
Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.781 produits)
- Apoptose(6.260 produits)
- Cycle cellulaire/point de contrôle(4.789 produits)
- Chromatine/Épigénétique(2.437 produits)
- Signalisation du cytosquelette(1.525 produits)
- Altération de l'ADN/réparation de l'ADN(2.967 produits)
- Endocrinologie/Hormones(3.706 produits)
- Enzyme(3.667 produits)
- GPCR/G-Protéine(9.000 produits)
- Immunologie et Inflammation(3.869 produits)
- Virus de la grippe(301 produits)
- Signalisation JAK/STAT(414 produits)
- Signalisation MAPK(1.249 produits)
- Transporteur membranaire/Canal ionique(3.029 produits)
- Métabolisme(10.207 produits)
- Microbiologie/Virologie(7.583 produits)
- Neuroscience(10.380 produits)
- Autres inhibiteurs(36.059 produits)
- Oxydation-Réduction(43 produits)
- Signalisation PI3K/Akt/mTOR(1.445 produits)
- Protéases/Protéasome(1.725 produits)
- Cellules souche et Dérivés(825 produits)
- Tyrosine Kinase/Adaptateurs(2.037 produits)
- Ubiquitination(1.716 produits)
Affichez 16 plus de sous-catégories
66687 produits trouvés pour "Inhibiteurs"
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Dihydroartemisinin
CAS :Dihydroartemisinin (Artenimol) is an antimalarial drug. High-Quality, Low-Cost!Formule :C15H24O5Degré de pureté :98% - 99.41%Couleur et forme :White SolidMasse moléculaire :284.35Lotilaner
CAS :Lotilaner is a parasiticide.Formule :C20H14Cl3F6N3O3SDegré de pureté :99.56%Couleur et forme :SolidMasse moléculaire :596.76Oxybutynin chloride
CAS :Oxybutynin chloride (Oxybutynin HCl) is an anticholinergic medication used to relieve urinary and bladder difficulties.Formule :C22H32ClNO3Degré de pureté :99.27% - >99.99%Couleur et forme :White PowderMasse moléculaire :393.96A-3 hydrochloride
CAS :<p>A-3 hydrochloride: potent, reversible kinase antagonist; permeable; inhibits PKC, CKI, PKA, CKII, MLCK; Ki: 4.3-80 μM.</p>Formule :C12H14Cl2N2O2SDegré de pureté :99.32%Couleur et forme :SolidMasse moléculaire :321.22Sulbentine
CAS :Sulbentine (Dibenzthione) is an antifungal agent.Formule :C17H18N2S2Degré de pureté :98.79%Couleur et forme :SolidMasse moléculaire :314.472',5'-Dideoxyadenosine
CAS :2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).Formule :C10H13N5O2Degré de pureté :99.55%Couleur et forme :White SolidMasse moléculaire :235.24Rivastigmine
CAS :Rivastigmine (Exelon) is a Cholinesterase Inhibitor, used for therapy of Alzheimer disease.Formule :C14H22N2O2Degré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :250.34Clofarabine
CAS :Clofarabine (Clofarex)m, a second generation purine nucleoside analog with antineoplastic activity, inhibits the enzymatic activities of ribonucleotideFormule :C10H11ClFN5O3Degré de pureté :99.94% - >99.99%Couleur et forme :White SolidMasse moléculaire :303.68Ropivacaine hydrochloride
CAS :Ropivacaine hydrochloride (Ropivacaine monohydrochloride) is the hydrochloride salt of ropivacaine, a local anesthetic of the amide type with analgesic activityFormule :C17H26N2O·HClDegré de pureté :99.85% - 99.95%Couleur et forme :SolidMasse moléculaire :310.86Oxytetracycline
CAS :Oxytetracycline (Terramycin) is a TETRACYCLINE analog isolated from the actinomycete STREPTOMYCES rimosus and used in a wide variety of clinical conditions.Formule :C22H24N2O9Degré de pureté :99.11%Couleur et forme :Light-Yellow Crystals Or Needles From Aqueous Meoh Physical Description Odorless Fluffy Yellow Solid Or Yellow Powder Bitter Taste (Ntp 1992)Masse moléculaire :460.43Diphenylacetonitrile
