Neuroscienza
Gli inibitori in neuroscienze sono composti progettati per modulare l'attività di proteine, enzimi o recettori specifici all'interno del sistema nervoso. Questi inibitori sono cruciali per studiare i meccanismi molecolari alla base della funzione neuronale, della trasmissione sinaptica e delle malattie neurodegenerative. Mirando ai recettori dei neurotrasmettitori, ai canali ionici e alle vie di segnalazione, gli inibitori in neuroscienze aiutano a esplorare la funzione cerebrale e a sviluppare strategie terapeutiche per disturbi neurologici come l'Alzheimer, il Parkinson e l'epilessia. Presso CymitQuimica, offriamo una vasta gamma di inibitori in neuroscienze di alta qualità per supportare la tua ricerca in neurobiologia, neurofarmacologia e scienze cognitive.
Sottocategorie di "Neuroscienza"
- recettore 5-HT(1.025 prodotti)
- ACK(1 prodotti)
- AChR(647 prodotti)
- Citrato liasi ATP(17 prodotti)
- Recettore adrenergico(3.024 prodotti)
- BACE(37 prodotti)
- Beta amiloide(230 prodotti)
- CaMK(73 prodotti)
- COX(602 prodotti)
- Recettore della dopamina(445 prodotti)
- Ricettore GABA(373 prodotti)
- Gamma-secretasi(62 prodotti)
- GluR(265 prodotti)
- GlyT(26 prodotti)
- Recettore dell'istamina(385 prodotti)
- LRRK2(43 prodotti)
- Recettore della melatonina(26 prodotti)
- NMDAR(10 prodotti)
- Recettore OX(41 prodotti)
- Recettore degli oppioidi(327 prodotti)
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Trovati 5637 prodotti di "Neuroscienza"
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VU0364770
CAS:VU0364770 (VU 0364770)(EC50=1.1 μM), a positive allosteric modulator(PAM) of mGlu4, shows insignificant activity at 68 other receptors, including other mGluFormula:C12H9ClN2OPurezza:99.65% - >99.99%Colore e forma:SolidPeso molecolare:232.67TAE-1
CAS:TAE-1 is an inhibitor of amyloid-β fibril formation and aggregation. It inhibits cholinesterases AChE and BuChE with IC50 of 0.3 μM and 3.9 μM, respectively.
Formula:C39H51I3N6O9Purezza:94.58%Colore e forma:SolidPeso molecolare:1128.57γ-Mangostin
CAS:Gamma-Mangostin (Normangostin) has free radical scavenging activity, and antiproliferative and apoptotic activity. Gamma-Mangostin is an antihypertensive agent.Formula:C23H24O6Purezza:98.55% - 99.08%Colore e forma:SolidPeso molecolare:396.434-Acetamidobutanoic acid
CAS:4-Acetamidobutanoic acid, a GABA derivative in eukaryotes, found in blood, feces, urine, and human prostate.Formula:C6H11NO3Purezza:98.51%Colore e forma:SolidPeso molecolare:145.16VUF 10166
CAS:VUF10166 is a novel, potent and competitive antagonist for 5-HT3A receptor with Ki of 0.04 nM, its affinity at 5-HT3AB receptor is significantly lower.Formula:C13H15ClN4Purezza:99.66%Colore e forma:SolidPeso molecolare:262.74(2S)-6-Prenylnaringenin
CAS:(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.Formula:C20H20O5Purezza:99.47%Colore e forma:SolidPeso molecolare:340.37SR 57227 hydrochloride
CAS:SR 57227A (SR 57227 hydrochloride) is a potent, orally active and selective 5-HT3 receptor agonist. It with ability to cross the blood brain barrier.Formula:C10H14ClN3·HClPurezza:99.89%Colore e forma:SolidPeso molecolare:248.15Semax acetate(80714-61-0 free base)
CAS:Semax acetate is a synthetic peptide analog of adrenocorticotropic hormone (ACTH) that has neuroprotective, analgesic, and anxiolytic properties.Formula:C39H55N9O12SPurezza:99.46%Colore e forma:SolidPeso molecolare:873.98MTEP hydrochloride
CAS:MTEP hydrochloride (MTEP) is non-competitive mGlu5 antagonist (IC50 and Ki of 5 nM and 16 nM, respectively)Formula:C11H9ClN2SPurezza:99.58%Colore e forma:SolidPeso molecolare:236.72Tiagabine hydrochloride
CAS:Tiagabine hydrochloride, a nipecotic acid derivative, is an anticonvulsant and selective GABA reuptake inhibitor.Formula:C20H25NO2S2·HClPurezza:99.09% - 99.77%Colore e forma:White To Off-White SolidPeso molecolare:412.01SB-649868
CAS:SB-649868 (GSK649868) is a potent and selective orally active antagonist of orexin(pKi =9.4 and 9.5 at the OX1 and OX2 receptor, respectively).Formula:C26H24FN3O3SPurezza:99.53%Colore e forma:SolidPeso molecolare:477.55Ref: TM-T5498
2mg34,00€5mg71,00€1mL*10mM (DMSO)86,00€10mg110,00€25mg225,00€50mg366,00€100mg587,00€200mg788,00€MPEP hydrochloride
CAS:MPEP hydrochloride is an effective and highly specific non-competitive antagonist at the mGlu5 receptor subtype (IC50: 36 nM).Formula:C14H12ClNPurezza:99.87% - >99.99%Colore e forma:SolidPeso molecolare:229.7Ladostigil hydrochloride
CAS:Ladostigil hydrochloride: oral dual cholinesterase and MAO-B/AChE inhibitor; IC50s: 37.1 & 31.8 μM; potential for depression and Alzheimer's research.Formula:C16H21ClN2O2Colore e forma:SolidPeso molecolare:308.8Azeliragon HCl
CAS:Azeliragon: potent oral RAGE inhibitor, blocks Alzheimer's-linked amyloid brain entry.Formula:C32H40Cl3N3O2Colore e forma:SolidPeso molecolare:605.04Eltoprazine
CAS:Eltoprazine(DU28853) is a serenic or antiaggressive agent which as an agonist at the 5-HT1A and 5-HT1B receptors and as an antagonist at the 5-HT2C receptor.Formula:C12H16N2O2Colore e forma:SolidPeso molecolare:220.27QNZ46
CAS:QNZ46 is a NR2C/NR2D-selective NMDA receptor non-competitive antagonist.
