Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.747 produits)
- Apoptose(6.181 produits)
- Cycle cellulaire/point de contrôle(4.805 produits)
- Chromatine/Épigénétique(2.567 produits)
- Signalisation du cytosquelette(1.498 produits)
- Altération de l'ADN/réparation de l'ADN(2.897 produits)
- Endocrinologie/Hormones(3.701 produits)
- Enzyme(3.671 produits)
- GPCR/G-Protéine(8.960 produits)
- Immunologie et Inflammation(3.692 produits)
- Virus de la grippe(296 produits)
- Signalisation JAK/STAT(414 produits)
- Signalisation MAPK(1.244 produits)
- Transporteur membranaire/Canal ionique(3.135 produits)
- Métabolisme(10.103 produits)
- Microbiologie/Virologie(7.550 produits)
- Neuroscience(10.300 produits)
- Autres inhibiteurs(35.771 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.400 produits)
- Protéases/Protéasome(1.670 produits)
- Cellules souche et Dérivés(742 produits)
- Tyrosine Kinase/Adaptateurs(1.922 produits)
- Ubiquitination(1.715 produits)
Affichez 16 plus de sous-catégories
66577 produits trouvés pour "Inhibiteurs"
Trier par
Degré de pureté (%)
0
100
|
0
|
50
|
90
|
95
|
100
UNC10217938A
CAS :UNC10217938A is a 3-deazapteridine analog, has strong oligonucleotide enhancing effects.Formule :C26H28N6O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :456.54Sulfuretin
CAS :Sulfuretin protects HepG2 cells from oxidative damage by scavenging ROS and activating HO-1 via Nrf2/ARE and JNK/ERK pathways.
Formule :C15H10O5Degré de pureté :98.91% - 99.86%Couleur et forme :SolidMasse moléculaire :270.24BpV(HOpic)
CAS :BpV(HOpic) (bpV (HOpic)) is a potent inhibitor of PTEN (IC50 of 14 nM).Formule :C6H4K2NO8VDegré de pureté :99.60%Couleur et forme :SolidMasse moléculaire :347.24BP 897
CAS :BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.Formule :C26H31N3O2Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :417.54Ref: TM-T9100
1mg80,00€5mg162,00€10mg227,00€25mg379,00€50mg540,00€100mg730,00€200mg938,00€1mL*10mM (DMSO)177,00€Murrayone
CAS :Murrayone from M. paniculata, a bioactive coumarin, prevents cancer metastasis and reduces ADP-induced platelet aggregation.Formule :C15H14O4Degré de pureté :98.01% - 98.79%Couleur et forme :SolidMasse moléculaire :258.27Ref: TM-TN1046
1mg84,00€5mg200,00€10mg340,00€25mg563,00€50mg795,00€100mg1.071,00€1mL*10mM (DMSO)177,00€Rimiducid
CAS :Rimiducid, a tacrolimus analogue, dimerizes FKBP domains to activate Caspase 9 and induce apoptosis; binds FKBP12 weakly.Formule :C78H98N4O20Degré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :1411.63Ref: TM-T14298
1mg129,00€2mg177,00€5mg285,00€10mg420,00€25mg692,00€50mg973,00€100mg1.305,00€500mg2.602,00€(S)-crizotinib
CAS :(S)-crizotinib (ent-crizotinib) （IC50 of 72 nM）, an effective MTH1 (NUDT1) inhibitor, is the (S)-enantiomer of crizotinib.Formule :C21H22Cl2FN5ODegré de pureté :98.52% - 99.47%Couleur et forme :SolidMasse moléculaire :450.34Tricaine methanesulfonate
CAS :Tricaine methanesulfonate (TMS/MS-222) is an anesthetic used in hatcheries and studies to immobilize fish for marking, transport, and invasive procedures.Formule :C10H15NO5SDegré de pureté :99.259% - 99.86%Couleur et forme :White PowderMasse moléculaire :261.30NADPH tetrasodium salt
