
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.687 produits)
- Apoptose(6.097 produits)
- Cycle cellulaire/point de contrôle(4.691 produits)
- Chromatine/Épigénétique(2.376 produits)
- Signalisation du cytosquelette(1.472 produits)
- Altération de l'ADN/réparation de l'ADN(2.921 produits)
- Endocrinologie/Hormones(3.611 produits)
- Enzyme(3.655 produits)
- GPCR/G-Protéine(8.755 produits)
- Immunologie et Inflammation(3.765 produits)
- Virus de la grippe(298 produits)
- Signalisation JAK/STAT(407 produits)
- Signalisation MAPK(1.230 produits)
- Transporteur membranaire/Canal ionique(2.947 produits)
- Métabolisme(9.940 produits)
- Microbiologie/Virologie(7.347 produits)
- Neuroscience(10.240 produits)
- Autres inhibiteurs(36.533 produits)
- Oxydation-Réduction(43 produits)
- Signalisation PI3K/Akt/mTOR(1.437 produits)
- Protéases/Protéasome(1.675 produits)
- Cellules souche et Dérivés(830 produits)
- Tyrosine Kinase/Adaptateurs(2.028 produits)
- Ubiquitination(1.682 produits)
Affichez 16 plus de sous-catégories
66582 produits trouvés pour "Inhibiteurs"
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Isoastragaloside II
CAS :<p>Isoastragaloside II (Astrasieversianin VII) is a derivative Astragaloside I, an ingredient in Astragalus membranaceus which have osteogenic properties.</p>Formule :C43H70O15Degré de pureté :98.59% - 99.73%Couleur et forme :SolidMasse moléculaire :827.01A-769662
CAS :A-769662 is an effective, reversible AMPK activator(EC50=0.8 μM).Formule :C20H12N2O3SDegré de pureté :97.52% - 99.58%Couleur et forme :SolidMasse moléculaire :360.39SB 415286
CAS :SB 415286 is a potent GSK3α inhibitor with IC50/Ki of 78 nM/31 nM with equally effective inhibition of GSK-3β.Formule :C16H10ClN3O5Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :359.72Asperuloside
CAS :Asperuloside (Asperulosid) has anti-inflammatory activity.Formule :C18H22O11Degré de pureté :99.42% - 99.99%Couleur et forme :SolidMasse moléculaire :414.36INCB032304
CAS :<p>INCB032304: Key for making Ruxolitinib, a JAK inhibitor, and Barretinib.</p>Formule :C15H21N5OSiDegré de pureté :99.26% - >99.99%Couleur et forme :SolidMasse moléculaire :315.45Magnocurarine
CAS :<p>Magnocurarine is a natural product from Magnolia officinalis.</p>Formule :C19H24NO3Degré de pureté :99.35% - >99.99%Couleur et forme :SolidMasse moléculaire :314.4Propaphos
CAS :<p>Propaphos (Kayaphos) is an organophosphorus-type insecticide.</p>Formule :C13H21O4PSDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :304.34AR-A014418
CAS :<p>AR-A014418 (GSK 3β inhibitor VIII) is an ATP-competitive, and selective GSK3β inhibitor.</p>Formule :C12H12N4O4SDegré de pureté :>99.99% - ≥95%Couleur et forme :SolidMasse moléculaire :308.31MHY-1685
CAS :<p>MHY-1685 is a mammalian target of rapamycin (mTOR) inhibitor and a senescence inhibitor that can rejuvenate senile hCSCs by modulating autophagy.</p>Formule :C11H8N2O4Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :232.19Vindesine sulfate
CAS :Vindesine sulfate, a vinca alkaloid derived from vinblastine, binds to spindle microtubules, causing cell death.Formule :C43H57N5O11SDegré de pureté :97.51%Couleur et forme :Amorphous SolidMasse moléculaire :852Sudan III
CAS :Sudan III (Solvent Red 23) is a solvent dye used to color nonpolar substances.Formule :C22H16N4ODegré de pureté :97.38%Couleur et forme :DrypowderMasse moléculaire :352.39Oxyfluorfen