Formula:C24H17N3O6Purezza:99.65%Colore e forma:SolidPeso molecolare:443.41Cinanserin
CAS:Cinanserin is a serotonin 5-HT2 antagonist.Formula:C20H24N2OSColore e forma:SolidPeso molecolare:340.483,5-Bis(4-nitrophenoxy)benzoic acid
CAS:3,5-Bis(4-nitrophenoxy)benzoic acid (Compound W) is an inhibitor of γ-secretase. It decreases the released levels of Aβ42 and notch-1 Aβ-like peptide 25.Formula:C19H12N2O8Purezza:99.14%Colore e forma:SolidPeso molecolare:396.31α-Conotoxin MII acetate
α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.Formula:C69H107N23O24S4Purezza:94.82% - 97.79%Colore e forma:SolidPeso molecolare:1770.99SSR504734
CAS:SSR504734 is a novel potent glycine transporter 1 (GlyT1) inhibitor.Formula:C20H20ClF3N2OColore e forma:SolidPeso molecolare:396.83YO-01027
CAS:YO-01027 (DBZ) is a potent γ-secretase inhibitor.Formula:C26H23F2N3O3Purezza:97.21% - 99.58%Colore e forma:SolidPeso molecolare:463.48(R)-baclofen
CAS:(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.Formula:C10H12ClNO2Purezza:97.20% - 98.94%Colore e forma:SolidPeso molecolare:213.666-fluoro-DL-Tryptophan
CAS:6-fluoro-DL-Tryptophan is an inhibitor of serotonin (5-HT) synthesis.Formula:C11H11FN2O2Purezza:99.25%Colore e forma:Off-White PowderPeso molecolare:222.22Nemifitide acetate(173240-15-8 free base)
Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.Formula:C35H47FN10O8Purezza:97.97%Colore e forma:SolidPeso molecolare:754.85Neurotensin TFA
Neurotensin TFA (39379-15-2) is a 13-amino acid neuropeptide with opioid-independent pain relief, acting in the CNS and gut, linked to numerous disorders.Formula:C80H122F3N21O22Purezza:99.41%Colore e forma:SolidPeso molecolare:1786.985-Benzyloxygramine
CAS:5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.Formula:C18H20N2OPurezza:99.13%Colore e forma:SolidPeso molecolare:280.36β-Amyloid 15-21 acetate
β-Amyloid 15-21 acetate (Beta-Amyloid (15-21) acetate) is a fragment of Amyloid-β peptide, maybe used in the research of neurological disease.Formula:C45H69N9O11Purezza:99.62%Colore e forma:SolidPeso molecolare:912.1FLI-06
CAS:FLI-06 is a Notch signaling inhibitor (EC50: 2.3 μM).Formula:C25H30N2O5Purezza:99.81% - ≥98%Colore e forma:SolidPeso molecolare:438.52Ref: TM-T3075
1mg34,00€2mg49,00€5mg71,00€1mL*10mM (DMSO)78,00€10mg94,00€25mg168,00€50mg295,00€100mg513,00€500mg1.125,00€Temgicoluril
CAS:Temgicoluril (mebikar) acts on GABA Receptor.Formula:C8H14N4O2Purezza:99.8%Colore e forma:SolidPeso molecolare:198.22Donepezil Hydrochloride
CAS:Donepezil HCl(Aricept) is a selective and effective AChE inhibitor for bAChE and hAChE (IC50: 8.12/11.6 nM).Formula:C24H29NO3·HClPurezza:99.55% - 99.8%Colore e forma:White To Off-White Crystalline SolidPeso molecolare:415.96Verubecestat
CAS:Verubecestat (MK-8931) (MK-8931) is an effective and specific β-secretase inhibitor and β-site APP-cleaving enzyme 1 inhibitor or BACE1 protein inhibitor.Formula:C17H17F2N5O3SPurezza:94.64% - 99.55%Colore e forma:SolidPeso molecolare:409.41Ref: TM-T7011
2mg38,00€5mg57,00€1mL*10mM (DMSO)63,00€10mg84,00€25mg144,00€50mg205,00€100mg334,00€500mg782,00€Dasotraline hydrochloride
CAS:Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.Formula:C16H16Cl3NPurezza:98.92% - 99.6%Colore e forma:SolidPeso molecolare:328.66Clozapine N-Oxide
CAS:View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.Formula:C18H19ClN4OPurezza:98.65% - 99.94%Colore e forma:SolidPeso molecolare:342.82SEN12333
CAS:SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonistFormula:C20H25N3O2Purezza:99.02%Colore e forma:SolidPeso molecolare:339.43Ref: TM-T23348
2mg37,00€5mg54,00€1mL*10mM (DMSO)59,00€10mg90,00€25mg164,00€50mg255,00€100mg409,00€200mg590,00€Frentizole
CAS:Frentizole, an immunosuppressive agent, is an inhibitor of the Aβ-ABAD interactionFormula:C15H13N3O2SPurezza:99.82%Colore e forma:SolidPeso molecolare:299.35Ritanserin
CAS:Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Formula:C27H25F2N3OSPurezza:99.77% - 99.89%Colore e forma:SolidPeso molecolare:477.57SSD114 HCl
CAS:SSD114 is a novel GABAB receptor positive allosteric modulator.Formula:C18H21ClF3N3OPurezza:99.03% - 99.95%Colore e forma:SolidPeso molecolare:387.83Ref: TM-T4522
2mg34,00€1mL*10mM (DMSO)46,00€5mg50,00€10mg75,00€25mg111,00€50mg172,00€100mg290,00€200mg419,00€LY2811376
CAS:LY2811376, an orally available non-peptidic β-secretase(BACE1) inhibitor (IC50: 239-249 nM), can decrease Aβ secretion (EC50: 300 nM).Formula:C15H14F2N4SPurezza:99% - 99.01%Colore e forma:SolidPeso molecolare:320.36Ref: TM-T2639
1mg50,00€2mg70,00€5mg116,00€1mL*10mM (DMSO)116,00€10mg195,00€25mg354,00€50mg530,00€100mg758,00€N-Desmethylclozapine
CAS:N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.Formula:C17H17ClN4Purezza:97.25% - 99.83%Colore e forma:Yellow Crystalline SolidPeso molecolare:312.8Ref: TM-T5158
2mg34,00€5mg48,00€1mL*10mM (DMSO)58,00€10mg79,00€25mg152,00€50mg235,00€100mg344,00€200mg490,00€L-745870 trihydrochloride
CAS:L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.Formula:C18H22Cl4N4Purezza:97.52%Colore e forma:SolidPeso molecolare:436.21Orexin 2 Receptor Agonist
CAS:Orexin 2 Receptor Agonist (OX2R) is an effective (EC50: 23 nM) and OX2R-selective (OX1R/OX2R EC50 ratio: 70) agonist.Formula:C32H34N4O5SPurezza:98.26% - 99.43%Colore e forma:SolidPeso molecolare:586.7Ref: TM-T3177
2mg39,00€5mg60,00€10mg75,00€1mL*10mM (DMSO)77,00€25mg130,00€50mg220,00€100mg323,00€200mg447,00€Syn-Ake acetate
CAS:Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.Formula:C19H29N5O3·2(C2H4O2)Purezza:99.60%Colore e forma:SolidPeso molecolare:495.58Azaphen
CAS:Azaphen (Pipofezin hydrochloride) is the reuptake of serotonin inhibitor.with antidepressant action and has sedative effects, suggesting antihistamine activity.Formula:C16H21Cl2N5OPurezza:97.62%Colore e forma:SolidPeso molecolare:370.28Piperazine
CAS:Piperazine (1,4-Diazacyclohexane), a gamma-aminobutyric acid (GABA) agonist, serves as a crucial building block and core component in a wide range of marketed drugs known for their varied pharmacological activities.Formula:C4H10N2Colore e forma:SolidPeso molecolare:86.14Chlorprothixene
CAS:Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.Formula:C18H18ClNSPurezza:98.77% - 99.756%Colore e forma:Pale Yellow Crystals SolidPeso molecolare:315.86NGB 2904
CAS:NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).Formula:C28H29Cl2N3OPurezza:98.79%Colore e forma:SolidPeso molecolare:494.46Ref: TM-T28167
500mgPrezzo su richiesta2mg38,00€5mg55,00€1mL*10mM (DMSO)72,00€10mg86,00€25mg155,00€50mg264,00€100mg374,00€Piperacetazine
CAS:Piperacetazine (Piperacetazinum), an antipsychotic prodrug, is used forschizophrenia.Formula:C24H30N2O2SPurezza:99.9% - 99.92%Colore e forma:SolidPeso molecolare:410.572'MeO6MF
CAS:2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functionalFormula:C17H14O3Purezza:99.28% - 99.63%Colore e forma:SolidPeso molecolare:266.29Ref: TM-T8887
1mg49,00€1mL*10mM (DMSO)96,00€5mg102,00€10mg152,00€25mg243,00€50mg340,00€100mg460,00€200mg627,00€A 582941 HCl (848591-90-2(free base))
A-582941 is a alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing propertiesFormula:C17H21ClN4Purezza:99.83%Colore e forma:SolidPeso molecolare:316.83Ref: TM-T8725
1mg58,00€1mL*10mM (DMSO)116,00€5mg118,00€10mg172,00€25mg281,00€50mg396,00€100mg537,00€200mg712,00€DMAB-anabaseine dihydrochloride
CAS:DMAB-anabaseine dihydrochloride (N,N-dimethyl-4-[(E)-(6-pyridin-3-yl-3,4-dihydro-2H-pyridin-5-ylidene)methyl]aniline;dihydrochloride) is an α7-containingFormula:C19H23Cl2N3Purezza:99.91%Colore e forma:SolidPeso molecolare:364.318-Hydroxy-DPAT hydrobromide
CAS:8-Hydroxy-DPAT hydrobromide (8-OH-DPAT hydrobromide) (8-OH-DPAT hydrobromide) is a potent and selective 5-HT1A agonist with a pIC50 of 8.19.Formula:C16H26BrNOPurezza:98.90% - 99.99%Colore e forma:SolidPeso molecolare:328.29Donepezil
CAS:Donepezil (Aricept) is a piperidine-based, potent, specific, and reversible inhibitor of acetylcholinesterase (AChE).
