
Apoptosi
Sottocategorie di "Apoptosi"
- ASK(9 prodotti)
- BCL(5 prodotti)
- Caspasi(151 prodotti)
- FOXO1(2 prodotti)
- IAP(67 prodotti)
- Mdm2(12 prodotti)
- PD-1/PD-L1(105 prodotti)
- PDK(9 prodotti)
- PERK(26 prodotti)
- Chinasi di serina/treonina(18 prodotti)
- Survivin(14 prodotti)
- TNF(58 prodotti)
- c-RET(61 prodotti)
- p53(63 prodotti)
Trovati 6043 prodotti di "Apoptosi"
tubuloside B
CAS:Tubuloside B from Cistanche salsa stems guards SH-SY5Y cells against TNFalpha-induced apoptosis.
Formula:C31H38O16Purezza:97.59% - 99.72%Colore e forma:SolidPeso molecolare:666.62ABT-737
CAS:ABT-737 is a BH3 mimetic and an inhibitor of Bcl-2, Bcl-xL, and Bcl-w. ABT-737 exhibits antitumor activity and anti-aging activity. Cost-effective and quality-assured.Formula:C42H45ClN6O5S2Purezza:98.15% - >99.99%Colore e forma:SolidPeso molecolare:813.43PF-4989216
CAS:PF-4989216 is a potent and selective PI3K inhibitor with IC50 of 2 nM, 142 nM, 65 nM, 1 nM, and 110 nM for p110α, p110β, p110γ, p110δ, and VPS34, respectively.Formula:C18H13FN6OSPurezza:99.85%Colore e forma:SolidPeso molecolare:380.4Ref: TM-T6938
2mg39,00€5mg65,00€10mg101,00€25mg187,00€50mg329,00€100mg398,00€200mg565,00€1mL*10mM (DMSO)67,00€JX06
CAS:JX06, a potent, selective and covalent PDK inhibitor, inhibits PDK1, PDK2 and PDK3 with IC50 of 49 nM, 101 nM and 313 nM respectively.Formula:C10H16N2O2S4Purezza:99.4%Colore e forma:SolidPeso molecolare:324.51Ref: TM-T22350
5mg48,00€10mg70,00€25mg133,00€50mg207,00€100mg335,00€200mg497,00€1mL*10mM (DMSO)52,00€WT-161
CAS:WT161 is a potent and selective inhibitor of HDAC6 (IC50:0.40 nM).Formula:C27H30N4O3Purezza:95.98% - 98.34%Colore e forma:SolidPeso molecolare:458.55Diosgenin glucoside
CAS:Diosgenin glucoside (Trillin) and other synthetic glycosides with similar activities may be of use in the management of hypercholesterolemia and atherosclerosis
Formula:C33H52O8Purezza:97.17% - 99.44%Colore e forma:SolidPeso molecolare:576.76MK-2206 dihydrochloride
CAS:MK-2206 dihydrochloride (MK-2206 2HCl) is a variant Akt inhibitor that inhibits Akt1, Akt2, and Akt3 (IC50=8/12/65 nM) with orally active, highly potent andFormula:C25H23Cl2N5OPurezza:99.228% - 99.94%Colore e forma:SolidPeso molecolare:480.39Ref: TM-T1952
2mg34,00€5mg49,00€10mg66,00€25mg90,00€50mg137,00€100mg205,00€200mg334,00€500mg552,00€1mL*10mM (DMSO)52,00€4,5-Dicaffeoylquinic acid
CAS:1.Formula:C25H24O12Purezza:98.86% - ≥95%Colore e forma:SolidPeso molecolare:516.45Ref: TM-T2S1158
1mg43,00€5mg84,00€10mg109,00€25mg172,00€50mg250,00€100mg326,00€200mg522,00€1mL*10mM (DMSO)102,00€AZ5576 racemate
CAS:AZ5576 racemate, potent Cdk9 inhibitor, oral, IC50 <5nM; disrupts RNAPII, aids AML treatment, kills MV411 cells.Formula:C21H24FN3O3Colore e forma:SolidPeso molecolare:385.43Geranyl acetate
CAS:Geranyl acetate is a monoterpene that has been found in C. sativa with diverse biological activities.Formula:C12H20O2Purezza:99.36%Colore e forma:Physical Description Clear Colorless Liquid With An Odor Of Lavender (Ntp 1992)Peso molecolare:196.29Pexidartinib
