Neuroscienza
Gli inibitori in neuroscienze sono composti progettati per modulare l'attività di proteine, enzimi o recettori specifici all'interno del sistema nervoso. Questi inibitori sono cruciali per studiare i meccanismi molecolari alla base della funzione neuronale, della trasmissione sinaptica e delle malattie neurodegenerative. Mirando ai recettori dei neurotrasmettitori, ai canali ionici e alle vie di segnalazione, gli inibitori in neuroscienze aiutano a esplorare la funzione cerebrale e a sviluppare strategie terapeutiche per disturbi neurologici come l'Alzheimer, il Parkinson e l'epilessia. Presso CymitQuimica, offriamo una vasta gamma di inibitori in neuroscienze di alta qualità per supportare la tua ricerca in neurobiologia, neurofarmacologia e scienze cognitive.
Sottocategorie di "Neuroscienza"
- recettore 5-HT(1.025 prodotti)
- ACK(1 prodotti)
- AChR(642 prodotti)
- Citrato liasi ATP(17 prodotti)
- Recettore adrenergico(2.998 prodotti)
- BACE(37 prodotti)
- Beta amiloide(217 prodotti)
- CaMK(73 prodotti)
- COX(598 prodotti)
- Recettore della dopamina(445 prodotti)
- Ricettore GABA(370 prodotti)
- Gamma-secretasi(57 prodotti)
- GluR(265 prodotti)
- GlyT(26 prodotti)
- Recettore dell'istamina(385 prodotti)
- LRRK2(43 prodotti)
- Recettore della melatonina(26 prodotti)
- NMDAR(10 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(325 prodotti)
Mostrare 12 più sottocategorie
Trovati 5445 prodotti di "Neuroscienza"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
CaM kinase II inhibitor TFA salt
CaM kinase II inhibitor TFA salt (Autocamtide-2-related inhibitory peptide (TFA)) is a highly specific and potent inhibitor of CaMKII with an IC50 of 40 nM.
Formula:C66H117F3N22O21Purezza:>99.99%Colore e forma:SolidPeso molecolare:1611.77Metoclopramide
CAS:Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.Formula:C14H22ClN3O2Purezza:99.75%Colore e forma:SolidPeso molecolare:299.80Ocinaplon
CAS:Ocinaplon (DOV 273547) is a GABAA receptors modulator.Formula:C17H11N5OPurezza:99.81%Colore e forma:SolidPeso molecolare:301.3PSEM 89S TFA
CAS:PSEM 89S TFA is a brain-penetrant and selective ion channels agonist, and is orthogonally selective for Q79G and L141F, respectively.Formula:C18H23F3N2O5Purezza:99.9%Colore e forma:SolidPeso molecolare:404.38Glycopyrrolate
CAS:Glycopyrrolate: muscarinic antagonist, antispasmodic for GI issues, reduces salivation with anesthesia.Formula:C19H28BrNO3Purezza:99.41% - 99.64%Colore e forma:SolidPeso molecolare:398.33Dihydroergocristine mesylate
CAS:DHEC mesylate is a vasodilator and α-adrenergic antagonist used for vascular dementia and as a geroprotector.Formula:C36H45N5O8SPurezza:98.9% - 99.79%Colore e forma:SolidPeso molecolare:707.84Rotundine
CAS:Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Formula:C21H25NO4Purezza:99.8% - 99.91%Colore e forma:Off-White SolidPeso molecolare:355.43VU0152099
CAS:VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).Formula:C18H17N3O3SPurezza:98.46%Colore e forma:SolidPeso molecolare:355.41Alprenolol benzoate
CAS:Alprenolol benzoate is the benzoate salt of Alprenolol -- a beta blocker.Formula:C22H29NO4Colore e forma:SolidPeso molecolare:371.48Nitrocaramiphen hydrochloride
CAS:Nitrocaramiphen hydrochloride is a selective M1 muscarinic antagonist and inhibits binding to sigma sites in brain.Formula:C18H27ClN2O4Purezza:99.74%Colore e forma:SolidPeso molecolare:370.87Ansofaxine hydrochloride