Formula:C24H29NO3Purezza:99.69%Colore e forma:White Or Almost White Crystal PowderPeso molecolare:379.493-MATIDA
CAS:3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a).Formula:C8H9NO4SPurezza:99.75% - 99.96%Colore e forma:SolidPeso molecolare:215.23Ref: TM-T3486
2mg34,00€5mg49,00€1mL*10mM (DMSO)49,00€10mg79,00€25mg145,00€50mg227,00€100mg339,00€200mg482,00€OXA (17-33) acetate
OXA (17-33) acetate is a more potent agonist of orexin-1 receptor (OX1, EC50 = 8.29 nM)) over OX2 (EC50 = 187 nM).Formula:C79H125N23O22Purezza:98.52%Colore e forma:SolidPeso molecolare:1748.98LP-922761 hydrate
LP-922761 hydrate: selective AAK1 inhibitor; IC50: 4.8 nM (enzyme), 7.6 nM (cellular); also inhibits BIKE (IC50: 24 nM); inert to GAK, opioids, α2, GABAa.Formula:C21H28N6O4Colore e forma:SolidPeso molecolare:414.98LOX-IN-3 dihydrochloride monohydrate
CAS:LOX-IN-3 dihydrochloride monohydrate is an oral lysyl oxidase inhibitor for research in fibrosis, cancer, and angiogenesis.Formula:C13H17Cl2FN2O3SColore e forma:SolidPeso molecolare:371.25ARC-239
CAS:ARC-239 is an agonist of α2-adrenergic receptor.Formula:C24H29N3O3Colore e forma:SolidPeso molecolare:407.51Cyclopentolate Hydrochloride
CAS:Cyclopentolate Hydrochloride is a muscarinic acetylcholine receptors antagonist with Kis of 1.62, 27.5, and 2.63 nM for M1, M2, and M3 receptors, respectively.Formula:C17H26ClNO3Purezza:99.91%Colore e forma:SolidPeso molecolare:327.85Pikamilone
CAS:Pikamilone (Picamilon) is an intelligent medicine.Formula:C10H12N2O3Purezza:99.38%Colore e forma:White Crystalline PowderPeso molecolare:208.21Loxapine hydrochloride
CAS:Loxapine hydrochloride, an oral anti-psychotic, inhibits dopamine and blocks 5-HT receptors.Formula:C18H19Cl2N3OColore e forma:SolidPeso molecolare:364.27Myristicin
CAS:Myristicin is a natural spice extract with antibacterial, anti-inflammatory, and hepatoprotective properties, and can induce apoptosis.
Formula:C11H12O3Purezza:99.828%Colore e forma:LiquidPeso molecolare:192.21Syk Inhibitor II dihydrochloride dihydrate
CAS:Potent, selective ATP-competitive Syk Inhibitor II (IC50: 41 nM), with anti-allergic properties, in dihydrochloride dihydrate form.Formula:C14H21Cl2F3N6O3Colore e forma:SolidPeso molecolare:449.26Hypidone hydrochloride
CAS:Hypidone hydrochloride (YL0919) is a novel antidepressant candidate with dual activity as a 5-HT1A receptor agonist and a selective serotonin reuptake inhibitorFormula:C18H23ClN2O2Purezza:99.82% - 99.93%Colore e forma:SolidPeso molecolare:334.84Dicyclomine
CAS:Dicyclomine: oral muscarinic antagonist, eases GI muscle spasms, high affinity for M1/M2 receptors, Ki of 5.1 nM/54.6 nM.Formula:C19H35NO2Colore e forma:SolidPeso molecolare:309.49Fesoterodine
CAS:Fesoterodine is an oral mAChR blocker (pKi: 7.3-8.0) for M1-M5, used to treat OAB.Formula:C26H37NO3Purezza:97.1%Colore e forma:SolidPeso molecolare:411.58m-Chlorophenylbiguanide hydrochloride
CAS:m-Chlorophenylbiguanide hydrochloride is a 5-HT3 receptor agonist.Formula:C8H11Cl2N5Purezza:99.43% - 99.87%Colore e forma:SolidPeso molecolare:248.11Xanthotoxol
CAS:Xanthotoxol (Psoralen) is a bioactive furocoumarin with anti-inflammatory, antioxidant, 5-HT antagonist, and neuroprotective properties.Formula:C11H6O4Purezza:98.44% - 99.97%Colore e forma:SolidPeso molecolare:202.16Solifenacin
CAS:Solifenacin (YM905 free base) (YM905 free base) is a novel muscarinic receptor antagonist, its pKis for M1, M2 and M3 receptors is of 7.6, 6.9 and 8.0,Formula:C23H26N2O2Purezza:99.87%Colore e forma:SolidPeso molecolare:362.46Propantheline
CAS:Propantheline: oral muscarinic receptor blocker for smooth muscle issues, hyperhidrosis, and bladder control.Formula:C23H30NO3Colore e forma:SolidPeso molecolare:368.494BP-TQS
CAS:4BP-TQS is an allosteric agonist of α7 nAChRs.Formula:C18H17BrN2O2SPurezza:99.96%Colore e forma:SolidPeso molecolare:405.31LY 2886721 Hydrochloride
CAS:Potent, selective BACE inhibitor; IC50 of 10.2 nM (BACE2) & 20.3 nM (BACE1). >5000x selectivity vs. other proteases. Lowers Aβ & sAPPβ in Alzheimer's mice.Formula:C18H17ClF2N4O2SColore e forma:SolidPeso molecolare:426.87Cyclopiazonic acid
CAS:Cyclopiazonic acid (CPA) is a neurotoxic secondary metabolite (SM) made by A.Formula:C20H20N2O3Purezza:99.27% - 99.80%Colore e forma:SolidPeso molecolare:336.38Ondansetron hydrochloride
CAS:Ondansetron hydrochloride (Zofran) is a serotonin 5-HT3 receptor antagonist, used to prevent nausea and vomiting caused by cancer chemotherapy, and radiationFormula:C18H19N3O·HClPurezza:99.78%Colore e forma:White PowderPeso molecolare:329.82Autocamtide 2 TFA(129198-88-5 free base)
Autocamtide 2 TFA, selective CaMKII peptide substrate, used in its activity assay.Formula:C67H119F3N22O22Purezza:98%Colore e forma:SolidPeso molecolare:1641.79Alosetron (Hydrochloride(1:X))
CAS:Alosetron Hydrochloride is a selective 5-HT3 antagonist for treating IBS.Formula:C17H18ClN4OColore e forma:SolidPeso molecolare:329.11691GALANTHAMINONE
CAS:Galanthaminone ((-)-Narwedine) is a cholinesterase (AChE) inhibitor, used for the treatment of mild to moderate Alzheimer's disease and other memory impairmentsFormula:C17H19NO3Purezza:99.93%Colore e forma:White To Off-White ChemicalPeso molecolare:285.34Ref: TM-T7114
2mg39,00€5mg58,00€1mL*10mM (DMSO)84,00€10mg93,00€25mg144,00€50mg200,00€100mg290,00€200mg414,00€Piboserod hydrochloride
CAS:Piboserod HCl is a selective antagonist of 5-HT4 and muscarinic receptor.Formula:C22H32ClN3O2Colore e forma:SolidPeso molecolare:405.96VU0238441
CAS:VU0238441 is agonist of Muscarinic acetylcholine receptor M5 (human) with EC50 of 2.1μM.Formula:C16H9ClF3NO2Purezza:100%Colore e forma:SolidPeso molecolare:339.7CRANAD 2