CAS:Pexidartinib (PLX-3397) is a capsule formulation containing a small-molecule receptor tyrosine kinase (RTK) inhibitor of KIT, CSF1R and FLT3 with potentialFormula:C20H15ClF3N5Purezza:98.34% - 99.45%Colore e forma:SolidPeso molecolare:417.81Ref: TM-T2115
5mg46,00€10mg58,00€25mg90,00€50mg114,00€100mg145,00€200mg192,00€500mg333,00€1mL*10mM (DMSO)49,00€Linalool
CAS:Linalool, in essential oils, offers antinociceptive, antimicrobial, and anti-inflammatory effects, protects the liver, and boosts plant defense.Formula:C10H18OPurezza:98.22%Colore e forma:Colorless Liquid Drypowder Liquid Othersolid LiquidPeso molecolare:154.25CIL56
CAS:CIL56 (CA3) is a small molecule that induces cellular ferroptosis through the production of iron-dependent reactive oxygen species (ROS).Formula:C23H27N3O5S2Purezza:99.46% - 99.91%Colore e forma:SolidPeso molecolare:489.61Ref: TM-T4309
1mg34,00€2mg49,00€5mg74,00€10mg109,00€25mg178,00€50mg284,00€100mg434,00€1mL*10mM (DMSO)81,00€TPEN
CAS:TPEN (TPEDA) is a specific cell-permeable heavy metal chelator.Formula:C26H28N6Purezza:98% - 99.72%Colore e forma:White Crystalline PowderPeso molecolare:424.54Rasagiline Mesylate
CAS:Rasagiline Mesylate (AGN1135) is a novel MAO-B inhibitor, which can treat idiopathic Parkinson's disease.Formula:C13H17NO3SPurezza:99.33%Colore e forma:White PowderPeso molecolare:267.342,5-dimethyl Celecoxib
CAS:2,5-dimethyl Celecoxib, a derivative targeting mPGES-1, inhibits PGE2 synthesis in inflammation.Formula:C18H16F3N3O2SPurezza:99.85%Colore e forma:SolidPeso molecolare:395.4Lanperisone
CAS:Lanperisone is a muscle relaxant.Formula:C15H18F3NOColore e forma:SolidPeso molecolare:285.3AT7519 Hydrochloride
CAS:AT7519 Hydrochloride (AT7519 HCl) is a multi-CDK inhibitor for CDK1, 2, 4, 6 and 9.Formula:C16H18Cl3N5O2Purezza:99.66% - 99.9%Colore e forma:SolidPeso molecolare:418.71G-749
CAS:G-749, a new-type FLT3 inhibitor, exhibits effective and sustained inhibition of the FLT3 wild type and mutants.Formula:C25H25BrN6O2Purezza:98.32% - 99.60%Colore e forma:SolidPeso molecolare:521.41Z-IETD-FMK
CAS:Z-IETD-FMK (Z-IE(OMe)TD(OMe)-FMK) is a selective caspase 8 inhibitor, which has cell permeable.Formula:C30H43FN4O11Purezza:95% - 99.81%Colore e forma:SolidPeso molecolare:654.68PhiKan 083
CAS:PhiKan 083 is a carbazole derivativeFormula:C16H18N2Purezza:98.37%Colore e forma:SolidPeso molecolare:238.33Ref: TM-T16523L
1mg34,00€5mg66,00€10mg105,00€25mg222,00€50mg313,00€100mg439,00€500mg954,00€1mL*10mM (DMSO)72,00€Hirsutine
CAS:Hirsutine induces apoptosis and is a potent Dengue virus inhibitor exhibiting low cytotoxicity.Hirsutine has anticancer, cardioprotective, anti-hypertensive andFormula:C22H28N2O3Purezza:99.36% - 99.98%Colore e forma:SolidPeso molecolare:368.47(Rac)-Antineoplaston A10
CAS:Antineoplaston A10 is the first identified human antineoplaston, naturally occurring with anti-proliferative properties.Formula:C13H14N2O3Purezza:98.41%Colore e forma:SolidPeso molecolare:246.26Ref: TM-T5379
1mg40,00€5mg88,00€10mg129,00€25mg210,00€50mg311,00€100mg449,00€200mg627,00€1mL*10mM (DMSO)95,00€A-1210477