CAS :NADPH tetrasodium salt is the reduced form of the electron acceptor nicotinamide adenine dinucleotide phosphate, which acts as an electron donor in a variety ofFormule :C21H26N7Na4O17P3Degré de pureté :97.15% - >99.99%Couleur et forme :SolidMasse moléculaire :833.35Camelliaside B
CAS :Camelliaside B possesses deglycosylation activity.Formule :C32H38O19Degré de pureté :95.92% - 99.92%Couleur et forme :SolidMasse moléculaire :726.63Enzastaurin 2HCl
CAS :Enzastaurin (DB-102/LY317615) is a macrocyclic bisindolemaleimide inhibiting protein kinase C beta to reduce tumor blood supply.Formule :C32H31Cl2N5O2Couleur et forme :SolidMasse moléculaire :588.53Cucurbitacin IIb
CAS :Cucurbitacin IIb is an active ingredient in Hemsleyadine, used to treat dysentery and other infections; it has anti-inflammatory effects.Formule :C30H48O7Degré de pureté :98.66% - >99.99%Couleur et forme :SolidMasse moléculaire :520.7Ref: TM-T4S1469
1mg96,00€5mg208,00€10mg359,00€25mg592,00€50mg837,00€100mg1.121,00€1mL*10mM (DMSO)240,00€2,4-D
CAS :2,4-D (Hedonal) is a synthetic auxin regulating plant growth and an herbicide disrupting root elongation.Formule :C8H6Cl2O3Degré de pureté :99.42%Couleur et forme :White To Yellow Crystalline Powder /Srp Yellow Color Is Phenolic Impurities/ Is Threat To The Environment Immediate Steps Should Be Taken To Limit Spread To The EnvironmentMasse moléculaire :221.04Chelidonic acid
CAS :Chelidonic acid, in Chelidonium majus, acts as an analgesic, antimicrobial, CNS sedative, and has anti-inflammatory properties.Formule :C7H4O6Degré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :184.10m-PEG7-alcohol
CAS :m-PEG7-alcohol (O-Methyl-heptaethylene glycol) is a PEG-based PROTAC linker. m-PEG7-alcohol can be used in the synthesis of PROTACs.Formule :C15H32O8Degré de pureté :96.02%Couleur et forme :SolidMasse moléculaire :340.41Methyl 3-aminopyrazine-2-carboxylate
CAS :Methyl 3-aminopyrazine-2-carboxylate: a pyrazine with methoxycarbonyl (2) and amino (3); an ester and aromatic amine, used in synthesis.Formule :C6H7N3O2Degré de pureté :99.34%Couleur et forme :Yellow Crystalline PowderMasse moléculaire :153.14Hyaluronic acid sodium
CAS :Hyaluronic acid sodium (Sodium Hyaluronate) is an anionic, nonsulfated glycosaminoglycan distributed throughout connective, epithelial, and neural tissues.Formule :C14H28O6Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :292.372Sarpogrelate hydrochloride
CAS :Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.
Formule :C24H32ClNO6Degré de pureté :99.73%Couleur et forme :Colorless LiquidMasse moléculaire :465.97Cloquintocet-mexyl
CAS :Cloquintocet-mexyl, a herbicide, targets and controls coarse annual grasses within the Poaceae family.Formule :C18H22ClNO3Degré de pureté :98.69%Couleur et forme :Light Brown Solid PowderMasse moléculaire :335.838-Fluoro-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-one
CAS :8-Fluoro-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-one serves as a pharmaceutical intermediate.