CAS:CRANAD-2, a near-infrared probe, detects amyloid-beta in vivo, increasing fluorescence 70x and shifting blue 90 nm upon binding.Formula:C23H25BF2N2O2Purezza:99.44%Colore e forma:Dark Blue To Black PowderPeso molecolare:410.27JI130
CAS:JI130 hinders Hes1 transcription repression; notably shrinks pancreatic tumor volume in mice.Formula:C23H24N2O3Purezza:99.61%Colore e forma:SolidPeso molecolare:376.45JNJ16259685
CAS:JNJ16259685 (TN.T 16259685) is a selective mGluR1 antagonist, and inhibits the synaptic activation of mGluR1 in a concentration-dependent manner with IC50 of 19Formula:C20H23NO3Purezza:98.31%Colore e forma:SolidPeso molecolare:325.4Ref: TM-T5512
1mg46,00€2mg62,00€5mg95,00€1mL*10mM (DMSO)95,00€10mg133,00€25mg278,00€50mg424,00€100mg620,00€Naratriptan hydrochloride
CAS:Naratriptan Hydrochloride, a selective 5-HT1 receptor agonist with anti-migraine effect, induces vasoconstriction and reduces inflammation in migraines.Formula:C17H25N3O2S·HClPurezza:99.17% - 99.93%Colore e forma:Beige SolidPeso molecolare:371.934,4'-DIMETHOXYBENZIL
CAS:4,4'-Dimethoxybenzil (p-Anisil) is a human intestinal carboxyl esterase (hiCE) inhibitor( Ki : 70 nM).Formula:C16H14O4Purezza:99.04%Colore e forma:Yellow Fine Crystalline PowderPeso molecolare:270.28Lu AF21934
CAS:Lu AF21934 is a brain-penetrant and selective mGlu4 receptor positive allosteric modulator (IC50: 500 nM, human).Formula:C14H16Cl2N2O2Purezza:99.79%Colore e forma:SolidPeso molecolare:315.2Rivanicline hemioxalate
Rivanicline hemioxalate is a selective α4β2 nicotinic receptor agonist (K i =26 nM), over 1,000x preference to α7 (K i =3.6 μM), with limited side effects.Formula:C12H16N2O4Purezza:98%Colore e forma:SolidPeso molecolare:207.23Flibanserin
CAS:Flibanserin (Girosa) is a serotonergic antidepressant used to treat hypoactive sexual desire disorder.
Formula:C20H21F3N4OPurezza:99.37% - 99.93%Colore e forma:White PowderPeso molecolare:390.4Trihexyphenidyl hydrochloride
CAS:Trihexyphenidyl hydrochloride (Benzhexol hydrochloride) is an antiparkinsonian agent of the antimuscarinic class.Formula:C20H32ClNOPurezza:99.65%Colore e forma:SolidPeso molecolare:337.927Isocorynoxeine
CAS:Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.Formula:C22H26N2O4Purezza:98% - 99.9%Colore e forma:SolidPeso molecolare:382.45Ref: TM-T6S0654
1mg62,00€2mg89,00€5mg132,00€1mL*10mM (DMSO)146,00€10mg226,00€25mg384,00€50mg557,00€100mg785,00€200mg1.054,00€Sumatriptan hydrochloride
CAS:Sumatriptan hydrochloride (GR 43175), an oral 5-HT1 receptor agonist, treats migraines; Ki: 5-HT1D - 17 nM, 5-HT1B - 27 nM, 5-HT1A - 100 nM.Formula:C14H22ClN3O2SColore e forma:SolidPeso molecolare:331.86L-838417 D9
CAS:L-838417 D9 (C-21191) is a novel deuterated subtype-selective GABAA positive allosteric modulator, acting as a partial agonist at α2, α3 and α5 subtypes[1].Formula:C19H10D9F2N7OPurezza:99.65%Colore e forma:SolidPeso molecolare:408.45Ref: TM-T22301
2mg34,00€5mg52,00€1mL*10mM (DMSO)58,00€10mg71,00€25mg128,00€50mg200,00€100mg323,00€200mg447,00€Acamprosate calcium
CAS:Acamprosate calcium (Campral EC) is a GABA receptor agonist and modulator of glutamatergic systems, used for treating alcohol dependence.Formula:C10H20CaN2O8S2Purezza:98% - 99.93%Colore e forma:White Odorless Or Nearly Odorless PowderPeso molecolare:400.48SB 242084
CAS:SB 242084 dihydrochloride hydrate is a psychoactive drug and research chemical which acts as a selective antagonist for the 5HT2C receptor.Formula:C21H19ClN4O2Purezza:99.75% - ≥98%Colore e forma:SolidPeso molecolare:394.85CALP1 acetate
CALP1 acetate is a calmodulin (CaM) agonist (Kd of 88 µM) that binds to the CaM EF-hand/Ca2+-binding site.
Formula:C42H79N9O12Purezza:99.63%Colore e forma:SolidPeso molecolare:902.13Pitofenone hydrochloride
CAS:Pitofenone hydrochloride (Pitophenone hydrochloride), a spasmolytic compound, inhibits the acetylcholinesterase (AChE) activity from bovine erythrocytes andFormula:C22H26ClNO4Purezza:99.97%Colore e forma:SolidPeso molecolare:403.9SB-200646
CAS:SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptorFormula:C15H14N4OPurezza:99.61%Colore e forma:SolidPeso molecolare:266.3Melperone
CAS:Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.Formula:C16H22FNOPurezza:98.84%Colore e forma:SolidPeso molecolare:263.35Quipazine maleate
CAS:Quipazine maleate is a 5-HT agonist affecting L-02 hepatocytes and raphe neurons, causing smooth muscle contracture and bronchospasm.Formula:C17H19N3O4Colore e forma:SolidPeso molecolare:329.356Cromoglicic acid
CAS:Cromoglicic acid prevents the release of inflammatory chemicals such as histamine from mast cells.
Formula:C23H16O11Purezza:99.55% - >99.99%Colore e forma:Colorless Crystals From Ethanol + Ether Physical Description Solid (Ntp 1992)Peso molecolare:468.37Duloxetine
CAS:Duloxetine is an inhibitor of serotonin-norepinephrine reuptake(Ki of 4.6 nM),with treatment of major depressive disorder and generalized anxiety disorder.Formula:C18H19NOSPurezza:99.71% - 99.89%Colore e forma:SolidPeso molecolare:297.41ST034307
CAS:ST034307 is an effective and selective inhibitor of adenylyl cyclase 1 (IC50: 2.3 μM).Formula:C10H4Cl4O2Purezza:99.28%Colore e forma:SolidPeso molecolare:297.95Ref: TM-T16938
1mg35,00€2mg50,00€5mg77,00€1mL*10mM (DMSO)84,00€10mg109,00€25mg224,00€50mg353,00€100mg567,00€200mg797,00€Sarpogrelate hydrochloride
CAS:Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.Formula:C24H32ClNO6Purezza:99.73%Colore e forma:Colorless LiquidPeso molecolare:465.97Rotigotine Hydrochloride
CAS:Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.
