Inhibiteurs
Les inhibiteurs sont des molécules qui se lient aux enzymes, récepteurs ou autres protéines pour réduire ou bloquer leur activité biologique. Ces composés sont largement utilisés en recherche pour étudier les voies biologiques, comprendre les mécanismes des maladies et développer des médicaments thérapeutiques. Les inhibiteurs jouent un rôle crucial dans le traitement de diverses maladies, y compris le cancer, les maladies cardiovasculaires et les infections. Chez CymitQuimica, nous offrons une large gamme d'inhibiteurs de haute qualité pour soutenir vos recherches en biochimie, biologie cellulaire et développement pharmaceutique.
Sous-catégories appartenant à la catégorie "Inhibiteurs"
- Angiogenèse(2.763 produits)
- Apoptose(6.205 produits)
- Cycle cellulaire/point de contrôle(4.812 produits)
- Chromatine/Épigénétique(2.553 produits)
- Signalisation du cytosquelette(1.520 produits)
- Altération de l'ADN/réparation de l'ADN(2.906 produits)
- Endocrinologie/Hormones(3.703 produits)
- Enzyme(3.671 produits)
- GPCR/G-Protéine(8.965 produits)
- Immunologie et Inflammation(3.749 produits)
- Virus de la grippe(297 produits)
- Signalisation JAK/STAT(414 produits)
- Signalisation MAPK(1.244 produits)
- Transporteur membranaire/Canal ionique(3.118 produits)
- Métabolisme(10.123 produits)
- Microbiologie/Virologie(7.569 produits)
- Neuroscience(10.314 produits)
- Autres inhibiteurs(35.804 produits)
- Oxydation-Réduction(40 produits)
- Signalisation PI3K/Akt/mTOR(1.411 produits)
- Protéases/Protéasome(1.681 produits)
- Cellules souche et Dérivés(752 produits)
- Tyrosine Kinase/Adaptateurs(1.947 produits)
- Ubiquitination(1.716 produits)
Affichez 16 plus de sous-catégories
66604 produits trouvés pour "Inhibiteurs"
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GSK256066 Trifluoroacetate
CAS :GSK 256066 Trifluoroacetate: selective PDE4 inhibitor, IC50: 3.2 pM for PDE4B, treats COPD.Formule :C29H27F3N4O7SCouleur et forme :SolidMasse moléculaire :632.61TCH-165
CAS :TCH-165 boosts 20S proteasome levels, enhancing IDP breakdown.Formule :C39H37N3O3Degré de pureté :98.2% - 98.75%Couleur et forme :SolidMasse moléculaire :595.73Ref: TM-T17011
1mg71,00€5mg152,00€10mg236,00€25mg432,00€50mg647,00€100mg888,00€200mg1.198,00€1mL*10mM (DMSO)193,00€Picotamide
CAS :Picotamide has anticoagulant and fibrinolytic properties.Formule :C21H20N4O3Degré de pureté :98.90%Couleur et forme :SolidMasse moléculaire :376.41Ref: TM-T9153
1mg38,00€5mg92,00€10mg147,00€25mg241,00€50mg349,00€100mg479,00€200mg657,00€1mL*10mM (DMSO)94,00€Nonapeptide-1
CAS :Nonapeptide-1 (Melanostatine™ 5) can inhibit the synthesis of melanin, which makes it of interest for treating certain skin conditions.Formule :C61H87N15O9SDegré de pureté :100%Couleur et forme :SolidMasse moléculaire :1206.5PUMA BH3 Free base
PUMA BH3 acetate (PUMA BH3 Free base) is a p53 positive regulator of apoptosis (PUMA) BH3 domain polypeptide that acts as a direct activator of Bak with a Kd ofFormule :C130H206N42O45SDegré de pureté :96.64%Couleur et forme :SolidMasse moléculaire :3109.35Esomeprazole potassium salt
CAS :Esomeprazole potassium, a potent oral proton pump inhibitor, curbs acid secretion in stomach cells, aiding GERD research.Formule :C17H18KN3O3SCouleur et forme :SolidMasse moléculaire :383.51TRAM-34
CAS :TRAM-34 (Triarylmethane-34), an effective and specific inhibitor of the intermediate-conductance Ca2+-activated K+ channel, does not block cytochrome P450.