CAS :Oxyfluorfen (Boxer), a herbicide of the nitrodiphenyl ether class, is used to control annual and perennial broad-leaved weeds and sedges in a variety of fieldFormule :C15H11ClF3NO4Degré de pureté :98.73% - 99.28%Couleur et forme :Orange Crystalline Solid At Room Temperature SolidMasse moléculaire :361.7EPZ004777 hydrochloride
CAS :EPZ004777 hydrochloride (EPZ004777 HCl) is a potent, selective DOT1L inhibitor with IC50 of 0.4 nM.Formule :C28H42ClN7O4Couleur et forme :SolidMasse moléculaire :576.13Nonacosane
CAS :Nonacosane is a straight-chain alkane comprising of 29 carbon atoms. It has a role as a plant metabolite and a volatile oil component.Formule :C29H60Degré de pureté :98.62% - ≥95%Couleur et forme :Orthorhombic Crystals From Petroleum Ether White FlakesMasse moléculaire :408.79Carabrone
CAS :Carabrone, a botanical bicyclic sesquiterpenic lactone, is a promising fungicidal agent that can effectively control G. tritici.Formule :C15H20O3Degré de pureté :99.72% - 99.9%Couleur et forme :SolidMasse moléculaire :248.32Bergamottin
CAS :<p>1.</p>Formule :C21H22O4Degré de pureté :97.59% - 99.99%Couleur et forme :SolidMasse moléculaire :338.4Nile Red
CAS :<p>Nile Red (Nile Blue A oxazone) is a strongly fluorescent stain used for the detection of intracellular lipid droplets in the presence of a hydrophobic</p>Formule :C20H18N2O2Degré de pureté :95.61% - 98.99%Couleur et forme :SolidMasse moléculaire :318.371-Octanol
CAS :<p>1-Octanol is a saturated fatty alcohol, inhibits T-type Ca²⁺ channels with a 4 μM IC50, and is a potential diesel-like biofuel.</p>Formule :C8H18ODegré de pureté :99.94%Couleur et forme :Colourless LiquidMasse moléculaire :130.23DI-N-OCTYL PHTHALATE
CAS :Phthalate ester: plasticizer/additive, studied for food contamination and toxicology.Formule :C24H38O4Degré de pureté :98.22%Couleur et forme :Clear Oily Liquid Penetrate The Soil And Contaminate Groundwater And Nearby Streams Eye Contact May ProduceMasse moléculaire :390.564',7-Dimethoxyisoflavone
CAS :4',7-Dimethoxyisoflavone (Daidzein dimethyl ether) , a kind of isoflavonoids, showed inhibitory effects on rat prostate testosterone 5α-reductase.Formule :C17H14O4Degré de pureté :98.23% - 98.39%Couleur et forme :SolidMasse moléculaire :282.29Biotinyl tyramide
CAS :Biotinyl tyramide, a biotin derivative, enhances in situ hybridization and immunohistochemical signals.Formule :C18H25N3O3SDegré de pureté :98.08% - 99.94%Couleur et forme :SolidMasse moléculaire :363.47Kaempferol-7-O-β-D-glucopyranoside
CAS :<p>Kaempferol-7-O-β-D-glucopyranoside (Kaempferol-7-O-D-glucopyranoside) , a novel supercoolant could be used to sub-zero non-freezing rat heart preservation.</p>Formule :C21H20O11Degré de pureté :99.91% - 99.96%Couleur et forme :SolidMasse moléculaire :448.38(-)-Dizocilpine maleate
CAS :<p>(-)-Dizocilpine maleate ((-)-MK 801 (Maleate)) is a potent, selective and non-competitive NMDA receptor antagonist with Kd of 37.2 nM in rat brain membranes.</p>Formule :C20H19NO4Degré de pureté :>99.99%Couleur et forme :White SolidMasse moléculaire :337.37Methoxyfenozide
CAS :Methoxyfenozide is an insect growth regulator. Methoxyfenozide used in the control of lepidopteran insect pests.Formule :C22H28N2O3Degré de pureté :99.59%Couleur et forme :White PowderMasse moléculaire :368.47Mibefradil dihydrochloride
CAS :<p>Mibefradil dihydrochloride (Ro 40-5967 (dihydrochloride)) is an blocker of calcium channel with moderate selectivity for T-type Ca2+ channels (T-type and L-type</p>Formule :C29H40Cl2FN3O3Degré de pureté :99.45% - 99.72%Couleur et forme :SolidMasse moléculaire :568.55Aficamten