Formule :C11H9FN2ODegré de pureté :99.21%Couleur et forme :SolidMasse moléculaire :204.2Remoxipride hydrochloride (hydrate)
CAS :Remoxipride hydrochloride (hydrate) is a potent D2DR (dopamine D2 receptor) antagonist and antipsychotic.Formule :C16H26BrClN2O4Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :425.75Grazoprevir hydrate
CAS :Grazoprevir: Hepatitis C protease inhibitor effective against various genotypes, including drug-resistant strains.Formule :C38H52N6O10SDegré de pureté :98%Couleur et forme :SolidMasse moléculaire :784.92MTEP hydrochloride
CAS :MTEP hydrochloride (MTEP) is non-competitive mGlu5 antagonist (IC50 and Ki of 5 nM and 16 nM, respectively)Formule :C11H9ClN2SDegré de pureté :99.58%Couleur et forme :SolidMasse moléculaire :236.72N-(Hydroxymethyl)nicotinamide
CAS :N-(Hydroxymethyl)nicotinamide (Bilamid) is an antimicrobial agent.Formule :C7H8N2O2Degré de pureté :99.9%Couleur et forme :White SolidMasse moléculaire :152.15N-p-trans-Coumaroyltyramine
CAS :N-p-trans-Coumaroyltyramine: natural AChE inhibitor, IC50 122 μM; anti-trypanosomal, IC50 13.3 μM vs T. brucei rhodesiense.Formule :C17H17NO3Degré de pureté :99.30% - 99.56%Couleur et forme :SolidMasse moléculaire :283.33Ref: TM-TN1030
1mg74,00€5mg177,00€10mg289,00€25mg485,00€50mg695,00€100mg945,00€1mL*10mM (DMSO)165,00€SRI-29329
CAS :SRI-29329 is a potent, specific inhibitor of CDC-like kinase (with IC50 of 78 nM, 16 nM and 86 nM for CLK1, CLK2 and CLK4, respectively).Formule :C20H26ClN7Degré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :399.92Argatroban Monohydrate
CAS :Argatroban Monohydrate is a specific thrombin inhibitor, which is a non-heparin anticoagulant, prevents the formation of thrombi.Formule :C23H38N6O6SDegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :526.65Dicyclanil
CAS :Dicyclanil, a regulator of insect growth, is a veterinary medicine for the protection against early-season myiasis.Formule :C8H10N6Degré de pureté :≥95%Couleur et forme :White Microcrystalline PowderMasse moléculaire :190.21A40926
CAS :A40926 (Dalbavancin Impurity) is effective against Gram positive bacteria.Formule :C83H88Cl2N8O29Degré de pureté :91.38% - 91.83%Couleur et forme :SolidMasse moléculaire :1732.53BIM-23190 aceate
BIM-23190 aceate, a somatostatin analog, a selective agonist of SSTR2 and SSTR5. BIM-23190 can be used in cancer and acromegaly studies.
Formule :C59H83N13O14S2Degré de pureté :99.7%Couleur et forme :SolidMasse moléculaire :1262.5Ganirelix Acetate
CAS :Ganirelix Acetate is a gonadotropin-releasing hormone (GnRH) receptor antagonistFormule :C82H117ClN18O15Degré de pureté :96.05%Couleur et forme :SolidMasse moléculaire :1630.4ODM-203
CAS :ODM-203, a Selective Inhibitor of FGFR and VEGFR, Shows Strong Antitumor Activity, and Induces Antitumor ImmunityFormule :C26H21F2N5O2SDegré de pureté :99.85%Couleur et forme :SolidMasse moléculaire :505.54Lanthanum(III) chloride heptahydrate
CAS :Lanthanum(III) chloride blocks divalent cation channels, useful for biochemical research.Formule :Cl3H14LaO7Degré de pureté :98%Couleur et forme :White Solid PowderMasse moléculaire :371.37Ref: TM-T22353
5mg46,00€10mg59,00€25mg87,00€50mg129,00€100mg178,00€200mg268,00€500mg460,00€1mL*10mM (DMSO)52,00€Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel-
CAS :Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel- is an estrogen receptor beta (ERβ) agonist.Formule :C18H18O3Degré de pureté :99.85% - 99.96%Couleur et forme :SolidMasse moléculaire :282.33Ref: TM-T9800
1mg93,00€5mg182,00€10mg269,00€25mg429,00€50mg610,00€100mg820,00€200mg1.099,00€1mL*10mM (DMSO)172,00€Dihydrokavain
CAS :Dihydrokavain, a major kavalactone in kava, significantly affects its anxiolytic properties.Formule :C14H16O3Degré de pureté :99.82% - ≥95%Couleur et forme :White PowderMasse moléculaire :232.27Adenosine 5'-diphosphate
CAS :Adenosine 5'-diphosphate (ADP) is a natural nucleotide derived from the dephosphorylation of ATP. ADP induces platelet aggregation. Cost effective and quality assured.Formule :C10H15N5O10P2Degré de pureté :99.5% - >99.99%Couleur et forme :SolidMasse moléculaire :427.26-TAMRA
CAS :6-TAMRA (6-Carboxytetramethylrhodamine) serves as a popular fluorophore for the creation of bioconjugates, particularly in the synthesis of fluorescentFormule :C25H22N2O5Degré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :430.45(25R)-Spirost-4-ene-3,12-dione
CAS :(25R)-Spirost-4-ene-3,12-dione is a natural product.Formule :C27H38O4Degré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :426.59Morroniside
CAS :Morroniside regulates liver inflammation, lipid metabolism, protects against diabetic kidney damage, and guards the brain from ischemic injury.Formule :C17H26O11Degré de pureté :99.70% - 99.84%Couleur et forme :SolidMasse moléculaire :406.38AT-56
CAS :AT56, a specific inhibitor of prostaglandin D2 synthase enzymatic activity, blunted adipogenic aldosterone effects.Formule :C25H27N5Degré de pureté :98.16% - 99.5%Couleur et forme :SolidMasse moléculaire :397.52Ref: TM-T1866
1mg37,00€5mg79,00€10mg119,00€25mg226,00€50mg378,00€100mg595,00€200mg833,00€1mL*10mM (DMSO)87,00€Pomalidomide-C5-COOH
Pomalidomide-C5-COOH, a CRBN-based ligand-linker for PROTAC tech.Formule :C19H21N3O6Degré de pureté :97.98%Couleur et forme :SolidMasse moléculaire :387.39Lactoferrin
CAS :Lactoferrin is secreted by mammals and displays extensive biological effects including boosting the cold tolerance of a well-applied probiotic strain.