Formule :C22H17ClN2Degré de pureté :99.01% - 99.91%Couleur et forme :SolidMasse moléculaire :344.84LP-935509
CAS :LP-935509 is a selective, brain-permeable, small molecule competitive inhibitor of articulin-2-associated kinase 1 (AAK1).Cost-effective and quality-assured.Formule :C20H24N6O3Degré de pureté :98.34% - 99.64%Couleur et forme :SolidMasse moléculaire :396.44Ref: TM-T15781
1mg39,00€2mg51,00€5mg84,00€10mg131,00€25mg251,00€50mg469,00€100mg683,00€1mL*10mM (DMSO)92,00€Uridine-5'-diphosphate disodium salt
CAS :UDP disodium salt is a P2Y6 agonist (EC50 = 13 nM), enhances inflammation, phagocytosis, vasoconstriction, and inhibits P2Y14.Formule :C9H12N2Na2O12P2Degré de pureté :98.76% - >99.99%Couleur et forme :White Fine CrystalsMasse moléculaire :448.12HSL-IN-3
CAS :HSL-IN-3 (HSL inhibitor 3) is a boronic acid derivative that is an inhibitor of hormone-sensitive lipase(HSL).Formule :C14H19BO4Degré de pureté :99.402%Couleur et forme :SolidMasse moléculaire :262.11Neurokinin A
CAS :Neurokinin A (NKA), formerly known as Substance K, is a neurologically active peptide translated from the pre-protachykinin gene.Formule :C50H80N14O14SDegré de pureté :>99.99%Couleur et forme :White To Off-White Lyophilized SolidMasse moléculaire :1133.32TRV-120027 acetate (1234510-46-3 free base)
CAS :TRV-120027 acetate: a β-arrestin-1-biased AT1 receptor agonist that inhibits G-protein signaling.Formule :C45H71N13O12Degré de pureté :99.34%Couleur et forme :SolidMasse moléculaire :986.14Echinacoside
CAS :Echinacoside: a polyphenol with anti-inflammatory, antioxidant, liver and nerve protection, NO scavenging, and vasodilation properties.Formule :C35H46O20Degré de pureté :99.59% - >99.99%Couleur et forme :White CrystalMasse moléculaire :786.73Ref: TM-T1716
5mg44,00€10mg55,00€25mg86,00€50mg111,00€100mg160,00€200mg227,00€500mg375,00€1mL*10mM (DMSO)66,00€Rosiglitazone potassium
CAS :Rosiglitazone (BRL 49653) is an oral PPARγ agonist (EC50: 60 nM), TRPC5 activator (EC50: 30 μM), and TRPM3 inhibitor, used in obesity and diabetes research.Formule :C18H18KN3O3SCouleur et forme :SolidMasse moléculaire :395.52Galanthamine
CAS :Galanthamine (Galantamine) is an acetylcholinesterase (AChE)inhibitor(IC50 : 500 nM), can reduce brain damage induced by hypoxia-ischemia.Formule :C17H21NO3Degré de pureté :98.03% - 99.87%Couleur et forme :Off-White SolidMasse moléculaire :287.35Rebaudioside A
CAS :Rebaudioside A (Reb A) is a novel agent of glycoside clathration of pharmacons, acts as α-glucosidase inhibitor.Formule :C44H70O23Degré de pureté :98.79% - 99.93%Couleur et forme :SolidMasse moléculaire :967.01Gadopentetic acid
CAS :Gadopentetic acid (Gd-DTPA), a gadolinium complex, is a paramagnetic MRI contrast agent used in bolus i.v. injections for DCE-MRI.Formule :C14H20GdN3O10Degré de pureté :98%Couleur et forme :White Crystalline PowderMasse moléculaire :547.57RU 24969 free base
CAS :RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.