CAS :<p>Aficamten is a Next-Generation Cardiac Myosin Inhibitor for the Treatment of Hypertrophic Cardiomyopathy.</p>Formule :C18H19N5O2Degré de pureté :99.19% - 99.57%Couleur et forme :SolidMasse moléculaire :337.382-Deoxy-2-sulfoamino-D-glucose sodium
CAS :2-Deoxy-2-sulfoamino-D-glucose sodium (GlcN-2S) is possible to effect reaction at arthritis.Formule :C6H12NNaO8SDegré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :281.22Nortrachelogenin-8'-O-β-glucoside
CAS :<p>Lignan 'Nortrachelogenin-8'-O-beta-glucoside with butyrolactone structure, found in Trachelospermum jasminoides leaves/stems.</p>Formule :C26H32O12Degré de pureté :97.05% - 98.46%Couleur et forme :SolidMasse moléculaire :536.53Biotin-PEG2-C2-iodoacetamide
CAS :Biotin-PEG2-C2-iodoacetamide (Biotin-PEG2-iodoacetamide) is a PEG-based PROTAC linker that can be used in PROTAC synthesis.Formule :C18H31IN4O5SDegré de pureté :98.01% - 99.85%Couleur et forme :SolidMasse moléculaire :542.43Aminohippurate sodium
CAS :Aminohippurate sodium (Sodium p-aminohippurate) is used as a diagnostic aid to measure effective renal plasma flow (ERPF) and excretory capacity.Formule :C9H9N2NaO3Degré de pureté :99.82%Couleur et forme :Beige Crystalline PowderMasse moléculaire :216.17Azido-PEG5-azide
CAS :Azido-PEG5-azide is a PEG-based PROTAC linker that can be used in PROTAC synthesis.Formule :C12H24N6O5Degré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :332.36Voglibose
CAS :<p>Voglibose (Glustat), an N-substituted derivative of valiolamine, exhibits excellent inhibitory activity against α-glucosidases and action against hyperglycemia</p>Formule :C10H21NO7Degré de pureté :98% - 99.90%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :267.28Kresoxim-Methyl
CAS :Kresoxim-methyl is a strobilurin fungicide,inhibits conidial germination of V. inaequalis isolates from apple orchards .Formule :C18H19NO4Degré de pureté :99.24%Couleur et forme :SolidMasse moléculaire :313.35Trabectedin
CAS :<p>Trabectedin (Ecteinascidin 743) has potent antitumor activity and the potential for soft tissue sarcoma and ovarian cancer research.</p>Formule :C39H43N3O11SDegré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :761.84iGOT1-01
CAS :<p>iGOT1-01 inhibits GOT1 enzyme, with IC50s of 84.6μM & 11.3μM in two assays, useful for cancer research.</p>Formule :C19H20N4ODegré de pureté :99.64% - 99.65%Couleur et forme :SolidMasse moléculaire :320.39Minoxidil sulfate
CAS :Minoxidil sulfate (U-58838) is the active metabolite required to exert the vasodilatory and hair growing effects of minoxidil.Formule :C9H15N5O4SDegré de pureté :99.01% - 99.72%Couleur et forme :White Crystalline SolidMasse moléculaire :289.3110074-G5
CAS :<p>10074-G5 is an inhibitor of c-Myc-Max dimerization.</p>Formule :C18H12N4O3Degré de pureté :99.51% - 99.67%Couleur et forme :SolidMasse moléculaire :332.31Shield-1
CAS :Shield-1 is a specific, high-affinity, and cell-permeable ligand for FK506-binding protein 12 (FKBP).Cost-effective and quality-assured.Formule :C42H56N2O10Degré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :748.9Bis-Tos-PEG4
CAS :Bis-Tos-PEG4 (PROTAC Linker 16) is a PEG-based PROTAC linker. Bis-Tos-PEG4 can be used in the synthesis of PROTACs.Formule :C22H30O9S2Degré de pureté :99.06%Couleur et forme :Colorless To YellowMasse moléculaire :502.6Tolfenpyrad
CAS :Tolfenpyrad is an effective insecticide[1], used against pests that are resistant to existing insecticides such as organophosphates and carbamates.[2]Formule :C21H22ClN3O2Degré de pureté :97%Couleur et forme :SolidMasse moléculaire :383.87Dipotassium glycyrrhizinate