Formule :C27H47N7O6Degré de pureté :96.61%Couleur et forme :SolidMasse moléculaire :565.71Boldine
CAS :Boldine (1,10-Dimethoxy-2,9-dihydroxyaporphine) is a natual product .Boldine displays anti-cancer, cytoprotective , anti-oxidant and anti-inflammatoryFormule :C19H21NO4Degré de pureté :97.78% - 98%Couleur et forme :SolidMasse moléculaire :327.37IACS-13909
CAS :IACS-13909 (BBP-398), a specific and potent allosteric inhibitor of SHP2, that suppresses signaling through the MAPK pathway.Formule :C17H18Cl2N6Degré de pureté :98.8%Couleur et forme :SolidMasse moléculaire :377.27Peptide YY (PYY) (3-36), human
CAS :Peptide YY (PYY) (3-36), human (Peptide YY (3-36)) is a gut hormone peptide. Peptide YY (PYY) (3-36), human acts as a Y2 receptor agonist to reduce appetite.Formule :C176H272N52O54Degré de pureté :97.76%Couleur et forme :SolidMasse moléculaire :3980.42Trilobatin
CAS :Trilobatin (P-Phlorizin) has anti-oxidant effect, can increase superoxide dismutase (SOD) activity.Trilobatin has anti-inflammatory effect, it potentiallyFormule :C21H24O10Degré de pureté :97.16%Couleur et forme :SolidMasse moléculaire :436.41Ref: TM-T2S0731
1mg50,00€5mg99,00€10mg141,00€25mg260,00€50mg385,00€100mg557,00€200mg790,00€1mL*10mM (DMSO)109,00€CCCP
CAS :CCCP blocks STING activation, TBK1, IRF3 signaling, and IFN-β production by disrupting MMP.Formule :C9H5ClN4Degré de pureté :97.15% - 99.64%Couleur et forme :Yellow To Orange PowderMasse moléculaire :204.62MLN8054 sodium
CAS :MLN8054 sodium is an Aurora A inhibitor.Formule :C25H14ClF2N4NaO2Couleur et forme :SolidMasse moléculaire :498.84L-Alanyl-L-glutamine
CAS :L-Alanyl-L-glutamine (Ala-Gln), a dipeptide composed of alanine and Gln, is an alternative supplement to L-glutamine in the production of biopharmaceuticals.Formule :C8H15N3O4Degré de pureté :99.71% - 99.97%Couleur et forme :SolidMasse moléculaire :217.22Coniferaldehyde
CAS :Coniferaldehyde (Ferulaldehyde) is a member of the class of cinnamaldehydes. Coniferaldehyde has a role as an antifungal agent and a plant metabolite.Formule :C10H10O3Degré de pureté :97.71% - 99.96%Couleur et forme :SolidMasse moléculaire :178.18Dobutamine
CAS :Dobutamine, a synthetic catecholamine, boosts cardiac output and improves blood flow, mainly targeting β1-AR.Formule :C18H23NO3Couleur et forme :SolidMasse moléculaire :301.38GR 125743
CAS :GR 125743 is a novel antagonist of 5-HT1B/1D receptor.Formule :C25H28N4O2Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :416.52Ref: TM-T8737
1mg40,00€2mg52,00€5mg84,00€10mg113,00€25mg222,00€50mg333,00€100mg495,00€1mL*10mM (DMSO)93,00€Encequidar
CAS :Encequidar (HM30181A) is a potent and selective P-glycoprotein inhibitor.Formule :C38H36N6O7Degré de pureté :99.93%Couleur et forme :SolidMasse moléculaire :688.73Ref: TM-T8426
1mg46,00€2mg62,00€5mg90,00€10mg137,00€25mg234,00€50mg360,00€100mg528,00€1mL*10mM (DMSO)127,00€Methyl 4-aminobutyrate HCl