Formule :C14H16N2ODegré de pureté :97.38%Couleur et forme :SolidMasse moléculaire :228.29SGX-523
CAS :SGX-523 is a selective Met inhibitor (IC50: 4 nM), no inhibitory to Abl, BRAFV599E, p38α, and c-Raf.
Formule :C18H13N7SDegré de pureté :99% - >99.99%Couleur et forme :SolidMasse moléculaire :359.41Isoeugenol
CAS :Isoeugenol (4-Propenylguaiacol), an essential oil constituent of nutmeg, clove, and cinnamon, shows antimicrobial activity.Formule :C10H12O2Degré de pureté :99.94%Couleur et forme :Oily Liquid; Easily Becomes Somewhat Yellow G / Cm3 °Ccurs In Ylang-Ylang Oil And Other Essential OilsMasse moléculaire :164.20Glycyl-L-valine
CAS :Glycyl-L-valine is a dipeptide composed of glycine and valine. It is an incomplete breakdown product of protein digestion or protein catabolism.Formule :C7H14N2O3Degré de pureté :≥95%Couleur et forme :SolidMasse moléculaire :174.2Tubastatin A Hydrochloride
CAS :Tubastatin A Hydrochloride (TSA HCl) is an effective and specific HDAC6 inhibitor (IC50: 15 nM).
Formule :C20H21N3O2·HClDegré de pureté :97.24% - 99.15%Couleur et forme :SolidMasse moléculaire :371.86CTCE 9908 acetate
CTCE 9908 acetate is an antagonist of CXCR4 and inhibits migration in CXCR4-expressing ovarian cancer cells.Formule :C88H151N27O25Degré de pureté :98.47%Couleur et forme :SolidMasse moléculaire :1987.31GSK591
CAS :GSK591 (GSK3203591), Alternative Names are EPZ015866, GSK3203591, is a potent selective inhibitor of the arginine methyltransferase PRMT5 (IC50=11 nM).Formule :C22H28N4O2Degré de pureté :99.35% - 99.45%Couleur et forme :SolidMasse moléculaire :380.48Ref: TM-T6853
1mg46,00€2mg58,00€5mg95,00€10mg137,00€25mg268,00€50mg404,00€100mg567,00€1mL*10mM (DMSO)101,00€Moexipril
CAS :Moexipril is an oral ACE inhibitor, lipid-soluble, targets plasma/tissue ACE, and is used for cardiovascular research.Formule :C27H34N2O7Couleur et forme :SolidMasse moléculaire :498.57Methyl 2-(1H-indol-3-yl)acetate
CAS :Methyl indole-3-acetate, in apples, is isolated from seeds of peas, Vicia, soybeans, and beans.Formule :C11H11NO2Degré de pureté :98.13%Couleur et forme :White To Yellow PowderMasse moléculaire :189.21N-terminally acetylated Leu-enkephalin
Leu-enkephalin, an endogenous 5-amino acid peptide, activates opioid receptors; its acetylated form exists.Formule :C30H39N5O8Degré de pureté :>99.99%Couleur et forme :SolidMasse moléculaire :597.66Cadazolid
CAS :Cadazolid (ACT-179811) is an oxazolidinone-type antibiotic, with activity against gram-positive bacteria, including Clostridium difficile.Formule :C29H29F2N3O8Degré de pureté :98.1% - 99.9%Couleur et forme :SolidMasse moléculaire :585.55BMS-1166
CAS :BMS-1166 is a potent PD-1/PD-L1 interaction inhibitor.
