
Inhibiteurs
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.762 produits)
- Apoptose(6.206 produits)
- Cycle cellulaire/point de contrôle(4.811 produits)
- Chromatine/Épigénétique(2.553 produits)
- Signalisation du cytosquelette(1.519 produits)
- Altération de l'ADN/réparation de l'ADN(2.906 produits)
- Endocrinologie/Hormones(3.703 produits)
- Enzyme(3.671 produits)
- GPCR/G-Protéine(9.002 produits)
- Immunologie et Inflammation(3.748 produits)
- Virus de la grippe(297 produits)
- Signalisation JAK/STAT(414 produits)
- Signalisation MAPK(1.244 produits)
- Transporteur membranaire/Canal ionique(3.106 produits)
- Métabolisme(10.125 produits)
- Microbiologie/Virologie(7.567 produits)
- Neuroscience(10.343 produits)
- Autres inhibiteurs(35.806 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.411 produits)
- Protéases/Protéasome(1.681 produits)
- Cellules souche et Dérivés(752 produits)
- Tyrosine Kinase/Adaptateurs(1.949 produits)
- Ubiquitination(1.716 produits)
66605 produits trouvés pour "Inhibiteurs"
Muvalaplin
CAS :Muvalaplin (LY3473329) is an orally active lipoprotein (a) Lp(a) reagent that inhibits Lp(a) formation by blocking apo(a)-apo B100 interactions.Formule :C42H54N4O6Degré de pureté :99.59% - 99.99%Couleur et forme :SoildMasse moléculaire :710.9Adarotene
CAS :Adarotene (ST1926) induces apoptosis, causes DNA damage, and has strong antiproliferative effects on human tumors.Formule :C25H26O3Degré de pureté :99.26%Couleur et forme :SolidMasse moléculaire :374.47Ref: TM-T14125
1mg35,00€2mg50,00€5mg77,00€10mg124,00€25mg230,00€50mg369,00€100mg537,00€500mg1.153,00€1mL*10mM (DMSO)78,00€BroMhexine IMpurity B
CAS :Bromhexine Impurity B reagent used in the preparation of Ambroxol and Bromhexine (B678600) metabolites Ambroxol EP Impurity E.Formule :C7H5Br2NODegré de pureté :99.20%Couleur et forme :Light Yellow Crystal PowderMasse moléculaire :278.93AZ084
CAS :AZ084 is a potent, selective, allosteric, and oral active CCR8 antagonist (Ki: 0.9 nM). It has the potential to treat asthma.Formule :C26H34N4O2Degré de pureté :97.12%Couleur et forme :SolidMasse moléculaire :434.57Ref: TM-T10425
1mg84,00€5mg161,00€10mg245,00€25mg406,00€50mg572,00€100mg772,00€200mg1.035,00€1mL*10mM (DMSO)172,00€ICA-27243
CAS :ICA-27243: Potent KCNQ2/Q3 opener, oral, EC50 0.38 μM; less effective on KCNQ4, KCNQ3/Q5; antiepileptic.Formule :C12H7ClF2N2ODegré de pureté :99.54%Couleur et forme :SolidMasse moléculaire :268.65MKC8866
CAS :MKC8866, a selective IRE1 RNase inhibitor with an IC50 of 0.29 μM, curbs breast and prostate cancer cell growth.Formule :C18H19NO7Degré de pureté :99.28% - 99.854%Couleur et forme :SolidMasse moléculaire :361.35Ref: TM-T15594
1mg88,00€2mgÀ demander5mg187,00€10mg264,00€25mg445,00€50mg588,00€100mg802,00€200mg1.074,00€1mL*10mM (DMSO)À demanderEmeramide
CAS :Emeramide (BDTH2) is a thiol-redox antioxidant. It is also a heavy metal chelator.Formule :C12H16N2O2S2Degré de pureté :98.73%Couleur et forme :SolidMasse moléculaire :284.4Flavone
CAS :Flavone (2-Phenyl-4-chromone) have effects on CYP (P450) activity which are enzymes that metabolize most drugs in the body.Formule :C15H10O2Degré de pureté :99.661% - 99.99%Couleur et forme :SolidMasse moléculaire :222.24Embeconazole
CAS :Embeconazole (R 120758) is a triazole antifungal agent with strong in vitro activity against clinically important fungi such as Candida and Aspergillus.Formule :C27H25F3N4O3SDegré de pureté :99.70% - 99.79%Couleur et forme :SolidMasse moléculaire :542.57Multifungin
CAS :Multifungin (Bromochlorosalicylanilide) is an antifungal that studies oral candidiasis.Formule :C13H9BrClNO2Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :326.57Ref: TM-T1043
2mg40,00€5mg60,00€10mg80,00€25mg140,00€50mg202,00€100mg305,00€500mg730,00€1mL*10mM (DMSO)47,00€5-CFDA
CAS :5-CFDA is a cell-permeable compound that, once inside cells, is converted to 5-carboxyfluorescein for labeling cells in fluorescence microscopy.Formule :C25H16O9Degré de pureté :97.16% - 97.51%Couleur et forme :SolidMasse moléculaire :460.39Rosiglitazone maleate
CAS :Rosiglitazone maleate (BRL 49653) is an oral antidiabetic and potential anticancer agent.Formule :C22H23N3O7SDegré de pureté :99.33% - 99.51%Couleur et forme :Off-White SolidMasse moléculaire :473.50FlutaMide Related CoMpound B
CAS :FlutaMide Related CoMpound B is used as pharmaceutical intermediates.Formule :C9H7F3N2O3Degré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :248.16Ethamsylate
CAS :Ethamsylate (Dicynene) 通常用作止血药,增加毛细血管内皮阻力和血小板粘附,抑制前列腺素的生物合成和作用。Formule :C10H17NO5SDegré de pureté :98.55%Couleur et forme :White Crystals Or Crystalline PowderMasse moléculaire :263.31Atazanavir
CAS :Atazanavir (BMS-232632)(BMS-232632) is an highly effective HIV-1 protease inhibitor.Formule :C38H52N6O7Degré de pureté :98% - 99.95%Couleur et forme :Crystalline SolidMasse moléculaire :704.86Diazinon
CAS :Diazinon (Dimpylate) is a thiophosphoric acid ester, functioning as a nonsystemic organophosphate insecticide that effectively targets and controls a variety ofFormule :C12H21N2O3PSDegré de pureté :97.07% - 98%Couleur et forme :Colorless Oil Ethanol/Xylene/Acetone With A Flash Point In The Range 82-105° FMasse moléculaire :304.35Trilaciclib hydrochloride
CAS :Trilaciclib hydrochloride (G1T28 hydrochloride) is an inhibitor of CDK4/6 (IC50s: 1 nM and 4 nM for CDK4 and CDK6).Formule :C24H32Cl2N8ODegré de pureté :99.69% - 99.89%Couleur et forme :SolidMasse moléculaire :519.472'-Deoxyadenosine monohydrate
CAS :Deoxyadenosine is a deoxyribonucleoside and adenosine derivative with a hydrogen replacing a hydroxyl group at ribose's 2' position.Formule :C10H15N5O4Degré de pureté :99.9% - 99.93%Couleur et forme :PowderMasse moléculaire :269.26Primaquine diphosphate
CAS :Primaquine diphosphate is the phosphate salt form of primaquine, a synthetic, 8-aminoquinoline derivative with antimalarial properties.Formule :C15H21N3O·2H3PO4Degré de pureté :99.73% - 99.82%Couleur et forme :Orange PowderMasse moléculaire :455.34Pitavastatin lactone
CAS :Pitavastatin lactone, a major human metabolite, potently inhibits HMG-CoA reductase with minimal hepatic microsome metabolism.Formule :C25H22FNO3Degré de pureté :98.18%Couleur et forme :White To Off-White PowderMasse moléculaire :403.45Ref: TM-T12490
5mg44,00€10mg62,00€25mg119,00€50mg178,00€100mg268,00€200mg401,00€1mL*10mM (DMSO)60,00€Dextromilnacipran
CAS :Dextromilnacipran (Levomilnacipran) is a selective serotonin and norepinephrine reuptake inhibitor.
