Enzimi inibitori
Gli inibitori enzimatici sono composti che riducono o arrestano l'attività degli enzimi legandosi specificamente ad essi. Questi inibitori svolgono un ruolo cruciale nella regolazione dei processi biologici e sono ampiamente utilizzati nella ricerca medica e nello sviluppo di farmaci. Bloccando l'attività enzimatica, consentono di studiare la funzione degli enzimi e di sviluppare trattamenti per diverse malattie. Presso CymitQuimica, offriamo un'ampia gamma di inibitori enzimatici di alta qualità per supportare la vostra ricerca in biologia e farmacologia.
Trovati 123 prodotti di "Enzimi inibitori"
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Nafamostat
CAS:Formula:C19H17N5O2Purezza:≥ 98.0%Colore e forma:White to off-white powderPeso molecolare:347.37Vildagliptin
CAS:Formula:C17H25N3O2Purezza:≥ 98.0%Colore e forma:White to off-white powderPeso molecolare:303.40IU1
CAS:Formula:C18H21FN2OPurezza:(TLC) ≥ 98%Colore e forma:Off-white to pale brown solidPeso molecolare:300.37Fumagillin
CAS:Formula:C26H34O7Purezza:≥ 95.0%Colore e forma:White, off-white or pale yellow to tan powderPeso molecolare:458.54Lactacystin
CAS:Formula:C15H24N2O7SPurezza:≥ 95.0%Colore e forma:White solid or powderPeso molecolare:376.43Nα-Tosyl-L-lysine chloromethyl ketone hydrochloride
CAS:Formula:C14H21ClN2O3S·HClPurezza:(HPLC) ≥ 98.0%Colore e forma:White powderPeso molecolare:369.31Bortezomib
CAS:Formula:C19H25BN4O4Purezza:≥ 98.0%Colore e forma:White to off-white powder or solidPeso molecolare:384.24E-64 protease inhibitor
CAS:Formula:C15H27N5O5Purezza:(HPLC) ≥ 98.0%Colore e forma:White crystalline powderPeso molecolare:357.40Bestatin hydrochloride
CAS:Formula:C16H24N2O4·HClPurezza:≥ 98.0% (dried basis)Colore e forma:White to almost white powderPeso molecolare:344.87Argatroban
CAS:Formula:C23H38N6O6SPurezza:(HPLC) ≥ 98%Colore e forma:White to off-white powderPeso molecolare:526.65AEBSF hydrochloride
CAS:Formula:C8H10FNO2S·HClPurezza:≥ 98.0%Colore e forma:White to off-white powder or solidPeso molecolare:239.69N-p-Tosyl-L-phenylalanine chloromethyl ketone
CAS:Formula:C17H18ClNO3SPurezza:(TLC) ≥ 98.0%Colore e forma:White to off-white powderPeso molecolare:351.85Z-VAD-FMK, cell permeable
CAS:Formula:C22H30FN3O7Purezza:≥ 95.0%Colore e forma:White to off-white solidPeso molecolare:467.5Elastatinal microbial
CAS:Formula:C21H36N8O7Purezza:~0.64μg/ml (IC50, pH8.8, 37°C)Colore e forma:White to light-yellow or tan powderPeso molecolare:512.60Pepstatin A
CAS:Formula:C34H63N5O9Purezza:≥ 98.0%Colore e forma:White to off-white powderPeso molecolare:685.90Suramin sodium salt
CAS:Formula:C51H34N6Na6O23S6Purezza:≥ 98%Colore e forma:White to off-white powderPeso molecolare:1429.16E-64d protease inhibitor
CAS:Formula:C17H30N2O5Purezza:≥ 95.0%Colore e forma:White powderPeso molecolare:342.43Carfilzomib
CAS:Formula:C40H57N5O7Purezza:(HPLC) ≥ 98.0%Colore e forma:White to off-white crystalline powder or crystalsPeso molecolare:719.91Phosphoramidon disodium salt
CAS:Formula:C23H32N3Na2O10PPurezza:≥ 97.0%Colore e forma:Colourless, transparent crystals or white to light yellow crystalline powderPeso molecolare:587.47Nafamostat mesylate
CAS:Formula:C19H17N5O2Purezza:≥ 99.0%Colore e forma:White to off-white or beige crystalline powderPeso molecolare:347.37DAPT
CAS:Formula:C23H26F2N2O4Purezza:(NMR) ≥ 98.0%Colore e forma:White to off-white solidPeso molecolare:432.50Leupeptin hemisulfate
CAS:Formula:C20H38N6O4·5H2SO4Purezza:≥ 95%Colore e forma:White to off-white powderPeso molecolare:475.59Z-Leu-Leu-Leu-al
CAS:Formula:C26H41N3O5Purezza:≥ 97.0%Colore e forma:White to off-white powder or solidPeso molecolare:475.63CP-10447