CAS:Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).Formula:C24H32ClNO3Purezza:99.57% - 99.77%Colore e forma:SolidPeso molecolare:417.97α-Thujone
CAS:α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.Formula:C10H16OPurezza:97.02% - 98.41%Colore e forma:Less Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996) Colorless Or Almost Colorless Liquid With A Menthol- Like Odor (Albert-Puleo 1978; Budavari 1996)Peso molecolare:152.23Azeliragon
CAS:Azeliragon (TTP488) is an antagonist at the Receptor for Advanced Glycation End products; is evaluated as a potential treatment for patients with mild-to-Formula:C32H38ClN3O2Purezza:96.7% - 98.33%Colore e forma:SolidPeso molecolare:532.12LY2119620
CAS:LY2119620 is a specific, and allosteric agonist of human M2 and M4 muscarinic acetylcholine receptors.Formula:C19H24ClN5O3SPurezza:99.7%Colore e forma:SolidPeso molecolare:437.94Isoflurane
CAS:Isoflurane (Forane) is a stable, non-explosive inhalation anesthetic that has been reported to induce caspase-3 activation.Formula:C3H2ClF5OPurezza:98%Colore e forma:Clear Colorless Liquid LiquidPeso molecolare:184.49PiB
CAS:PiB (Pittsburgh Compound-B) is a standard for analysis of 11C-PiB. 11C-PiB is a β-amyloid PET imaging tracer for Alzheimer's disease diagnosis.
Formula:C14H12N2OSPurezza:97.02%Colore e forma:SolidPeso molecolare:256.32Tiagabine hydrochloride
CAS:Tiagabine hydrochloride, a nipecotic acid derivative, is an anticonvulsant and selective GABA reuptake inhibitor.Formula:C20H25NO2S2·HClPurezza:99.09% - 99.77%Colore e forma:White To Off-White SolidPeso molecolare:412.01VU0155094
CAS:VU0155094 (ML 397) is a positive allosteric modulator with differential activity at the various group III mGluRs.Formula:C24H24N2O4SPurezza:97.21%Colore e forma:SolidPeso molecolare:436.52Ref: TM-T9011
1mg62,00€5mg110,00€10mg161,00€25mg269,00€50mg371,00€100mg537,00€200mg710,00€1mL*10mM (DMSO)127,00€FLI-06
CAS:FLI-06 is a Notch signaling inhibitor (EC50: 2.3 μM).Formula:C25H30N2O5Purezza:99.81% - ≥98%Colore e forma:SolidPeso molecolare:438.52Ref: TM-T3075
1mg34,00€2mg49,00€5mg71,00€10mg94,00€25mg168,00€50mg295,00€100mg513,00€500mg1.125,00€1mL*10mM (DMSO)78,00€SSD114 HCl
CAS:SSD114 is a novel GABAB receptor positive allosteric modulator.Formula:C18H21ClF3N3OPurezza:99.03% - 99.95%Colore e forma:SolidPeso molecolare:387.83Ref: TM-T4522
2mg34,00€5mg50,00€10mg75,00€25mg111,00€50mg172,00€100mg290,00€200mg419,00€1mL*10mM (DMSO)46,00€Cyclopentolate Hydrochloride
CAS:Cyclopentolate Hydrochloride is a muscarinic acetylcholine receptors antagonist with Kis of 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively.Formula:C17H26ClNO3Purezza:99.91%Colore e forma:SolidPeso molecolare:327.85Hypidone hydrochloride
CAS:Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitorFormula:C18H23ClN2O2Purezza:99.82% - 99.93%Colore e forma:SolidPeso molecolare:334.84Pempidine HCl
CAS:Pempidine HCl, a nicotinic antagonist and former hypertension treatment, now mainly serves as a lab tool.Formula:C10H22ClNColore e forma:SolidPeso molecolare:191.74(+)-Kavain
CAS:(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.Formula:C14H14O3Purezza:97% - ≥95%Colore e forma:White Fine PowderPeso molecolare:230.26Isopropamide Iodide
CAS:Isopropamide iodide: long-acting anticholinergic, treats peptic ulcers, GI disorders, Alzheimer's.