Formule :C15H22N2ODegré de pureté :98.95% - >99.99%Couleur et forme :SolidMasse moléculaire :246.35Chloramphenicol
CAS :Chloramphenicol (Chloromycetin) is a broad-spectrum antibiotic that inhibits the biosynthesis of bacterial proteins. Cost-effective and quality-assured.
Formule :C11H12Cl2N2O5Degré de pureté :99.6% - 99.84%Couleur et forme :Needles Or Elongated Plates From Water Or Ethylene Dichloride SolidMasse moléculaire :323.13LSP-249
CAS :LSP-249 is a plasma kallikrein inhibitor under the study for angioedema, with an EC50 less than 100 nM in cell.Formule :C24H22ClN5ODegré de pureté :99.51%Couleur et forme :SolidMasse moléculaire :431.92ATPγS tetralithium salt
CAS :ATPγS tetralithium salt is a good substrate for RNA-stimulated nucleotide hydrolysis and RNA unwinding activity of eIF4A.Cost-effective and quality-assured.Formule :C10H12Li4N5O12P3SDegré de pureté :90% - ≥98%Couleur et forme :White PowderMasse moléculaire :546.98Sodium citrate dihydrate
CAS :Sodium citrate dihydrate (Trisodium citrate dihydrate) is an anticoagulant, and also used as a buffer and food preservatives.Formule :C6H9Na3O9Degré de pureté :≥98%Couleur et forme :Solid CrystallineMasse moléculaire :294.1Pamicogrel
CAS :Pamicogrel (KBT3022) is an inhibitor of COX.Formule :C25H24N2O4SDegré de pureté :99.83%Couleur et forme :SolidMasse moléculaire :448.53AV-412
CAS :AV-412 (MP412) is an EGFR inhibitor (EGFR, EGFR T790M, EGFR L858R, EGFR L858R/T790M and ErbB2 with IC50s of 0.75, 0.79, 0.5, 2.3, 19 nM).Formule :C41H44ClFN6O7S2Degré de pureté :99.85% - 99.92%Couleur et forme :SolidMasse moléculaire :851.41Ref: TM-T10419
1mg42,00€2mg55,00€5mg90,00€10mg137,00€25mg240,00€50mg403,00€100mg582,00€1mL*10mM (DMSO)129,00€Tocainide
CAS :Tocainide is a blocker of the sodium channel and used for the treatment of tinnitus.Formule :C11H16N2ODegré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :192.26GATA4-NKX2-5-IN-1
CAS :GATA4-NKX2-5-IN-1 inhibits GATA4-NKX2-5 synergy (IC50=3μM), doesn't affect related kinases, and modulates cardiac gene expression.Formule :C21H23N3O2Degré de pureté :99.00%Couleur et forme :SolidMasse moléculaire :349.43Ref: TM-T11368
1mg62,00€5mg135,00€10mg178,00€25mg284,00€50mg380,00€100mg509,00€200mg698,00€1mL*10mM (DMSO)149,00€2-Phenylbutanoic acid
CAS :2-Phenylbutanoic acid (2-Phenylbutyric acid) is used as an industrial intermediate.Formule :C10H12O2Degré de pureté :98.25%Couleur et forme :SolidMasse moléculaire :164.2Imidazolidinyl urea
CAS :Imidazolidinyl urea (Imidurea) is an antimicrobial preservative used in cosmetics.Formule :C11H16N8O8Degré de pureté :98.6%Couleur et forme :White Fluid Powder With Slight Characteristic OdorMasse moléculaire :388.29FFN 511
CAS :Fluorescent false neurotransmitter (FFN)Formule :C17H20N2O2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :284.35Rovalpituzumab
CAS :Rovalpituzumab: humanized antibody against DLL3, forms ADCs, treats small cell lung cancer.Degré de pureté :> 95%Couleur et forme :LiquidMasse moléculaire :145.02 kDaIslatravir
CAS :Islatravir (MK-8591) is an effective anti-HIV-1 agent.Formule :C12H12FN5O3Degré de pureté :98.77%Couleur et forme :SolidMasse moléculaire :293.25Ref: TM-T16098
1mg80,00€5mg170,00€10mg259,00€25mg454,00€50mg615,00€100mg827,00€200mg1.111,00€1mL*10mM (DMSO)182,00€Phloracetophenone
CAS :Phloracetophenone combats obesity, lowers lipids by slowing fat absorption via pancreatic lipase inhibition.Formule :C8H8O4Degré de pureté :99.57%Couleur et forme :Light Yellow CrystalMasse moléculaire :168.15Astressin acetate
Astressin acetate is an antagonist of corticotropin releasing factor (CRF) with low affinity for the CRF binding protein and high affinity for the clonedFormule :C163H273N49O44Degré de pureté :96.87%Couleur et forme :SolidMasse moléculaire :3623.21Isohomovanillic acid
CAS :Isohomovanillic acid (Homoisovanillic acid is used as pharmaceutical intermediates.
Formule :C9H10O4Degré de pureté :99.04%Couleur et forme :SolidMasse moléculaire :182.17Flunixin meglumine
CAS :Flunixin meglumine (Banamine) is an effective inhibitor of the enzyme cyclooxygenase with anti-inflammatory and antipyretic activity.Formule :C21H28F3N3O7Degré de pureté :99.57% - >99.99%Couleur et forme :SolidMasse moléculaire :491.46Nabumetone
CAS :Nabumetone (BRL14777)(BRL14777) is a non-steroidal anti-inflammatory drug and its active metabolite 6MNA inhibits the enzymes cyclo-oxygenase I and II.Formule :C15H16O2Degré de pureté :97.59% - 99.61%Couleur et forme :White /Almost White Crystalline PowderMasse moléculaire :228.29Diazoxide
CAS :Diazoxide (Proglycem) is a benzothiadiazine derivative that is a peripheral vasodilator used for hypertensive emergencies.Formule :C8H7ClN2O2SDegré de pureté :99% - 99.83%Couleur et forme :SolidMasse moléculaire :230.67Traxanox
CAS :Traxanox: oral diuretic, boosts phagocytosis in mice/rats, reverses antibody production inhibition in BALB/c mice.Formule :C13H6ClN5O2Degré de pureté :98.37%Couleur et forme :SolidMasse moléculaire :299.67Nortriptyline hydrochloride
CAS :Nortriptyline HCl, a metabolite of amitriptyline, treats major and atypical depression, dysthymia.Formule :C19H22ClNDegré de pureté :99.85% - ≥95%Couleur et forme :SolidMasse moléculaire :299.84Paprotrain
CAS :Paprotrain ((alphaZ)-alpha-(3-Pyridinylmethylene)-1H-indole-3-acetonitrile) inhibits the ATPase activity of MKLP-2 with an IC50 of 1.35 μM and a Ki of 3.36 μM.Formule :C16H11N3Degré de pureté :99.91%Couleur et forme :SolidMasse moléculaire :245.28Ref: TM-T12359
5mg46,00€10mg58,00€25mg92,00€50mg160,00€100mg236,00€200mg353,00€500mg580,00€1mL*10mM (DMSO)49,00€Fudosteine
CAS :Fudosteine is a novel mucoactive agent and a MUC5AC mucin hypersecretion inhibitor.
