Proteasi/Proteasoma
Gli inibitori delle proteasi e del proteasoma sono composti che bloccano l'attività delle proteasi e del proteasoma, che sono coinvolti nella degradazione e nel turnover delle proteine. Questi inibitori sono fondamentali per studiare la regolazione dell'omeostasi proteica, il controllo del ciclo cellulare e l'apoptosi. Gli inibitori delle proteasi e del proteasoma vengono anche utilizzati nel trattamento di malattie come il cancro, dove la degradazione anomala delle proteine svolge un ruolo nella progressione della malattia. Inibendo le proteasi o il proteasoma, questi composti possono indurre la morte cellulare nelle cellule tumorali e sono strumenti critici sia per la ricerca di base che per lo sviluppo terapeutico. Presso CymitQuimica, offriamo una vasta gamma di inibitori delle proteasi e del proteasoma di alta qualità per supportare la tua ricerca in biochimica, biologia cellulare e sviluppo di farmaci.
Sottocategorie di "Proteasi/Proteasoma"
- Acetil-CoA carbossilasi(36 prodotti)
- Cisteina proteasi(110 prodotti)
- DPP-4(20 prodotti)
- Glutaminasi(44 prodotti)
- Proteasi HIV(506 prodotti)
- PAI-1(26 prodotti)
- Inibitori della proteasi(50 prodotti)
- Ricettore attivato dalla proteasi(54 prodotti)
- Proteasoma(95 prodotti)
- Proteasi serina(55 prodotti)
- p97(15 prodotti)
Mostrare 3 più sottocategorie
Trovati 1093 prodotti di "Proteasi/Proteasoma"
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Rilpivirine HCl
CAS:Rilpivirine HCl (Rilpivirine hydrochloride) is an NNRTI inhibitor with antiviral activity that inhibits the HIV virus.Formula:C22H19ClN6Purezza:99.48%Colore e forma:SolidPeso molecolare:402.88(R)-Trolox
CAS:(R)-Trolox is a selective tyrosinase inhibitor used in food, cosmetics, and pharmaceutical products.Formula:C14H18O4Purezza:99.88%Colore e forma:SolidPeso molecolare:250.29Methylchloroisothiazolinone/Methylisothiazolinone Mixture
CAS:Methylchloroisothiazolinone/Methylisothiazolinone Mixture (Kathon 886MW),a preservative, activates MMPs in human bronchial epithelial cells.Formula:C8H9ClN2O2S2Purezza:99.76%Colore e forma:SolidPeso molecolare:264.75KP-457
CAS:KP-457 is a ADAM17 and a TNFα converting enzyme TACE inhibitor that blocks the production of soluble TNF (sTNF).Formula:C21H24N2O7S2Purezza:98.33%Colore e forma:SolidPeso molecolare:480.56Ref: TM-T77778
1mg92,00€5mg216,00€10mg354,00€25mg655,00€50mg1.035,00€100mg1.406,00€1mL*10mM (DMSO)230,00€Sitagliptin phosphate monohydrate
CAS:Sitagliptin phosphate monohydrate (MK-0431 phosphate monohydrate) is a potent inhibitor of DPP-IV with IC50 of 19 nM in Caco-2 cell extracts.Formula:C16H15F6N5O·H3PO4·H2OPurezza:99.85% - 99.98%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:523.33Teneligliptin
CAS:Teneligliptin (MP-513), potent DPP-4 inhibitor, IC50 ~1 nM, blocks DPP-4 in human/rat plasma and recombinant forms.Formula:C22H30N6OSPurezza:99.73%Colore e forma:SolidPeso molecolare:426.58Ledipasvir
CAS:Ledipasvir (GS-5885) is a Hepatitis C Virus NS5A Inhibitor.Formula:C49H54F2N8O6Purezza:99.96%Colore e forma:SolidPeso molecolare:889Ref: TM-T6200
1mg38,00€2mg49,00€5mg79,00€10mg88,00€25mg159,00€50mg256,00€100mg444,00€500mg1.017,00€1mL*10mM (DMSO)88,00€(1S,2R)-Alicapistat