CAS:A-1210477 is an effective and specific MCL-1 and Bcl-2 inhibitor (Ki/IC50: 0.454/26.2 nM).Formula:C46H55N7O7SPurezza:99.17% - 99.37%Colore e forma:SolidPeso molecolare:850.04Pseudolaric Acid B
CAS:Pseudolaric acid B, a natural diterpenoid compound, is isolated from Pseudolarix kaempferi.Formula:C23H28O8Purezza:98.91% - 99.84%Colore e forma:SolidPeso molecolare:432.46Z-YVAD-FMK
CAS:AA-Z-YVAD-FMK is a Irreversible caspase-1 inhibitor,with anti-inflammatory and anti-tumor activities.Formula:C31H39FN4O9Purezza:98.00%Colore e forma:SolidPeso molecolare:630.66Loganin
CAS:Loganin inhibits Cox-1, suppresses TNF-α, and has antioxidant and anti-melanogenic properties.Formula:C17H26O10Purezza:99.01% - 99.9%Colore e forma:White PowderPeso molecolare:390.38SHR0302
CAS:SHR0302 (ARQ252) is a JAK inhibitor that binds JAK1 with stronger affinity than others (Selectivity for JAK1 is more than 10 times for JAK2, 77 times for JAK3,Formula:C18H22N8O2SPurezza:99.11%Colore e forma:SolidPeso molecolare:414.48Ref: TM-T9195
1mg80,00€5mg183,00€10mg298,00€25mg512,00€50mg817,00€100mg1.311,00€1mL*10mM (DMSO)167,00€L-Threonic acid magnesium salt
CAS:L-Threonic acid magnesium salt (L-TAMS) increases synapse density and memory ability in both aged rats and late stage Alzheimer’s disease (AD) model mice.Formula:C8H14MgO10Purezza:99.73%Colore e forma:SolidPeso molecolare:294.5RET V804M-IN-1
CAS:RET V804M-IN-1 (RETV804M kinase inhibitor) is a wt-RET -selective RETV804M kinase inhibitors(IC50 = 20 nM).Formula:C19H16N6OPurezza:97.94% - 99.62%Colore e forma:SolidPeso molecolare:344.37Ref: TM-T8467
1mg35,00€2mg50,00€5mg74,00€10mg90,00€25mg157,00€50mg236,00€100mg334,00€200mg495,00€1mL*10mM (DMSO)82,00€NVP-HSP990
CAS:NVP-HSP990 (HSP990) is an effective and specific HSP90α/β inhibitor (IC50: 0.6 /0.8 nM).Formula:C20H18FN5O2Purezza:98.03% - 99.32%Colore e forma:SolidPeso molecolare:379.39GSK2982772
CAS:GSK2982772 is an inhibitor of receptor interacting serine/threonine kinase 1 (RIPK1)with IC50 values of 16 nM and 20 nM for human and monkey RIP1, respectively.Formula:C20H19N5O3Purezza:99.27% - 99.31%Colore e forma:SolidPeso molecolare:377.4GSK3179106
CAS:GSK3179106 is RET kinase inhibitor with an IC50 of 0.4 nMFormula:C22H21F4N3O4Purezza:99.8% - 99.90%Colore e forma:SolidPeso molecolare:467.41GSK547
CAS:GSK547 (GSK'547) is a highly selective and potent inhibitor of RIP1 kinase,inhibits macrophage-mediated adaptive immune tolerance in pancreatic cancer.Formula:C20H18F2N6OPurezza:99.17%Colore e forma:SolidPeso molecolare:396.39Cabozantinib S-malate
CAS:Cabozantinib S-malate (XL184) is the salt form of cabozantinib, an orally bioavailable, small molecule RTK inhibitor with potential antineoplastic activity.Formula:C32H30FN3O10Purezza:98% - >99.99%Colore e forma:SolidPeso molecolare:635.59PP121
CAS:PP-121 inhibits PDGFR, Hck, mTOR, VEGFR2, Src, Abl, and DNA-PK with IC50 values ranging from 2 to 60 nM.Formula:C17H17N7Purezza:98.45% - 99.93%Colore e forma:SolidPeso molecolare:319.36MK-8745
CAS:MK-8745 is a potent and selective Aurora A inhibitor.