Formule :C6H13NO3SDegré de pureté :99.59%Couleur et forme :Off-White CrystallineMasse moléculaire :179.24KHK-IN-1
CAS :KHK-IN-1: Ketohexokinase inhibitor, IC50=12 nM, permeable, inhibits F1P in HepG2 cells, potential for obesity/diabetes research.Formule :C21H26N8SDegré de pureté :99.00%Couleur et forme :SolidMasse moléculaire :422.55Filorexant
CAS :Filorexant (MK-6096) is an orally bioavailable effective and selective reversible antagonist of OX1 and OX2 receptor with (Ki <3 nM).Formule :C24H25FN4O2Degré de pureté :98.88%Couleur et forme :SolidMasse moléculaire :420.481-Aminohydantoin hydrochloride
CAS :1-Aminohydantoin HCl, a metabolite of furantoin, binds to proteins, releases in acid, and is detectable in meat/milk for drug residue tests.Formule :C3H6ClN3O2Degré de pureté :99.64%Couleur et forme :Pale Yellow PowderMasse moléculaire :151.555α-Cholestan-3-one
CAS :5α-Cholestan-3-one (Coprostanone) is an intermediate product in cholesterol metabolism, which is elevated in the case of cerebrotendinous xanthomatosis.Formule :C27H46ODegré de pureté :99.84% - 99.97%Couleur et forme :SolidMasse moléculaire :386.65γ-DGG acetate(6729-55-1 free base)
CAS :gamma-DGG acetate(6729-55-1 free base) (γ-D-Glutamylglycine) is a competitive blocker of AMPA receptor.Formule :C9H16N2O7Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :264.23(R)-CR8
CAS :(R)-CR8 ((R)-Isomer) is a potent and selective CDK inhibitor.
Formule :C24H29N7ODegré de pureté :98.41%Couleur et forme :SolidMasse moléculaire :431.53DDAO
CAS :DDAO: NIR red fluorescent probe, λem 656 nm, excitation 600-650 nm, detects various enzymes.Formule :C15H11Cl2NO2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :308.16Vinpocetine
CAS :Vinpocetine (RGH-4405) is a selective inhibitor of cyclic GMP phosphodiesterase (PDE).Formule :C22H26N2O2Degré de pureté :99.85% - 99.98%Couleur et forme :White Crystalline SolidMasse moléculaire :350.45Pamidronate Disodium
CAS :Pamidronate Disodium (CGP 23339A), a nitrogen-containing bisphosphonate, can help to strengthen bones.Formule :C3H9NNa2O7P2Degré de pureté :99.86% - 99.93%Couleur et forme :White CrystalsMasse moléculaire :279.03Auristatin E
CAS :Auristatin E, MMAE analog, blocks tubulin polymerisation, has cytotoxic and potent antitumor effects, used in ADCs.Formule :C40H69N5O7Degré de pureté :98.81%Couleur et forme :SolidMasse moléculaire :732.01Vitamin K
CAS :Vitamin K (Kephton) has blood coagulation action and is important for coagulation factors, matrix-Gla protein, and osteocalcin.Degré de pureté :97.00% - 99.79%Couleur et forme :SolidAdipic acid
CAS :Adipic acid is a precursor for the production of nylon.Formule :C6H10O4Degré de pureté :99.59%Couleur et forme :White Solid CrystallineMasse moléculaire :146.14BPK-29 hydrochloride
CAS :"BPK-29 hydrochloride targets NR0B1, altering C274 and hinders KEAP1-mutant cancer cell growth."Formule :C26H33Cl2N3O3Degré de pureté :99.06%Couleur et forme :SolidMasse moléculaire :506.46Ref: TM-T13586L
5mg34,00€10mg56,00€25mg102,00€50mg180,00€100mg260,00€200mg370,00€1mL*10mM (DMSO)37,00€Trapidil
CAS :Trapidil (Avantrin) is a coronary vasodilator agent.Formule :C10H15N5Degré de pureté :99.42%Couleur et forme :SolidMasse moléculaire :205.26Letaxaban
CAS :Letaxaban (TAK-442) is a small molecule Xa factor inhibitor that can be used to study polar coronary syndromes and thrombotic blockages.Formule :C22H26ClN3O5SDegré de pureté :99.13% - 99.87%Couleur et forme :SolidMasse moléculaire :479.98Dicoumarol
CAS :Dicoumarol: an anticoagulant from moldy sweet-clover, depletes vitamin K, inhibits clotting enzymes.
Formule :C19H12O6Degré de pureté :99.75% - 99.9%Couleur et forme :White Or Creamy White Crystalline Powder SolidMasse moléculaire :336.31-(2-Hydroxyethyl)imidazolidine-2-thione
CAS :1-(2-Hydroxyethyl)imidazolidine-2-thione is used as pharmaceutical intermediates.Formule :C5H10N2OSDegré de pureté :99.63%Couleur et forme :White CrystalMasse moléculaire :146.21Dropropizine
CAS :Dropropizine (UCB-1967), a racemic non-opiate antitussive agent, is served as a cough suppressant.
Formule :C13H20N2O2Degré de pureté :99.38%Couleur et forme :White Or Almost White PowderMasse moléculaire :236.31Nitroxazepine
CAS :Nitroxazepine (CIBA 2330Go), a tricyclic antidepressant, inhibits serotonin and norepinephrine reuptake, used in depression research.Formule :C18H19N3O4Degré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :341.36Ref: TM-T12232
1mg82,00€5mg168,00€10mg293,00€25mg442,00€50mg610,00€100mg827,00€500mg1.603,00€1mL*10mM (DMSO)177,00€Atovaquone
CAS :Atovaquone (Atavaquone) is a hydroxynaphthoquinone that has antimicrobial activity and is being used in antimalarial protocols.Formule :C22H19ClO3Degré de pureté :98% - 99.85%Couleur et forme :Yellow To Orange Crystalline SolidMasse moléculaire :366.84L002
CAS :L002 is a potent inhibitor of acetyltransferase p300 with an IC50 of 1.98 μM, blocking histone and p53 acetylation, and may treat cardiac hypertrophy.Formule :C15H15NO5SDegré de pureté :98.59%Couleur et forme :SolidMasse moléculaire :321.35Xl-281
CAS :XL-281: potent oral RAF kinase inhibitor, effective on wild-type and mutants, reduces tumor growth and cell proliferation, increases apoptosis.Formule :C24H19ClN4O4Degré de pureté :95.77% - 98.83%Couleur et forme :SolidMasse moléculaire :462.895-Fluorouracil
CAS :5-Fluorouracil (5-FU) is a uracil analog, an inhibitor of DNA synthesis.Formule :C4H3FN2O2Degré de pureté :98% - >99.99%Couleur et forme :White To Practically White Crystalline Powder Neoplastic Drug Chemosterilant For Insects (Epa 1998)Masse moléculaire :130.08Chlorpropamide
CAS :Chlorpropamide (Diabinese) is a sulfonylurea hypoglycemic agent used in the treatment of non-insulin-dependent diabetes mellitus not responding to dietaryFormule :C10H13ClN2O3SDegré de pureté :98.90%Couleur et forme :Crystals From Dil Ethanol Physical Description White Crystalline Powder With A Slight Odor (Ntp 1992)Masse moléculaire :276.74Danicamtiv
CAS :Danicamtiv (MYK-491) is an inotropic agent and it also is a selective allosteric activator of cardiac myosin.Formule :C16H20F3N5O4SDegré de pureté :99.38%Couleur et forme :SolidMasse moléculaire :435.42Ref: TM-T15050
1mg136,00€5mg274,00€10mg454,00€25mg750,00€50mg1.026,00€100mg1.406,00€1mL*10mM (DMSO)303,00€BMS-195270
CAS :BMS-195270 is a bio-active chemical.Formule :C15H9ClF3N3O2Degré de pureté :98.7%Couleur et forme :SolidMasse moléculaire :355.7Dinitolmide
CAS :Dinitolmide (Zoalene), a poultry feed additive, is a coccidiostat for poultry.Formule :C8H7N3O5Degré de pureté :97.27%Couleur et forme :Crystals From Dilute AlcoholMasse moléculaire :225.16Phleomycin
CAS :Phleomycin is one of the anticancer glycopeptide antibiotics which cause DNA cleavage.Formule :C48H69N17O20S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :1268.29Sesamin
CAS :Sesamin (Fsesamin) is a lignan extracted from Sesamum indicum L.