Formule :C36H33ClN2O7Degré de pureté :99.22%Couleur et forme :SolidMasse moléculaire :641.11SQ22536
CAS :SQ22536, a tetrahydrofuryl adenosine analogue, inhibits adenylate cyclase in catfish and rat hepatocytes non-competitively.Formule :C9H11N5ODegré de pureté :99.18%Couleur et forme :Off-White SolidMasse moléculaire :205.22Ref: TM-T2172
2mg35,00€5mg51,00€10mg79,00€25mg160,00€50mg274,00€100mg411,00€200mg615,00€1mL*10mM (DMSO)57,00€Dymanthine
CAS :Dymanthine (ADMA 18) is an agent of veterinary anthelmintic.Formule :C20H43NDegré de pureté :99.85%Couleur et forme :Colorless To White Solid Or Semi-Solid Or LiquidMasse moléculaire :297.56Apitolisib
CAS :Apitolisib (RG 7422) is a PI3K inhibitor, used in cancer trials, targeting PI3Kα, β, δ, γ (IC50= 5, 27, 7, 14 nM).Formule :C23H30N8O3SDegré de pureté :98.28% - 99.64%Couleur et forme :SolidMasse moléculaire :498.6SSAA09E3
CAS :SSAA09E3 is a novel inhibitor of SARS-CoV replication, acting by preventing fusion of the viral membrane with the host cellular membrane.Formule :C21H13NO3Degré de pureté :99.59%Couleur et forme :SolidMasse moléculaire :327.33NSC 185058
CAS :NSC 185058 is an inhibitor of ATG4B, a major cysteine protease. It also can attenuate the autophagic activity.Formule :C11H9N3SDegré de pureté :99.27%Couleur et forme :SolidMasse moléculaire :215.271-Undecanol
CAS :1-Undecanol (1-Hendecanol) is a natural product in many foods such as fruits, butter, eggs and cooked pork, is used as a flavoring ingredient.Formule :C11H24ODegré de pureté :98%Couleur et forme :Colourless LiquidMasse moléculaire :172.31NB-598 Maleate
CAS :NB-598 Maleate is a competitive squalene epoxidase (SE) inhibitor.Formule :C31H35NO5S2Degré de pureté :98%Couleur et forme :SolidMasse moléculaire :565.74Org 25543
CAS :Org 25543 is the development of an N-Acyl amino acid that selectively inhibits the glycine transporter 2 to produce analgesia in a rat model of chronic pain.Formule :C24H32N2O4Degré de pureté :99.13%Couleur et forme :SolidMasse moléculaire :412.52Ref: TM-T50082
1mg55,00€5mg114,00€10mg170,00€25mg274,00€50mg371,00€100mg522,00€200mg687,00€1mL*10mM (DMSO)129,00€Acetylshikonin
CAS :Acetylshikonin, an AChE inhibitor and a non-selective cytochrome P450 inhibitor, is derived from Comfrey and has anticancer and anti-inflammatory properties.Formule :C18H18O6Degré de pureté :92.45% - 99.74%Couleur et forme :SolidMasse moléculaire :330.33Ref: TM-T5S2343
1mg42,00€5mg88,00€10mg135,00€25mg255,00€50mg378,00€100mg560,00€500mg1.216,00€1mL*10mM (DMSO)88,00€Succinic acid
CAS :Succinic acid (1, 2-ethanedicarboxylic acid) is a product of anaerobic metabolism and an intermediate of the tricarboxylic acid cycle. High-Quality, Low-Cost!Formule :C4H6O4Degré de pureté :99.55%Couleur et forme :Solid CrystallineMasse moléculaire :118.09Ac-RYYRIK-NH2 acetate
Ac-RYYRIK-NH2 acetate is an agonist at nociceptin/orphanin FQ(noc/OFQ) receptors, affecting spontaneous locomotor activity.Formule :C46H74N14O11Degré de pureté :99.84%Couleur et forme :SolidMasse moléculaire :999.17Glycochenodeoxycholic Acid