Formula:C20H19ClFN5OSPurezza:99.09% - 99.79%Colore e forma:SolidPeso molecolare:431.91AS1842856
CAS:AS1842856 is a Foxo1 inhibitor that blocks the transcriptional activity of Foxo1. AS1842856 has autophagy inhibitory activity. Cost-effective and quality-assured.Formula:C18H22FN3O3Purezza:99.36% - >99.99%Colore e forma:SolidPeso molecolare:347.38Scopoletin
CAS:Scopoletin (Esculetin 6-methyl ether) is a plant growth factor derived from the root of Scopolia carniolica, inhibits of acetylcholinesterase (AChE).Formula:C10H8O4Purezza:97.06% - 99.88%Colore e forma:Yellow To Beige Crystalline PowderPeso molecolare:192.17Kinsenoside
CAS:Kinsenoside ((+)-Kinsenoside) shows significant antihepatotoxic, and anti-inflammatory activities.Formula:C10H16O8Purezza:99.2% - 99.92%Colore e forma:SolidPeso molecolare:264.235-Geranoxy-7-methoxycoumarin
CAS:5-Geranoxy-7-methoxycoumarin shows antifungal activity.Formula:C20H24O4Purezza:98.94% - 99.99%Colore e forma:SolidPeso molecolare:328.4Ref: TM-TN3110
1mg104,00€5mg245,00€10mg361,00€25mg607,00€50mg845,00€100mg1.169,00€1mL*10mM (DMSO)Prezzo su richiestaFX1
CAS:FX1 is an effective and selective BCL6 inhibitor (IC50: 35 μM).Formula:C14H9ClN2O4S2Purezza:97.59%Colore e forma:SolidPeso molecolare:368.82ASK1-IN-2
CAS:ASK1-IN-2: oral ASK1 inhibitor, IC50 32.8 nM, potential ulcerative colitis treatment.Formula:C19H17FN6OPurezza:98.79%Colore e forma:SolidPeso molecolare:364.38Mimosine
CAS:L-Mimosine (Leucenol) is an antineoplastic alanine-substituted pyridine derivative isolated from Leucena glauca and acts as an iron chelator.Formula:C8H10N2O4Purezza:99.2% - 99.84%Colore e forma:Crystals From Water SolidPeso molecolare:198.18Indinavir sulfate
CAS:Indinavir sulfate (L735524 sulfate) is a HIV protease inhibitor.It inhibits the HIV-1 protease with an IC50 value of 0.41 nM and Ki value of 0.24 nM.
Formula:C36H49N5O8SPurezza:99.75% - >99.99%Colore e forma:White PowderPeso molecolare:711.87Etomoxir sodium salt
CAS:Etomoxir sodium salt ((R)-Etomoxir sodium salt) is a carnitine palmitoyltransferase 1a (CPT-1a) inhibitor that blocks fatty acid synthesis.Formula:C15H18ClO4·NaPurezza:99.34% - 99.82%Colore e forma:SolidPeso molecolare:320.74Ref: TM-T4535
1mg34,00€2mg40,00€5mg57,00€10mg93,00€25mg144,00€50mg250,00€100mg409,00€200mg602,00€1mL*10mM (DMSO)63,00€KY-05009
CAS:KY-05009 blocks TGF-β1 EMT in lung cancer cells, inhibits TNIK, Wnt genes, induces apoptosis, and is an ATP-competitive TNIK inhibitor (Ki = 100 nM).Formula:C18H16N4O2SPurezza:99.89%Colore e forma:SolidPeso molecolare:352.41Ref: TM-T11793
5mg48,00€10mg67,00€25mg111,00€50mg161,00€100mg231,00€200mg335,00€1mL*10mM (DMSO)49,00€Capmatinib 2HCl
CAS:Capmatinib 2HCl (INC-280 2HCl), a c-MET inhibitor, is potent (IC50 = 0.13 nM), highly specific, and induces apoptosis in tumor cells.Formula:C23H19Cl2FN6OPurezza:98.80%Colore e forma:SolidPeso molecolare:485.34Ref: TM-T4260
2mg34,00€5mg49,00€10mg64,00€25mg84,00€50mg92,00€100mg126,00€500mg303,00€1mL*10mM (DMSO)58,00€ASP3026