CAS :<p>Dipotassium glycyrrhizinate is an anionic surfactant having anti-allergic and anti-inflammatory activities.</p>Formule :C42H60K2O16Degré de pureté :98.74%Couleur et forme :White Crystalline PowderMasse moléculaire :899.12Curcumol
CAS :Curcumol ((-)-Curcumol), a pure monomer isolated extracted from Rhizoma Curcumaeis, has antitumor activities.Formule :C15H24O2Degré de pureté :98.99% - 99.87%Couleur et forme :SolidMasse moléculaire :236.35Tetanus toxin 830-843 acetate
Tetanus toxin 830-843 acetate (119260-99-0) is a T cell epitope from toxoid, triggering T-cell activation for vaccine aid.Formule :C76H122N18O24Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1671.89Danicopan
CAS :<p>Danicopan (ACH-4471), an oral factor D inhibitor, binds strongly (Kd 0.54 nM) and may treat PNH and aHUS.</p>Formule :C26H23BrFN7O3Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :580.41Tenovin-3
CAS :Tenovin-3 acts as a p53 activator.Formule :C18H21N3OSDegré de pureté :99.72% - ≥95%Couleur et forme :SolidMasse moléculaire :327.44Carnosic acid
CAS :Carnosic acid is a lipid absorption inhibitor, endowed with antioxidative, antimicrobial, photoprotective potential, and antiproliferative properties.Formule :C20H28O4Degré de pureté :98.31% - 99.5%Couleur et forme :Yellow PowderMasse moléculaire :332.433-Aminobutanoic acid
CAS :3-Aminobutanoic acid (DL-3-AMINOBUTYRIC ACID) is a natural product.Formule :C4H9NO2Degré de pureté :98.48% - 99.96%Couleur et forme :White PowderMasse moléculaire :103.12Danusertib
CAS :<p>Danusertib (PHA-739358) is a small-molecule 3-aminopyrazole derivative with potential antineoplastic activity.</p>Formule :C26H30N6O3Degré de pureté :97.88% - 98.79%Couleur et forme :White PowderMasse moléculaire :474.55HATU
CAS :HATU, with Hünig's base DIPEA, forms amide bonds in peptide synthesis by activating carboxylic acids.Formule :C10H15F6N6OPDegré de pureté :99.87%Couleur et forme :White Crystal PowderMasse moléculaire :380.23m-Toluoyl chloride
CAS :<p>m-Toluoyl chloride is a bioactive chemical.</p>Formule :C8H7ClODegré de pureté :≥95%Couleur et forme :Clear Colorless To Light Brown LiquidMasse moléculaire :154.594(3H)-Quinazolinone
CAS :4(3H)-Quinazolinone (4-Hydroxyquinazoline) is a chemically synthesized masonry block, a biologically active nitrogen heterocyclic compound.Formule :C8H6N2ODegré de pureté :99.23%Couleur et forme :White SolidMasse moléculaire :146.15Iron sucrose
CAS :<p>Iron sucrose (Sucroferric oxyhydroxide) is treatment of iron deficiency anemia.</p>Formule :C18H24Fe2O24Degré de pureté :99.97%Couleur et forme :SolidMasse moléculaire :736.1AM-0902
CAS :<p>AM-0902 is a potent and specific TRPA1 antagonist (IC50s: 71/131 nM for rTRPA1 and hTRPA1).</p>Formule :C17H15ClN6O2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :370.79Cysteamine hydrochloride
CAS :<p>Cysteamine hydrochloride (Thioethanolamine Hydrochloride) is an agent for the treatment of nephropathic cystinosis and an antioxidant.</p>Formule :C2H7NS·HClDegré de pureté :99.34% - 99.87%Couleur et forme :White Crystalline Powder With A Strong And Disagreeable SmellMasse moléculaire :113.61Thalidomide-O-amido-PEG2-C2-NH2 TFA
CAS :<p>Thalidomide-based E3 ligase ligand-linker for PROTAC with PEG2 bridge; cereblon-targeted.</p>Formule :C23H27F3N4O10Degré de pureté :95.74% - 99%Couleur et forme :SolidMasse moléculaire :576.48Fargesin