CAS:(1S,2R)-Alicapistat inhibits calpains 1 and 2, shows promise for Alzheimer's, and has an IC50 of 395 nM.Formula:C25H27N3O4Purezza:99.60%Colore e forma:SoildPeso molecolare:433.5Ref: TM-T60150
1mg67,00€5mg150,00€10mg208,00€25mg316,00€50mg423,00€100mg567,00€1mL*10mM (DMSO)170,00€PSI
CAS:PSI is a proteasome inhibitor.Formula:C32H50N4O8Purezza:97% - 98.33%Colore e forma:SolidPeso molecolare:618.76Danoprevir
CAS:Danoprevir (RG7227) is a peptidomimetic inhibitor of the NS3/4A protease(IC50=0.2-3.5 nM) of hepatitis C virus (HCV).Formula:C35H46FN5O9SPurezza:98% - 99.80%Colore e forma:SolidPeso molecolare:731.83Nelfinavir
CAS:Nelfinavir (AG1341), with Ki=2 nM, is an HIV treatment and broad-spectrum anticancer drug.Formula:C32H45N3O4SPurezza:98.16% - 99.5%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:567.78Triton X-45(n=4)
CAS:Triton X-45: nonionic, low HLB surfactant, dispersible in water, high Krafft point, relevant for HCV research.Formula:C22H38O5Colore e forma:SolidPeso molecolare:382.53Isecarosmab
CAS:Isecarosmab (M6495) is a monoclonal antibody targeting ADAMTS-5, protect cartilage and inhibit ADAMTS-5-mediated degradation of aggrecan,osteoarthritis (OA).Purezza:95% - 98.0% (SDS-PAGE); 96.7% (SEC-HPLC)Colore e forma:LiquidZampilimab
CAS:Zampilimab (UCB-7858) is a humanised monoclonal antibody targeting TGM2, inhibits the cross-linking transamidase activity of TG2, renal fibrosis.Purezza:95%Colore e forma:LiquidLanadelumab
CAS:Lanadelumab (SHP643), a humanized IgG1 antibody, inhibits plasma kallikrein and its interaction with HMWK, supporting hereditary angioedema research.Purezza:95% - 97.4% (SDS-PAGE); 99.2% (SEC-HPLC)Colore e forma:LiquidAnti-Human/Mouse denatured collagen type-I Antibody
Anti-Human/Mouse denatured collagen type-I Antibody (XL313) is an IgG1, κ inhibitor derived from mice, targeting denatured collagen type-I in both human and mouse.Colore e forma:Odour LiquidGalegenimab
CAS:Galegenimab (RG 6147) is an Fab targeting HtrA1, capable of blocking proteolytic cleavage of biglycan (an HtrA1 substrate), suitable for AMD research.Purezza:95% - 95.8% (SDS-PAGE); 99.7% (SEC-HPLC)Colore e forma:LiquidKZR-504
CAS:KZR-504 is a selective inhibitor of immunoproteasome low molecular mass polypeptide 2 (LMP2) (IC50s: 51 nM, 4.274 μM for LMP2 and LMP7, respectively).Formula:C21H23N3O6Colore e forma:SolidPeso molecolare:413.42Anti-Matriptase Antibody
Anti-Matriptase Antibody is a human-derived antibody expressed in CHO cells, targeting Matriptase. It features a huIgG1 heavy chain and huκ light chain, with a predicted molecular weight (MW) of 150 kDa. The isotype control for Anti-Matriptase Antibody can be found in HumanIgG1kappa, Isotype Control.HCV-IN-30
CAS:HCV-IN-30 is an HCV NS5A replication complex inhibitor (IC50s: 901 and 102 nM for genotypes 1a and 1b replicons).Formula:C36H44N6O4Purezza:99.6%Colore e forma:SolidPeso molecolare:624.77S 2160
CAS:S 2160 is a synthetic chromogenic substrate for thrombin.Formula:C33H40N8O6Colore e forma:SolidPeso molecolare:644.72Carboxypeptidase G2 (CPG2) Inhibitor
CAS:Carboxypeptidase G2 (CPG2) Inhibitor (CPG2 Inhibitor) is a new CPG2 Inhibitor with antitumor activity.Formula:C13H15NO6SPurezza:99.96%Colore e forma:SolidPeso molecolare:313.33Cathepsin Inhibitor 1