CAS:ASP3026 has been used in trials studying the treatment of Solid Tumor, B-Cell Lymphoma, Advanced Malignancies,and Positive for Anaplastic Lymphoma Kinase.Formula:C29H40N8O3SPurezza:98.78% - 99.81%Colore e forma:SolidPeso molecolare:580.74BTZO-1
CAS:BTZO-1 is an antioxidant response element (ARE) activator with cardioprotective activity.Formula:C13H8N2OSPurezza:99.46%Colore e forma:SolidPeso molecolare:240.28Ref: TM-T7845
2mg34,00€5mg50,00€10mg85,00€25mg154,00€50mg222,00€100mg331,00€200mg470,00€1mL*10mM (DMSO)56,00€Salidroside
CAS:Salidroside is a bioactive phenolic glycoside compound isolated from Rhodiola rosea and is a prolyl endopeptidase inhibitor.Cost-effective and quality-assured.Formula:C14H20O7Purezza:97.81%Colore e forma:Red-Brown Fine PowderPeso molecolare:300.30Ref: TM-T2717
2mg34,00€5mg50,00€10mg81,00€25mg130,00€50mg178,00€100mg268,00€200mg408,00€1mL*10mM (DMSO)55,00€Tomatine
CAS:Tomatine (lycopersicin) is an antiproliferatve agent of breast adenocarcinoma cells.Formula:C50H83NO21Purezza:98.42% - 99.94%Colore e forma:White To Light YellowPeso molecolare:1034.19MG-101
CAS:MG-101 (Calpain inhibitor I) is a cell-permeable and potent inhibitor of cysteine proteases including calpains and lysosomal cathepsins.Formula:C20H37N3O4Purezza:98% - ≥98%Colore e forma:SolidPeso molecolare:383.53Kahweol
CAS:Kahweol has anticarcinogenic, anti-angiogenic,and anti-inflammatory activities, it can block the LPS-induced activation of NF-kappaB by preventing IkappaBFormula:C20H26O3Purezza:99.26% - 99.86%Colore e forma:Off-White To Yellow SolidPeso molecolare:314.42BC-1258
CAS:BC-1258 is a unique small molecule F-box/LRR-repeat protein 2 (FBXL2) activator.Formula:C22H22N4S2Purezza:97.48% - 99.64%Colore e forma:SolidPeso molecolare:406.57LY2857785
CAS:LY2857785 is a type I competitive and reversible ATP kinase inhibitor against CDK7/CDK8/CDK9 (IC50s: 246 nM/16 nM/11 nM).Formula:C26H36N6OPurezza:99.68%Colore e forma:Solid PowderPeso molecolare:448.6Ref: TM-TQ0060
1mg50,00€2mg71,00€5mg105,00€10mg170,00€25mg334,00€50mg537,00€100mg863,00€1mL*10mM (DMSO)117,00€B-AP15
CAS:B-AP15 (NSC-687852) selectively inhibits 26S proteasome enzymes Usp14 and UCHL5, blocking their activity.
Formula:C22H17N3O6Purezza:91.43% - 98.77%Colore e forma:SolidPeso molecolare:419.39Citronellyl acetate
CAS:Citronellyl acetate is a natural productFormula:C12H22O2Purezza:98%Colore e forma:LiquidPeso molecolare:198.30PS 48
CAS:PS 48 has been shown to be a PKB Kinase (PDK1) activator (Kd: 10.3 μM). This compound selectively binds to the PIF-binding pocket of PKB Kinase (PDK1).Formula:C17H15ClO2Purezza:99.96% - ≥95%Colore e forma:SolidPeso molecolare:286.75R406 free base
CAS:R406 free base (R406 (free base)) is a potent Syk inhibitor.Formula:C22H23FN6O5Purezza:97.64% - 99.11%Colore e forma:SolidPeso molecolare:470.45Ref: TM-T2467
1mg44,00€5mg66,00€10mg92,00€25mg177,00€50mg319,00€100mg507,00€500mg1.063,00€1mL*10mM (DMSO)69,00€PR-619
CAS:PR-619 (2,6-Diamino-3,5-dithiocyanopyridine) is a DUB inhibitor. PR-619 induces endoplasmic reticulum stress and activates autophagy. Cost-effective and quality-assured.Formula:C7H5N5S2Purezza:97.25% - >99.99%Colore e forma:SolidPeso molecolare:223.28Benzonitrile, 3,3'-[(2-oxo-1,3-cyclohexanediylidene)dimethylidyne]bis-