CAS :Methyl 4-aminobutyrate HCl (GABA methyl ester) is a methyl ester compound derived from the condensation of aminobutyric acid and methanol.Formule :C5H12ClNO2Degré de pureté :99.99%Couleur et forme :SolidMasse moléculaire :153.61BMS 182874 hydrochloride
CAS :BMS 182874 hydrochloride is a nonpeptide endothelin (El) receptor antagonist.Formule :C17H20ClN3O3SDegré de pureté :97.01%Couleur et forme :SolidMasse moléculaire :381.88Ref: TM-T21790
1mg77,00€2mg92,00€5mg140,00€10mg205,00€25mg343,00€50mg477,00€100mg665,00€200mg897,00€1mL*10mM (DMSO)146,00€MUN36378
CAS :MUN36378 is a FTO inhibitor for treatment of leukemia.Formule :C18H15Cl2N3O2Degré de pureté :99.70%Couleur et forme :SolidMasse moléculaire :376.24Angiotensin I/II (1-5)
CAS :Angiotensin I/II (1-5) is a peptide (ASP-ARG-VAL-TYR-ILE) that contains the amino acids 1-5 and is converted from Angiotensin I/II.Formule :C30H48N8O9Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :664.75Ossirene
CAS :Ossirene (AS101), a potent in vitro and in vivo immunomodulator, is a novel inhibitor of IL-1beta converting enzyme.Formule :C2H4Cl3O2Te·H4NDegré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :312.05Ref: TM-T6761
2mg39,00€5mg58,00€10mg93,00€25mg138,00€50mg197,00€100mg294,00€200mg437,00€1mL*10mM (DMSO)66,00€AZD1208 hydrochloride
CAS :AZD1208 hydrochloride is a highly selective, potent and orally active PIM inhibitor.Formule :C21H22ClN3O2SCouleur et forme :SolidMasse moléculaire :415.94Lenacil
CAS :Lenacil (634 Hexilure) is an agent of herbicide.Lenacil can inhibit photosynthesis.Formule :C13H18N2O2Degré de pureté :99.65%Couleur et forme :Less Crystals Colorless CrystalsMasse moléculaire :234.29Sudan IV
CAS :Sudan IV (Solvent Red 24) is a lysochrome (fat-soluble dye) diazo dye used for the staining of triglycerides，lipids and lipoproteins on frozen paraffin sections
Formule :C24H20N4OCouleur et forme :Dark Red Solid PowderMasse moléculaire :380.445-Hydroxymethyldeoxyuridine
CAS :5-Hydroxymethyldeoxyuridine: anticancer/antiviral; inhibits S180 and Ehrlich cells (ED50=8.5/4 μM) & leukemia lines (IC50=1.7-5.8 μM).Formule :C10H14N2O6Degré de pureté :99.80%Couleur et forme :SolidMasse moléculaire :258.23MS-049 oxalate salt
CAS :MS-049 oxalate salt is a potent and selective inhibitor of protein arginine methyltransferases (PRMTs) PRMT 4 and PRMT6.Formule :C17H26N2O5Couleur et forme :SolidMasse moléculaire :338.4Gamabufotalin
CAS :Gamabufotalin, a Chansu bufadienolide, treats COX-2 diseases and cancer with high stability and low side effects.Formule :C24H34O5Degré de pureté :99.18% - 99.51%Couleur et forme :SolidMasse moléculaire :402.52Prexasertib
CAS :Prexasertib (LY2606368) is a selective checkpoint kinase 1 (CHK1) inhibitor (Ki 0.9 nM, IC50<1 nM). antitumor activity. High-Quality, Low-Cost!Formule :C18H19N7O2Degré de pureté :97.3% - 98.23%Couleur et forme :SolidMasse moléculaire :365.39N-Acetylornithine
CAS :N-Acetylornithine is found in human blood plasma (avg. 1.1±0.4 μmol/L) and urine (~1 μmol/day).Formule :C7H14N2O3Degré de pureté :99.86% - ≥95%Couleur et forme :SolidMasse moléculaire :174.2TM5441