Formula:C23H33IN2OPurezza:99.67%Colore e forma:SolidPeso molecolare:480.43Zacopride
CAS:Zacopride is a selective agonist of inward rectifier potassium current (I K1) channel, inhibiting ventricular arrhythmias without affecting atrial arrhythmias.Formula:C15H20ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:309.79Drofenine
CAS:Drofenin: anticonvulsant, anticholinergic, neurotropic, musculotropic, FIASMA.Formula:C20H31NO2Colore e forma:SolidPeso molecolare:317.47GSK2578215A
CAS:GSK2578215A is a potent and selective LRRK2 kinase inhibitor.Formula:C24H18FN3O2Purezza:99.57% - 99.94%Colore e forma:SolidPeso molecolare:399.42VU0119498
CAS:VU0119498 is a M1 muscarinic receptor agonist (EC50 = 3.1 μM) and pan mAChR M3, M5 positive allosteric modulator (PAM),and is a neuroprotective agent.Formula:C15H10BrNO2Purezza:97.56%Colore e forma:SolidPeso molecolare:316.15Olanzapine HCl
CAS:Olanzapine HCl, an FDA-approved atypical antipsychotic for schizophrenia and bipolar disorder, resembles clozapine and quetiapine.Formula:C17H21ClN4SColore e forma:SolidPeso molecolare:348.89Pirenperone
CAS:Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.Formula:C23H24FN3O2Purezza:99.2%Colore e forma:SolidPeso molecolare:393.457-Amino-4-(trifluoromethyl)coumarin
CAS:7-Amino-4-(trifluoromethyl)coumarin (Coumarin 151) is a 5-Hydroxytryptamine Receptor Subtype 1E (HTR1E) antagonist.Formula:C10H6F3NO2Purezza:97.31% - 97.84%Colore e forma:Yellow PowderPeso molecolare:229.16Cerlapirdine hydrochloride
CAS:Cerlapirdine/SAM-531, potent 5-HT6 antagonist, targets Alzheimer's and schizophrenia cognitive issues; phase II trials, promising efficacy, safe profile.Formula:C22H24ClN3O3SColore e forma:SolidPeso molecolare:445.96Tandospirone citrate
CAS:Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)Formula:C27H37N5O9Purezza:97.84% - 99.90%Colore e forma:SolidPeso molecolare:575.61RU 24969 free base
CAS:RU 24969 (5-methoxy-3-(1,2,3,6-tetrahydropyridin-4-yl)-1H-indole) is a selective agonist of 5-HT1A and 5-HT1B receptors.Formula:C14H16N2OPurezza:97.38%Colore e forma:SolidPeso molecolare:228.29Oxotremorine sesquifumarate
CAS:Oxotremorine sesquifumarate is a muscarinic agonist.
Formula:C12H18N2OC4H4O4Purezza:97.94%Colore e forma:SolidPeso molecolare:380.39SKF89976A HCl
CAS:SKF89976A: GABA uptake inhibitor, selective for GAT-1, passes blood-brain barrier, active in vivo (IC50: 0.13 μM hGAT-1).Formula:C22H25NO2Colore e forma:SolidPeso molecolare:335.44Hemicholinium 3
CAS:Hemicholinium 3 is a potent and selective choline uptake blocker.Formula:C24H34Br2N2O4Purezza:98% - 99.95%Colore e forma:SolidPeso molecolare:574.35Revefenacin
CAS:Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.Formula:C35H43N5O4Purezza:98.12%Colore e forma:SolidPeso molecolare:597.75Miltirone
CAS:Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.Formula:C19H22O2Purezza:99.22% - 99.66%Colore e forma:SolidPeso molecolare:282.38Flibanserin
CAS:Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.