Formule :C20H18O6Degré de pureté :99.38% - 99.86%Couleur et forme :White Or Light Yellow Fine PowderMasse moléculaire :354.35Sunitinib
CAS :Sunitinib (SU 11248) is a multi-targeted receptor tyrosine kinase (RTK) inhibitor that inhibits VEGFR2 and PDGFRβ (IC50=80/2 nM).Formule :C22H27FN4O2Degré de pureté :98% - 99.67%Couleur et forme :Yellow SolidMasse moléculaire :398.47Levonorgestrel
CAS :Levonorgestrel (D-Norgestrel) is a Progestin and Progestin-containing Intrauterine Device.Formule :C21H28O2Degré de pureté :99.42% - 99.44%Couleur et forme :Crystals From Methanol SolidMasse moléculaire :312.45Itopride hydrochloride
CAS :Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.Formule :C20H27ClN2O4Degré de pureté :99.59%Couleur et forme :White Or Pale Brownish CrystalMasse moléculaire :394.9(±)-N-3-Benzylnirvanol
CAS :(±)-N-3-Benzylnirvanol is a racemic mixture of (+)-N-3-Benzylnirvanol and (-) -n-3-Benzylnirvanoll.Formule :C18H18N2O2Degré de pureté :98.31%Couleur et forme :SolidMasse moléculaire :294.35Naringin dihydrochalcone
CAS :Naringin dihydrochalcone (Naringin DC) is an inhibitor of CYP enzymes, used as an artificial sweetener.Formule :C27H34O14Degré de pureté :99.07% - 99.73%Couleur et forme :Solid PowderMasse moléculaire :582.55NS-2028
CAS :NS-2028 is a selective sGC inhibitor, affecting both basal and NO-activated activities; used in nitric oxide research.Formule :C9H5BrN2O3Degré de pureté :99.44%Couleur et forme :A Crystalline SolidMasse moléculaire :269.05Ref: TM-T16344
1mg39,00€5mg88,00€10mg143,00€25mg250,00€50mg378,00€100mg543,00€200mg738,00€1mL*10mM (DMSO)87,00€BNC105
CAS :BNC105 is a tubulin polymerization inhibitor. It has potent antiproliferative and tumor vascular disrupting properties.Formule :C20H20O7Degré de pureté :96.57%Couleur et forme :SolidMasse moléculaire :372.37Ref: TM-T14694
1mg79,00€5mg152,00€10mg215,00€25mg351,00€50mg494,00€100mg665,00€200mg893,00€1mL*10mM (DMSO)167,00€LCH-7749944
CAS :LCH-7749944 suppresses human gastric cancer cell growth, induces apoptosis, and inhibits PAK4 with IC50 of 14.93 μM.Formule :C20H22N4O2Degré de pureté :99.48%Couleur et forme :SolidMasse moléculaire :350.41Ref: TM-T11826
1mg50,00€5mg103,00€10mg156,00€25mg269,00€50mg403,00€100mg583,00€200mg785,00€1mL*10mM (DMSO)110,00€Cefpiramide acid
CAS :Cefpiramide acid (Cefpiramidum) is a third-generation cephalosporin antibiotic.Formule :C25H24N8O7S2Degré de pureté :97.40%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :612.64Orphenadrine Citrate
CAS :Orphenadrine Citrate (Flexon) is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.Formule :C18H23NO·C6H8O7Degré de pureté :99.58%Couleur et forme :White SolidMasse moléculaire :461.5Procarbazine hydrochloride
CAS :Procarbazine hydrochloride (NSC-77213 HCl) is the hydrochloride salt of a methylhydrazine derivative with antineoplastic and mutagenic activities.Formule :C12H19N3O·HClDegré de pureté :96.99% - ≥98%Couleur et forme :(Ntp 1992)Masse moléculaire :257.76Lexatumumab
CAS :Lexatumumab (GHS-ETR2), a human antibody, targets TRAILR2 for anticancer effects and apoptosis in mesothelioma.
Degré de pureté :> 95%Couleur et forme :LiquidMasse moléculaire :143.48 kDaTLR1
CAS :TLR1 is a cell-penetrating Toll/IL-1 receptor/resistance (TIR) domain/BB-Loop mimic and inhibits IL-1 receptor-mediated responses.Formule :C18H26N2O2Degré de pureté :98.7%Couleur et forme :SolidMasse moléculaire :302.41Ref: TM-T13932
1mg52,00€5mg116,00€10mg172,00€25mg278,00€50mg371,00€100mg513,00€200mg680,00€1mL*10mM (DMSO)123,00€Vixarelimab
CAS :Vixarelimab (KPL-716) is an anti-OSM antibody that blocks IL-31/OSM signaling, for severe itch and pulmonary fibrosis study.
Degré de pureté :SDS-PAGE:96.2%;SEC-HPLC:97.3%Couleur et forme :LiquidMasse moléculaire :144.99 kDaSalbutamol
CAS :Salbutamol (Albuterol) stimulates beta2-adrenergic receptors in the lungs, thereby activating the enzyme adenylate cyclase that catalyzes the conversion of ATP to cyclic-3', 5'-adenosine monophosphate (cAMP).Formule :C13H21NO3Degré de pureté :91.59% - 99.9%Couleur et forme :White To Off-White Crystalline Solid SolidMasse moléculaire :239.31Ly-295501
CAS :Ly-295501 (ILX-295501) showed antitumor and anticancer activity in human pancreatic cancer xenotransplantation model.Formule :C15H12Cl2N2O4SDegré de pureté :98.23%Couleur et forme :SolidMasse moléculaire :387.24Tilavonemab
CAS :Tilavonemab (ABBV-8E12), a humanized anti-tau antibody, halts tau uptake in neurons and may help with Alzheimer's research.Degré de pureté :95.2% (SDS-PAGE); 96.6% (SEC-HPLC) - 95.2% (SDS-PAGE); 96.6% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :145.73kDa7-O-Methyleriodictyol
CAS :7-O-Methyleriodictyol is a flavanone isolated from Artemisia monosperma and shows biological effects on rat isolated smooth muscles.Formule :C16H14O6Degré de pureté :98.10%Couleur et forme :SolidMasse moléculaire :302.28MMV390048
CAS :MMV390048 is an antimalarial agent and is a representative of a new chemical class of Plasmodium PI4K inhibitor (Kdapp=0.3 μM).Formule :C18H14F3N3O2SDegré de pureté :97.48%Couleur et forme :SolidMasse moléculaire :393.38Ref: TM-T16125
2mg34,00€5mg50,00€10mg77,00€25mg138,00€50mg215,00€100mg330,00€200mg470,00€1mL*10mM (DMSO)55,00€2,3-Dihydrobenzofuranyl-5-acetic acid
CAS :2,3-Dihydro-5-benzofuranacetic Acid is used as Pharmaceutical material and intermeidates.Formule :C10H10O3Degré de pureté :99.6%Couleur et forme :White To Light Yellow Crystal PowderMasse moléculaire :178.18Amorolfine hydrochloride
CAS :Amorolfine hydrochloride (Amorolfine HCl) is an antifungal reagent.Formule :C21H36ClNODegré de pureté :99.05% - >99.99%Couleur et forme :White PowderMasse moléculaire :353.97Luteolin
CAS :Luteolin (Luteolol) belongs to the flavonoid group of natural products and is a Nrf2 inhibitor, PDE inhibitor.Formule :C15H10O6Degré de pureté :96.61% - 99.71%Couleur et forme :SolidMasse moléculaire :286.24Carbadox
CAS :Carbadox, an antibacterial for swine dysentery and growth promotion, is banned in the UK due to carcinogen and mutagen risks.Formule :C11H10N4O4Degré de pureté :98.38% - 99.73%Couleur et forme :Minute Yellow Crystals Yellow CrystalsMasse moléculaire :262.22Hydrocortisone acetate
CAS :Hydrocortisone acetate (Cortisol 21-acetate) is the synthetic acetate salt form of hydrocortisone, a corticosteroid with anti-inflammatory and immunosuppressive
Formule :C23H32O6Degré de pureté :98.89% - 99.22%Couleur et forme :White To Off-White Crystalline PowderMasse moléculaire :404.5Samuraciclib hydrochloride
CAS :Samuraciclib HCl is an oral CDK7 inhibitor (IC50: 41 nM), 45-230x selective over CDK1/2/5/9, inhibiting breast cancer growth (GI50: 0.2-0.3 μM).Formule :C22H31ClN6ODegré de pureté :98.99% - 99.8%Couleur et forme :SolidMasse moléculaire :430.97Ref: TM-T10898