CAS :TM5441 is an orally bioavailable fibrinogen activator inhibitor-1 inhibitor that inhibits several cancer cell lines with IC50 values ranging from 13.9 to 51.1 μM.Cost-effective and quality-assured.Cost-effective and quality-assured.Formule :C21H17ClN2O6Degré de pureté :97.62% - 99.09%Couleur et forme :SolidMasse moléculaire :428.82Mini Gastrin I, human acetate
Mini Gastrin I, human acetate is a shorter version of human gastrin, consists of amino acids 5-17 of the parent peptide.Formule :C76H103N15O28SDegré de pureté :99.35% - 99.82%Couleur et forme :SolidMasse moléculaire :1706.78Coixol
CAS :Coixol (MBOA) is a muscle relaxant, anti-convulsant, enhances vole reproduction, stimulates ovulation, and regulates mucin in airway cells.Formule :C8H7NO3Degré de pureté :97.96% - 99.87%Couleur et forme :SolidMasse moléculaire :165.15Quisinostat dihydrochloride
CAS :Quisinostat dihydrochloride (JNJ26854165(Quisinostat) 2HCl) 是一种有口服活性，高效的 pan-HDAC 抑制剂，具有广泛的抗肿瘤活性。它对 HDAC1、HDAC2、HDAC4、HDAC10和HDAC11 的IC50值分别为 0.11 nM、0.33 nM、0.64 nM、0.46 nM 和 0.37 nM。Formule :C21H28Cl2N6O2Degré de pureté :97.13%Couleur et forme :SolidMasse moléculaire :467.39Ref: TM-T6865
1mg62,00€5mg120,00€10mg170,00€25mg294,00€50mg411,00€100mg573,00€200mg807,00€1mL*10mM (DMSO)123,00€PF-562271 besylate
CAS :PF-562271 besylate: potent, ATP-competitive FAK inhibitor, IC50 1.5 nM, 10x less effective on Pyk2, highly selective vs other kinases.Formule :C21H20F3N7O3S·C6H6O3SDegré de pureté :97.65% - 99.01%Couleur et forme :SolidMasse moléculaire :665.66Ref: TM-T6177
1mg35,00€5mg74,00€10mg94,00€25mg138,00€50mg198,00€100mg296,00€200mg427,00€1mL*10mM (DMSO)89,00€Leucokinin VIII acetate
Leucokinin VIII acetate (Leucokinin 8) is an diuretic octapeptide isolated form head extracts of the cockroach.
Formule :C44H56N10O13Degré de pureté :98.52%Couleur et forme :SolidMasse moléculaire :932.99Isosilybin A
CAS :Isosilybin A is a partial PPARγ agonist, it significantly induced ABCA1 protein expression, it inhibited both monophenolase (IC50=1.7-7.6μM) and diphenolase (Formule :C25H22O10Degré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :482.44N,N-Bis(2-hydroxyethyl)-p-phenylenediami
CAS :N,N-Bis(2-hydroxyethyl)-p-phenylenediamine is an intermediate compound.Formule :C10H18N2O6SDegré de pureté :92.96%Couleur et forme :White Crystal PowderMasse moléculaire :294.32Octapeptide-2 Acetate
Octapeptide-2 Acetate, a stable hair growth promoter, activates stem cells in follicles for improved growth.Formule :C40H64N10O18SDegré de pureté :98.47%Couleur et forme :SolidMasse moléculaire :1005.06Aureusimine B
CAS :Aureusimine B, a Calpain inhibitor, is produced by Staphylococcus aureus biofilms and could be a potential biomarker for S. aureus biofilm-based infections.Formule :C14H16N2ODegré de pureté :99.95%Couleur et forme :SolidMasse moléculaire :228.29Ref: TM-T37753
1mg93,00€2mg117,00€5mg177,00€10mg269,00€25mg429,00€50mg610,00€100mg820,00€200mg1.071,00€1mL*10mM (DMSO)164,00€FIPI HCl