Formula:C19H26ClNOSPurezza:99.53% - 99.56%Colore e forma:Almost White To White Crystalline PowderPeso molecolare:351.93Jagged-1 (188-204) TFA(219127-21-6 free base)
Jagged-1 (188-204) TFA, a JAG-1 skin protein fragment, induces epidermal maturation and keratinocyte stratification.Formula:C95H128F3N25O28S3Purezza:99.48%Colore e forma:SolidPeso molecolare:2221.37PRX-07034 hydrochloride
CAS:PRX-07034 hydrochloride is a selective antagonist of 5-HT6 receptor. It has cognition and memory-enhancing properties and decreases body weight in rodents.Formula:C21H29Cl2N3O4SPurezza:98.5%Colore e forma:SolidPeso molecolare:490.44pyridostigmine
CAS:Pyridostigmine(Regonol) is an acetylcholinesterase inhibitor that can treat myasthenia gravis by increasing acetylcholine at the postsynaptic motor endplate.Formula:C9H13N2O2Purezza:98.10%Colore e forma:SolidPeso molecolare:181.21Ref: TM-T8631
1mg84,00€1mL*10mM (DMSO)159,00€5mg167,00€10mg245,00€25mg404,00€50mg567,00€100mg767,00€200mg1.018,00€Temanogrel hydrochloride
CAS:Temanogrel hydrochloride is a serotonin antagonist and anti-platelet agent.Formula:C24H29ClN4O4Colore e forma:SolidPeso molecolare:472.97MDL 72527
CAS:MDL 72527 (N1,N4-Di(buta-2,3-dien-1-yl)butane-1,4-diamine dihydrochloride) is a polyamine oxidase (POA) inhibitorFormula:C12H22Cl2N2Purezza:98.98%Colore e forma:SolidPeso molecolare:265.22Ref: TM-T22965
1mg38,00€2mg50,00€1mL*10mM (DMSO)82,00€5mg84,00€10mg119,00€25mg236,00€50mg385,00€100mg575,00€Thiocolchicoside
CAS:Thiocolchicoside, a muscle relaxant, has anti-inflammatory and analgesic properties; not for seizure-prone people.Formula:C27H33NO10SPurezza:99.11% - 99.39%Colore e forma:SolidPeso molecolare:563.62IGS-1.76
CAS:IGS-1.76 binds strongly to hNCS-1, modulates its Ric8a interaction, and inhibits the hNCS-1/Ric8a complex.Formula:C22H18N2OSPurezza:98.18% - 98.56%Colore e forma:SolidPeso molecolare:358.46SKF-83566
CAS:SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.Formula:C17H18BrNOPurezza:95.00% - 99.82%Colore e forma:SolidPeso molecolare:332.23LRRK2-IN-1
CAS:LRRK2-IN-1 is an effective and selective LRRK2 inhibitor.Formula:C31H38N8O3Purezza:98% - 98.82%Colore e forma:SolidPeso molecolare:570.69VU0155094
CAS:VU0155094 (ML 397) is a positive allosteric modulator with differential activity at the various group III mGluRs.Formula:C24H24N2O4SPurezza:97.21%Colore e forma:SolidPeso molecolare:436.52Ref: TM-T9011
1mg62,00€5mg110,00€1mL*10mM (DMSO)127,00€10mg161,00€25mg269,00€50mg371,00€100mg537,00€200mg710,00€Acephate
CAS:Acephate (Orthene) is an anticholinesterase insecticide with a weak inhibitory effect on AChE in rats, but it can effectively inhibit AChE in cockroaches.Formula:C4H10NO3PSPurezza:≥98%Colore e forma:Colorless Crystals Acephate Is A White Solid Used As A Contact And Systemic InsecticidePeso molecolare:183.17Encenicline
CAS:Encenicline (EVP-6124), a selective α7 nAChRs agonist, targets cognitive impairment in schizophrenia and Alzheimer's.Formula:C16H17ClN2OSPurezza:99.20%Colore e forma:SolidPeso molecolare:320.84Ref: TM-T7193
1mg70,00€5mg133,00€1mL*10mM (DMSO)144,00€10mg207,00€25mg349,00€50mg495,00€100mg675,00€200mg888,00€BRL 54443
CAS:BRL 54443 is a potent 5-HT1E/1F receptor agonist (pKi values are 8.7 and 8.9 respectively).Formula:C14H18N2OPurezza:98.07%Colore e forma:SolidPeso molecolare:230.31Semagacestat
CAS:Semagacestat (LY450139) (LY450139) is a γ-secretase blocker for Aβ42/Aβ40/Aβ38 (IC50: 10.9/12.1/12.0 nM) and also inhibits Notch signaling (IC50: 14.1 nM).Formula:C19H27N3O4Purezza:97.1% - 99.9%Colore e forma:SolidPeso molecolare:361.44Verubecestat tosylate
CAS:Verubecestat (MK-8931/SCH 900931) is a potent BACE1 inhibitor, promising for Alzheimer’s, reducing Aβ in CSF by up to 92%.Formula:C25H26N4O4S2Colore e forma:SolidPeso molecolare:510.627GSK2578215A
CAS:GSK2578215A is a potent and selective LRRK2 kinase inhibitor.Formula:C24H18FN3O2Purezza:99.57% - 99.94%Colore e forma:SolidPeso molecolare:399.42VU0361737
CAS:VU0361737 (ML-128) is a mGlu4 PAM; EC50 is 240 nM (human) and 110 nM (rat), weak at mGlu5/8, inactive at mGlu1/2/3/6/7, CNS-penetrant.Formula:C13H11ClN2O2Purezza:99.60% - 99.85%Colore e forma:SolidPeso molecolare:262.69Olanzapine HCl
CAS:Olanzapine HCl, an FDA-approved atypical antipsychotic for schizophrenia and bipolar disorder, resembles clozapine and quetiapine.Formula:C17H21ClN4SColore e forma:SolidPeso molecolare:348.89GSK-1034702 HCl
CAS:GSK-1034702 HCl is a potent M1 receptor allosteric agonist.Formula:C18H25ClFN3O2Colore e forma:SolidPeso molecolare:369.87MDL 100009
CAS:MDL 100009, the S-enantiomer of MDL 100151 and the opposite enantiomer of MDL 100907, is a selective antagonist of 5-HT2A.Formula:C22H28FNO3Purezza:98.96%Colore e forma:SolidPeso molecolare:373.46Ref: TM-T22359
1mg99,00€5mg187,00€1mL*10mM (DMSO)222,00€10mg280,00€25mg434,00€50mg585,00€100mg775,00€200mg1.054,00€Dinotefuran
CAS:Dinotefuran (MTI-446), a neonicotinoid insecticide, targets pests by blocking their nervous system.Formula:C7H14N4O3Purezza:99.89%Colore e forma:White Crystalline PowderPeso molecolare:202.21Sofpironium bromide
CAS:Sofpironium bromide (BBI4000) belongs to a class of drugs called anticholinergics, which exert their effect by blocking the action of acetylcholine.Formula:C22H32BrNO5Purezza:98.85%Colore e forma:SolidPeso molecolare:470.4Ref: TM-T28827
1mg74,00€5mg160,00€1mL*10mM (DMSO)165,00€10mg250,00€25mg452,00€50mg680,00€100mg1.008,00€200mg1.349,00€Revefenacin
CAS:Revefenacin (TD-4208) is a mAChR antagonist has a high affinity on M3 receptor( Ki : 0.18 nM),and potentially useful for the treatment of respiratory disease.Formula:C35H43N5O4Purezza:98.12%Colore e forma:SolidPeso molecolare:597.75SKF89976A hydrochloride
CAS:SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) andFormula:C22H26ClNO2Purezza:98.02%Colore e forma:SolidPeso molecolare:371.9Ref: TM-T12930
1mg34,00€5mg65,00€1mL*10mM (DMSO)71,00€10mg89,00€25mg167,00€50mg264,00€100mg409,00€200mg590,00€Prucalopride Succinate
CAS:Prucalopride Succinate is a 5-HT4 receptor agonist with Ki 2.5 nM (5-HT4a) and 8 nM (5-HT4b).Formula:C18H26ClN3O3·C4H6O4Purezza:99.24%Colore e forma:SolidPeso molecolare:485.96CCMI
CAS:CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.Formula:C19H15Cl2N3O2Purezza:>99.99%Colore e forma:SolidPeso molecolare:388.25AF-353
CAS:AF-353 (Ro-4), an effective and orally bioavailable antagonist of the P2X3/P2X2/3 receptor, inhibits human and rat P2X3 (pIC50= 8.0).Formula:C14H17IN4O2Purezza:92.98% - 99.356%Colore e forma:SolidPeso molecolare:400.21Avagacestat
CAS:Avagacestat (BMS-708163) (BMS-708163) is a potent, selective, orally bioavailable γ-secretase inhibitor of Aβ40 and Aβ42 with IC50 of 0.3 nM and 0.27 nM,Formula:C20H17ClF4N4O4SPurezza:98.87% - 99.73%Colore e forma:SolidPeso molecolare:520.89Ref: TM-T6249
1mg38,00€5mg77,00€1mL*10mM (DMSO)88,00€10mg116,00€25mg215,00€50mg310,00€100mg450,00€200mg605,00€Lurasidone
CAS:Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6Formula:C28H36N4O2SPurezza:99.78% - 99.91%Colore e forma:SolidPeso molecolare:492.68Amyloid β-Protein 10-20 acetate
Amyloid β-Protein 10-20 acetate (Amyloid β-Protein 10-20 acetate (152286-31-2 free base)) is a fragment of Amyloid-β peptide, maybe used in the research ofFormula:C73H103N17O18Purezza:97.23%Colore e forma:SolidPeso molecolare:1506.65CGP52432
CAS:CGP52432 is a very potent antagonist of GABAB receptors (IC50 = 85 nM).Formula:C15H24Cl2NO4PPurezza:98.75%Colore e forma:SolidPeso molecolare:384.24TBPB
CAS:TBPB is an allosteric M1 mAChR agonist.
