Proteasi/Proteasoma
Gli inibitori delle proteasi e del proteasoma sono composti che bloccano l'attività delle proteasi e del proteasoma, che sono coinvolti nella degradazione e nel turnover delle proteine. Questi inibitori sono fondamentali per studiare la regolazione dell'omeostasi proteica, il controllo del ciclo cellulare e l'apoptosi. Gli inibitori delle proteasi e del proteasoma vengono anche utilizzati nel trattamento di malattie come il cancro, dove la degradazione anomala delle proteine svolge un ruolo nella progressione della malattia. Inibendo le proteasi o il proteasoma, questi composti possono indurre la morte cellulare nelle cellule tumorali e sono strumenti critici sia per la ricerca di base che per lo sviluppo terapeutico. Presso CymitQuimica, offriamo una vasta gamma di inibitori delle proteasi e del proteasoma di alta qualità per supportare la tua ricerca in biochimica, biologia cellulare e sviluppo di farmaci.
Sottocategorie di "Proteasi/Proteasoma"
- Acetil-CoA carbossilasi(36 prodotti)
- Cisteina proteasi(110 prodotti)
- DPP-4(24 prodotti)
- Glutaminasi(44 prodotti)
- Proteasi HIV(495 prodotti)
- PAI-1(26 prodotti)
- Inibitori della proteasi(50 prodotti)
- Ricettore attivato dalla proteasi(54 prodotti)
- Proteasoma(87 prodotti)
- Proteasi serina(51 prodotti)
- p97(15 prodotti)
Mostrare 3 più sottocategorie
Trovati 992 prodotti di "Proteasi/Proteasoma"
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MMP-12 Inhibitor
CAS:MMP-12 Inhibitor is a selective inhibitor of MMP-12 with IC50s of 2, 160, 320, and 22.3 nM for human, mouse, rat, and sheep MMP-12.
Formula:C19H20N2O7SPurezza:97.51% - 99.96%Colore e forma:SoildPeso molecolare:420.44RXP470
CAS:RXP470 is a potent and selective MMP-12 inhibitor (Ki 0.24 nM).Formula:C35H35BrClN4O10PColore e forma:SolidPeso molecolare:818MMP Inhibitor 4
MMP Inhibitor4 (compound 4 B) is an effective MMP inhibitor with anti-proliferative properties. It induces cell cycle arrest at the subG1 phase and reduces the mRNA expression of MMP2, MMP9, and VEGFA.Formula:C16H18BrClN2O5Colore e forma:SolidPeso molecolare:433.68Histatin 5 TFA
Histatin 5 TFA effectively inhibits host matrix metalloproteinases (MMP-2) and (MMP-9), demonstrating inhibition concentrations (IC 50s) of 0.57 μM and 0.25 μMFormula:C135H196N51F3O35Colore e forma:SolidPeso molecolare:3150.31Acetyl-Calpastatin (184-210)(human) acetate
Acetyl-Calpastatin acetate inhibits µ-calpain (Ki=0.2nM) and cathepsin L (Ki=6μM) selectively and reversibly.
Formula:C144H234N36O46SPurezza:97.84% - 98.16%Colore e forma:SolidPeso molecolare:3237.68Cathepsin L-IN-3
CAS:Cathepsin L-IN-3, a tripeptide-sized inhibitor of cathepsin L, effectively targets this specific enzyme.Formula:C41H49N7O4SColore e forma:SolidPeso molecolare:735.94Pseudostellarin G
CAS:Pseudostellarin G, a naturally occurring cyclo-octapeptide, exhibits inhibitory activity against tyrosinase and suppresses melanin production.Formula:C42H56N8O9Colore e forma:SolidPeso molecolare:816.94RJS308