CAS :Diphenylacetonitrile (Dipan) is used as herbicide and industrial intermediate.Formule :C14H11NDegré de pureté :98.56%Couleur et forme :White CrystalMasse moléculaire :193.24Lanraplenib
CAS :Lanraplenib (GS-9876) is a highly selective and orally active SYK inhibitor (IC50=9.5 nM) in development for the treatment of inflammatory diseases.Formule :C23H25N9ODegré de pureté :98.35%Couleur et forme :SolidMasse moléculaire :443.5Mifepristone
CAS :Mifepristone (C-1073) is a progesterone-receptor (IC50=0.2 nM) and glucocorticoid-receptor antagonist (IC50=2.6 nM). High-Quality, Low-Cost!Formule :C29H35NO2Degré de pureté :98.9% - ≥95%Couleur et forme :Pale Yellow SolidMasse moléculaire :429.593,4-Dimethoxyphenylacetic acid
CAS :3,4-Dimethoxyphenylacetic acid (Homoveratrumic acid) is the papaverine intermediate, used to synthesis cardiovascular drugs.Formule :C10H12O4Degré de pureté :99.63%Couleur et forme :SolidMasse moléculaire :196.2Bromhexine hydrochloride
CAS :Bromhexine hydrochloride (Bisolvon) is a mucolytic agent used in the treatment of respiratory disorders associated with viscid or excessive mucus.Formule :C14H21Br2ClN2Degré de pureté :99.98%Couleur et forme :White SolidMasse moléculaire :412.59Ethylenediaminetetraacetic acid trisodium salt
CAS :Ethylenediaminetetraacetic acid trisodium salt (EDTA Trisodium) used to bind metal ions in the chelation therapy.Formule :C10H13N2Na3O8Degré de pureté :99.92% - 99.96%Couleur et forme :White CrystalsMasse moléculaire :358.19Desbenzyl Donepezil Hydrochloride
CAS :Desbenzyl Donepezil Hydrochloride is an impurity of Donepezil.Formule :C17H24ClNO3Degré de pureté :99.39%Couleur et forme :SolidMasse moléculaire :325.83Tigecycline
CAS :<p>Tigecycline (GAR-936), a broad-spectrum glycylcycline, disrupts protein synthesis by binding the 30S ribosomal subunit.</p>Formule :C29H39N5O8Degré de pureté :98.81% - >99.99%Couleur et forme :PowderMasse moléculaire :585.65Zileuton
CAS :Zileuton (A 64077) inhibits 5-lipoxygenase, reduces leukotrienes, aids bronchodilation, lessens mucus/edema, and helps manage asthma symptoms.Formule :C11H12N2O2SDegré de pureté :98.72% - 99.43%Couleur et forme :Crystalline SolidMasse moléculaire :236.294'-Demethylepipodophyllotoxin
CAS :4'-Demethylepipodophyllotoxin (DMEP) is a potent inhibitor of microtubule assembly.Formule :C21H20O8Degré de pureté :98.49% - 99.72%Couleur et forme :White Crystalline PowderMasse moléculaire :400.38Deoxycholic acid
CAS :Deoxycholic acid (Cholanoic Acid) is a bile acid formed by bacterial action from cholate.Formule :C24H40O4Degré de pureté :99.91% - 99.91%Couleur et forme :Crystals From Alc SolidMasse moléculaire :392.57BLT-1
CAS :<p>BLT-1 is a scavenger receptor BI (SR-BI)inhibitor.</p>Formule :C12H23N3SDegré de pureté :97.97%Couleur et forme :SolidMasse moléculaire :241.4Nufenoxole
CAS :Nufenoxole is an orally active and antidiarrhoeal compound that inhibits fluid secretion in the human jejunum.Formule :C25H29N3ODegré de pureté :98.84%Couleur et forme :SolidMasse moléculaire :387.52Pancreatin
CAS :Pancreatin (pancrelipase) is a mixture of several digestive enzymes secreted by the exocrine cells of the pancreas.Degré de pureté :98%Couleur et forme :SolidProcurcumadiol
CAS :Procurcumadiol (5-Hydroxyprocurcumenol) is a natural product found in Curcuma longa and Curcuma phaeocaulis.Formule :C15H22O3Degré de pureté :99.88%Couleur et forme :SolidMasse moléculaire :250.33ARP-100
CAS :ARP-100 (MMP-2 Inhibitor III) is a potent and selective matrix metalloproteinase MMP-2 inhibitor (IC50=12 nM).Formule :C17H20N2O5SDegré de pureté :97.18%Couleur et forme :SolidMasse moléculaire :364.42Zolmitriptan