Formula:C25H32N4OPurezza:97.87% - 99.9%Colore e forma:SolidPeso molecolare:404.55FITM
CAS:FITM is a potent negative allosteric modulator of mGlu1 receptor(Ki : 2.5 nM).Formula:C18H18FN5OSPurezza:97.25% - 99.23%Colore e forma:SolidPeso molecolare:371.43Ref: TM-T7292
1mg34,00€2mg44,00€1mL*10mM (DMSO)62,00€5mg66,00€10mg92,00€25mg177,00€50mg268,00€100mg394,00€Orexin B, rat, mouse Acetate
Orexin B, rat, mouse Acetate (Rat orexin B) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively.Formula:C128H219N45O36SPurezza:94.61%Colore e forma:SolidPeso molecolare:2996.45rac-BHFF
CAS:rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.Formula:C17H21F3O3Purezza:99.69% - >99.99%Colore e forma:SolidPeso molecolare:330.34Ref: TM-T4176
2mg43,00€5mg60,00€1mL*10mM (DMSO)71,00€10mg96,00€25mg187,00€50mg311,00€100mg472,00€200mg657,00€Loxapine
CAS:Loxapine, a dibenzoxazepine antipsychotic, treats schizophrenia by blocking D2/D4 and serotonin receptors. Related to clozapine.Formula:C18H18ClN3OPurezza:99.88%Colore e forma:Pale Yellowish Crystals From Petroleum Ether SolidPeso molecolare:327.81Imidazenil
CAS:Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion threshold.Formula:C18H12BrFN4OPurezza:98.4% - 99.85%Colore e forma:SolidPeso molecolare:399.22Ref: TM-T8971
100mgPrezzo su richiesta1mg93,00€5mg177,00€1mL*10mM (DMSO)178,00€10mg281,00€25mg475,00€50mg677,00€Tiaprofenic acid
CAS:Tiaprofenic acid (Acido tiaprofenico) is a non-steroidal anti-inflammatory drug used to treat pain, especially arthritic pain.Formula:C14H12O3SPurezza:99.51%Colore e forma:SolidPeso molecolare:260.31Phenylbiguanide
CAS:Phenylbiguanide (N-Phenylbiguanide) is a 5-HT3 receptor selective agonist(EC50 : 3.0±0.1 μM)Formula:C8H11N5Purezza:99.54%Colore e forma:SolidPeso molecolare:177.21LY900009
CAS:LY900009 is a small molecule inhibitor of Notch signalling via selective inhibition of the γ-secretase protein.Formula:C23H27N3O4Purezza:97.07%Colore e forma:SolidPeso molecolare:409.48Ref: TM-T9015
1mg35,00€5mg80,00€1mL*10mM (DMSO)87,00€10mg112,00€25mg197,00€50mg290,00€100mg420,00€200mg590,00€BQCA
CAS:BQCA (benzylquinolone carboxylic acid) a highly selective allosteric M1 mAChR modulator.Formula:C18H15NO4Purezza:97.22%Colore e forma:SolidPeso molecolare:309.32Songorine
CAS:Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.Formula:C22H31NO3Purezza:98% - 99.92%Colore e forma:SolidPeso molecolare:357.49Dihydroergocristine mesylate
CAS:DHEC mesylate is a vasodilator and α-adrenergic antagonist used for vascular dementia and as a geroprotector.Formula:C36H45N5O8SPurezza:98.9% - 99.79%Colore e forma:SolidPeso molecolare:707.84Glycopyrrolate
CAS:Glycopyrrolate: muscarinic antagonist, antispasmodic for GI issues, reduces salivation with anesthesia.Formula:C19H28BrNO3Purezza:99.41% - 99.64%Colore e forma:SolidPeso molecolare:398.33SAX-187
CAS:SAX-187 (SAX-187) has high-affinity binding at the human 5-HT6 receptor.Formula:C15H13ClN4O2S2Purezza:97.82% - 98%Colore e forma:SolidPeso molecolare:380.87Ref: TM-T3183
1mg79,00€5mg152,00€1mL*10mM (DMSO)166,00€10mg245,00€25mg398,00€50mg532,00€100mg735,00€200mg973,00€Rotundine
CAS:Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.Formula:C21H25NO4Purezza:99.8% - 99.91%Colore e forma:Off-White SolidPeso molecolare:355.43Isocarboxazid
CAS:Isocarboxazid: a monoamine oxidase inhibitor used for various depression and anxiety disorders.Formula:C12H13N3O2Purezza:98.32% - 99.94%Colore e forma:SolidPeso molecolare:231.25Ref: TM-T4559
1mg34,00€2mg49,00€5mg74,00€1mL*10mM (DMSO)82,00€10mg90,00€25mg164,00€50mg235,00€100mg350,00€500mg795,00€MTEP
CAS:MTEP: potent, selective mGluR5 antagonist; IC50=5 nM, Ki=16 nM; may have antidepressant/anxiolytic effects; useful in Parkinson's research.Formula:C11H8N2SColore e forma:SolidPeso molecolare:200.26PF3274167
CAS:PF3274167 (Cligosiban) is a potent and selective, high-affinity nonpeptide oxytocin receptor antagonist.Formula:C19H19ClFN5O3Purezza:99.67% - 99.88%Colore e forma:SolidPeso molecolare:419.84Fluralaner
CAS:Fluralaner (A1443) is an isoxazoline ectoparasiticide.Formula:C22H17Cl2F6N3O3Purezza:99.72% - 99.99%Colore e forma:Solid PowderPeso molecolare:556.29Melatonin
CAS:Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.Formula:C13H16N2O2Purezza:98% - 99.89%Colore e forma:Pale Yellow Leaflets From Benzene SolidPeso molecolare:232.28Jujuboside A
CAS:Jujuboside A: glycoside from Semen Ziziphi Spinosae, may treat Alzheimer's, has neuro-inhibitory effects.Formula:C58H94O26Purezza:98% - >99.99%Colore e forma:SolidPeso molecolare:1207.35Perospirone hydrochloride
CAS:Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.Formula:C23H31ClN4O2SPurezza:99.37%Colore e forma:White SolidPeso molecolare:463RAGE antagonist peptide acetate
RAGE antagonist peptide acetate blocks RAGE-ligands like HMGB-1, has anti-tumor, and anti-inflammatory effects.Formula:C59H105N13O19SPurezza:97.17%Colore e forma:SolidPeso molecolare:1332.61FTIDC
CAS:FTIDC: potent, selective mGluR1 allosteric antagonist, weak on mGluR5. IC50: human 5.8 nM, mouse 3.1 nM. Noncompetitive.Formula:C18H23FN6OPurezza:94.58%Colore e forma:SolidPeso molecolare:358.41Ref: TM-T3483
1mg100,00€2mg145,00€5mg215,00€1mL*10mM (DMSO)236,00€10mg340,00€25mg565,00€50mg797,00€100mg1.071,00€SCH-23390 hydrochloride
CAS:SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).Formula:C17H19Cl2NOPurezza:98% - 99.83%Colore e forma:SolidPeso molecolare:324.24Ref: TM-T4369
1mg39,00€2mg50,00€5mg78,00€1mL*10mM (DMSO)78,00€10mg97,00€25mg195,00€50mg369,00€100mg550,00€(RS)-3-Hydroxyphenylglycine