CAS :FIPI: Selective phospholipase D inhibitor, blocks mercury-induced lipid signals, protects aortic cells.Formule :C23H25ClFN5O2Couleur et forme :SolidMasse moléculaire :457.93AMD 3465 hexahydrobromide
CAS :AMD 3465 hexahydrobromide (GENZ-644494 (hexahydrobromide)) is a CXCR4 receptor antagonist with potential anticancer and anti-HIV activity.Formule :C24H44Br6N6Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :896.072-O-α-D-Glucopyranosyl-L-ascorbic Acid
CAS :2-O-α-D-Glucopyranosyl-L-ascorbic Acid (ASCORBYL GLUCOSIDE) is a glucoside derivative of ascorbic acid that can be enzymatically hydrolysed to ascorbic acid.Formule :C12H18O11Degré de pureté :98.56% - 99.73%Couleur et forme :SolidMasse moléculaire :338.26Gilteritinib
CAS :Gilteritinib (ASP2215) is a potent inhibitor at the FMS-related tyrosine kinase 3 (FLT3) and AXL tyrosine kinase receptors (IC50 = 0.29 nM and <1 nM,Formule :C29H44N8O3Degré de pureté :97.75% - 99.90%Couleur et forme :SolidMasse moléculaire :552.71Ref: TM-T4409
1g1.288,00€1mg38,00€2mg52,00€5mg85,00€10mg114,00€25mg177,00€50mg261,00€100mg411,00€500mg954,00€W-7 hydrochloride
CAS :W-7 hydrochloride (W-7 HCl), a calmodulin antagonist, inhibits Ca2+-calmodulin-dependent myosin light chain kinase and phosphodiesterase, W-7 hydrochlorideFormule :C16H22Cl2N2O2SDegré de pureté :99.63%Couleur et forme :White Crystalline SolidMasse moléculaire :377.324-Propionamidophenol
CAS :4-Propionamidophenol is a kind of analog of p-acetamidophenol.Formule :C9H11NO2Degré de pureté :99.64%Couleur et forme :Pale Purple SolidMasse moléculaire :165.19Quercetin-3-O-glucose-6''-acetate
CAS :Quercetin-3-O-glucose-6''-acetate (6"-O-Acetylisoquercitrin) is an inhibitor of NADPH oxidase. Quercetin-3-O-glucose-6''-acetate has antioxidant activities.Formule :C23H22O13Degré de pureté :97.48%Couleur et forme :SolidMasse moléculaire :506.41Phenelzine
CAS :Phenelzine is a MAOI antidepressant, boosting brain catecholamines, effective for endogenous depression.Formule :C8H12N2Degré de pureté :98%Couleur et forme :LiquidMasse moléculaire :136.19Ref: TM-T9540
5mgÀ demander10mgÀ demander25mgÀ demander50mgÀ demander100mgÀ demander200mgÀ demander500mgÀ demanderCucurbitacin IIA
CAS :1.Formule :C32H50O8Degré de pureté :98.62% - 99.87%Couleur et forme :SolidMasse moléculaire :562.73Acetyl-L-lysine
CAS :Acetyl-L-lysine: N-acetylated amino acid, normally found in trace urine amounts, elevated in aminoacylase I deficiency.Formule :C8H16N2O3Degré de pureté :99.40% - 99.83%Couleur et forme :SolidMasse moléculaire :188.22Maohuoside A
CAS :Maohuoside A promotes osteogenesis of rat mesenchymal stem cells via BMP and MAPK signaling pathways.Formule :C27H32O12Degré de pureté :98.91% - 99.57%Couleur et forme :SolidMasse moléculaire :548.54Ref: TM-TN2081
1mg52,00€5mg116,00€10mg172,00€25mg266,00€50mg353,00€100mg803,00€200mg1.063,00€1mL*10mM (DMSO)142,00€BIBR 1532
CAS :BIBR 1532 is an effective, specific and non-competitive telomerase inhibitor (IC50: 100 nM, in a cell-free assay).