RJS308 is a PROTAC degrader of cyclosporin A (cyclosporin A) with a DC50 of 284 nM. It exhibits antiviral activity by inhibiting the replication of HIV-1 and HCV. (Pink: ligand for target protein CypA ligand-2; Black: linker; Blue: ligand for E3 ligase VHL (S,R,S)-AHPC-Me)Formula:C63H75N13O11SColore e forma:SolidPeso molecolare:1222.42TR-107
CAS:TR-107 (Anticancer agent 230) is a mitochondrial protease ClpP activator that inhibits tumor growth in the MDA-MB-231 xenograft model.Formula:C22H19ClN4OColore e forma:SoildPeso molecolare:390.87Rivulariapeptolides 1155
Rivulariapeptolides 1155 inhibits chymotrypsin (41.84 nM), elastase (4.94 nM), and proteinase K (56.54 nM).Formula:C59H81N9O15Colore e forma:SolidPeso molecolare:1156.33GSK2818713
CAS:GSK2818713 is a novel Hepatitis C NS5A replication complex inhibitor.Formula:C46H56N8O8Colore e forma:SolidPeso molecolare:849.002Ecallantide TFA
Ecallantide (DX-88) TFA, a specific recombinant plasma kallikrein inhibitor, directly inhibits bradykinin production and is indicated for the prevention ofColore e forma:Odour SolidBenzamidine
CAS:Benzamidine is a reversible competitive inhibitor of trypsin with a Ki of 19 μM. It also exhibits inhibitory activity on an enzyme in homogenized porcine sperm acrosome, with a Ki of 4 μM.Formula:C7H8N2Colore e forma:SolidPeso molecolare:120.15L 659286
CAS:L 659286 is one kind of cephalosporin derivative.Formula:C17H21N5O7S2Colore e forma:SolidPeso molecolare:471.51JC-10
CAS:JC-10 is a potent inhibitor of metalloproteinases and is often used as a probe.Formula:C25H29Cl2IN4Purezza:95%Colore e forma:SolidPeso molecolare:583.34Z-Arg-Arg-βNA acetate
CAS:Z-Arg-Arg-βNA acetate serves as a sensitive dipeptide substrate for Cathepsin B protease, while demonstrating resistance to proteases H and L. This compound is crucial for differentiating non-Cathepsin B type proteins.Formula:C32H43N9O6Colore e forma:SolidPeso molecolare:649.74Sofosbuvir impurity H
Sofosbuvir impurity H, an diastereoisomer of Sofosbuvir, is the impurity of Sofosbuvir.Formula:C29H33FN3O10PPurezza:98%Colore e forma:SolidPeso molecolare:633.56Leptosin D
CAS:Leptosin D, a thiodiketopiperazine alkaloid derived from mushrooms, effectively inhibits tyrosinase activity, demonstrating an inhibition concentration (IC50)Formula:C25H24N4O3S2Colore e forma:SolidPeso molecolare:492.61VAMP
VAMP is a tetrapeptide that acts as a competitive dipeptidyl peptidase IV (DPP-IV) inhibitor, exhibiting an IC50 of 1.00 μM and a Kd of 6.89 μM. It effectively targets the DPP-IV-GLP-1 axis and is utilized in the research of type 2 diabetes.Formula:C18H32N4O5SColore e forma:SolidPeso molecolare:416.535Linagliptin Methyldimer
CAS:Linagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.Formula:C50H56N16O4Purezza:99.91%Colore e forma:SolidPeso molecolare:945.08Plasma kallikrein-IN-1
CAS:Plasma kallikrein-IN-1 is a PKK inhibitor with an IC 50 value of 0.5 nM.Formula:C23H25F2N7OColore e forma:SolidPeso molecolare:453.498Cathepsin K inhibitor 7
Cathepsin K Inhibitor7 (compound 7) is an inhibitor of Cathepsin K, exhibiting a pKi value of 7.3. It is utilized in research on osteoporosis.Colore e forma:Odour SolidAla-Phe-Pro-pNA TFA