CAS:<p>Cathepsin Inhibitor 1 is an inhibitor of Cathepsin (L, L2, S, K, B) with pIC50 of 7.9, 6.7, 6.0, 5.5 and 5.2, respectively.</p>Formula:C20H24ClN5O2Purezza:99.78%Colore e forma:SolidPeso molecolare:401.89MMP-2/9-IN-1
CAS:MMP-2/9-IN-1 (Compound 4a) is a potent dual inhibitor of MMP-2 (IC50: 56 nM) and MMP-9 (IC50: 38 nM). leading to DNA fragmentation.Formula:C14H16IN7SColore e forma:SolidPeso molecolare:441.29PK44 phosphate
CAS:PK44 phosphate is a potent inhibitor of dipeptidyl peptidase IV (DPP-IV) (IC50: 15.8 nM).Formula:C17H19F5N7O5PColore e forma:SolidPeso molecolare:527.349(R)-ND-336
CAS:(R)-ND-336: potent, selective MMP-9 inhibitor (K i = 19 nM); inhibits MMP-2 (127 nM), MMP-14 (119 nM); studied for diabetic foot ulcers.Formula:C16H18ClNO3S2Colore e forma:SolidPeso molecolare:371.89VEL-0230
CAS:VEL-0230 (NC-2300) is a cathespin K inhibitor boosting bone growth and reducing loss, targeting bone diseases and developed by Velcura Therapeutics.Formula:C14H24NNaO5Colore e forma:SolidPeso molecolare:309.33L-873724
CAS:L-873724: Selective, reversible cathepsin K inhibitor; IC50s—cat K: 0.2 nM, cat S: 178 nM, cat L: 264 nM, cat B: 5239 nM; inhibits bone resorption.Formula:C23H26F3N3O3SPurezza:98%Colore e forma:SolidPeso molecolare:481.53JO146
CAS:JO146为针对沙眼衣原体高温需要蛋白A(CtHtrA)的蛋白酶抑制剂，其对CtHtrA和人中性粒细胞弹性蛋白酶(HNE)的IC50值分别为21.86 μM和1.15 μM，可应用于细菌感染的抑制。Formula:C31H44N3O7PColore e forma:SolidPeso molecolare:601.67Alicapistat
CAS:Alicapistat (ABT-957) is a human calpains 1 and 2 inhibitor. It can potentially be used to treat Alzheimer's disease (AD).Formula:C25H27N3O4Purezza:98%Colore e forma:SolidPeso molecolare:433.5Tyrosinase-IN-6
CAS:Tyrosinase-IN-6 (4B) is a potent tyrosinase inhibitor (IC50=3.80 μM) with good antioxidant activity.Formula:C24H31N3O2Colore e forma:SolidPeso molecolare:393.52Immunoproteasome inhibitor 1
CAS:Potent, reversible immunoproteasome inhibitor; Ki: β5c 1.18 μM, β1i 0.27 μM, β5i 1.91 μM; potential in treating cancer.Formula:C20H26N2O4Colore e forma:SolidPeso molecolare:358.43CAA0225
CAS:CAA0225 is a selective inhibitor of cathepsin L. CAA0225 is a probe for autophagic proteolysis.Formula:C28H29N3O5Colore e forma:SolidPeso molecolare:487.55MDL 27399
CAS:MDL 27399 suppresses human neutrophil cathepsin G.Formula:C26H36N4O8Colore e forma:SolidPeso molecolare:532.59Anticancer agent 82
CAS:Anticancer agent 82, a FiVe1 derivative, selectively targets VIM in cancer cells to disrupt mitosis, with improved oral bioavailability.Formula:C19H18Cl2N4OColore e forma:SolidPeso molecolare:389.28AM 4299 B
CAS:AM 4299 B is a novel inhibitor of a thiol protease.Formula:C16H27N3O7Purezza:98%Colore e forma:SolidPeso molecolare:373.4Calpain Inhibitor XI
CAS:Calpain Inhibitor XI, a reversible covalent inhibitor of calpain-1, is utilized in the research of neurodegenerative disorders.Formula:C26H40N4O6Colore e forma:SolidPeso molecolare:504.62Tyrosinase-IN-3
CAS:Tyrosinase-IN-3 inhibits melanin production; potential for skin whitening and food preservation.Formula:C21H23NO5Colore e forma:SolidPeso molecolare:369.41HCV-IN-35
CAS:HCV-IN-35 is a potent inhibitor of HCV and shows potential for infectious disease research.Formula:C30H36ClN5Colore e forma:SolidPeso molecolare:502.09Calpain-2-IN-1