CAS:<p>Applications CP-10447 is an inhibitor apolipoprotein B (apoB) and triglyceride secretion in human hepatoma cells (HepG2) by inhibiting MTP activity and stimulating the early ER degradation of apoB. It is useful tool for further study of the mechanisms of apoB secretion and triglyceride-rich lipoprotein assembly.<br>References Haghpassand, M. et al.: J. Lipid. Res., 37, 1468 (1996); Pan, M. et al.: J. Biol. chem., 275, 27399 (2000);<br></p>Formula:C16H13BrN2OColore e forma:NeatPeso molecolare:329.192-(Hydroxyamino)acetic Acid
CAS:Prodotto controllato<p>Applications 2-(Hydroxyamino)acetic Acid is a novel lactase inhibitor.<br>References Hattori, M., et al.: J. Insect Physiol., 51, 1359 (2005); Murao, S., et al.: Biosci. Biotech. Biochem., 56, 987 (1992)<br></p>Formula:C2H5NO3Colore e forma:NeatPeso molecolare:91.07(3S,4S,3’S)-Ezetimibe
CAS:<p>Applications (3S,4S,3’S)-Ezetimbe is a 3-epimer impurity of Ezetimibe (E975000), a cholesterol absorption inhibitor.<br>References van Heek, M., at al.: J. Pharmacol. Exp. Ther., 283, 157 (1997), van Heek, M., at al.: Brit. J. Pharmacol., 129, 1748 (2000)<br></p>Formula:C24H21F2NO3Colore e forma:Off-WhitePeso molecolare:409.43LCZ696
CAS:<p>Applications LCZ696 is a novel dual-acting inhibitor of angiotensin II receptor and neprilysin, which can be used for blood pressure reduction.<br>References Ruilope, L.M.; et al.: Lancet, 375, 1255 (2010)<br></p>Formula:C24H28NO5·C24H27N5O3·3Na·x(H2O)Colore e forma:MixturePeso molecolare:479.48 + (433.47) + x(18.02)Abamine
CAS:Prodotto controllato<p>Applications Abamine is an inhibitor of 9-Cis-Epoxycarotenoid dioxygenase (NCED), the key regulatory enzyme in the plant hormone abscisic acid (ABA) biosynthesis pathway.<br>References Kitahata, N., et al.: Bioorg. Med. Chem., 14, 5555 (2006); Han, S., et al.: Bioorg. Med. Chem. Lett., 14, 3033 (2004)<br></p>Formula:C21H24FNO4Colore e forma:NeatPeso molecolare:373.423'-Deoxyadenosine 5’-Diphosphate Triethylamine Salt (>90%)
CAS:<p>Stability Hygroscopic<br>Applications 3'-Deoxyadenosine 5’-Diphosphate Triethylamine Salt, is a nucleotide and was proposed to be a possible inhibitor of DNA synthesis.<br>References Frederiksen, Sune.: Biochimica et Biophysica Acta, 76(3), 366-71 (1963)<br></p>Formula:C10H15N5O9P2•xC6H15NPurezza:>90%Colore e forma:NeatPeso molecolare:411.20 + x(101.19)Teneligliptin Hydrobromide (2:5)
CAS:Prodotto controllato<p>Applications Teneligliptin Hydrobromide (2:5) is a dipeptidyl peptidase-4 (DPP-4) inhibitor that is used to treat type 2 diabetes. It is eliminated via excretion, and has a half-life of 24.2 hours in the human body.<br>References Goda, M. & Kadowaki, T.: Drugs Today, 49, 615 (2013); Kishimoto, M.: Diabetes Metab. Syndr. Obes., 6, 187 (2012)<br></p>Formula:C22H32·5Br2·5N6OSColore e forma:NeatPeso molecolare:628.86Daidzein Diglucuronide
CAS:Prodotto controllatoFormula:C27H26O16Colore e forma:White To Off-WhitePeso molecolare:606.49(3S,5S)-Atorvastatin Calcium Salt
CAS:Prodotto controllato<p>Impurity Atorvastatin Related Compound E<br>Applications Impuritiy of Atorvaststin (A791750), a selective, competitive HMG-CoA reductase inhibitor. Atorvastatin is the only drug in its class specfically indicated for lowering both elevated LDL-cholesterol and triglycerides in patients with hypercholesterolemia. Atorvastatin Related Compound E<br>References Kearney, A.S., et al.: Pharm. Res., 10, 1461 (1993), Heinonen, T.M., et al.: Clin. Ther., 18, 853 (1996), Whitfield, L.R., et al.: Eur. J. Drug Metab. Pharmacokinet., 25, 97 (2000),<br></p>Formula:C33H34FN2O5·CaColore e forma:NeatPeso molecolare:1155.34N-(2-Hydroxyethyl)-1-deoxy-L-idonojirimycin Hydrochloride