1mg108,00€2mg147,00€5mg222,00€10mg335,00€25mg595,00€50mg847,00€100mg1.153,00€1mL*10mM (DMSO)245,00€Isothiuronium
CAS :Isothiouronium, a functional group, is the acid salt of isothiourea.Formule :C12H25IN2SDegré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :356.31Butamben
CAS :Butamben (Butyl 4-aminobenzoate) is a long-duration local anesthetic used for the treatment of chronic pain.Formule :C11H15NO2Degré de pureté :99.43%Couleur et forme :Crystals From Alc Physical Description Yellow Powder Insoluble In Water (Ntp 1992)Masse moléculaire :193.24Darifenacin hydrobromide
CAS :Darifenacin hydrobromide (UK-88525) is a selective muscarinic receptor antagonist used to treat urinary incontinence and overactive bladder syndrome.Formule :C28H31BrN2O2Degré de pureté :99.75% - >99.99%Couleur et forme :SolidMasse moléculaire :505.45Oxaliplatin
CAS :Oxaliplatin (L-OHP) is a DNA alkylating agent, an inhibitor of DNA synthesis.Formule :C8H14N2O4PtDegré de pureté :97% - 99.93%Couleur et forme :SolidMasse moléculaire :397.29Candesartan
CAS :Candesartan (CV 11974) is an angiotensin II receptor blocker used widely in the therapy of hypertension and heart failure.Formule :C24H20N6O3Degré de pureté :98.3% - 99.55%Couleur et forme :Colorless Solid CrystallineMasse moléculaire :440.47Casanthranol
CAS :Casanthranol: a stimulant laxative from cascara sagrada bark, eases constipation by boosting intestinal muscle contractions.Formule :C21H22O10Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :434.397Rocuronium bromide
CAS :Rocuronium bromide (ORG 9426) is a muscle relaxant or aminosteroid non-depolarizing neuromuscular blocker, which is used to provide skeletal muscle relaxation.Formule :C32H53BrN2O4Degré de pureté :99.77% - >99.99%Couleur et forme :White Or Off-White PowderMasse moléculaire :609.68Octocrylene
CAS :Octocrylene, found in sunscreens and cosmetics, penetrates skin, acting as a photosensitizer to increase free radicals when exposed to light.Formule :C24H27NO2Degré de pureté :99.21%Couleur et forme :Physical Description Yellow Viscous Liquid Insoluble In Water (Ntp 1992)Masse moléculaire :361.48Dibenzosuberol
CAS :Dibenzosuberol is used as a Pharmaceutical intermediate.Formule :C15H14ODegré de pureté :98.73%Couleur et forme :White Fluffy PowderMasse moléculaire :210.27Chlorhexidine
CAS :Chlorhexidine is a biguanide antiseptic targeting bacteria, damaging cell membranes and causing cell death, more effective against gram-positive types.Formule :C22H30Cl2N10Degré de pureté :98% - 99.85%Couleur et forme :Crystals From Methanol SolidMasse moléculaire :505.45Cloxiquine
CAS :Cloxiquine (Dermofongin) is a monohalogenated 8-hydroxyquinoline with activity against bacteria, fungi, and protozoa.Formule :C9H6ClNODegré de pureté :99.82% - 99.87%Couleur et forme :Light Yellow CrystalsMasse moléculaire :179.6p-Ethynylphenylalanine hydrochloride
CAS :p-Ethynylphenylalanine hydrochloride (4-Ethynyl-L-phenylalanine HCL) is a novel, potent and specific inhibitor of TPH[1].Formule :C11H12ClNO2Degré de pureté :99.03%Couleur et forme :SolidMasse moléculaire :225.67Verubulin hydrochloride
CAS :Verubulin hydrochloride (MPC-6827 hydrochloride) is an agent of blood brain barrier permeable microtubule-disrupting, with potent and broad-spectrum cytotoxicFormule :C17H18ClN3ODegré de pureté :98.29% - 99.77%Couleur et forme :SolidMasse moléculaire :315.8Ref: TM-T13298
5mg50,00€10mg78,00€25mg145,00€50mg210,00€100mg300,00€200mg434,00€1mL*10mM (DMSO)56,00€Iminostilbene
CAS :Iminostilbene (Dibenzazepine) (Dibenzazepine) is a chemical precursor of carbamazepine which is used primarily in the treatment of epilepsy and neuropathic painFormule :C14H11NDegré de pureté :98.50%Couleur et forme :Yellow To Brown PowderMasse moléculaire :193.24Miltefosine
CAS :Miltefosine (HePC), effective oral drug for both visceral and cutaneous leishmaniasis, in clinical trials worldwide.Formule :C21H46NO4PDegré de pureté :98% - 99.94%Couleur et forme :White To Off-White PowderMasse moléculaire :407.57NI-42
CAS :NI-42, a BRPFs inhibitor: IC50(BRPF1/2/3)=7.9/48/260 nM, Kd(BRPF1/2/3)=40/210/940 nM; selective for class IV BRDs.Formule :C18H15N3O3SDegré de pureté :99.18%Couleur et forme :SolidMasse moléculaire :353.39Efalizumab
CAS :Efalizumab: humanized monoclonal antibody CD11a; modulates T cell activation/adhesion; for plaque psoriasis, psoriatic arthritis research.Degré de pureté :SDS-PAGE:95% SEC-HPLC:98.77%Couleur et forme :LiquidMasse moléculaire :146.14 kDaBrivudine
CAS :Brivudine (BVDU), an antiviral medicine, is used in the therapy of herpes zoster.Formule :C11H13BrN2O5Degré de pureté :99.51% - 99.85%Couleur et forme :SolidMasse moléculaire :333.14SLU-PP-332
CAS :SLU-PP-332 is a pan-estrogen receptor-related receptor (ERR) agonist with high affinity for ERRα, ERRβ, and ERRγ with EC50 values of 98, 230, and 430 nM,Formule :C18H14N2O2Degré de pureté :97.53% - 98.60%Couleur et forme :SoildMasse moléculaire :290.324-Amino-5-Chloro-2-Methoxybenzoic Acid
CAS :4-Amino-5-Chloro-2-Methoxybenzoic Acid (Metoclopramide EP Impurity C) is a Metoclopramide metabolite.Formule :C8H8ClNO3Degré de pureté :99.78%Couleur et forme :White To Slightly Beige PowderMasse moléculaire :201.61Uracil
CAS :Uracil, a pyrimidine in RNA, pairs with adenine, becomes thymine when methylated, and aids enzyme synthesis.Formule :C4H4N2O2Degré de pureté :99.51% - 99.97%Couleur et forme :Fine Off-White Crystalline PowderMasse moléculaire :112.09Ethisterone
CAS :Ethisterone (17α-Ethynyltestosterone) is a progestogen hormone.Formule :C21H28O2Degré de pureté :97.96% - 99.50%Couleur et forme :Off-White PowderMasse moléculaire :312.45Nacubactam
CAS :Nacubactam (OP0595 free acid) is a potent inhibitor of non-β-lactam-β-lactamase with activity against class A and class C β-lactamases.Formule :C9H16N4O7SDegré de pureté :98.93%Couleur et forme :SolidMasse moléculaire :324.31Ref: TM-T12166
1mg59,00€5mg126,00€10mg207,00€25mg414,00€50mg622,00€100mg885,00€1mL*10mM (DMSO)140,00€Aripiprazole
CAS :Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.Formule :C23H27Cl2N3O2Degré de pureté :99.43% - 99.62%Couleur et forme :Colourless Flake Crystalline SolidMasse moléculaire :448.39Minocycline hydrochloride
CAS :Minocycline HCl: tetracycline antibiotic, treats bacterial infections and acne, may cause acute or chronic hepatitis.Formule :C23H28ClN3O7Degré de pureté :99.28% - >99.99%Couleur et forme :Bright Yellow-Orange Amorphous Solid Crystalline YellowMasse moléculaire :493.94ETC-206
CAS :ETC-206 is a selective inhibitor of MNK1 and MNK2 (IC50s: 64 nM and 86 nM).