CAS:Benzonitrile, 3,3'-[(2-oxo-1,3-cyclohexanediylidene)dimethylidyne]bis- (9CI) is an inhibitor of p53 with an IC50 value of 0.35 μMFormula:C22H16N2OPurezza:99.18%Colore e forma:SolidPeso molecolare:324.38Ref: TM-T9129
1mg52,00€5mg107,00€10mg158,00€25mg259,00€50mg374,00€100mg523,00€200mg710,00€1mL*10mM (DMSO)111,00€Pilaralisib analogue
CAS:Pilaralisib analogue (XL147 analogue) is a selective and reversible class I PI3K inhibitor for PI3Kα/δ/γ.Formula:C21H16N6O2S2Purezza:99.3% - 99.72%Colore e forma:SolidPeso molecolare:448.52Ref: TM-T2377
2mg35,00€5mg52,00€10mg84,00€25mg132,00€50mg205,00€100mg354,00€200mg460,00€1mL*10mM (DMSO)93,00€Roquinimex
CAS:Roquinimex (FCF89) (Linomide) is a quinoline derivative immunostimulant which increases NK cell activity and macrophage cytotoxicity; inhibits angiogenesis andFormula:C18H16N2O3Purezza:97.69%Colore e forma:SolidPeso molecolare:308.33Toyocamycin
CAS:Toyocamycin (Vengicide) is an adenosine analog produced by Actinomycete, acts as an XBP1 inhibitor, inhibits IRE1α-induced ATP-dependent XBP1 mRNA cleavage (Formula:C12H13N5O4Purezza:98.1% - 99.44%Colore e forma:SolidPeso molecolare:291.26Ref: TM-T17143
5mg47,00€10mg65,00€25mg113,00€50mg202,00€100mg354,00€500mg825,00€1mL*10mM (DMSO)50,00€Adalimumab
CAS:Adalimumab (anti-TNF-alpha) is the first fully human recombinant IgG1 monoclonal antibody that specifically targets human TNF-alpha.Purezza:95% - >95.0% (SDS-PAGE)Colore e forma:LiquidPeso molecolare:145.4 kDatrans-Chalcone
CAS:trans-Chalcone (Chalkone) is an aromatic ketone that forms the central core for a variety of important biological compounds, which are known collectively asFormula:C15H12OPurezza:99.89%Colore e forma:SolidPeso molecolare:208.26Solasodine
CAS:Solasodine, a toxic alkaloid from Solanaceae, kills HeLa cervical cancer and U937 leukemia cells.Formula:C27H43NO2Purezza:99.64% - 99.94%Colore e forma:SolidPeso molecolare:413.64Se-Methylselenocysteine
CAS:Se-Methylselenocysteine (Se-MSC) is a potent chemopreventive agent in many test systems and has been shown to inhibit tumor promotion and induce apoptosis.Formula:C4H9NO2SePurezza:99.49% - 99.87%Colore e forma:White To Slightly Yellow PowderPeso molecolare:182.08Divalproex Sodium
CAS:Divalproex Sodium (Valproate semisodium) binds to and inhibits gamma-aminobutyric acid (GABA) transaminase and its anticonvulsant activity may be exerted byFormula:C8H16O2·C8H15O2·NaPurezza:99.87%Colore e forma:A White Powder With A Characteristic OdorPeso molecolare:310.41Ref: TM-T6474
10mg39,00€25mg55,00€50mg79,00€100mg116,00€200mg188,00€500mg335,00€1mL*10mM (DMSO)55,00€Tamibarotene
CAS:Tamibarotene (Amnolake) is an orally active, synthetic retinoid, developed to overcome all-trans retinoic acid (ATRA) resistance, with potential antineoplasticFormula:C22H25NO3Purezza:98.55% - 99.73%Colore e forma:Crystalline SolidPeso molecolare:351.44Ref: TM-T6694
1g350,00€10mg44,00€25mg60,00€50mg74,00€100mg92,00€200mg144,00€500mg235,00€1mL*10mM (DMSO)44,00€PCI-34051
CAS:PCI-34051 is an effective and selective HDAC8 inhibitor (IC50: 10 nM).