Ala-Phe-Pro-pNA TFA serves as a chromogenic substrate for tripeptidyl peptidase and can be utilized to assess the enzyme's activity.Colore e forma:Odour SolidSofosbuvir impurity K
CAS:Sofosbuvir impurity K is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.Formula:C22H29ClN3O9PPurezza:98%Colore e forma:SolidPeso molecolare:545.91Enzyme-IN-1
CAS:Enzyme-IN-1（compound 1）为基于肽的N端亲核试剂（Ntn）水解酶抑制剂，特别针对20S蛋白酶体的糜胰蛋白酶样活性（CT-L）进行抑制，可能展现出抗炎特性。Formula:C36H50N4O7Colore e forma:SolidPeso molecolare:650.8CRA-2059 hydrochloride
CRA-2059 hydrochloride is a highly specific and selective tryptase inhibitor, with a Ki of 620 pM for recombinant human tryptase-β (rHTβ)[1][2].Colore e forma:SolidN-CBZ-Phe-Arg-AMC
CAS:Z-FR-AMC substrate for serine proteases; cathepsins, kallikrein, plasmin. Substrate: 330/390 nm; Product: 342/441 nm.Formula:C33H36N6O6Purezza:98%Colore e forma:White To Off-White PowderPeso molecolare:612.68CL 82198 hydrochloride
CAS:CL 82198 hydrochloride selectively inhibits MMP-13, not MMP-1/9/TACE, and blocks HP75 invasion and neurotoxicity in zebrafish.Formula:C17H23ClN2O3Colore e forma:SolidPeso molecolare:338.83Sofosbuvir impurity A
CAS:Sofosbuvir impurity A is an diastereoisomer of Sofosbuvir. Sofosbuvir is anHCV RNA replication inhibitor ,with potent anti-hepatitis C virus activity.Formula:C22H29FN3O9PPurezza:98%Colore e forma:SolidPeso molecolare:529.45Cajaninstilbene acid
CAS:Cajaninstilbene acid is a useful organic compound for research related to life sciences. The catalog number is T124035 and the CAS number is 87402-84-4.Formula:C21H22O4Colore e forma:SolidPeso molecolare:338.403TAPI1 acetate
TAPI1 acetate (TNF-α processing inhibitor-1) is a TACE (ADAM17) inhibitor that inhibits shedding of TNF-α cytokine receptors; MMP inhibitor .Formula:C28H41N5O7Purezza:98.82% - 99.94%Colore e forma:SolidPeso molecolare:559.65CRA-2059 TFA
CRA-2059 is a highly specific and selective tryptase inhibitor, with a Ki of 620 pM for recombinant human tryptase-β (rHTβ)[1][2].Colore e forma:SolidDPP8/9-IN-1
DPP8/9-IN-1 (Compound 16) is a selective covalent inhibitor of dipeptidyl peptidase 8 and 9 (DPP8/9), with IC50 values of 14 nM and 298 nM, respectively. It irreversibly binds to the active site serine (such as S730 in DPP9) through a phosphate ester warhead, blocking substrate binding and inhibiting DPP8/9-mediated protein processing. DPP8/9-IN-1 holds potential for research in cancer and inflammatory diseases.Colore e forma:Odour SolidTiprelestat
CAS:Tiprelestat: strong inhibitor of human neutrophil elastase, anti-inflammatory, antimicrobial, used in inflammation/immune research.
Formula:C254H416N72O75S10Colore e forma:SolidPeso molecolare:5999.09Z-Leu-Tyr-Chloromethylketone
CAS:Z-Leu-Tyr-Chloromethylketone is a calpain inhibitor [1].Formula:C24H29ClN2O5Colore e forma:SolidPeso molecolare:460.95N-CBZ-Phe-Arg-AMC TFA
N-CBZ-Phe-Arg-AMC TFA (Z-FR-AMC TFA) is a fluorescent substrate for serine proteases. assess the activity of trypsin, plasmin, and cathepsin.Formula:C35H37F3N6O8Purezza:99.88%Colore e forma:SolidPeso molecolare:726.7PSI-7409
CAS:PSI-7409 is the active 5'-triphosphate metabolite of Sofosbuvir (PSI-7977).