CAS:(RS)-3-Hydroxyphenylglycine is a PI-linked metabotropic glutamate receptors agonist.Formula:C8H9NO3Purezza:99.29%Colore e forma:SolidPeso molecolare:167.16(-)-(S)-B-973B
CAS:(-)-(S)-B-973B is an effective allosteric agonist and a positive allosteric modulator of α7 nAChR.Formula:C24H26F2N6OPurezza:99.52%Colore e forma:SolidPeso molecolare:452.5E4CPG
CAS:E4CPG is a novel group I/II metabotropic glutamate receptor antagonist, more potent than (RS)-MCPG.Formula:C11H13NO4Purezza:99.96%Colore e forma:SolidPeso molecolare:223.23Cariprazine hydrochloride
CAS:Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)Formula:C21H33Cl3N4OPurezza:99.78% - >99.99%Colore e forma:SolidPeso molecolare:463.87Methylbenactyzium Bromide
CAS:Methylbenactyzium Bromide (Semulgin) is an anticonvulsant that is the active metabolite of trimethadione.Formula:C21H28BrNO3Purezza:99.29%Colore e forma:SolidPeso molecolare:422.36CZC-54252
CAS:CZC-54252 is a potent inhibitor of LRRK2.Formula:C22H25ClN6O4SPurezza:99.39%Colore e forma:SolidPeso molecolare:504.99Chelidamic acid
CAS:Chelidamic acid is a heterocyclic organic acid with a pyran skeleton. Chelidamic acid is inhibitors of glutamate decarboxylase, with a Ki of 33 μM.Formula:C7H5NO5Purezza:98.11%Colore e forma:Pale Yellow PowderPeso molecolare:183.12Lerisetron
CAS:Lerisetron is an antagonist of serotonin type 3 (5-HT3) receptor, with antiemetic activity.Formula:C18H20N4Purezza:99.15% - 99.82%Colore e forma:SolidPeso molecolare:292.38Basmisanil
CAS:Basmisanil (RG1662) is a negative allosteric modulator/inverse agonist of GABAAα5 receptors.Formulations containing basmisanil are in clinical trials for theFormula:C21H20FN3O5SPurezza:99.21% - 99.42%Colore e forma:SolidPeso molecolare:445.46Ref: TM-T7165
2mg35,00€1mL*10mM (DMSO)49,00€5mg52,00€10mg74,00€25mg116,00€50mg187,00€100mg356,00€500mg802,00€Atracurium besylate
CAS:Atracurium besylate (51W89) is a short-acting, non-depolarizing muscle relaxant, not affecting the heart or reliant on kidneys.Formula:C65H82N2O18S2Purezza:98.94% - 99.71%Colore e forma:SolidPeso molecolare:1243.49Afloqualone
CAS:Afloqualone (HQ-495) is a GABA Receptor agonist with sedative and muscle-relaxant properties.Formula:C16H14FN3OPurezza:99.72%Colore e forma:SolidPeso molecolare:283.3RTI-55 Hydrochloride
CAS:Prodotto controllatoStability Very Hygroscopic
Applications RTI-55 is a semi-synthetic alkaloid that is a cocaine analogue belonging to the phenyltropane group. RTI-55 acts as a dopamine reuptake inhibitor (DRI) with siginificant abuse potential. RTI-55 is used to assess the rate of dopamine neuron degradation in the brains of patients with Parkinson’s disease.
References Fujita, M. et al.: J. Chem. Neuroanat., 7, 13 (1994); Elmer, G.I. et al.: Pharmacol. Biochem. Behav., 53, 911 (1996); Coulter, C.L. et al.: Brain Res., 690, 217 (1995);Formula:C16H20INO2·ClHColore e forma:NeatPeso molecolare:421.7Riluzole
CAS:Riluzole (RP-54274) is an anticonvulsant, glutamate antagonist, and prolongs ALS patient survival.Formula:C8H5F3N2OSPurezza:99.71% - 99.88%Colore e forma:PowderPeso molecolare:234.2HTT-D3
CAS:HTT-D3 is a Huntington splicing regulator that induces HTT mRNA degradation, leading to a reduction in HTT protein levels.
Formula:C23H25FN6Purezza:99.31%Colore e forma:SolidPeso molecolare:404.48SB 243213
CAS:SB 243213 is a 5-HT2C receptor antagonist with anxiolytic and antidepressant activity used in schizophrenia and movement disorders.Formula:C22H19F3N4O2Purezza:98.78% - 99.86%Colore e forma:SolidPeso molecolare:428.41Pipecuronium bromide
CAS:Pipecuronium bromide (RGH-1106) is an nAChR antagonist that also acts as a non-depolarising steroidal neuromuscular blocker that causes muscle relaxation.Formula:C35H62Br2N4O4Purezza:>99.99%Colore e forma:PowderPeso molecolare:762.7(R)-Mirtazapine
CAS:(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.Formula:C17H19N3Purezza:99.75%Colore e forma:SolidPeso molecolare:265.35Ketanserin tartrate
CAS:Ketanserin tartrate (KJK-945 tartrate) is a 5-HT2A receptor and α1-adrenergic receptor antagonist for the study of systemic sclerosis.Formula:C26H28FN3O9Purezza:99.68%Colore e forma:SolidPeso molecolare:545.51γ-Secretase modulator 13
CAS:γ-Secretase modulator 13 is a γ-secretase modulator (GSMs) that can be used to study Alzheimer's disease and tumors.Formula:C22H23FN6SPurezza:99.79%Colore e forma:SolidPeso molecolare:422.52WAY-100635 maleate
CAS:WAY-100635 Maleate is a specific and effective 5-HT receptor antagonist (IC50=0.95 nM).Formula:C25H34N4O2·xC4H4O4Purezza:99.96%Colore e forma:White SolidPeso molecolare:538.645Ref: TM-T3453
2mg43,00€5mg63,00€1mL*10mM (DMSO)74,00€10mg89,00€25mg150,00€50mg215,00€100mg316,00€500mg765,00€3-Methoxy Dopamine-d4 Hydrochloride (Major)
CAS:Prodotto controllatoApplications A labelled metabolite of Dopamine.
Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package
References Pellmar, T., et al.: Toxicol. Sci., 49, 29 (1999), Ejnik, J., et al.: J. Pharm. Biomed. Anal., 24, 227 ( 2000), Priest, N., et al.: Lancet, 357, 244 (2001), Institoris, L., et al.: Toxicology, 178, 161 (2002),Formula:C92H4H9NO2·ClHColore e forma:NeatPeso molecolare:207.69LP-533401 hydrochloride
CAS:LP-533401 hydrochloride is a peripheral Tph inhibitor that does not cross the BBB and can be used to study periodontal disease and hepatic steatosis.Formula:C27H23ClF4N4O3Purezza:98%Colore e forma:SolidPeso molecolare:562.94Oxazolam
CAS:Prodotto controllatoApplications A psychotropic agent with anxiolytic, anticonvulsant, sedative and skeletal muscle relaxant properties. It is a precursor to the active substance Desmethyldiazepam (D291595).