Formula:C17H16N2O3Purezza:97.219% - 98.29%Colore e forma:SolidPeso molecolare:296.32MI-136
CAS:MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.Formula:C23H21F3N6SPurezza:98.63% - 99.12%Colore e forma:SolidPeso molecolare:470.51Ref: TM-T6889
1mg47,00€5mg87,00€10mg147,00€25mg279,00€50mg472,00€100mg730,00€200mg1.017,00€1mL*10mM (DMSO)97,00€Rapanone
CAS:Rapanone (2,5-Dihydroxy-3-tridecyl-[1,4]benzoquinone) is a natural benzoquinone that is a potent and selective inhibitor of human synovial PLA2.Formula:C19H30O4Purezza:99.56%Colore e forma:SolidPeso molecolare:322.44HS-173
CAS:HS-173 is an effective PI3Kα inhibitor (IC50: 0.8 nM).Formula:C21H18N4O4SPurezza:99.33% - 99.64%Colore e forma:SolidPeso molecolare:422.46Ref: TM-T2308
2mg34,00€5mg52,00€10mg77,00€25mg128,00€50mg200,00€100mg296,00€200mg425,00€1mL*10mM (DMSO)52,00€Fidaxomicin
CAS:Fidaxomicin (Tiacumicin B) is a semisynthetic macrolide antibiotic used to treat Clostridium difficile-associated diarrhea in adults.Formula:C52H74Cl2O18Purezza:99.76% - 99.82%Colore e forma:SolidPeso molecolare:1058.04Ref: TM-T6194
1g414,00€10mg46,00€25mg56,00€50mg77,00€100mg117,00€200mg167,00€500mg268,00€1mL*10mM (DMSO)52,00€Leachianone A
CAS:Leachianone A (Isokurarinone) is a potential antitoxic agent, it shows inhibitory effects on cadmium- Induced cytotoxicity.Formula:C26H30O6Purezza:98.53% - 99.79%Colore e forma:SolidPeso molecolare:438.51Kevetrin hydrochloride
CAS:Kevetrin hydrochloride (4-Isothioureidobutyronitrile hydrochloride) is a small molecule and activator of the tumor suppressor protein p53, with potentialFormula:C5H10ClN3SPurezza:99.32% - 99.93%Colore e forma:SolidPeso molecolare:179.67PS210
CAS:PS210 selectively activates PDK1 (Kd: 3 μM), doesn't affect PDK1 downstream kinases. Prodrug PS423 inhibits PDK1-mediated S6K phosphorylation.
Formula:C19H15F3O5Purezza:99.78%Colore e forma:SolidPeso molecolare:380.31Alofanib
CAS:Alofanib (RPT835) selectively inhibits FGFR2 in KATO III cells with IC50 <10 nM; doesn’t affect FGFR1/3 or FGF2-FGFR2 binding.Formula:C19H15N3O6SPurezza:99.53% - 99.81%Colore e forma:SolidPeso molecolare:413.4Everolimus
CAS:Everolimus (SDZ-RAD) is a potent mTOR inhibitor that binds to FKBP-12. It is used alone or in combination with calcineurin inhibitors.
Formula:C53H83NO14Purezza:97.76% - 99.78%Colore e forma:Off-White To Light Yellow PowdPeso molecolare:958.22Galgravin
CAS:Galgravin combats inflammation, safeguards neurons, promotes neurite growth, and resists Abeta25-35 and MPP+ toxicity.
Formula:C22H28O5Purezza:99.75% - 99.88%Colore e forma:SolidPeso molecolare:372.45Dinoprost tromethamine salt
CAS:Dinoprost tromethamine salt (PGF2α THAM) is a naturally occurring prostaglandin used in medicine to induce labor and as an abortifacient.Formula:C24H45NO8Purezza:99.73%Colore e forma:Natural Form Crystals SolidPeso molecolare:475.62Sanguinarine
CAS:Sanguinarine (Pseudochelerythrine) is a specific inhibitor of Rac1b with anti-microbial, anti-oxidant and anti-inflammatory properties.Formula:C20H14NO4Purezza:99.04% - 99.76%Colore e forma:SolidPeso molecolare:332.33Clovamide
CAS:Trans-Clovamide (trans-Clovamide) is a naturally occurring caffeoyl conjugate identified in the antioxidant polyphenolic fraction of cocoa (T.Formula:C18H17NO7Purezza:97.12% - 97.68%Colore e forma:SolidPeso molecolare:359.33Salermide
CAS:Salermide is an inhibitor of Sirt1 and Sirt2, causing strong cancer-specific apoptotic cell death.Formula:C26H22N2O2Purezza:97.09% - 99.55%Colore e forma:SolidPeso molecolare:394.47Piperlongumine
CAS:Piperlongumine (Piplartine) is a natural alkaloid from Piper longum L.Formula:C17H19NO5Purezza:97.03% - 99.90%Colore e forma:SolidPeso molecolare:317.34LY2409881 trihydrochloride
CAS:LY2409881 trihydrochloride is a novel specific inhibitor of IKK2 (IC50: 30 nM); IC50 for IKK1 and other common kinases is at least one log higher.Formula:C24H32Cl4N6OSPurezza:≥95%Colore e forma:SolidPeso molecolare:594.43Cycleanine
CAS:Cycleanine has potent antibacterial, antifungal, antiplasmodial, and cytotoxic activities.