CAS :<p>Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, alleviating migraines.</p>Formule :C16H21N3O2Degré de pureté :99.69% - 99.91%Couleur et forme :White Or Kind Of White PowderMasse moléculaire :287.36Larazotide acetate
CAS :Larazotide acetate is a synthetic peptide. It functions as a tight junction regulator and reverses leaky junctions to their normally closed state.Formule :C34H59N9O12Degré de pureté :95.53% - 99.425%Couleur et forme :SolidMasse moléculaire :785.89Chlorhexidine
CAS :Chlorhexidine is a biguanide antiseptic targeting bacteria, damaging cell membranes and causing cell death, more effective against gram-positive types.Formule :C22H30Cl2N10Degré de pureté :98% - 99.85%Couleur et forme :Crystals From Methanol SolidMasse moléculaire :505.45Roxithromycin
CAS :Roxithromycin (RU-28965) is a semi-synthetic derivative of the macrolide antibiotic erythromycin with antibacterial and anti-malarial activities.Formule :C41H76N2O15Degré de pureté :99.29% - 99.98%Couleur et forme :White Crystalline PowderMasse moléculaire :837.05Imrecoxib
CAS :Imrecoxib (BAP-909) is a novel and selective cyclooxygenase 2 (COX-2) inhibitor (IC50: 18 nM).Formule :C21H23NO3SDegré de pureté :99.87%Couleur et forme :SolidMasse moléculaire :369.48HBX 19818
CAS :<p>HBX 19818 is a specific ubiquitin-specific protease 7 (USP7) inhibitor (IC50: 28.1 μM).</p>Formule :C25H28ClN3ODegré de pureté :97.71%Couleur et forme :SolidMasse moléculaire :421.96Orotic acid
CAS :<p>Orotic acid (Vitamin B13) is an intermediate product in pyrimidine metabolism.</p>Formule :C5H4N2O4Degré de pureté :99.42%Couleur et forme :Crystals Physical Description White Crystals Or Crystalline Powder (Ntp 1992)Masse moléculaire :156.1Cisplatin
CAS :Cisplatin (CDDP) is a DNA cross-linking agent.Formule :Cl2H6N2PtDegré de pureté :97.13% - 99.63%Couleur et forme :Orange-Yellow To Deep Yellow Solid Or PowderMasse moléculaire :300.04Allopurinol
CAS :Allopurinol (Zyloric) is a Xanthine Oxidase Inhibitor. The mechanism of action of allopurinol is as a Xanthine Oxidase Inhibitor.Formule :C5H4N4ODegré de pureté :99.36% - 99.96%Couleur et forme :Fluffy White To Off-White Powder Physical Description Odorless Tasteless White Microcrystalline Powder (Ntp 1992)Masse moléculaire :136.11AES-135
CAS :AES-135 is a potent HDAC inhibitor, inhibits HDAC3, HDAC6, HDAC11 (IC50s: 654, 190, and 636 nM) with anti-tumor activity.Formule :C33H29F6N3O5SDegré de pureté :97.72%Couleur et forme :SolidMasse moléculaire :693.66DUPA(OtBu)-OH
CAS :DUPA(OtBu)-OH, a DUPA precursor, targets PSMA with high affinity (Ki=8nM) to deliver Docetaxel for prostate cancer therapy.Formule :C23H40N2O9Degré de pureté :97.29%Couleur et forme :SolidMasse moléculaire :488.57ACT-389949
CAS :<p>ACT-389949: Potent, selective FPR2/ALX agonist; EC50 3 nM; potential inflammatory disorder treatment.</p>Formule :C20H18F2N6O3Degré de pureté :99.4%Couleur et forme :SolidMasse moléculaire :428.39Dibenzosuberone
CAS :Dibenzosuberone, pharmaceutical intermediates, is used for the synthesis of drug amitriptyline.Formule :C15H12ODegré de pureté :99.83%Couleur et forme :Clear To Yellow LiquidMasse moléculaire :208.26Solabegron
CAS :Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-ARFormule :C23H23ClN2O3Degré de pureté :97.89%Couleur et forme :SolidMasse moléculaire :410.89Isomaltose
CAS :Isomaltose (D-Isomaltose) is a reducing disaccharide, similar to maltose, but with an α-(1-6)-linkage instead of the α-(1-4)-linkage.Formule :C12H22O11Degré de pureté :99.98% - ≥95%Couleur et forme :Coloured SolutionMasse moléculaire :342.30trans-C75