Formula:C20H21F3N4OPurezza:99.37% - 99.93%Colore e forma:White PowderPeso molecolare:390.4L-838417 D9
CAS:L-838417 D9 (C-21191) is a novel deuterated subtype-selective GABAA positive allosteric modulator, acting as a partial agonist at α2, α3 and α5 subtypes[1].Formula:C19H10D9F2N7OPurezza:99.65%Colore e forma:SolidPeso molecolare:408.45Ref: TM-T22301
2mg34,00€5mg52,00€10mg71,00€25mg128,00€50mg200,00€100mg323,00€200mg447,00€1mL*10mM (DMSO)58,00€Phenibut (hydrochloride)
CAS:Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.Formula:C10H14ClNO2Purezza:99.93%Colore e forma:White Crystalline PowderPeso molecolare:215.68W-84 dibromide
CAS:W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.Formula:C32H44Br2N4O4Purezza:95.56%Colore e forma:SolidPeso molecolare:708.52Edrophonium chloride
CAS:Edrophonium chloride is an acetylcholinesterase (AChE) inhibitor that is known to prevent the breakdown of the neurotransmitter acetylcholine by bindingFormula:C10H16ClNOPurezza:97.41%Colore e forma:LiquidPeso molecolare:201.69Opiranserin hydrochloride
CAS:Opiranserin (VVZ-149) hydrochloride is a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A), with IC50s of 0.86 and 1.3 μMFormula:C21H35ClN2O5Purezza:99.33%Colore e forma:SolidPeso molecolare:430.97Ref: TM-T9833
1mg90,00€5mg215,00€10mg340,00€25mg618,00€50mg879,00€100mg1.224,00€500mg2.457,00€1mL*10mM (DMSO)236,00€Avagacestat
CAS:Avagacestat (BMS-708163) (BMS-708163) is a potent, selective, orally bioavailable γ-secretase inhibitor of Aβ40 and Aβ42 with IC50 of 0.3 nM and 0.27 nM,Formula:C20H17ClF4N4O4SPurezza:98.87% - 99.73%Colore e forma:SolidPeso molecolare:520.89Ref: TM-T6249
1mg38,00€5mg77,00€10mg116,00€25mg215,00€50mg310,00€100mg450,00€200mg605,00€1mL*10mM (DMSO)88,00€Clozapine N-Oxide
CAS:View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.Formula:C18H19ClN4OPurezza:98.65% - 99.94%Colore e forma:SolidPeso molecolare:342.82Orexin B, rat, mouse Acetate
Orexin B, rat, mouse Acetate (Rat orexin B) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.Formula:C128H219N45O36SPurezza:94.61%Colore e forma:SolidPeso molecolare:2996.45Eptapirone
CAS:Eptapirone (F 11440) is a highly effective and selective 5-HT1A receptor agonist with marked antidepressant and anxiolytic potential.Formula:C16H23N7O2Purezza:99.39% - 99.65%Colore e forma:SolidPeso molecolare:345.4Almotriptan
CAS:Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.Formula:C17H25N3O2SPurezza:99.85%Colore e forma:Light Yellow Or White PowerPeso molecolare:335.46Bitopertin
CAS:Bitopertin (Paliflutine) (RG1678, RO-4917838) is a potent inhibitor of glycine transporter 1 (GlyT1), with Ki of 8.1 nM for human hGlyT1b and IC50 of 22-25 nMFormula:C21H20F7N3O4SPurezza:98.57% - 98.71%Colore e forma:SolidPeso molecolare:543.46Rizatriptan benzoate
CAS:Rizatriptan benzoate (MK-462 Benzoate) selectively binds to and activates serotonin (5-HT) 1B receptors and 5-HT 1D receptors providing relief of migraineFormula:C22H25N5O2Purezza:99% - 99.79%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:391.47Ref: TM-T1512
10mg44,00€25mg74,00€50mg119,00€100mg173,00€200mg259,00€500mg437,00€1mL*10mM (DMSO)48,00€Trazodone
CAS:Trazodone (AF-1161), a 5-HT 2A/2C receptor antagonist, is used as an antidepressant for treating major anxiety disorders and depressive disorder.Formula:C19H22ClN5OPurezza:99.79% - 99.92%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:371.86Isocarboxazid