CAS:Prodotto controllato<p>Stability Hygroscopic<br>Applications α-Glycosidase inhibitor.<br>References van de Water, F., et al.: Drug Metab. Rev., 37, 443 (2005), Koepsell, H., et al.: Pharm. Res., 24, 1227 (2007), Jappar, D., et al.: Pharm. Res., 26, 172 (2009),<br></p>Formula:C8H18ClNO5Colore e forma:NeatPeso molecolare:243.69N-(2-Hydroxyethyl)-1-deoxy-L-altronojirimycin Hydrochloride Salt
CAS:Prodotto controllato<p>Stability Hygroscopic<br>Applications α-Glycosidase inhibitor.<br>References Jefferies, I., et al.: Bioorg. Med. Chem. Lett., 7, 1171 (1997), Hassan, A., et al.: Carbohydr. Res., 339, 1565 (2004),<br></p>Formula:C8H18ClNO5Colore e forma:NeatPeso molecolare:243.6852Aprotinin Hydrochloride
CAS:<p>Applications Aprotinin is used in cardiac surgery to minimize bleeding and reduce exposure to blood products.<br>References Mangano, D. et al.: New Eng. J. Med., 354, 353 (2006); Fergusson, D. et al.: New. Eng. J. Med., 358, 2319 (2008);<br></p>Formula:C284H432N84O79S7·x(ClH)Colore e forma:White SolidPeso molecolare:6511.51(free amine)Nitromifene Citrate (E/Z mixture)
CAS:Prodotto controllato<p>Applications Nitromifene citrate is a non-steroidal estrogen antagonist. It is structurally similar to Tamoxifen (T006000) which is a selective estrogen response modifier (SERM).<br>References Rudick, C., et al.: Endorcrinol., 144, 179 (2003); Sutherland, R., et al.: Nature, 267, 434 (1977)<br></p>Formula:C33H36N2O11Colore e forma:Yellow To OrangePeso molecolare:636.65Galacto-PUGNAc (>90%)
CAS:Prodotto controllato<p>Stability Moisture and Temperature Sensitive<br>Applications Galacto-PUGNAc is a highly selective inhibitor for β-hexosaminidases HEXA and HEXB is cell-permeable. Galacto-PUGNAc is able to modulate the activity of HEXA and HEXB in tissue culture, increasing ganglioside GM2 levels in neuroblastoma cells<br>References Stubbs, K.A. et al.: Angew. Chem. Int. Ed., 48, 1300 (2009);<br></p>Formula:C15H19N3O7Purezza:>90%Colore e forma:NeatPeso molecolare:353.332,5-Dideoxy-2,5-imino-D-mannitol
CAS:Prodotto controllato<p>Stability Hygroscopic<br>Applications A glucosidase inhibitor.<br>References Fellows, L.E.: Pestic. Sci., 17, 602 (1986)<br></p>Formula:C6H13NO4Colore e forma:Off White SolidPeso molecolare:163.17Vitamin B12 e-Monocarboxylic Acid
CAS:<p>Stability Hygroscopic<br>Applications Vitamin B12 Monocarboxylic Acid is an impurity of Vitamin B12 (V676005) which is a water-soluble vitamin with a key role in the normal functioning of the brain and nervous system, and for the formation of blood.<br>References Rickes, et al.: Science, 107, 396 (1948); Kirschbaum, J., et al.: Anal. Profiles Drug Subs., 10, 183 (1981); Grasbeck, R., et al.: Clin. Biochem., 17, 99 (1984)<br></p>Formula:C63H87CoN13O15PColore e forma:Dark Red SolidPeso molecolare:1356.35tert-Butyl (2S,4S)-4-[4-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]-2-[(1,3-thiazolidin-3-yl)carbonyl]pyrrolidine-1-carboxylate
CAS:Prodotto controllato<p>Applications tert-Butyl (2S,4S)-4-[4-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]-2-[(1,3-thiazolidin-3-yl)carbonyl]pyrrolidine-1-carboxylate is an orally anti-diabetic agent as a inhibitors of dipeptidylpeptidase IV (DPP-4).<br>References Yoshida, T., et al.: Bioorg. Med. Chem., 20, 5705-5719 (2012);<br></p>Formula:C27H38N6O3SColore e forma:NeatPeso molecolare:526.69
![tert-Butyl (2S,4S)-4-[4-(3-Methyl-1-phenyl-1H-pyrazol-5-yl)piperazin-1-yl]-2-[(1,3-thiazolidin-3-y…](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTR%2Fthumb-webp%2FB807705.webp&w=3840&q=75)