.49Ref: TM-T11200
1mg39,00€5mg97,00€10mg150,00€25mg283,00€50mg469,00€100mg735,00€200mg938,00€1mL*10mM (DMSO)94,00€Guaifenesin
CAS :Guaifenesin (Guaiphenesin) is an expectorant that also has some muscle relaxing action. It is used in many cough preparations.Formule :C10H14O4Degré de pureté :99.73% - 99.96%Couleur et forme :Minute Rhombic Prisms From Ether Drypowder Liquid OthersolidMasse moléculaire :198.22Metacavir
CAS :Metacavir, a reverse transcriptase inhibitor, is used potentially for the treatment of HBV infection.Formule :C11H15N5O3Degré de pureté :>99.99% - >99.99%Couleur et forme :SolidMasse moléculaire :265.272-Pyridinecarbohydrazide
CAS :2-Pyridinecarbohydrazide (2-Picolinyl hydrazide) is an effective inhibitor of Catalase-peroxidase-NAPDH.Formule :C6H7N3ODegré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :137.146PPD-Q
CAS :6PPD-Q (6PPD-Quinone) is an environmental pollutant that can target CNR2, CNR1, AA2AR, LCAT and TRPA1. High-Quality, Low-Cost!Formule :C18H22N2O2Degré de pureté :98.43% - 99.40%Couleur et forme :SolidMasse moléculaire :298.38MC3482
CAS :MC3482 is a specific inhibitor of sirtuin5 (SIRT5).Formule :C33H38N4O8Degré de pureté :98% - 99.90%Couleur et forme :SoildMasse moléculaire :618.68Ref: TM-T11962
1mg52,00€2mg74,00€5mg111,00€10mg180,00€25mg283,00€50mg445,00€100mg723,00€500mg1.454,00€Oxiracetam
CAS :<p>Oxiracetam (ISF2522), a cyclic derivative of gamma-aminobutyric acid (GABA), is utilized for the treatment of cognitive impairments.</p>Formule :C6H10N2O3Degré de pureté :99.67%Couleur et forme :White Crystalline PowderMasse moléculaire :158.16(R)-ADX-47273
CAS :<p>(R)-ADX-47273 is a potent mGluR5 positive allosteric modulator(EC50 of 168 nM for potentiation ).</p>Formule :C20H17F2N3O2Degré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :369.36Niacin
CAS :Niacin is a water-soluble B vitamin with antihyperlipidemic effects, found in food and converted to niacinamide for coenzyme activity.Formule :C6H5NO2Degré de pureté :99.68% - 99.96%Couleur et forme :White Solid PowderMasse moléculaire :123.11OMDM-1
CAS :OMDM-1 ((Z)-N-[(2S)-1-hydroxy-3-(4-hydroxyphenyl)propan-2-yl]octadec-9-enamide) is a selective and metabolically stable anandamide cellular uptake (ACU)Formule :C27H45NO3Degré de pureté :99.57%Couleur et forme :SolidMasse moléculaire :431.65Taurocholic acid
CAS :Taurocholic acid (N-Choloyltaurine) is a bile acid involved in the emulsification of fats.Taurocholic acid is cytoprotective, preventing tumor necrosis factor-Formule :C26H45NO7SDegré de pureté :99.59% - 99.85%Couleur et forme :Clusters Of Slender Four-Sided Prisms From Alcohol + Ether SolidMasse moléculaire :515.7Erythrosine B
CAS :Erythrosine B: red food dye for cherries, fish; dental plaque indicator; cell stain; similar to thyroxine.Formule :C20H6I4Na2O5Degré de pureté :97.29%Couleur et forme :Maroon PowderMasse moléculaire :879.86Ro 10-5824 dihydrochloride
CAS :Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).Formule :C17H22Cl2N4Degré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :353.29ZEN-3694
CAS :ZEN-3694 (ZEN 3694) is a bromo-structural domain extra-terminal inhibitor (BETi) with activity in androgen signaling inhibitor (ASI) resistance models and canFormule :C19H19N5ODegré de pureté :98.94% - 99.76%Couleur et forme :SolidMasse moléculaire :333.39Trastuzumab deruxtecan
CAS :<p>Trastuzumab deruxtecan (T-DXd) is an ADC with anticancer and antitumour activity that has been shown to improve gastric cancer.</p>Degré de pureté :95% - SEC-HPLC:98.49%Couleur et forme :LiquidMasse moléculaire :145 kDa (average)Lurtotecan
CAS :<p>Lurtotecan (GI147211) is a semisynthetic Camptothecin analog. Lurtotecan is a topoisomerase I inhibitor with anticancer effects.</p>Formule :C28H30N4O6Degré de pureté :99.18%Couleur et forme :SoildMasse moléculaire :518.56Neohesperidin
CAS :Neohesperidin (NSC-31048) with antioxidant and neuroprotective properties.Formule :C28H34O15Degré de pureté :96.73% - 98.53%Couleur et forme :White Solid Solid Particulate/PowderMasse moléculaire :610.56Sodium butanoate
CAS :<p>Sodium butanoate (Sodium Butyrate) is the sodium salt of butyrate with potential antineoplastic activity.</p>Formule :C4H7NaO2Degré de pureté :98.02% - 99.79%Couleur et forme :White PowderMasse moléculaire :110.09Benzydamine hydrochloride
CAS :Benzydamine hydrochloride (AF864), a locally-acting nonsteroidal anti-inflammatory drug, has local anaesthetic and analgesic properties.Formule :C19H23N3O·HClDegré de pureté :99.01%Couleur et forme :The White Crystalline PowderMasse moléculaire :345.87DL-Carnitine
CAS :DL-Carnitine: found in liver/muscle, used therapeutically for pancreatic/gastric secretions and hyperlipoproteinemia treatment.Formule :C7H15NO3Degré de pureté :99.75%Couleur et forme :SolidMasse moléculaire :161.2Cericlamine
CAS :Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.Formule :C12H17Cl2NODegré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :262.18Clindamycin phosphate
CAS :Clindamycin phosphate: a broad-spectrum chlorinated antibiotic, modified from lincomycin, used topically.Formule :C18H34ClN2O8PSDegré de pureté :98.15%Couleur et forme :White SolidMasse moléculaire :504.96Tirzepatide monosodium salt
Tirzepatide sodium salt (LY3298176 sodium salt) is a GIP and GLP-1 receptor agonist with neuroprotective activity and can be used to treat obesity.Formule :C225H347N48O68NaDegré de pureté :99.69%Couleur et forme :SoildMasse moléculaire :4835.51Nitisinone
CAS :<p>Nitisinone (SC0735)(SC0735) is an enzyme 4-hydroxyphenylpyruvate dioxygenase inhibitor.</p>Formule :C14H10F3NO5Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :329.23