Formule :C25H20N4O2Degré de pureté :99.72% - 99.79%Couleur et forme :SolidMasse moléculaire :408.45Mezagitamab
CAS :Mezagitamab (TAK-079) is a fully humanized IgG1λ monoclonal antibody against CD38 with high affinity for cells expressing CD38.Degré de pureté :97.5% (SDS-PAGE); 99.1% (SEC-HPLC) - 97.5% (SDS-PAGE); 99.1% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :144.4 kDaD-AP5
CAS :D-AP5 (D-APV) is a NMDA receptor antagonist.Formule :C5H12NO5PDegré de pureté :98.77% - >99.99%Couleur et forme :White Fine Crystalline PowderMasse moléculaire :197.13Perhexiline maleate
CAS :Perhexiline maleate is an orally active inhibitor of CPT1 and CPT2 that reduces fatty acid metabolism.Formule :C23H39NO4Degré de pureté :99.77% - ≥98%Couleur et forme :SolidMasse moléculaire :393.56Ref: TM-T12408
1mg42,00€2mg52,00€5mg85,00€10mg115,00€25mg202,00€50mg299,00€100mg447,00€200mg610,00€1mL*10mM (DMSO)90,00€Sulfamethazine sodium
CAS :Sulfamethazine sodium (Sulfadimethyldiazine Sodium Salt) salt is a sodium salt form of sulfamethazine, a sulfonamide antibiotic used in the livestock industry.Formule :C12H13N4NaO2SDegré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :300.31BETd-260
CAS :BETd-260, a PROTAC linked by a Cereblon ligand and a BET ligand, has an inhibitory effect on BRD4 protein in leukemic cell lines.Formule :C43H46N10O6Degré de pureté :96.76%Couleur et forme :SolidMasse moléculaire :798.89Diclofenac
CAS :Diclofenac: a nonsteroidal compound inhibiting COX-1 and COX-2, reducing pro-inflammatory prostaglandins.Formule :C14H11Cl2NO2Degré de pureté :99.69% - 99.97%Couleur et forme :Crystals From Ether-Petroleum Ether SolidMasse moléculaire :296.15Elotuzumab
CAS :Elotuzumab targets SLAMF7, activates NK cells, induces cytotoxicity, and treats multiple myeloma with lenalidomide and dexamethasone.
Degré de pureté :SDS-PAGE:97.4%;SEC-HPLC:98.1%Couleur et forme :LiquidMasse moléculaire :145.4 kDaAzatadine dimaleate
CAS :Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).
Formule :C28H30N2O8Degré de pureté :99.7% - >99.99%Couleur et forme :PowderMasse moléculaire :522.55(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid
CAS :(1R,5S,6r)-N-(2-methyl-1-((3-methylpyridin-2-yl)oxy)propan-2-yl)-3-azabicyclo[3.1.0]hexane-6-carboxamide L(+)-Tartaric acid is a potential SSTR4 agonist.Formule :C20H29N3O8Degré de pureté :99.72%Couleur et forme :SoildMasse moléculaire :439.46Relatlimab
CAS :Relatlimab (BMS-986016), a monoclonal antibody, blocks LAG-3/MHC II and LAG-3/FGL1, treating advanced melanoma with Nivolumab.
Degré de pureté :SDS-PAGE:96.8%;SEC-HPLC:97.2%Couleur et forme :LiquidMasse moléculaire :145.2 kDaCyproheptadine hydrochloride sesquihydrate
CAS :Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.Formule :C21H24ClNODegré de pureté :99.77% - >99.99%Couleur et forme :White To Slightly Yellowish Crystalline SolidMasse moléculaire :341.88UK-124114
CAS :Selamectin, a derivative of ivermectin, is a macrocyclic lactone that enhances chloride channels in nematodes, inhibiting H. contortus larval growth.Formule :C43H63NO11Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :769.96Itraconazole
CAS :Itraconazole (R51211) is a triazole antifungal agent that inhibits cytochrome P-450-dependent enzymes required for ERGOSTEROL synthesis.Formule :C35H38Cl2N8O4Degré de pureté :98% - 99.90%Couleur et forme :Off-White Crystalline SolidMasse moléculaire :705.63Axatilimab
CAS :Axatilimab (SNDX-6352) is a human IgG4 antibody that targets CSF-1R and can be used to study immune system diseases and respiratory diseases.Degré de pureté :97.9% (SDS-PAGE); 97% (SEC-HPLC) - 97.9% (SDS-PAGE); 97% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :147.17 kDaDC-05
CAS :DC-05 is an inhibitor of DNA methyltransferase 1 (DNMT1) (IC50 and a Kd: 10.3 μM and 1.09 μM, respectively).
Formule :C25H25N3ODegré de pureté :98.95%Couleur et forme :SolidMasse moléculaire :383.49Prilocaine hydrochloride
CAS :Prilocaine HCl: local amino amide anesthetic, blocks voltage-gated sodium channels in neurons, inhibits Na+ permeability.Formule :C13H21ClN2ODegré de pureté :99.97%Couleur et forme :Needles White Or Off White Crystalline PowderMasse moléculaire :256.77Cholesteryl Acetate
CAS :Cholesteryl Acetate is a cholesterol ester obtained from the esterification of the hydroxyl group of cholesterol with acetic acid.Formule :C29H48O2Degré de pureté :99.94%Couleur et forme :SolidMasse moléculaire :428.69Imipenem monohydrate
CAS :Imipenem monohydrate (Imipenem) is a β lactam antibiotic. Imipenem monohydrate acts on the bacterial cell wall. Cost-effective and quality-assured.Formule :C12H19N3O5SDegré de pureté :98.77% - 99.94%Couleur et forme :Off-White Nonhygroscopic CrytalsMasse moléculaire :317.36Elezanumab
CAS :Elezanumab (ABT-555) is a human anti-RGMa antibody blocking BMP signaling via SMAD1/5/8; IC50 ~97 pM. It aids neuroregeneration and repairs neuronal damage.Degré de pureté :SDS-PAGE:97.4%;SEC-HPLC:98.7%Couleur et forme :LiquidMasse moléculaire :143.43 kDaToltrazuril
CAS :Toltrazuril (Toltrazurilo), an antiprotozoal agent, has effect on Coccidia parasites.Formule :C18H14F3N3O4SDegré de pureté :99.32%Couleur et forme :PowderMasse moléculaire :425.38Ordesekimab
CAS :Ordesekimab (AMG 714) is a human anti-IL-15 IgG1 κ monoclonal antibody for studying NRCD.Degré de pureté :> 95%Couleur et forme :LiquidMasse moléculaire :145.12 kDaTroxerutin
CAS :Troxerutin (Trihydroxyethylrutin), a natural bioflavonoid, is isolated from Sophora japonica. It has many benefits and medicinal properties.Formule :C33H42O19Degré de pureté :98.28% - 99.24%Couleur et forme :Light Yellow PowderMasse moléculaire :742.68Thymol methyl ether
CAS :Thymol methyl ether is a volatile substance present in the rhizomes of Arnica with potential antibacterial and anticancer antioxidant activity.Formule :C11H16ODegré de pureté :99.79%Couleur et forme :SolidMasse moléculaire :164.24Nefopam hydrochloride
CAS :Nefopam hydrochloride (Nefopam HCl) is the hydrochloride salt form of nefopam, a centrally-acting, non-opioid benzoxazocine with analgesic activity.Formule :C17H20ClNODegré de pureté :99.32% - 99.85%Couleur et forme :SolidMasse moléculaire :289.8(R)-Ketorolac
CAS :(R)-Ketorolac ((+)-Ketorolac) is the R-enantiomer of Ketorolac, with potent analgesic activity.