Formula:C10H16FN2O14P3Purezza:98%Colore e forma:SolidPeso molecolare:500.16Tyrosinase/elastase-IN-1
Tyrosinase/elastase-IN-1, a triterpenoid extracted from the leaves of Rubus fraxinifolius, exhibits inhibitory activities against both tyrosinase and elastaseFormula:C33H52O5Colore e forma:SolidPeso molecolare:528.76Peptide 74
CAS:Peptide 74 is a synthetic peptide. It also inhibits the activated form of this enzyme.Formula:C62H107N23O20S2Purezza:98%Colore e forma:SolidPeso molecolare:1558.79Micropeptin 478A
CAS:Micropeptin 478A is a plasmin inhibitor from the Cyanobacterium Microcystis aeruginosa.Formula:C40H62ClN9O15SPurezza:98%Colore e forma:SolidPeso molecolare:976.49MK-6169
CAS:MK-6169 is an effective Pan-Genotype Hepatitis C Virus NS5A inhibitor. It also has Optimized Activity against Common Resistance-Associated Substitutions.Formula:C54H62FN9O8SPurezza:98%Colore e forma:SolidPeso molecolare:1016.2PM 102
CAS:Peptide that reverses the anticoagulant effect of heparin. Potently binds heparin (Kd = 36 nM in vitro).Formula:C235H425N111O64Purezza:98%Colore e forma:SolidPeso molecolare:5830[Asp371]-Tyrosinase (369-377), human
CAS:Tyrosinase (369-377,YMDGTMSQV) originates from tyrosinase and needs TAP and proteosome for cell presentation.Formula:C42H66N10O16S2Purezza:98%Colore e forma:SolidPeso molecolare:1031.16Stevia Powder
Stevia Powder, a natural sweetener, possesses antioxidant properties. It regulates antifibrotic pathways in cirrhotic rats, demonstrated by a reduction in hepatic stellate cells and decreased expression of matrix metalloproteinases MMP2 and MMP13. Furthermore, it increases the antifibrotic molecule Smad7, which helps prevent the elevation of serum necrosis and bile retention markers, thereby inhibiting the progression of liver fibrosis.Colore e forma:Odour SolidRoseltide rT1
CAS:Roseltide rT1 is a neutrophil elastase inhibitor (IC50=0.47 μM) and is rich in cysteine, classified as one of the Roseltides (rT1-rT8). It has the potential to inhibit related diseases by improving neutrophil elastase-stimulated cAMP accumulation in vitro.Formula:C110H177N31O31S6Colore e forma:SolidPeso molecolare:2622.16Pirmitegravir
CAS:Pirmitegravir (STP0404) is a potent ALLINI, blocks LEDGF/p75 site, shows antiviral action against HIV.
Formula:C27H31ClN4O3Purezza:99.79% - 99.79%Colore e forma:SolidPeso molecolare:495.01Phaeosphaone D
CAS:Phaeosphaone D, a thiodiketopiperazine from Phaeosphaeria fuckelii fungus, inhibits mushroom tyrosinase (IC50 = 33.2 μM).Formula:C20H27N3O3S2Colore e forma:SolidPeso molecolare:421.58OM-7D3-B3
OM-7D3-B3 is a monoclonal antibody that targets human tight junction protein 1 (CLDN1) with a dissociation constant (Kd) of 4 nM. This antibody inhibits the role of CLDN1 in the cellular entry of the hepatitis C virus (HCV) and holds potential for research into HCV infection.Colore e forma:Odour LiquidElastatinal
CAS:Elastatinal is an elastase inhibitor. It is found in culture filtrates of various species of actinomyces.Formula:C21H36N8O7Colore e forma:Yellowish SolidPeso molecolare:512.56GPLGLAGGWGERDGS
CAS:GPLGLAGGWGERDGS is a polypeptide with MMP enzyme responsiveness and tumor-targeting properties, suitable for research on enzyme-guided nanoparticle assembly within tumors.Formula:C61H93N19O21Colore e forma:SolidPeso molecolare:1428.51Z-Pro-Pro-aldehyde-dimethyl acetal
CAS:Z-Pro-Pro-aldehyde-dimethyl acetal is a potent prolyl endopeptidase (PREP) inhibitor, effectively impeding the activity of this cytoplasmic serine endoproteaseFormula:C20H28N2O5Purezza:98%Colore e forma:SolidPeso molecolare:376.45Nostosin G
Nostosin G, a linear peptide with Hpla, Hty, and argininal, inhibits trypsin effectively (IC50 = 0.1 μM).Formula:C25H33N5O6Colore e forma:SolidPeso molecolare:499.56Dutogliptin tartrate
CAS:Dutogliptin tartrate is an effective and selective oral dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.Formula:C14H26BN3O9Purezza:98%Colore e forma:SolidPeso molecolare:391.18LMP7/LMP2-IN-1
CAS:LMP7/LMP2-IN-1 (Compound 19) is an orally effective inhibitor targeting the immunoproteasome subunits LMP7 and LMP2, with respective IC50 values of 257 and 10 nM. This compound reduces the production of antibodies and downregulates the B cells in the germinal centers of the spleen and plasma cells in NP-OVA immunized mice. It has potential applications in the study of autoimmune diseases.Formula:C16H27BN4O3Colore e forma:SoildPeso molecolare:334.22HIV-1 inhibitor-6