CAS :trans-C75 ((±)-C75) is an enantiomer of C75. C75 is an inhibitor of fatty-acid synthase (FASN).Formule :C14H22O4Degré de pureté :98.88% - 99.57%Couleur et forme :White To Off-White SolidMasse moléculaire :254.32Aliskiren hemifumarate
CAS :<p>Aliskiren hemifumarate (CGP60536B) is an orally active nonpeptide renin inhibitor with antihypertensive activity.</p>Formule :C30H53N3O6C4H4O4Degré de pureté :96.18% - 99.21%Couleur et forme :SolidMasse moléculaire :1219.6Nampt activator-1
CAS :NAMPT Activator-1, EC50: 3.3-3.7 µM, specific niacinamide phosphotransferase stimulant, shields cells, potential neuroprotectant.Formule :C16H17N3O3Degré de pureté :99.84% - 99.98%Couleur et forme :SoildMasse moléculaire :299.32Nitazoxanide
CAS :Nitazoxanide (NSC-697855) is a synthetic benzamide antiprotozoal; it disrupts pyruvate electron transfer reactions.Formule :C12H9N3O5SDegré de pureté :99% - 99.93%Couleur et forme :SolidMasse moléculaire :307.28Chlorpheniramine maleate
CAS :Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.Formule :C20H23ClN2O4Degré de pureté :99.64% - 99.98%Couleur et forme :Odorless White Crystalline Solid Or White Powder With A Bitter TasteMasse moléculaire :390.87Bicalutamide
CAS :<p>Bicalutamide (ICI-176334), a synthetic, nonsteroidal antiandrogen, competitively binds to cytosolic androgen receptors in target tissues, thereby inhibiting the</p>Formule :C18H14F4N2O4SDegré de pureté :98% - 99.87%Couleur et forme :Off-White Crystalline SolidMasse moléculaire :430.37Orphenadrine hydrochloride
CAS :Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.Formule :C18H23NO·HClDegré de pureté :99.88%Couleur et forme :Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)Masse moléculaire :305.85Arjungenin
CAS :Arjungenin, a triterpene derived from Terminalia arjuna, exhibits insect feeding-deterrent and growth inhibitory properties.Formule :C30H48O6Degré de pureté :99.76%Couleur et forme :SolidMasse moléculaire :504.70Pomisartan 2HCl
<p>Pomisartan 2HCl (BIBR363 2HCL) is a small molecule AT1R antagonist used to study heart failure and hypertension.</p>Formule :C31H32Cl2N4O2Degré de pureté :99.88%Couleur et forme :SoildMasse moléculaire :563.52Fostemsavir Tris
CAS :Fostemsavir Tris (BMS-663068 Tris) is the prodrug of BMS-626529,is a oral, safe and effective inhibitor of HIV-1 attachment.Formule :C29H37N8O11PDegré de pureté :99.45%Couleur et forme :SolidMasse moléculaire :704.62MRT-83
CAS :MRT-83 is a potent Smo antagonist.Formule :C31H30N4O5Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :538.59Ciliobrevin D
CAS :Ciliobrevin D is a AAA+ ATPase motor cytoplasmic dynein inhibitor.Formule :C17H8Cl3N3O2Degré de pureté :98.09%Couleur et forme :SolidMasse moléculaire :392.62Metamizole sodium hydrate
CAS :Metamizole sodium hydrate (Analgin) is a potent analgesic drug that has been demonstrated to inhibit cyclooxygenase (COX).Formule :C13H18N3NaO5SDegré de pureté :99.69% - 99.89%Couleur et forme :White Or Light Yellow Crystalline Powder Odorless Tiny BitterMasse moléculaire :351.36Dexchlorpheniramine Maleate
CAS :Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.Formule :C20H23ClN2O4Degré de pureté :99.58%Couleur et forme :White Or Almost White Crystalline PowderMasse moléculaire :390.86Isotretinoin
CAS :Isotretinoin (13-cis-Retinoic acid) binds to and activates nuclear retinoic acid receptors (RARs); activated RARs serve as transcription factors that promoteFormule :C20H28O2Degré de pureté :97.01% - 98.06%Couleur et forme :Reddish-Orange Plates From Isopropyl Alcohol (Ntp 1992)Masse moléculaire :300.44Sonepcizumab