CAS:Isocarboxazid: a monoamine oxidase inhibitor used for various depression and anxiety disorders.Formula:C12H13N3O2Purezza:98.32% - 99.94%Colore e forma:SolidPeso molecolare:231.25Ref: TM-T4559
1mg34,00€2mg49,00€5mg74,00€10mg90,00€25mg164,00€50mg235,00€100mg350,00€500mg795,00€1mL*10mM (DMSO)82,00€Puerarin
CAS:Puerarin (Kakonein), also known as Kakonein, is a member of the class of compounds known as isoflavonoid C-glycosides. It is a 5-HT2C receptor antagonist.Formula:C21H20O9Purezza:98.90% - 99.21%Colore e forma:Yellow Brown Fine PowderPeso molecolare:416.38Tasimelteon
CAS:Tasimelteon (BMS-214778) is a melatonin receptor agonist that is used for the treatment of non-24 hour sleep-wake disorder in blind individuals.Formula:C15H19NO2Purezza:98.93% - 99.93%Colore e forma:SolidPeso molecolare:245.32ARN2966
CAS:ARN2966 is an inhibitor of amyloid precursor protein (APP)and amyloid-β (Aβ) secretion.Formula:C12H12N2OPurezza:99.52% - 99.86%Colore e forma:SolidPeso molecolare:200.24Ref: TM-T7490
1mg34,00€5mg74,00€10mg113,00€25mg222,00€50mg358,00€100mg530,00€500mg1.153,00€1mL*10mM (DMSO)82,00€Syk Inhibitor II dihydrochloride dihydrate
CAS:Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.Formula:C14H21Cl2F3N6O3Colore e forma:SolidPeso molecolare:449.26(-)-(S)-B-973B
CAS:(-)-(S)-B-973B is an effective allosteric agonist and a positive allosteric modulator of α7 nAChR.Formula:C24H26F2N6OPurezza:99.52%Colore e forma:SolidPeso molecolare:452.5Naratriptan
CAS:Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.Formula:C17H25N3O2SPurezza:99.08%Colore e forma:SolidPeso molecolare:335.47Ref: TM-T8666
1mg39,00€2mg50,00€5mg73,00€10mg92,00€25mg166,00€50mg240,00€100mg360,00€1mL*10mM (DMSO)88,00€Alosetron (Hydrochloride(1:X))
CAS:Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.Formula:C17H18ClN4OColore e forma:SolidPeso molecolare:329.11691Fluralaner
CAS:Fluralaner (A1443) is an isoxazoline ectoparasiticide.Formula:C22H17Cl2F6N3O3Purezza:99.72% - 99.99%Colore e forma:Solid PowderPeso molecolare:556.29Ginsenoside Rc
CAS:Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.
Formula:C53H90O22Purezza:98.83% - 99.56%Colore e forma:White PowderPeso molecolare:1079.27Cinanserin
CAS:Cinanserin is a serotonin 5-HT2 antagonist.Formula:C20H24N2OSColore e forma:SolidPeso molecolare:340.48IPSU
CAS:IPSU is an antagonist of OX2 receptor. IPSU Exhibits approximately six-fold selectivity for OX2 versus OX1 receptors.Formula:C23H27N5O2Purezza:97.05%Colore e forma:SolidPeso molecolare:405.49Ref: TM-T5503
2mg51,00€5mg86,00€10mg97,00€25mg200,00€50mg299,00€100mg432,00€200mg662,00€1mL*10mM (DMSO)92,00€Ipratropium Bromide
CAS:Ipratropium Bromide (Sch 1000) is an antagonist of muscarinic receptors and is used in COPD and asthma studies.Formula:C20H30BrNO3Purezza:99.92%Colore e forma:SolidPeso molecolare:412.37SCH-23390 hydrochloride
CAS:SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Formula:C17H19Cl2NOPurezza:98% - 99.83%Colore e forma:SolidPeso molecolare:324.24Ref: TM-T4369
1mg39,00€2mg50,00€5mg78,00€10mg97,00€25mg195,00€50mg369,00€100mg550,00€1mL*10mM (DMSO)78,00€GNE-7915
CAS:GNE-7915 is a highly potent, selective and brain-penetrable leucine-rich repeat kinase 2 (LRRK2) inhibitor.Formula:C19H21F4N5O3Purezza:98% - ≥95%Colore e forma:SolidPeso molecolare:443.4Ref: TM-T1945
5mg44,00€10mg58,00€25mg108,00€50mg177,00€100mg299,00€200mg389,00€500mg645,00€1mL*10mM (DMSO)48,00€MK-0752
CAS:MK-0752, a γ-secretase inhibitor, reduces Aβ40 production(IC50=5 nM).