CAS :Glycochenodeoxycholic Acid (Lithocholylglycine) is a glycine conjugate of lithocholic acid, a bile acid.Formule :C26H43NO5Degré de pureté :97% - 99.97%Couleur et forme :SolidMasse moléculaire :449.62Ref: TM-T4588
5mg34,00€10mg49,00€25mg79,00€50mg104,00€100mg154,00€200mg220,00€500mg374,00€1mL*10mM (DMSO)54,00€Phenyl-β-D-glucopyranoside
CAS :Phenyl-β-D-glucopyranoside (PHENYL-B-D-GLUCOPYRANOSIDE) is a component of Phellodendron amurense with anti-cancer and anti-inflammatory activities.Formule :C12H16O6Degré de pureté :98.5% - 98.95%Couleur et forme :White PowderMasse moléculaire :256.25Olsalazine
CAS :Olsalazine (Dipentium), an anti-inflammatory drug, is used in the treatment of inflammatory bowel disease. It is also a novel DNA hypomethylating agent.Formule :C14H10N2O6Degré de pureté :99.31%Couleur et forme :SolidMasse moléculaire :302.24Chrysosplenetin
CAS :Chrysosplenetin is a metabolic inhibitor of artemisinin.Formule :C19H18O8Degré de pureté :97.43% - 98.4%Couleur et forme :SolidMasse moléculaire :374.34Ref: TM-TJS1159
1mg57,00€5mg120,00€10mg178,00€25mg329,00€50mg485,00€100mg692,00€500mg1.404,00€1mL*10mM (DMSO)215,00€DAPT
CAS :DAPT (LY-374973) is a γ-secretase inhibitor that inhibits total Aβ and Aβ42 (IC50=115/200 nM) and is orally active.Formule :C23H26F2N2O4Degré de pureté :98.06% - 99.81%Couleur et forme :White SolidMasse moléculaire :432.46Ref: TM-T6202
2mg38,00€5mg55,00€10mg94,00€25mg157,00€50mg264,00€100mg358,00€200mg490,00€1mL*10mM (DMSO)56,00€Luliconazole
CAS :Luliconazole (NND 502) is an Azole Antifungal. The mechanism of action of luliconazole is as a Cytochrome P450 2C19 Inhibitor.Formule :C14H9Cl2N3S2Degré de pureté :98.27% - 99.83%Couleur et forme :SolidMasse moléculaire :354.28IPSU
CAS :IPSU is an antagonist of OX2 receptor. IPSU Exhibits approximately six-fold selectivity for OX2 versus OX1 receptors.Formule :C23H27N5O2Degré de pureté :97.05%Couleur et forme :SolidMasse moléculaire :405.49Ref: TM-T5503
2mg51,00€5mg86,00€10mg97,00€25mg200,00€50mg299,00€100mg432,00€200mg662,00€1mL*10mM (DMSO)92,00€Amentoflavone
CAS :Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.Formule :C30H18O10Degré de pureté :98.21% - 99.22%Couleur et forme :Odourless Whitish SolidMasse moléculaire :538.46Ref: TM-T3417
2mg34,00€5mg50,00€10mg80,00€25mg126,00€50mg215,00€100mg349,00€200mg512,00€1mL*10mM (DMSO)59,00€Mesaconic acid
CAS :Mesaconic acid (Methylfumaric acid) is used as a fire retardant, as recent studies revealed this acid is a competitive inhibitor of fumarate reduction.Formule :C5H6O4Degré de pureté :99.68%Couleur et forme :SolidMasse moléculaire :130.1Phaseoloidin
CAS :Phaseoloidin, a homogentisic acid glucoside from Nicotiana attenuata trichomes, contributes to the plant's resistance against lepidopteran herbivores.Formule :C14H18O9Degré de pureté :99.32% - ≥95%Couleur et forme :SolidMasse moléculaire :330.29Ref: TM-T5777
2mg35,00€5mg52,00€10mg77,00€25mg111,00€50mg164,00€100mg240,00€200mg344,00€1mL*10mM (DMSO)40,00€