References Ochs, H.R. et al.: J. Clin. Pharmacol., 24, 446 (1984); Takagi, H. et al.: Nip. Yakur. Zas., 66, 134 (1970);Formula:C18H17ClN2O2Colore e forma:NeatPeso molecolare:328.79EasyStep Human EFNA1(Ephrin A1) ELISA Kit
The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Human EFNA1, and the Human EFNA1 standard plate wells that pre-coated using protein-related techniques are provided separately. Standard/Sample Diluent Buffer or samples are added to the appropriate microtiter plate wells ,then added a HRP-conjugated antibody specific to Human EFNA1. After TMB substrate solution is added, only those wells that contain Human EFNA1 and HRP-conjugated antibody will exhibit a change in color. The enzyme-substrate reaction is terminated by the addition of sulphuric acid solution and the color change is measured spectrophotometrically at a wavelength of 450nm ± 10nm. The concentration of Human EFNA1 in the samples is then determined by comparing the OD of the samples to the standard curve.Colore e forma:Colourless TransparentliquidUCM 608
CAS:UCM 608 (2-Phenylmelatonin) is an antagonist of melatonin-induced contractile responses at low concentrations and induces an increase in GDP-GTP exchange.Formula:C19H20N2O2Purezza:98.88%Colore e forma:SolidPeso molecolare:308.37RO7185876
CAS:RO7185876 is a selective gamma secretase modulator, which can be used in the study of Alzheimer's disease.Formula:C25H28F3N7Purezza:99.50%Colore e forma:SolidPeso molecolare:483.532Tandospirone
CAS:Tandospirone (SM-3997) is a 5-HT1A receptor partial agonist with anxiolytic and antidepressant activity used in the study of central nervous system disorders.Formula:C21H29N5O2Purezza:99.94%Colore e forma:SolidPeso molecolare:383.49Ref: TM-TQ0315
2mg37,00€5mg54,00€1mL*10mM (DMSO)59,00€10mg87,00€25mg141,00€50mg193,00€100mg308,00€200mg441,00€4-Hydroxyindole
CAS:4-Hydroxyindole: aromatic, antioxidant, used in cancer treatment and preventing neurodegenerative diseases.Formula:C8H7NOPurezza:97.05% - 98.13%Colore e forma:Off-White Cyrstalline SolidPeso molecolare:133.15EasyStep Human BNP(Brain Natriuretic Peptide) ELISA Kit
The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Human BNP, and the Human BNP standard plate wells that pre-coated using protein-related techniques are provided separately. Standard/Sample Diluent Buffer or samples are added to the appropriate microtiter plate wells ,then added a HRP-conjugated antibody specific to Human BNP. After TMB substrate solution is added, only those wells that contain Human BNP and HRP-conjugated antibody will exhibit a change in color. The enzyme-substrate reaction is terminated by the addition of sulphuric acid solution and the color change is measured spectrophotometrically at a wavelength of 450nm ± 10nm. The concentration of Human BNP in the samples is then determined by comparing the OD of the samples to the standard curve.Colore e forma:Colourless TransparentliquidEasyStep Human GH(Growth Hormone) ELISA Kit
The test principle applied in this kit is Sandwich enzyme immunoassay. The microtiter plate provided in this kit has been pre-coated with an antibody specific to Human GH, and the Human GH standard plate wells that pre-coated using protein-related techniques are provided separately. Standard/Sample Diluent Buffer or samples are added to the appropriate microtiter plate wells ,then added a HRP-conjugated antibody specific to Human GH. After TMB substrate solution is added, only those wells that contain Human GH and HRP-conjugated antibody will exhibit a change in color. The enzyme-substrate reaction is terminated by the addition of sulphuric acid solution and the color change is measured spectrophotometrically at a wavelength of 450nm ± 10nm. The concentration of Human GH in the samples is then determined by comparing the OD of the samples to the standard curve.Colore e forma:Colourless TransparentliquidGSK-1034702
CAS:GSK-1034702 is an M1 mAChR agonist that improves cognitive deficits and may be useful in the study of neurologic disorders.Formula:C18H24FN3O2Purezza:99.41%Colore e forma:SolidPeso molecolare:333.4(S)-4CPG
CAS:(S)-4CPG ((S)-4-Carboxyphenylglycine) is a competitive mGlu1 receptor antagonist that attenuates nociceptive hypersensitivity and nociceptive abnormalities associated with sciatic nerve constriction injuries in rats, and may be used in the study of neurological disorders.Formula:C9H9NO4Purezza:99.96%Colore e forma:SolidPeso molecolare:195.173,4-Dihydroxyphenylacetic Acid-13C,18O2
CAS:Applications A labelled metabolite of Dopamine.
References Johnson, S., et al.: J. Physiol., 450, 455 (1992), Kolesnikov, Y., et al.: Eur. J. Pharmacol., 296, 17 (1996), Leshner, A., et al.: Science, 278, 45 (1997), Li, J., et al.: Acta Pharmacol. Sin., 20, 375 (1999), Gibson, D., et al.: Brain Res., 952, 71 (2002), Volpicelli, L., et al.: Pharmacol. Biochem. Behav., 64, 487 (1999),Wei, X., et al.: Eur. J. Pharmacol., 515, 99 (2005)Formula:C713CH8O218O2Colore e forma:NeatPeso molecolare:173.14RAD 140
CAS:Applications RAD 140 is a potent, orally bio-available, and non-steroidal selective androgen receptor modulator (SARM).
References Miller, C.P., et al.: ACS Med. Chem. Lett., 2, 124-129 (2011)Formula:C20H16ClN5O2Colore e forma:NeatPeso molecolare:393.8L-368,899 hydrochloride
CAS:L-368,899 hydrochloride is an OXTR antagonist that prevents oxytocin-induced antiabnormal pain and anti-nausea, and may be used in the study of depression.Formula:C26H43ClN4O5S2Purezza:99.59%Colore e forma:SolidPeso molecolare:591.23Ref: TM-T11794
2mg105,00€5mg147,00€1mL*10mM (DMSO)200,00€10mg230,00€25mg439,00€50mg685,00€100mg964,00€(S)-Mirtazapine
CAS:(S)-Mirtazapine ((S)-Org3770) is a 5-HT2 receptor antagonist with pro-nociceptive effects that can be used to study depression.Formula:C17H19N3Purezza:99.37%Colore e forma:SolidPeso molecolare:265.35Rizatriptan
CAS:Rizatriptan (Risatriptan) is a selective 5-hydroxytryptamine 1B/1D receptor agonist used in the study of migraine.Formula:C15H19N5Purezza:99.74%Colore e forma:SolidPeso molecolare:269.356-Cyano-7-nitroquinoxaline-2,3-dione
CAS:Prodotto controllatoStability Store Tightly Sealed at RT
Applications A potent, competitive kainate/quisqualate (non-NMDA) receptor antagonist. IC50 of tritiated ligands to rat cortical membranes by CNQX: AMPA, Kainate and CPP are 0.3mM, 1.5mM, and 25mM, respectively.
References Honore, et al. Science, 241, 701 (1988),Haas, H.S., et al.: Int. J. Oncol., 27, 867 (2005), Kobayashi, K., et al.: J. Pharmacol. Sci., 108, 517 (2008), Shabat-Simon, M., et al.: J. Neurosci., 28, 8406 (2008), Cruz, L.A., et al.: J. Med. Chem., 51, 5856 (2008),Formula:C9H4N4O4Colore e forma:NeatPeso molecolare:232.15Monepantel
CAS:Monepantel (AAD1566) is an organic anthelmintic and an antagonist of nAChRs from roundworms and esophageostomy.Formula:C20H13F6N3O2SPurezza:99.83%Colore e forma:White PowderPeso molecolare:473.39Ref: TM-T16126
1mg93,00€5mg236,00€1mL*10mM (DMSO)259,00€10mg340,00€25mg670,00€50mg964,00€100mg1.378,00€Velufenacin
CAS:Velufenacin is an antagonist of muscarinic receptor[1].Formula:C19H20ClFN2O2Purezza:99.65%Colore e forma:SolidPeso molecolare:362.83Ref: TM-T9771
1mg47,00€5mg96,00€1mL*10mM (DMSO)105,00€10mg156,00€25mg270,00€50mg370,00€100mg522,00€200mg687,00€Darigabat
CAS:Darigabat (PF-06372865) is a GABAA receptor modulator with anxiolytic activity that inhibits α2, α1 PAM, and α2 PAM.Formula:C22H21FN4O3SPurezza:98.42% - 99.29%Colore e forma:SolidPeso molecolare:440.49Setiptiline
CAS:Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.Formula:C19H19NPurezza:98.05% - 98.07%Colore e forma:SolidPeso molecolare:261.36