CAS:HIV-1 inhibitor-6 (3-Pyridinecarboxamide, 1,4-dihydro-1-methyl-N-(5-nitro-1,2-benzisothiazol-3-yl)-4-oxo-) is a potent HIV-1 pre-mRNA selective splicingFormula:C14H10N4O4SPurezza:99.33%Colore e forma:SolidPeso molecolare:330.32Ref: TM-T9854
1mg75,00€5mg169,00€10mg284,00€25mg452,00€50mg645,00€100mg867,00€500mgPrezzo su richiestaSofosbuvir impurity J
CAS:Sofosbuvir impurity J is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.Formula:C22H30FN4O8PPurezza:98%Colore e forma:SolidPeso molecolare:528.47Arabinosylhypoxanthine
CAS:Arabinosylhypoxanthine inhibits Ns5b polymerase in hepatitis C virus and can be used in biochemical experiments and organic synthesis.Formula:C10H12N4O5Purezza:99.71%Colore e forma:SolidPeso molecolare:268.23Retagliptin
CAS:Retagliptin is a DPP-4 inhibitor potentially used to treat Type 2 diabetes.Formula:C19H18F6N4O3Colore e forma:SolidPeso molecolare:464.36Diprotin A TFA
CAS:Diprotin A (TFA) is an inhibitor of dipeptidyl peptidase IV (DPP-IV).Formula:C19H32F3N3O6Colore e forma:SolidPeso molecolare:455.47Urokinase
CAS:Urokinase (uPA) is a serine protease that activates plasminogen to plasmin, crucial for thrombolysis and ECM degradation.Colore e forma:SolidTanaproget
CAS:Tanaproget is an orally available, high-affinity, non-steroidal progesterone receptor (PR) agonist with an IC50 of 1.7 nM for hPR.Formula:C16H15N3OSPurezza:98%Colore e forma:SolidPeso molecolare:297.38Ubenimex
CAS:Formula:C16H24N2O4Purezza:>98.0%(HPLC)Colore e forma:White to Almost white powder to crystalPeso molecolare:308.382'-β-C-Ethynyladenosine
CAS:2'-β-C-Ethynyladenosine is a nucleoside analog that potently inhibits hepatitis C virus (HCV) replication by targeting the viral NS5B polymerase.Formula:C12H13N5O4Colore e forma:SolidPeso molecolare:291.26Anguizole
CAS:Anguizole, a small molecule, effectively inhibits Hepatitis C Virus (HCV) replication by modifying the subcellular distribution of NS4B.Formula:C17H11ClF2N4O2SColore e forma:SolidPeso molecolare:408.81Saxagliptin hydrochloride
CAS:Saxagliptin: oral DPP-4 inhibitor, enhances incretins, manages type 2 diabetes by reducing glucose levels.Formula:C18H26ClN3O2Colore e forma:SolidPeso molecolare:351.87Sivelestat Sodium Tetrahydrate
CAS:Formula:C20H21N2NaO7S·4H2OPurezza:>95.0%(T)(HPLC)Colore e forma:White to Light yellow powder to crystalPeso molecolare:528.50Alogliptin (13CD3)
CAS:Alogliptin (SYR-322) 13CD3 is the deuterium-labeled Alogliptin. Alogliptin is a selective inhibitor of DPP-4.Formula:C18H21N5O2Purezza:98%Colore e forma:SolidPeso molecolare:343.4(-)-Gallocatechin Gallate
CAS:Formula:C22H18O11Purezza:>95.0%(HPLC)Colore e forma:White to Light yellow powder to crystalPeso molecolare:458.38Pepstatin A
CAS:Formula:C34H63N5O9Purezza:>90.0%(HPLC)Colore e forma:White to Light yellow powder to crystalPeso molecolare:685.90CTS-1027
CAS:CTS-1027 is a small molecule inhibitor of MMPs (IC50s: 0.3 nM, 0.5 nM for MMP2, MMP13). It has > 1,000 fold selectivity over MMP1.Formula:C19H20ClNO6SColore e forma:SolidPeso molecolare:425.88H-Pro-Lys-OH TFA
H-Pro-Lys-OH TFA is a dipeptide composed of proline and lysine, serving as a substrate for imino dipeptidase (prolinase). Additionally, it can be utilized in peptide synthesis.Formula:C13H22F3N3O5Colore e forma:SolidPeso molecolare:357.33LN5P45
LN5P45, an OTUB2 inhibitor (IC50: 2.3 μM), promotes monoubiquitination of OTUB2 at lysine 31 and is utilized in the study of tumor progression and metastasis [1Formula:C13H15ClN2O2Colore e forma:SolidPeso molecolare:266.726-Chloro-7-deazapurine-2F-β-D-arabinofuranose
CAS:6-Chloro-7-deazapurine-2F-β-D-arabinofuranose is a Nucleoside - 7-deazapurine nucleoside, fluoronucleoside, halo nucleoside; Arabino-nucleoside.Formula:C11H11ClFN3O3Colore e forma:SolidPeso molecolare:287.67Ref: TM-TNU0055
5mgPrezzo su richiesta10mgPrezzo su richiesta25mgPrezzo su richiesta50mgPrezzo su richiesta100mgPrezzo su richiesta500mgPrezzo su richiestaPSI-6206 13C,d3
CAS:PSI-6206 13CD3 is the deuterium labeled PSI-6206. PSI-6206 is a potent and selective HCV NS5B polymerase inhibitor.