Formula:C21H21ClF2O4SPurezza:98% - 99.55%Colore e forma:SolidPeso molecolare:442.9Vilazodone Hydrochloride
CAS:Vilazodone Hydrochloride (EMD 68843) , a partial agonist of 5-HT1A receptors and specific serotonin reuptake inhibitor (SSRI), is utilized in treating of theFormula:C26H27N5O2·HClPurezza:99.56% - >99.99%Colore e forma:SolidPeso molecolare:477.99lumateperone Tosylate
CAS:lumateperone Tosylate (ITI-007) is a 5-HT2A receptor antagonist, a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors.Formula:C31H36FN3O4SPurezza:95.83% - 99.95%Colore e forma:SolidPeso molecolare:565.7A-484954
CAS:A-484954 (A 484954) is a highly specific eukaryotic elongation factor-2 (eEF2, IC50: 280 nM) inhibitor.Formula:C13H15N5O3Purezza:97.47% - 99.86%Colore e forma:SolidPeso molecolare:289.29Ref: TM-TQ0137
1mg43,00€2mg56,00€5mg88,00€10mg144,00€25mg305,00€50mg543,00€100mg775,00€1mL*10mM (DMSO)103,00€Dihydroergotoxine mesylate
CAS:Dihydroergotoxine mesylate (Ergoloid mesylates) is mainly used to improve symptoms and physical symptoms of mental degeneration related to aging.Formula:C20H29N3O5SPurezza:99.39% - ≥95%Colore e forma:SolidPeso molecolare:423.53Metoclopramide hydrochloride hydrate
CAS:Metoclopramide hydrochloride hydrate (Metoclopramide monohydrochloride monohydrate) is a dopamine D2 antagonist that is a drug used for digestive dysfunction.Formula:C14H25Cl2N3O3Purezza:99.33%Colore e forma:SolidPeso molecolare:354.27MK-1064
CAS:MK-1064 (Urokinase inhibitor 1) is a selective orexin 2 receptor antagonist (2-SORA).Formula:C24H20ClN5O3Purezza:99.19% - 99.82%Colore e forma:SolidPeso molecolare:461.9Vortioxetine hydrobromide
CAS:Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33Formula:C18H22N2S·HBrPurezza:98.85% - 99.98%Colore e forma:SolidPeso molecolare:379.36Citalopram
CAS:Citalopram (Lu 10-171), a serotonin and 5-HT reuptake inhibitor.Citalopram has antidepressant activity and may be used to study dementia.Formula:C20H21FN2OPurezza:99.78% - 99.89%Colore e forma:SolidPeso molecolare:324.39HTT-D3
CAS:HTT-D3 is a Huntington splicing regulator that induces HTT mRNA degradation, leading to a reduction in HTT protein levels.