Formula:C38H42N2O6Purezza:98.04% - 99.57%Colore e forma:SolidPeso molecolare:622.75AMAROGENTIN
CAS:Amarogentin, extracted from Swertia/Gentiana roots, aids liver cancer prevention/treatment by affecting cell cycle and apoptosis.Formula:C29H30O13Purezza:99.98% - ≥95%Colore e forma:SolidPeso molecolare:586.54Epothilone B
CAS:Epothilone B (EPO 906) is a compound isolated from the myxobacterium Sorangium cellulosum.Formula:C27H41NO6SPurezza:99.79% - 99.84%Colore e forma:White PowderPeso molecolare:507.68Ref: TM-T6075
1mg35,00€2mg50,00€5mg66,00€10mg99,00€25mg215,00€50mg389,00€100mg567,00€1mL*10mM (DMSO)73,00€Pitavastatin calcium
CAS:Pitavastatin calcium (NK-104), a inhibitor of HMG-CoA reductase, lowers both total cholesterol and low-density lipoprotein cholesterol in animals and humans.Formula:C50H46CaF2N2O8Purezza:98.89% - >99.99%Colore e forma:White To Off-White PowderPeso molecolare:880.98RIPGBM
CAS:RIPGBM is a selective inducer of apoptosis in glioblastoma multiforme cancer stem cells (EC50: ≤500 nM).Formula:C26H21FN2O3Purezza:99.45%Colore e forma:SolidPeso molecolare:428.45Ref: TM-T16754
2mg35,00€5mg54,00€10mg93,00€25mg177,00€50mg318,00€100mg530,00€200mg677,00€1mL*10mM (DMSO)60,00€L-Glutamic acid
CAS:L-Glutamic acid is an agonist of glutamate receptors, including metabotropic glutamate receptors (mGluR), AMPA, NMDA, and KA. High-Quality, Low-Cost!Formula:C5H9NO4Purezza:99.14% - 99.55%Colore e forma:White Solid CrystallinePeso molecolare:147.13Pectolinarin
CAS:Pectolinarin is a Cirsium isolate with anti-inflammatory activity.Formula:C29H34O15Purezza:98% - 99.79%Colore e forma:SolidPeso molecolare:622.57SC144
CAS:SC144 is an orally active small-molecule gp130 inhibitor.Formula:C16H11FN6OPurezza:99.20%Colore e forma:SolidPeso molecolare:322.3PND-1186
CAS:PND-1186 (VS-4718) is a reversible and specific FAK inhibitor (IC50: 1.5 nM).Formula:C25H26F3N5O3Purezza:99.14% - 99.75%Colore e forma:SolidPeso molecolare:501.5SIRT7 inhibitor 97491
CAS:SIRT7 inhibitor 97491 is an HDAC inhibitor with high specificity for SIRT7 (IC50 = 325 nM). SIRT7 inhibitor 97491 promotes apoptosis through caspase pathway.Formula:C15H12ClN3OPurezza:99.79%Colore e forma:SolidPeso molecolare:285.73Ref: TM-T39233
1mg96,00€5mg235,00€10mg354,00€25mg597,00€50mg852,00€100mg1.159,00€1mL*10mM (DMSO)259,00€Bafetinib
CAS:Bafetinib (INNO-406): Dual Bcr-Abl/Lyn inhibitor; IC50: 5.8/19 nM; ineffective against T315I mutant, less on c-Kit/PDGFR.Formula:C30H31F3N8OPurezza:94.16% - 99.68%Colore e forma:SolidPeso molecolare:576.62Ref: TM-T6311
1mg34,00€2mg49,00€5mg74,00€10mg98,00€25mg150,00€50mg178,00€100mg333,00€200mg432,00€1mL*10mM (DMSO)95,00€PHT-427
CAS:PHT-427 (CS-0223) is a dual Akt (Ki: 2.7 μM) and PDPK1 (Ki: 5.2 μM) inhibitor (high-affinity binding for the PH domains of Akt and PDPK1).Formula:C20H31N3O2S2Purezza:97.54% - >99.99%Colore e forma:SolidPeso molecolare:409.61