Formula:C10H13FN2O5Purezza:98%Colore e forma:SolidPeso molecolare:264.23MMP-8 Inhibitor I
CAS:MMP-8 Inhibitor I is a selective inhibitor of the neutrophil collagenase matrix metalloproteinase-8 (MMP-8) with an IC50 value of 4 nM.Formula:C17H18N2O5SColore e forma:SolidPeso molecolare:362.4E-64d [for Biochemical Research]
CAS:Formula:C17H30N2O5Purezza:>95.0%(HPLC)Colore e forma:White to Almost white powder to crystalPeso molecolare:342.44Sitagliptin fenilalanil
CAS:Sitagliptin fenilalanil is a dipeptidyl aminopeptidase (DPP-4) inhibitor.Formula:C25H24F6N6O2Colore e forma:SolidPeso molecolare:554.49Ubenimex Hydrochloride [for Biochemical Research]
CAS:Formula:C16H24N2O4·HClPurezza:>97.0%(HPLC)Colore e forma:White to Almost white powder to crystalPeso molecolare:344.84Glutaminase-IN-3
CAS:Glutaminase-IN-3 is a potent Glutaminase 1 inhibitor with potential antitumor activity and inhibits GLS1 for cancer research.Formula:C19H19F3N6O2SPurezza:98.51%Colore e forma:SolidPeso molecolare:452.45PKSI-527
CAS:PKSI-527 inhibits plasma kallikrein (Ki=0.81μM), selective vs. glandular kallikrein/thrombin/urokinase/Xa, reduces bradykinin, affects clotting times.Formula:C25H32ClN3O4Colore e forma:SolidPeso molecolare:473.99Tilpisertib
CAS:Tilpisertib is a serine/threonine kinase inhibitor (WO2017007689).Formula:C33H33ClN8OColore e forma:SolidPeso molecolare:593.13Tomeglovir
CAS:Tomeglovir is a potent anti-CMV agent, inhibiting the processing of viral DNA-concatemers (IC50s: 0.34/0.039 μM for HCMV and MCMV).Formula:C23H27N3O4SPurezza:98%Colore e forma:SolidPeso molecolare:441.54H-Arg-4MβNA
CAS:H-Arg-4MβNA (H-Arg-4MbNA) is a peptide that serves as a substrate for cathepsin H. The enzyme activity is often detected in gel electrophoresis.Formula:C17H23N5O2Purezza:99.98%Colore e forma:SolidPeso molecolare:329.4BAY-677
CAS:BAY-677, an inactive counterpart to BAY-678, inhibits human neutrophil elastase with 20 nM IC50 and is an SGC-nominated probe.Formula:C20H15F3N4O2Colore e forma:SolidPeso molecolare:400.35(Arg)9
CAS:(Arg)9 (Nona-L-arginine;Peptide R9) is a cell-penetrating peptide,and exhibits neuroprotective activity(IC50 of 0.78 μM, in the glutamic acid model).Formula:C54H110N36O10Colore e forma:SolidPeso molecolare:1423.69PD-166793
CAS:PD-166793 is an MMP inhibitor with inhibitory effects on MMP-2, MMP-3 and MMP-13.PD-166793 improves myocardial ischemia in a rat heart failure model.Formula:C17H18BrNO4SPurezza:99.86%Colore e forma:SolidPeso molecolare:412.3Ref: TM-T20563
5mg42,00€10mg60,00€25mg112,00€50mg175,00€100mg261,00€200mg368,00€1mL*10mM (DMSO)46,00€Dabigatran ethyl ester
CAS:Dabigatran ethyl ester (Dabigatran (ethyl ester)) is an emerging oral anticoagulant and it also is a direct inhibitor of thrombin activity.Formula:C27H29N7O3Purezza:99.98%Colore e forma:SolidPeso molecolare:499.56DMP 777
CAS:DMP 777 is an orally active inhibitor of human leukocyte elastase.Formula:C31H40N4O6Colore e forma:SolidPeso molecolare:564.67Ilomastat