CAS :Fargesin may act as a β1AR antagonist to shield rat hearts from ischemia/reperfusion damage and can also enhance dyslipidemia and hyperglycemia.Formule :C21H22O6Degré de pureté :99.82% - 99.93%Couleur et forme :SolidMasse moléculaire :370.40Aurothiomalate sodium
CAS :<p>Sodium aurothiomalate (Miochrysin) inhibits PKC-ι, TrxR; used as an anti-rheumatic and has anti-tumor properties.</p>Formule :C4H3AuNa2O4SDegré de pureté :99.66%Couleur et forme :SoildMasse moléculaire :390.07D-(+)-Fucose
CAS :1. D-(+)-Fucose is a hexose deoxy sugar found on N-linked glycans that appears on the cell surface of mammalian and plant cells.Formule :C6H12O5Degré de pureté :99.26% - 99.87%Couleur et forme :White PowderMasse moléculaire :164.16Dapagliflozin ((2S)-1,2-propanediol, hydrate)
CAS :<p>Dapagliflozin ((2S)-1,2-propanediol, hydrate) (BMS-512148 (2S)-1,2-propanediol, hydrate) is a selective, orally active inhibitor of the renal sodium-glucose co-</p>Formule :C24H35ClO9Degré de pureté :99.88% - 99.94%Couleur et forme :SolidMasse moléculaire :502.98Fasentin
CAS :Fasentin (N-[4-chloro-3-(trifluoromethyl)phenyl]-3-oxobutanamide) is an inhibitor of GluT1.Formule :C11H9ClF3NO2Degré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :279.64NFAT Inhibitor-2
CAS :NFAT Inhibitor-2 is a compound used as a molecular building block.Formule :C22H20F2N2O4SDegré de pureté :97.37%Couleur et forme :SolidMasse moléculaire :446.47Sodium 2-hydroxybutanoate
CAS :<p>Sodium 2-hydroxybutanoate, a by-product of alpha-ketobutyrate, is formed via LDH or alphaHBDH-catalyzed reactions.</p>Formule :C4H7NaO3Degré de pureté :98.92% - 99.96%Couleur et forme :SolidMasse moléculaire :126.09Rhapontigenin 3'-O-glucoside
CAS :Rhapontigenin 3'-O-glucoside, a derivative of Rhapontigenin, functions as a P450 1A1 inhibitor and is utilized in cancer prevention.Formule :C21H24O9Degré de pureté :99.66% - >99.99%Couleur et forme :SolidMasse moléculaire :420.41WM-8014
CAS :WM-8014 (MOZ-IN-3) is an inhibitor of MOZ(IC50=55 nM), a member of histone acetyltransferases.Formule :C20H17FN2O3SDegré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :384.42Thymopentin
CAS :<p>Thymopentin (TP5), a synthetic peptide of amino acids 32-36 of thymopoietin, is an active immunomodulator studied for rheumatoid arthritis and AIDS.</p>Formule :C30H49N9O9Degré de pureté :99.35% - 99.94%Couleur et forme :WhiteMasse moléculaire :679.77Sudan I
CAS :Sudan I (Solvent Yellow 14) is an organic compound, typically classified as an azo dye.Formule :C16H12N2ODegré de pureté :97.18%Couleur et forme :Orange To Orange Red Solid Solid Particulate/PowderMasse moléculaire :248.28Ginkgetin
CAS :Ginkgetin: antiviral, antifungal, anti-inflammatory; COX-2 reducer; STAT3 inhibitor; pro-apoptotic in cancer; neuroprotective in Parkinson's.Formule :C32H22O10Degré de pureté :98.63% - 99.94%Couleur et forme :SolidMasse moléculaire :566.51Dermorphin TFA
CAS :Dermorphin TFA is a new class of opioids-like peptidesFormule :C42H51F3N8O12Degré de pureté :98% - >99.99%Couleur et forme :SolidMasse moléculaire :916.89DASA-58
CAS :DASA-58 is a specific and potent Pyruvate kinase M2 (PKM2) activator.Formule :C19H23N3O6S2Degré de pureté :96.96% - 99.28%Couleur et forme :SolidMasse moléculaire :453.53JNJ-47965567
CAS :JNJ-47965567 (JNJ-479655) is a selective antagonist of the purinergic receptor P2X subtype 7 (P2X7), a ligand-gated ion channel(with pKis of 7.9 and 8.7 forFormule :C28H32N4O2SDegré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :488.643-Methylglutaric acid