Formule :C15H13NO3Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :255.27Cinepazide maleate
CAS :Cinepazide maleate (MD-67350), a maleate salt form of cinepazide, is a vasodilator.
Formule :C22H31N3O5·C4H4O4Degré de pureté :99.9% - 99.97%Couleur et forme :White Or Off-White Crystalline PowderMasse moléculaire :533.57Tisotumab
CAS :Tisotumab (Anti-Human F3 Recombinant Antibody) is a human IgG1 monoclonal antibody against tissue factor (TF).Degré de pureté :SDS-PAGE:95% SEC-HPLC:99.08%Couleur et forme :LiquidMasse moléculaire :144.66 kDaAQ-13 dihydrochloride
CAS :AQ-13 dihydrochloride is an antimalarial drug. It is effective against drug-resistant strains of Plasmodium falciparum.Formule :C16H24Cl3N3Degré de pureté :99.81%Couleur et forme :SolidMasse moléculaire :364.74Ref: TM-T10356
1mg34,00€5mg71,00€10mg104,00€25mg203,00€50mg304,00€100mg434,00€500mg945,00€1mL*10mM (DMSO)79,00€(3aR,9aR)-Fluparoxan
CAS :(3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmentalFormule :C10H10FNO2Degré de pureté :97.82%Couleur et forme :SoildMasse moléculaire :195.199-Cyclopentyladenine
CAS :9-Cyclopentyladenine (NSC-19486) is an adenylate cyclase inhibitor that blocks cellular morphological differentiation and phosphorylation of specific signalingFormule :C10H13N5Degré de pureté :99.98%Couleur et forme :SolidMasse moléculaire :203.24Sophocarpine monohydrate
CAS :Sophocarpine monohydrate, a major ingredient of Sophora alopecuroides, has a wide range of pharmacological effects.Formule :C15H22N2ODegré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :246.35Nitazoxanide
CAS :Nitazoxanide (NSC-697855) is a synthetic benzamide antiprotozoal; it disrupts pyruvate electron transfer reactions.Formule :C12H9N3O5SDegré de pureté :99% - 99.93%Couleur et forme :SolidMasse moléculaire :307.28Miconazole
CAS :Miconazole (R18134) is an imidazole antifungal agent that is used topically and by intravenous infusion.Formule :C18H14Cl4N2ODegré de pureté :98% - 99.89%Couleur et forme :SolidMasse moléculaire :416.13(R)-Elagolix
CAS :(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing hormone receptor.Formule :C32H30F5N3O5Degré de pureté :99.08%Couleur et forme :SolidMasse moléculaire :631.59Ref: TM-T11174
5mg50,00€10mg75,00€25mg137,00€50mg195,00€100mg306,00€200mg452,00€1mL*10mM (DMSO)70,00€Asenapine Maleate
CAS :Asenapine Maleate (Org 5222 maleate) is a second generation (atypical) antipsychotic agent that is taken sublingually.Formule :C21H20ClNO5Degré de pureté :99.28%Couleur et forme :SolidMasse moléculaire :401.84MRTX-1257
CAS :MRTX-1257: selective, irreversible KRAS G12C inhibitor; IC50 of 900 pM; 31% bioavailable in mice; 77% target engagement.Formule :C33H39N7O2Degré de pureté :97.3% - 99.07%Couleur et forme :SolidMasse moléculaire :565.71Ref: TM-T16143
1mg64,00€2mg89,00€5mg131,00€10mg207,00€25mg371,00€50mg540,00€100mg785,00€200mgÀ demander1mL*10mM (DMSO)170,00€Tranexamic acid
CAS :Tranexamic acid (Amstat) is an Antifibrinolytic Agent. The physiologic effect of tranexamic acid is by means of Decreased Fibrinolysis.Formule :C8H15NO2Degré de pureté :99.64% - 99.79%Couleur et forme :White Crystalline PowderMasse moléculaire :157.21SLC26A3-IN-1
CAS :"SLC26A3-IN-1 inhibits SLC26A3, an anion transporter linked to diarrhea, with 340 nM IC50."Formule :C23H18O4Degré de pureté :99.02%Couleur et forme :SolidMasse moléculaire :358.39TBK1/IKKε-IN-2
CAS :TBK1/IKKε-IN-2 is a dual inhibitor of TBK1 and IKKε.Formule :C26H27N5O3Degré de pureté :98.89%Couleur et forme :SolidMasse moléculaire :457.52Ref: TM-T15559
1mg87,00€5mg178,00€10mg289,00€25mg462,00€50mg625,00€100mg802,00€1mL*10mM (DMSO)178,00€Burfiralimab
CAS :Burfiralimab (hzVSF-v13) is a monoclonal immunoglobulin (IgG4) directed against waveform proteins and can be used to study rheumatoid arthritis.Degré de pureté :90%Couleur et forme :LiquidMasse moléculaire :144.6 kDaSarizotan 2HCl
CAS :Sarizotan 2HCl is an hERG channel inhibitor and 5-hydroxytryptamine 5-HT1A receptor agonist with potential antidepressant effects for the study of Parkinsonian movement disorders.Formule :C22H23Cl2FN2ODegré de pureté :98.83%Couleur et forme :SoildMasse moléculaire :421.34Picenadol
CAS :Picenadol (LY 150720) is a racemic mixture of N-methyl-4-phenylpiperidine derivatives with agonist-antagonist opioid properties.Picenadol has central analgesicFormule :C16H25NODegré de pureté :97.10%Couleur et forme :SolidMasse moléculaire :247.38GW-870086
CAS :GW-870086 is an effective anti-inflammatory agent.Formule :C31H39F2NO6Degré de pureté :99.86%Couleur et forme :SolidMasse moléculaire :559.64Ref: TM-T15451
2mg33,00€5mg50,00€10mg75,00€25mg111,00€50mg198,00€100mg296,00€200mg427,00€1mL*10mM (DMSO)60,00€Olsalazine disodium
CAS :Olsalazine disodium (Dipentum) is bioconverted to 5-aminosalicylic acid (5-ASA) in the colon and has anti-inflammatory activity in ulcerative colitis.Formule :C14H8N2Na2O6Degré de pureté :99.47% - 99.52%Couleur et forme :Yellow Crystalline PowderMasse moléculaire :346.2CP-809101 hydrochloride
CAS :CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).Formule :C15H18Cl2N4ODegré de pureté :99.5%Couleur et forme :SolidMasse moléculaire :341.24Zinc pyrithione
CAS :Zinc pyrithione (OM-1563), an antibacterial and antifungal agent can disrupt membrane transport by blocking the proton pump.Formule :C10H8N2O2S2ZnDegré de pureté :99.09% - 99.47%Couleur et forme :Off-White To Tan PowderMasse moléculaire :317.71DHPG
CAS :DHPG is a potent Group I mGluR agonist; doesn't affect Group II/III; linked to phospholipase D.Formule :C8H9NO4Degré de pureté :99.55%Couleur et forme :SolidMasse moléculaire :183.16Bezafibrate
CAS :Bezafibrate (BM15075) is an antilipemic agent that lowers CHOLESTEROL and TRIGLYCERIDES.Formule :C19H20ClNO4Degré de pureté :99.56% - 99.82%Couleur et forme :SolidMasse moléculaire :361.82(R)-BI-2852
CAS :(R)-5-hydroxy isoindolin-1-one is an RAS protein inhibitor with antiproliferative and antitumor properties.Formule :C31H28N6O2Degré de pureté :97.80%Couleur et forme :SoildMasse moléculaire :516.59ART558
CAS :ART558 is a potent, selective, low molecular weight, allosteric DNA polymerase activity of Polθ inhibitor (IC50=7.9 nM).Formule :C21H21F3N4O2Degré de pureté :99.18% - 99.67%Couleur et forme :SolidMasse moléculaire :418.41Fludazonium chloride