Formule :C21H17NO3Degré de pureté :98.49% - 98.90%Couleur et forme :SolidMasse moléculaire :331.36PXS-4728A
CAS :BI-1467335 HCl(BI 1467335) is a selective, orally active inhibitor of semicarbazide-sensitive amine oxidase (SSAO) that helps improve chronic obstructiveFormule :C15H22ClFN2O2Degré de pureté :98.61%Couleur et forme :SolidMasse moléculaire :316.8Zearalenone
CAS :Zearalenone (F2 toxin) is a mycotoxin produced mainly by fungi belonging to the genus Fusarium in foods and feeds.Formule :C18H22O5Degré de pureté :98.39% - 99.11%Couleur et forme :This Chemical May Be Sensitive To Prolonged Exposure To Air Insoluble In Water Physical Description White Micr°Crystals Or White Powder (Ntp 1992)Masse moléculaire :318.36dBET1
CAS :dBET1 fuses (+)-JQ1 with thalidomide, degrades BET proteins via cereblon (EC50: 430 nM), and triggers apoptosis.Formule :C38H37ClN8O7SDegré de pureté :98.02% - 99.3%Couleur et forme :SolidMasse moléculaire :785.27Ref: TM-T4495
1mg50,00€5mg99,00€10mg161,00€25mg268,00€50mg427,00€100mg650,00€200mg888,00€1mL*10mM (DMSO)145,00€EST73502 HCl
CAS :EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of σ1 receptor (Ki = 118 nM). EST73502 displays antinociceptive activity.Formule :C19H27ClF2N2O2Degré de pureté :99.96%Couleur et forme :SolidMasse moléculaire :388.88Ref: TM-T39284
1mg96,00€5mg172,00€10mg244,00€25mg403,00€50mg567,00€100mg750,00€200mg1.018,00€1mL*10mM (DMSO)187,00€LY2409881 trihydrochloride
CAS :LY2409881 trihydrochloride is a novel specific inhibitor of IKK2 (IC50: 30 nM); IC50 for IKK1 and other common kinases is at least one log higher.Formule :C24H32Cl4N6OSDegré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :594.43Maprotiline
CAS :Maprotiline blocks norepinephrine uptake, has antidepressant properties, and fights cancer by inducing apoptosis and inhibiting ERK and CRABP1.Formule :C20H23NCouleur et forme :SolidMasse moléculaire :277.4Gypsogenin
CAS :Gypsogenin (639-14-5) is a naturally occurring biochemical that shows anti-ABL1 kinase and anti-chronic Myelogenous Leukemia activities.Formule :C30H46O4Degré de pureté :99.73%Couleur et forme :SolidMasse moléculaire :470.68Ref: TM-T25476
1mg134,00€5mg315,00€10mg469,00€25mg748,00€50mg1.064,00€100mg1.415,00€1mL*10mM (DMSO)349,00€SN-38
CAS :SN-38 (NK012) is the active metabolite of Irinotecan, a DNA topoisomerase I (Topo I) inhibitor, which inhibits DNA and RNA synthesis (IC50=0.077/1.3 μM).Formule :C22H20N2O5Degré de pureté :98% - 99.97%Couleur et forme :Light-Yellow SolidMasse moléculaire :392.4PAR-2 Activating Peptide acetate
PAR-2 Activating Peptide acetate (SLIGRL-NH2 acetate) is an agonist of Protease-Activated Receptor-2 (PAR-2).Formule :C31H60N10O9Degré de pureté :98.5% - 99.92%Couleur et forme :SolidMasse moléculaire :716.885,7-Dimethoxyluteolin
CAS :5,7-Dimethoxyluteolin is a natural product from Hovenia acerba. 5,7-Dimethoxyluteolin is a dopamine transporter (DAT) activator with an EC50 of 3.417 μM.Formule :C17H14O6Degré de pureté :99.27%Couleur et forme :SolidMasse moléculaire :314.29Alovudine
CAS :3'-Fluoro-3'-deoxythymidine (3'-Deoxy-3'-fluorothymidine) is a marker of DNA synthesis,which is less susceptible to inflammatory changes than FDG.Formule :C10H13FN2O4Degré de pureté :99.41%Couleur et forme :Less Solid Colourless SolidMasse moléculaire :244.22Epothilone B
CAS :Epothilone B (EPO 906) is a compound isolated from the myxobacterium Sorangium cellulosum.Formule :C27H41NO6SDegré de pureté :99.79% - 99.84%Couleur et forme :White PowderMasse moléculaire :507.68Ref: TM-T6075
1mg35,00€2mg50,00€5mg66,00€10mg99,00€25mg215,00€50mg389,00€100mg567,00€1mL*10mM (DMSO)73,00€
![8-Fluoro-1,3,4,5-tetrahydro-6H-azepino[5,4,3-cd]indol-6-one](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT4698.webp&w=3840&q=75)
![Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel-](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT9800.webp&w=3840&q=75)