CAS :Methylglutaric acid, a leucine byproduct, is linked to two metabolic disorders, detected in patient urine.Formule :C6H10O4Degré de pureté :98.64%Couleur et forme :SolidMasse moléculaire :146.14MT-DADMe-ImmA
CAS :<p>MT-DADMe-ImmA (MTDIA) is an inhibitor of human 5'-methylthioadenosine phosphorylase (MTAP, Ki: 90 pM).</p>Formule :C13H19N5OSDegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :293.39Filastatin
CAS :Filastatin is a long-lasting inhibitor of Candida albicans filamentation, and has potent antifungal effect.Formule :C18H18ClN3O3Degré de pureté :99.64%Couleur et forme :SolidMasse moléculaire :359.81Alrestatin
CAS :<p>Alrestatin (AY-22284) is a specific inhibitor of aldose reductase and attenuates glucose-induced angiotensin II production in rat vascular smooth muscle in</p>Formule :C14H9NO4Degré de pureté :99.23%Couleur et forme :SolidMasse moléculaire :255.2256Pimecrolimus
CAS :<p>Pimecrolimus, a calcineurin inhibitor, binds FKBP-12, blocking calcium-dependent signals.</p>Formule :C43H68ClNO11Degré de pureté :99.53% - 99.87%Couleur et forme :White Crystalline PowderMasse moléculaire :810.45Benzenepentacarboxylic Acid
CAS :Benzenepentacarboxylic Acid (Pentacarboxybenzene) is a novel fluorescent probe to detect and scavenge HO-.Formule :C11H6O10Degré de pureté :98.29%Couleur et forme :SolidMasse moléculaire :298.16Regorafenib monohydrate
CAS :<p>Regorafenib Monohydrate is a novel oral multikinase inhibitor with IC50 values of 13, 4.2, 46, 22, 7, 1.5, 2.5, 28, 19 nM for VEGFR1, murine VEGFR2, murine</p>Formule :C21H17ClF4N4O4Degré de pureté :99.69%Couleur et forme :SolidMasse moléculaire :500.83PF-3845
CAS :PF-3845 is a potent, selective and irreversible FAAH inhibitor with Ki of 230 nM, showing negligible activity against FAAH2.Formule :C24H23F3N4O2Degré de pureté :99.54% - 99.58%Couleur et forme :SolidMasse moléculaire :456.46Ethylhydrocupreine hydrochloride
CAS :<p>Ethylhydrocupreine hydrochloride (Optochin hydrochloride) is a derivative of quinine with antimicrobial activity against Streptococcus pneumoniae.</p>Formule :C21H29ClN2O2Degré de pureté :99.73% - 99.86%Couleur et forme :SolidMasse moléculaire :376.92Alobresib
CAS :Alobresib (Vorolanib) is an inhibitor of BET bromodomain,is an antineoplastic drug candidate.Formule :C26H23N5O2Degré de pureté :97.63%Couleur et forme :SolidMasse moléculaire :437.49Flavokawain A
CAS :NSC-37445 shows anti-tumor properties; Flavokawain A may reduce inflammation by hindering specific signaling in macrophages.Formule :C18H18O5Degré de pureté :97.1% - 99.72%Couleur et forme :SolidMasse moléculaire :314.332EDO-S101
CAS :EDO-S101 (Tinostamustine) is a pan HDAC inhibitor with IC50 values of 9, 9 and 25 nM for HDAC1, HDAC2 and HDAC3 , respectively.Formule :C19H28Cl2N4O2Degré de pureté :98.02% - 99.44%Couleur et forme :SolidMasse moléculaire :415.36Thalidomide-O-COOH
CAS :<p>Thalidomide-O-COOH is a Cereblon ligand for CRBN protein recruitment and PROTAC construction with a linker.</p>Formule :C15H12N2O7Degré de pureté :98% - 98.29%Couleur et forme :SolidMasse moléculaire :332.27S-trityl-L-Cysteine
CAS :<p>S-trityl-L-Cysteine is a potent inhibitor of human mitotic kinesin Eg5</p>Formule :C22H21NO2SDegré de pureté :97.02%Couleur et forme :Almost White To Light Yellow Granular PowderMasse moléculaire :363.47m-3M3FBS
CAS :m-3M3FBS is a phospholipase C (PLC) activator.Formule :C16H16F3NO2SDegré de pureté :99.66%Couleur et forme :SolidMasse moléculaire :343.36Benzotript
CAS :<p>Benzotript is an gastrin-receptor antagonist, with anti-gastrinic.</p>Formule :C18H15ClN2O3Degré de pureté :97.82%Couleur et forme :SolidMasse moléculaire :342.776SMER28