CAS :Fludazonium chloride (NSC-351149) is an antifungal agent.Formule :C26H20Cl5FN2O2Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :588.71Ref: TM-T12264
1mg215,00€5mg430,00€10mg587,00€25mg892,00€50mg1.198,00€100mg1.575,00€200mg2.133,00€1mL*10mM (DMSO)532,00€Hydroquinidine
CAS :Hydroquinidine ((+)-Hydroquinidine) is an organic compound, used as an antiarrhythmic agent.Formule :C20H26N2O2Degré de pureté :98.61% - 99.68%Couleur et forme :SolidMasse moléculaire :326.43(E)-Cardamonin
CAS :(E)-Cardamonin (Alpinetin chalcone) is a chalconoid that has been isolated from several plants including Alpinia katsumadai and Alpinia conchigera.Formule :C16H14O4Degré de pureté :99.07% - 99.84%Couleur et forme :SolidMasse moléculaire :270.28Spartalizumab
CAS :"Spartalizumab (PDR001), a humanized IgG4 monoclonal antibody, targets PD-1 to inhibit PD-L1/L2 interactions, useful in ATC research."Degré de pureté :SDS-PAGE:95.2%;SEC-HPLC:96.3%Couleur et forme :LiquidMasse moléculaire :145.74 kDaBMVC-8C3O
CAS :BMVC-8C3O is a DNA G-quadruplex (G4) ligand.Cost-effective and quality-assured.Formule :C42H53I3N4O3Degré de pureté :99.72%Couleur et forme :SolidMasse moléculaire :1042.61Ref: TM-T13584
1mg101,00€5mg192,00€10mg285,00€25mg462,00€50mg623,00€100mg858,00€200mg1.153,00€1mL*10mM (DMSO)371,00€NVP-2
CAS :NVP-2 selectively inhibits CDK9 (IC50: 0.514 nM), prompts apoptosis, and affects other CDKs (IC50: 0.584-0.706 μM).Formule :C27H37ClN6O2Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :513.07Ref: TM-T16363
1mg52,00€2mg74,00€5mg113,00€10mg192,00€25mg416,00€50mg615,00€100mg875,00€1mL*10mM (DMSO)128,00€Voriconazole
CAS :Voriconazole (UK-109496) is a triazole antifungal agent that specifically inhibits STEROL 14-ALPHA-DEMETHYLASE and CYTOCHROME P-450 CYP3A.Formule :C16H14F3N5ODegré de pureté :98% - 99.91%Couleur et forme :White To Off White Crystalline PowderMasse moléculaire :349.31Ref: TM-T0120
10mg35,00€25mg55,00€50mg78,00€100mg110,00€200mg158,00€500mg253,00€1mL*10mM (DMSO)40,00€INCB-9471
CAS :INCB-9471 is a CCR5 antagonist with anti-HIV activity and inhibits the interaction between HIV-1 gp120.Formule :C30H40F3N5O2Degré de pureté :98.80%Couleur et forme :SolidMasse moléculaire :559.666Mebhydrolin napadisylate
CAS :Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergicFormule :C19H20N2C10H8O6S2Degré de pureté :99.35% - 99.96%Couleur et forme :White Or Almost White CrystallineMasse moléculaire :420.52O-Desmethyl gefitinib
CAS :O-Desmethyl gefitinib is an active EGFR inhibitor (IC50: 36 nM), a metabolite of Gefitinib, formed by CYP2D6.Formule :C21H22ClFN4O3Degré de pureté :97.17%Couleur et forme :SolidMasse moléculaire :432.88Ref: TM-T16369
1mg52,00€5mg105,00€10mg167,00€25mg324,00€50mg518,00€100mg742,00€1mL*10mM (DMSO)114,00€Sacituzumab
CAS :Sacituzumab is an IgG1 monoclonal antibody, a naked antibody to Sacituzumab govitecan, with potential anti-tumor activity for the study of tumors.Degré de pureté :95% - >95.3% (SEC-HPLC); 96.7% (SDS-PAGE)Couleur et forme :LiquidMasse moléculaire :145.51 kDaAmylase
CAS :Amylase (Diastase) is any one of a group of enzymes which catalyses the breakdown of starch into maltose.Formule :NADegré de pureté :98%Couleur et forme :SolidMasse moléculaire :N/AAmifostine
CAS :Amifostine (Ethyol) anhydrous is a cytoprotective agent, acts as a free radical scavenging activity.Formule :C5H15N2O3PSDegré de pureté :99.59%Couleur et forme :White SolidMasse moléculaire :214.225-TAMRA-SE
CAS :5-TAMRA-SE binds amines, gives stable orange-red fluorescence, exc/em ~546/579nm, pH-insensitive.Formule :C29H25N3O7Degré de pureté :97.96%Couleur et forme :SolidMasse moléculaire :527.53Loxoribine
CAS :Loxoribine (RWJ 21757), a guanosine analog, is an oral TLR7 agonist with antiviral and antitumor properties.Formule :C13H17N5O6Degré de pureté :99.11%Couleur et forme :SolidMasse moléculaire :339.3CMS-121
CAS :CMS-121, a quinolone derivative, is an orally active acetyl-CoA carboxylase 1 (ACC1) inhibitor.Formule :C20H19NO3Degré de pureté :98.71%Couleur et forme :SolidMasse moléculaire :321.37Utomilumab
CAS :Utomilumab, a humanized IgG2 against T-cell receptor 4-1BB/CD137, shows antitumor effects in advanced cancers.Formule :C17H24N8O3Degré de pureté :95% - 95.1% (SDS-PAGE); 98.5% (SEC-HPLC)Couleur et forme :LiquidMasse moléculaire :142.77 kDaTK216
CAS :TK216 is a potent inhibitor of E26 transformation-specific (ETS) with anticancer activity.Formule :C19H15Cl2NO3Degré de pureté :97.22%Couleur et forme :SolidMasse moléculaire :376.23Fluorothyl
CAS :Fluorothyl (Bis(2,2,2-trifluoroethyl) ether) is a convulsant used in experimental animals.Formule :C4H4F6ODegré de pureté :98%Couleur et forme :Clear Colorless LiquidMasse moléculaire :182.06KGA-2727
CAS :KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity over SGLT2 for diabetes treatment.Formule :C26H40N4O8Degré de pureté :98.46%Couleur et forme :SolidMasse moléculaire :536.62Ref: TM-T15656
1mg109,00€2mg158,00€5mg260,00€10mg430,00€25mg710,00€50mg973,00€100mg1.333,00€1mL*10mM (DMSO)305,00€DPTN dihydrochloride
CAS :DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.Formule :C22H20Cl2N4OSDegré de pureté :99.95%Couleur et forme :SoildMasse moléculaire :459.39Dasatinib
CAS :Dasatinib (BMS-354825) is a tyrosine kinase inhibitor that inhibits Src and Bcr-Abl (Ki=16/30 pM) and is orally active and ATP-competitive.Formule :C22H26ClN7O2SDegré de pureté :99.59% - 99.86%Couleur et forme :Pale-Yellow SolidMasse moléculaire :488.01L-Arabinopyranose
CAS :L-Arabinopyranose (Pectinose) is an aldopentose, including an aldehyde (CHO) functional group.
Formule :C5H10O5Degré de pureté :99.86% - 99.91%Couleur et forme :White To Off White Crystalline PowderMasse moléculaire :150.13KPLH1130
CAS :KPLH1130, a PDK inhibitor, boosts glucose tolerance and reduces inflammation in high-fat diet mice.
Formule :C15H13N3O3Degré de pureté :99.07%Couleur et forme :SolidMasse moléculaire :283.28Bambuterol hydrochloride
CAS :Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.Formule :C18H30ClN3O5Degré de pureté :99.53% - 99.61%Couleur et forme :White SolidMasse moléculaire :403.91Isosulfan blue
CAS :Isosulfan blue, a blue dye used in lymphangiography and sentinel node biopsies, may cause allergies.Formule :C27H31N2NaO6S2Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :566.66Ref: TM-T15598
2mg35,00€5mg50,00€10mg74,00€25mg137,00€50mg190,00€100mg265,00€200mg376,00€1mL*10mM (DMSO)63,00€