CAS :<p>Sonepcizumab, a human monoclonal antibody, targets S1P to combat cancer and prevent post-glaucoma eye scarring.</p>Degré de pureté :SDS-PAGE:95% SEC-HPLC:98.90%Couleur et forme :LiquidMasse moléculaire :146.43 kDaT-0156
CAS :T-0156 is a PEG5 inhibitor that inhibits the hydrolysis of cyclic guanosine monophosphate (cGMP) with low affinity for PDE6, PDE1, PDE2, PDE3 and PDE4.Formule :C31H29N5O7Degré de pureté :98.53% - 98.76%Couleur et forme :SoildMasse moléculaire :583.59Sunitinib
CAS :Sunitinib (SU 11248) is a multi-targeted receptor tyrosine kinase (RTK) inhibitor that inhibits VEGFR2 and PDGFRβ (IC50=80/2 nM).Formule :C22H27FN4O2Degré de pureté :98% - 99.67%Couleur et forme :Yellow SolidMasse moléculaire :398.47Ozagrel
CAS :<p>Ozagrel (Domenan) is a selective thromboxane A(2) (TXA(2)) synthetase inhibitor with IC50 of 11 nM for rabbit platelet, used for the improvement of</p>Formule :C13H12N2O2Degré de pureté :97.90% - 99.38%Couleur et forme :White PowderMasse moléculaire :228.25Febantel
CAS :Febantel is an anthelmintic. It is used for veterinary use on dogs, cats, cattle, sheep, goats, pig, and poultry against roundworms and tapeworms.Formule :C20H22N4O6SDegré de pureté :99.85%Couleur et forme :White To Off-White PowderMasse moléculaire :446.48Capreomycin sulfate
CAS :Capreomycin sulfate (Capastat sulfate) , a cyclic peptide antibiotic, binds to the 70S ribosomal unit leading to inhibition of protein synthesis.Formule :C25H46N14O11SDegré de pureté :98% - 99.54%Couleur et forme :White PowderMasse moléculaire :752.76Clopidogrel
CAS :Clopidogrel (SR-25990C), a P2Y12 receptor antagonist, decreases platelet aggregation.Formule :C16H16ClNO2SDegré de pureté :98.23% - 98.83%Couleur et forme :White PowderMasse moléculaire :321.82Retagliptin Phosphate
CAS :Retagliptin Phosphate (SP 2086) is pharmaceutical composition of DPP-4 inhibitor, for treating type-2 diabetes.Formule :C19H21F6N4O7PDegré de pureté :98.70%Couleur et forme :SolidMasse moléculaire :562.36Moguisteine
CAS :Moguisteine (BBR-2173) is a new-type peripheral non-narcotic antitussive drug.Formule :C16H21NO5SDegré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :339.41NH2-PEG6-Boc
CAS :NH2-PEG6-Boc is a PEG-based PROTAC linker that can be used in PROTAC synthesis[1].Formule :C19H39NO8Degré de pureté :≥98%Couleur et forme :SolidMasse moléculaire :409.51BI-1935
CAS :<p>BI-1935 is an inhibitor of soluble epoxide hydrolase (sEH). For diseases related to cardiovascular disease.</p>Formule :C24H21F3N6O3Degré de pureté :97.55%Couleur et forme :SolidMasse moléculaire :498.46Gluconate Calcium
CAS :Gluconate Calcium (Gluconic acid hemicalcium salt) is the calcium salt of gluconic acid, used as a calcium replenisher in hypocalcemic states.Formule :C12H22CaO14Degré de pureté :99.57% - 99.81%Couleur et forme :Crystals Granules Or PowderMasse moléculaire :430.37KukoaMine B
CAS :Kukoamine B, as a constituent of Lycii Cortex, exhibits anti-acute inflammatory, anti-oxidant, and anti-diabetic characteristics.Formule :C28H42N4O6Degré de pureté :95% - 99.59%Couleur et forme :SolidMasse moléculaire :530.66Broxyquinoline
CAS :Broxyquinoline (5,7-Dibromo-8-hydroxyquinoline) is an antiprotozoal agent, and it can release oxygen free radicals from the water in mucous membranes.Formule :C9H5Br2NODegré de pureté :99.71%Couleur et forme :Almost White PowderMasse moléculaire :302.95Aminophylline
CAS :<p>Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.</p>Formule :C7H8O2·C2H8N2Degré de pureté :99.31%Couleur et forme :White Or Slightly Yellowish Granules Or Powder SolidMasse moléculaire :420.43MK-8719