CAS :SMER28 triggers autophagy in cells without mTOR, blocking amyloid beta buildup.Formule :C11H10BrN3Degré de pureté :99.94% - >99.99%Couleur et forme :SolidMasse moléculaire :264.12RG108
CAS :RG108 (N-Phthalyl-L-tryptophan) is an DNA methyltransferase inhibitor(IC50=115 nM).Formule :C19H14N2O4Degré de pureté :98% - 99.43%Couleur et forme :SolidMasse moléculaire :334.33BMP signaling agonist sb4
CAS :<p>BMP signaling agonist sb4 (SB 4) is an agonist of benzoxazole bone morphogenetic protein (BMP) signaling (EC50 :74 nM)</p>Formule :C14H10BrNOSDegré de pureté :99.48% - 99.805%Couleur et forme :SolidMasse moléculaire :320.2Carbenoxolone
CAS :<p>Carbenoxolone (Biogastrone) is an inhibitor of 11β-HSD and gap junction connexin channels.</p>Formule :C34H50O7Degré de pureté :99.75%Couleur et forme :White Crystalline PowderMasse moléculaire :570.76Proteinase K
CAS :Proteinase K (Protease K) is a non-specific serine protease. Proteinase K hydrolyzes peptide bonds and is used for protein digestion. Cost-effective and quality-assured.Formule :C29H27N2O12PDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :626.511Potassium 2-hydroxy-2-methylsuccinate
CAS :<p>Potassium 2-hydroxy-2-methylsuccinate ((±)-2-Hydroxy-2-methylsuccinic acid dipotassium salt) is a type of endogenous metabolite.</p>Formule :C5H6K2O5Degré de pureté :99.96% - ≥98%Couleur et forme :SolidMasse moléculaire :224.29BA 1 acetate(183241-31-8 free base)
<p>BA 1 acetate: bombesin agonist, IC50s: 0.26/1.55/2.52 nM (BB1/BB2/BB3), boosts glucose transport, promotes lung cancer cell growth in vitro.</p>Formule :C59H80N14O13Degré de pureté :95.3%Couleur et forme :SolidMasse moléculaire :1193.35Tenacissoside G
CAS :Tenacissoside G, a C21 steroid derived from the stems of Marsdenia tenacissima, can reverse multidrug resistance in cancer cells exhibiting overexpression of P-Formule :C42H64O14Degré de pureté :96.18% - 97.03%Couleur et forme :SolidMasse moléculaire :792.95[Arg8]-Vasotocin acetate(113-80-4 free base)
CAS :[Arg8]-Vasotocin acetate is a hormone present in the neurohypophysis of nonmammalian vertebrates that is related to vasopressin and oxytocin.Formule :C45H71N15O14S2Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :1110.27PS-1145
CAS :<p>PS-1145 (IKK Inhibitor X) is a specific IKK inhibitor with IC50 of 88 nM.</p>Formule :C17H11ClN4ODegré de pureté :98.81% - >99.99%Couleur et forme :SolidMasse moléculaire :322.75RO4929097
CAS :<p>RO4929097 (RG-4733), a γ secretase inhibitor (IC50: 4 nM), inhibits cellular processing of Aβ40 and Notch (EC50: 14/5 nM).</p>Formule :C22H20F5N3O3Degré de pureté :98.5% - 99.51%Couleur et forme :SolidMasse moléculaire :469.41-Oleoyl lysophosphatidic acid sodium
CAS :1-Oleoyl lysophosphatidic acid sodium (1-Oleoyl lysophosphatidic acid sodium salt) salt is an Endogenous agonist of LPA1 and LPA2Formule :C21H40O7P·NaDegré de pureté :98.75% - 99.24%Couleur et forme :SolidMasse moléculaire :458.51Gnetol
CAS :Gnetol inhibits butyrylcholinesterase (IC50: 1.3 μM), tyrosinase, melanin synthesis in B16 cells, and AA-induced platelet aggregation.Formule :C14H12O4Degré de pureté :98.55% - ≥95%Couleur et forme :SolidMasse moléculaire :244.24Telotristat Etiprate
CAS :Telotristat Etiprate (LX 1606 Hippurate) is an orally bioavailable, tryptophan hydroxylase (TPH) inhibitor with potential antiserotonergic activity.Formule :C27H26ClF3N6O3·C9H9NO3Degré de pureté :99.21% - 99.83%Couleur et forme :White SolidMasse moléculaire :754.15