Formula:C23H25FN6Purezza:99.31%Colore e forma:SolidPeso molecolare:404.48γ-Secretase modulator 13
CAS:γ-Secretase modulator 13 is a γ-secretase modulator (GSMs) that can be used to study Alzheimer's disease and tumors.Formula:C22H23FN6SPurezza:99.79%Colore e forma:SolidPeso molecolare:422.52RTI-55 Hydrochloride
CAS:Prodotto controllatoStability Very Hygroscopic
Applications RTI-55 is a semi-synthetic alkaloid that is a cocaine analogue belonging to the phenyltropane group. RTI-55 acts as a dopamine reuptake inhibitor (DRI) with siginificant abuse potential. RTI-55 is used to assess the rate of dopamine neuron degradation in the brains of patients with Parkinson’s disease.
References Fujita, M. et al.: J. Chem. Neuroanat., 7, 13 (1994); Elmer, G.I. et al.: Pharmacol. Biochem. Behav., 53, 911 (1996); Coulter, C.L. et al.: Brain Res., 690, 217 (1995);Formula:C16H20INO2·ClHColore e forma:NeatPeso molecolare:421.7Ketanserin tartrate
CAS:Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.Formula:C26H28FN3O9Purezza:99.68%Colore e forma:SolidPeso molecolare:545.516-Cyano-7-nitroquinoxaline-2,3-dione
CAS:Prodotto controllatoStability Store Tightly Sealed at RT
Applications A potent, competitive kainate/quisqualate (non-NMDA) receptor antagonist. IC50 of tritiated ligands to rat cortical membranes by CNQX: AMPA, Kainate and CPP are 0.3mM, 1.5mM, and 25mM, respectively.
References Honore, et al. Science, 241, 701 (1988),Haas, H.S., et al.: Int. J. Oncol., 27, 867 (2005), Kobayashi, K., et al.: J. Pharmacol. Sci., 108, 517 (2008), Shabat-Simon, M., et al.: J. Neurosci., 28, 8406 (2008), Cruz, L.A., et al.: J. Med. Chem., 51, 5856 (2008),Formula:C9H4N4O4Colore e forma:NeatPeso molecolare:232.15EasyStep Human GH(Growth Hormone) ELISA Kit
The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Human GH, and the Human GH standard plate wells that pre-coated using protein-related techniques are provided separately. Standard/Sample Diluent Buffer or samples are added to the appropriate microtiter plate wells ,then added a HRP-conjugated antibody specific to Human GH. After TMB substrate solution is added, only those wells that contain Human GH and HRP-conjugated antibody will exhibit a change in color. The enzyme-substrate reaction is terminated by the addition of sulphuric acid solution and the color change is measured spectrophotometrically at a wavelength of 450nm ± 10nm. The concentration of Human GH in the samples is then determined by comparing the OD of the samples to the standard curve.Colore e forma:Colourless TransparentliquidMonepantel
CAS:Monepantel (AAD1566) is an organic anthelmintic and an antagonist of nAChRs from roundworms and esophageostomy.Formula:C20H13F6N3O2SPurezza:99.83%Colore e forma:White PowderPeso molecolare:473.39Ref: TM-T16126
1mg93,00€5mg236,00€10mg340,00€25mg670,00€50mg964,00€100mg1.378,00€1mL*10mM (DMSO)259,00€EasyStep Human EFNA1(Ephrin A1) ELISA Kit
The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Human EFNA1, and the Human EFNA1 standard plate wells that pre-coated using protein-related techniques are provided separately. Standard/Sample Diluent Buffer or samples are added to the appropriate microtiter plate wells ,then added a HRP-conjugated antibody specific to Human EFNA1. After TMB substrate solution is added, only those wells that contain Human EFNA1 and HRP-conjugated antibody will exhibit a change in color. The enzyme-substrate reaction is terminated by the addition of sulphuric acid solution and the color change is measured spectrophotometrically at a wavelength of 450nm ± 10nm. The concentration of Human EFNA1 in the samples is then determined by comparing the OD of the samples to the standard curve.Colore e forma:Colourless TransparentliquidSetiptiline
CAS:Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.Formula:C19H19NPurezza:98.05% - 98.07%Colore e forma:SolidPeso molecolare:261.36Hordenine-d6
CAS:Prodotto controllatoApplications A labelled phenethylamine alkaloid with antibacterial and antibiotic properties found mainly in plants from the cactaceae family. It showed effects similar to Cytosine (C998950) and acted as a depressant on the central nervous system (CNS) during animal testing.