CAS :MK-8719 is a highly potent and selective inhibitor of O-GlcNAcase (OGA) (hOGA, Ki=7.9 nM) .Formule :C9H14F2N2O3SDegré de pureté :99.67%Couleur et forme :SolidMasse moléculaire :268.28Ketorolac tromethamine salt
CAS :Ketorolac tromethamine salt (Ketorolac tris salt) non-selective inhibits the enzymes cyclooxygenase 1 (COX-1) and COX-2with anti-inflammatory, analgesic, andFormule :C19H24N2O6Degré de pureté :99.48% - 99.85%Couleur et forme :CrystallineMasse moléculaire :376.4NE 10790
CAS :NE 10790, similar to risedronate, is a mild bone resorption inhibitor but poorly blocks FPP synthase.Formule :C8H10NO6PDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :247.14L-SelenoMethionine
CAS :L-Selenomethionine is a natural amino acid boosting cell growth and antioxidant enzyme levels.Formule :C5H11NO2SeDegré de pureté :99.5% - 99.67%Couleur et forme :White To Off-WhitepowderMasse moléculaire :196.11Quinine
CAS :Quinine is a natural cinchona alkaloid that has been used for centuries in the prevention and therapy of malaria.Formule :C20H24N2O2Degré de pureté :99.93% - 99.97%Couleur et forme :White Solid PowderMasse moléculaire :324.42Lin28-let-7a antagonist 1
CAS :Lin28-let-7a antagonist 1, with an IC50 of 4.03 μM for Lin28A-let-7a-1 interaction,and shows a clear antagonistic effect against the Lin28-let-7a interaction.Formule :C31H29N5O7Degré de pureté :99.44%Couleur et forme :SolidMasse moléculaire :583.59Diammonium Glycyrrhizinate
CAS :Diammonium Glycyrrhizinate, a licorice-derived anti-inflammatory, metabolizes to glycyrrhetinic acid, affecting corticosteroid metabolism & blood pressure.Formule :C42H62O16·2H3NDegré de pureté :90% - 99.93%Couleur et forme :SolidMasse moléculaire :857β-Cyclodextrin
CAS :β-Cyclodextrin (NSC 269471) is a member of the class of compounds known as oligosaccharides.Formule :C42H70O35Degré de pureté :97.13% - 99.92%Couleur et forme :White Solid PowderMasse moléculaire :1134.98Lycorine hydrochloride
CAS :<p>Lycorine hydrochloride (Narcissine hydrochloride) is VE-cadherin inhibitor,and has IC50 of 1.2μM in Hey1B cell.It is an HCV inhibitor with strong activity.</p>Formule :C16H18ClNO4Degré de pureté :99.45% - 99.49%Couleur et forme :Fine Crystal PowderMasse moléculaire :323.77DREADD agonist 21
CAS :DREADD agonist 21 is a potent agonist of human muscarinic acetylcholine M3 receptors (EC50=1.7 nM).Formule :C17H18N4Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :278.35Gboxin
CAS :Gboxin is an inhibitor of oxidative phosphorylation that targets glioblastoma,inhibits the activity of F0F1 ATP synthase, with antitumour activity.Formule :C22H33ClN2O2Degré de pureté :99.96% - >99.99%Couleur et forme :SolidMasse moléculaire :392.96AZD7624
CAS :AZD7624 is an p38 inhibitor. It has potent anti-inflammatory activity.Formule :C27H30FN5O3Degré de pureté :98.82%Couleur et forme :SolidMasse moléculaire :491.56Tramiprosate
CAS :<p>Tramiprosate (Alzhemed) is an orally active, BBB-crossing, naturally occurring amino acid that binds soluble Aβ and maintains it in a non-protofibrillar form.</p>Formule :C3H9NO3SDegré de pureté :99%Couleur et forme :White Crystals Or Crystalline PowerMasse moléculaire :139.17Ascorbyl palmitate
CAS :<p>Ascorbyl palmitate (L-Ascorbic acid 6-hexadecanoate), an ester formed from ascorbic acid and palmitic acid, produces a fat-soluble form of vitamin C.</p>Formule :C22H38O7Degré de pureté :99.52%Couleur et forme :White Or Yellowish White Powder White Or Yellowish-White Powder With A Citrus-Like OdourMasse moléculaire :414.535,6-Dihydro-5-methyluracil