CAS:Formula:C20H28N4O4Purezza:>95.0%(HPLC)(qNMR)Colore e forma:White to Light yellow powder to crystalPeso molecolare:388.475-Amino-8-hydroxyquinoline
CAS:5-Amino-8-hydroxyquinoline(5A8HQ),Proteasome inhibitor. Potential anticancer agent.Formula:C9H8N2OPurezza:99.69%Colore e forma:SolidPeso molecolare:160.17Teneligliptin D8
CAS:Teneligliptin D8 a deuterium labeled Teneligliptin (MP-513). Teneligliptin is a potent, orally available, competitive, and long-lasting inhibitor of DPP-4.Formula:C22H30N6OSPurezza:98%Colore e forma:SolidPeso molecolare:434.63Trisodium Hydrogen Ethylenediaminetetraacetate Hydrate [for Biochemical Research]
CAS:Formula:C10H13N2Na3O8·xH2OPurezza:>98.0%(T)Colore e forma:White to Almost white powder to crystalPeso molecolare:358.19 (as Anhydrous)Thrombin inhibitor 5
CAS:Thrombin inhibitor 5 (compound 385), IC50: 0.1-1 μM, used in venous thromboembolism studies.Formula:C11H9FN4O3Purezza:99.58%Colore e forma:SolidPeso molecolare:264.21Ref: TM-T9845
2mg35,00€5mg56,00€10mg86,00€25mg154,00€50mg224,00€100mg320,00€200mg434,00€1mL*10mM (DMSO)55,00€ML-345
CAS:ML-345, Selective IDE inhibitor (IC50=188 nM) targeting Cys819, for type 2 diabetes and Alzheimer's research.Formula:C21H22FN3O5S2Purezza:99.21%Colore e forma:SolidPeso molecolare:479.55Ref: TM-T35802
1mg39,00€5mg84,00€10mg120,00€25mgPrezzo su richiesta50mgPrezzo su richiesta100mg434,00€1mL*10mM (DMSO)Prezzo su richiestaGW280264X
CAS:GW280264X (Carbamic acid) is an inhibitor of ADAM17 .Formula:C28H41N5O6SPurezza:99.51%Colore e forma:SolidPeso molecolare:575.72Ref: TM-T8961
1mg156,00€5mg319,00€10mg477,00€25mg773,00€50mg1.063,00€100mg1.431,00€1mL*10mM (DMSO)404,00€UAMC00039 dihydrochloride
CAS:UAMC00039 dihydrochloride is a potent, reversible and competitive dipeptidyl peptidase II inhibitor with an IC50 of 0.48 nM.Formula:C16H26Cl3N3OPurezza:>99.99%Colore e forma:SolidPeso molecolare:382.76Chlorcyclizine
CAS:CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.Formula:C18H21ClN2Purezza:98.75%Colore e forma:SolidPeso molecolare:300.83Ledipasvir hydrochloride
CAS:Ledipasvir hydrochloride, a hepatitis C NS5A inhibitor, has EC50 of 34 pM (1a) and 4 pM (1b), also inhibits SARS-CoV 3CL pro (IC50 1.62 µM).Formula:C49H55ClF2N8O6Colore e forma:SolidPeso molecolare:925.46KGP94
CAS:KGP94 is a potent, selective, and competitive inhibitor of the lysosomal endopeptidase enzyme.Formula:C14H12BrN3OSPurezza:99.6%Colore e forma:SolidPeso molecolare:350.23Ref: TM-T27730
1mg65,00€5mg138,00€10mg215,00€25mg359,00€50mg510,00€100mg692,00€200mg928,00€1mL*10mM (DMSO)152,00€Alloxan monohydrate
CAS:Alloxan Monohydrate is a glucose analog used to induce diabetes by destroying beta-cells.
Formula:C4H4N2O5Purezza:99.01% - 99.42%Colore e forma:Off-White To Beige-Yellowish Crystalline PowderPeso molecolare:160.09
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