References Aliev, K.U. et al.: Med. Zhur. Uzbek., 8, 71 (1966); Ghosal, S. et al. Planta Medica, 22, 434 (1972); Starha, R. et al.: Biochem. Sys. Ecol., 27, 839 (1999);Formula:C10H9D6NOColore e forma:Light Beige To Light BrownPeso molecolare:171.27Riluzole
CAS:Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.
Formula:C8H5F3N2OSPurezza:99.71% - 99.88%Colore e forma:PowderPeso molecolare:234.2Latrepirdine dihydrochloride
CAS:Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.Formula:C21H25N3·2HClPurezza:98.45%Colore e forma:SolidPeso molecolare:392.37Darigabat
CAS:Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.Formula:C22H21FN4O3SPurezza:98.42% - 99.29%Colore e forma:SolidPeso molecolare:440.49Citalopram-d6
CAS:Prodotto controllatoApplications Labelled Citalopram (C505000), an inhibitor of serotonin (5-HT) uptake. Used as an antidepressant.
References Christensen, A.V., et al.: Eur. J. Pharmacol., 41, 153 (1977), Keller, M.B., et al.: J. Clin. Psychiatry, 61, 896 (2000), Von Moltke, L.L., et al.: Drug Metab. Dispos., 29, 1102 (2001),Formula:C202H6H15FN2OColore e forma:NeatPeso molecolare:330.43Oxazolam
CAS:Prodotto controllatoApplications A psychotropic agent with anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant properties. It is a precursor to the active substance Desmethyldiazepam (D291595).
References Ochs, H.R. et al.: J. Clin. Pharmacol., 24, 446 (1984); Takagi, H. et al.: Nip. Yakur. Zas., 66, 134 (1970);Formula:C18H17ClN2O2Colore e forma:NeatPeso molecolare:328.79SB 243213
CAS:SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.Formula:C22H19F3N4O2Purezza:98.78% - 99.86%Colore e forma:SolidPeso molecolare:428.41Tandospirone
CAS:Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.Formula:C21H29N5O2Purezza:99.94%Colore e forma:SolidPeso molecolare:383.49Ref: TM-TQ0315
2mg37,00€5mg54,00€10mg87,00€25mg141,00€50mg193,00€100mg308,00€200mg441,00€1mL*10mM (DMSO)59,00€L-368,899 hydrochloride
CAS:L-368,899 hydrochloride is an OXTR antagonist that prevents oxytocin-induced antiabnormal pain and anti-nausea, and may be used in the study of depression.Formula:C26H43ClN4O5S2Purezza:99.59%Colore e forma:SolidPeso molecolare:591.23Ref: TM-T11794
2mg105,00€5mg147,00€10mg230,00€25mg439,00€50mg685,00€100mg964,00€1mL*10mM (DMSO)200,00€RO7185876
CAS:RO7185876 is a selective gamma secretase modulator, which can be used in the study of Alzheimer's disease.Formula:C25H28F3N7Purezza:99.50%Colore e forma:SolidPeso molecolare:483.532(R)-Mirtazapine
CAS:(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.Formula:C17H19N3Purezza:99.75%Colore e forma:SolidPeso molecolare:265.35WAY-100635 maleate
CAS:WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).Formula:C25H34N4O2·xC4H4O4Purezza:99.96%Colore e forma:White SolidPeso molecolare:538.645Ref: TM-T3453
2mg46,00€5mg66,00€10mg95,00€25mg159,00€50mg226,00€100mg334,00€500mg807,00€1mL*10mM (DMSO)79,00€4-Hydroxyindole
CAS:4-Hydroxyindole: aromatic, antioxidant, used in cancer treatment and preventing neurodegenerative diseases.Formula:C8H7NOPurezza:97.05% - 98.13%Colore e forma:Off-White Cyrstalline SolidPeso molecolare:133.15