CAS :<p>5,6-Dihydro-5-methyluracil (Dihydrothymine) is an intermediate breakdown product of thymine.</p>Formule :C5H8N2O2Degré de pureté :98.53%Couleur et forme :SolidMasse moléculaire :128.13Chlorindione
CAS :<p>Chlorindione (chlophenadione) is a vitamin K antagonist, a potent anticoagulant compound.</p>Formule :C15H9ClO2Degré de pureté :97.23% - 99.67%Couleur et forme :SolidMasse moléculaire :256.68NK-252
CAS :NK-252 is a potential activator of Nrf2. It has great Nrf2-activating potential.Formule :C13H11N5O3Degré de pureté :98.32%Couleur et forme :SolidMasse moléculaire :285.26Ziprasidone hydrochloride
CAS :Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychoticFormule :C21H22CL2N4OSDegré de pureté :97.97% - 99.82%Couleur et forme :SolidMasse moléculaire :449.4(Rac)-Telinavir
CAS :<p>N1 compound with anti-HIV activity; contains dimethyl, phenyl, quinoline groups.</p>Formule :C33H44N6O5Degré de pureté :99.30%Couleur et forme :SolidMasse moléculaire :604.742-(1-Piperazinyl)pyrimidine
CAS :2-(1-Piperazinyl)pyrimidine is used as an anti-anxiety drug.Formule :C8H12N4Degré de pureté :98.46%Couleur et forme :Liquid - Crystal - LumpMasse moléculaire :164.21Lapatinib
CAS :Lapatinib (GW572016) is an inhibitor of ErbB2 and EGFR (IC50=9.2/10.8 nM) with oral activity.Formule :C29H26ClFN4O4SDegré de pureté :99.00% - 99.81%Couleur et forme :PowderMasse moléculaire :581.066-Methoxy-2-naphthoic acid
CAS :6-Methoxy-2-naphthoic acid (6-Methoxy-2-naphthalenecarboxylic acid) is an modulator of NMDAR.Formule :C12H10O3Degré de pureté :99.25%Couleur et forme :White To Off-White Powder Crystals Crystalline Powder And/Or ChunksMasse moléculaire :202.21Endovion
CAS :Endovion (NS3728) is a pharmacological anion channel and an Anoctamin-1 (ANO 1) channel inhibitor. Endovion is also the specific VRAC/VSOAC blocker.Formule :C16H9BrF6N6ODegré de pureté :98.51%Couleur et forme :SolidMasse moléculaire :495.18Phthalic acid mono-2-ethylhexyl ester
CAS :Phthalic acid mono-2-ethylhexyl ester (Phthalic Acid Monooctyl Ester is a major bioactive metabolite of DEHP, which inhibits the 17, 20 lyase activity of CYP17.Formule :C16H22O4Degré de pureté :98.01%Couleur et forme :Physical Description Clear Colorless To Cloudy White Viscous Liquid (Ntp 1992)Masse moléculaire :278.34Sulfalene
CAS :Sulfalene (SMP2), a long-acting sulfonamide antibiotic, is used for the therapy of chronic bronchitis, urinary tract infections, and malaria.Formule :C11H12N4O3SDegré de pureté :99.24% - 99.52%Couleur et forme :White Or Slightly Yellow Crystal PowderMasse moléculaire :280.3Cirsiumaldehyde
CAS :Cirsiumaldehyde is a compound isolated from the mature fruits of Lobelia chinensis, Cornus officinalis, and the fruits of Hippophae rhamnoides.CirsiumaldehydeFormule :C12H10O5Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :234.2IAXO-102
CAS :IAXO-102 is a TLR4 antagonist that negatively regulates TLR4 signaling.Formule :C35H71NO5Degré de pureté :98.17%Couleur et forme :SolidMasse moléculaire :585.94Amphotericin B
CAS :Amphotericin B (NSC-527017) is a polyene antifungal agent with broad-spectrum activity against many fungal species.Formule :C47H73NO17Degré de pureté :99.75% - ≥98%Couleur et forme :Deep Yellow Prisms Or Needles From N N-Dimethylformamide Physical Description Bright Yellow Powder (Ntp 1992)Masse moléculaire :924.08XEN723
CAS :XEN723 is a potent thiazolylimidazolidinone Stearoyl-CoA Desaturase (SCD1) inhibitor(IC50s of 45 and 524 nM in mouse and HepG2 cell, respectively).Formule :C21H20FN5O2SDegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :425.48