CAS:Calpain-2-IN-1 is a selective calpain-2 inhibitor with Ki values of 181 nM for calpain-1 and 7.8 nM for calpain-2, applicable for neurodegenerative diseases a.Formula:C28H37N3O7Colore e forma:SolidPeso molecolare:527.61Tyrosinase-IN-10
CAS:Tyrosinase-IN-10 serves as a partially competitive inhibitor of tyrosinase, demonstrating an inhibition concentration (IC50) value of 1.6 μM against the enzyme'Formula:C16H12O4Colore e forma:SolidPeso molecolare:268.26TAPI-0
CAS:TAPI-0 is a matrix metalloprotease (MMP) and TACE inhibitor.Formula:C24H32N4O5Colore e forma:SolidPeso molecolare:456.53NAAA-IN-2
CAS:<p>NAAA-IN-2, a selective inhibitor with 50 nM IC50, targets NAAA, an enzyme hydrolyzing PEA/OEA, and may aid inflammation and pain studies.</p>Formula:C11H13N3O2SColore e forma:SolidPeso molecolare:251.3Gü2602
CAS:Gü2602 inhibits the cathepsin K zymogen autocatalytic activation that is a potent, reversible inhibitor of cathepsin K (CatK) with a Ki of 0.013 nM for matureFormula:C16H22N4O3Colore e forma:SolidPeso molecolare:318.37MMP-1-IN-1
MMP-1-IN-1 is a highly potent MMP-1 inhibitor with an IC 50 of 0.034 μM .Formula:C14H17ClN2O3Colore e forma:SolidPeso molecolare:296.75(3S,4S)-A2-32-01
(3S,4S)-A2-32-01, a less active (S,S)-enantiomer of A2-32-01. A2-32-01 is a potent caseinolytic protein proteases (ClpP) inhibitor .Formula:C19H27NO2Colore e forma:SolidPeso molecolare:301.42Azo-Resveratrol
CAS:Azo-Resveratrol is an analog of Resveratrol used as a potent tyrosinase inhibitor.Formula:C12H10N2O3Colore e forma:SolidPeso molecolare:230.22HCV-IN-34
CAS:HCV-IN-35, an oral HCV blocker, has an EC50 of 0.010 μM and a CC50 of 7.5 μM, indicating strong antiviral effects.Formula:C31H36ClN5Colore e forma:SolidPeso molecolare:514.1HCV-IN-33
CAS:HCV-IN-33 (Compound (S)-3i) is an inhibitor of HCV entry.Formula:C31H36ClN5Colore e forma:SolidPeso molecolare:514.1Tyrosinase-IN-7
CAS:Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.Formula:C15H10O5Purezza:99%Colore e forma:SolidPeso molecolare:270.24JNJ-10329670
CAS:JNJ 10329670 is a highly potent (Ki of approximately 30 nM), nonpeptidic, noncovalent inhibitor of human cathepsin S with immunosuppressive activity.Formula:C30H34ClF3N6O3SColore e forma:SolidPeso molecolare:651.14BC-05
CAS:BC-05, an orally active inhibitor targeting CD13 and the proteasome, displays potent inhibition with IC50 values of 0.13 μM against human CD13 and 1.39 μM forFormula:C21H29BN2O9Purezza:98%Colore e forma:SolidPeso molecolare:464.27RID-F
CAS:RID-F is an inhibitor of the nonpeptidic proteasome.Formula:C38H50N2O2Purezza:98%Colore e forma:SolidPeso molecolare:566.82AL-9
CAS:AL-9 is a GT-1b and GT-2a replication inhibitor.Formula:C23H22N4O3Purezza:98%Colore e forma:SolidPeso molecolare:402.45PMPA sodium
CAS:PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) inhibitor.Formula:C6H11Na4O7PPurezza:98%Colore e forma:SolidPeso molecolare:318.08Tyrosinase-IN-11
CAS:Tyrosinase-IN-11: potent inhibitor, IC50 - 50nM/64nM (L-tyrosinase/L-dopa), antioxidant, low toxicity, for hyperpigmentation study.Formula:C15H14O5Colore e forma:SolidPeso molecolare:274.27Kallikrein 5-IN-2
CAS:Kallikrein 5-IN-2 inhibits KLK5 (pIC50=7.1); may normalize skin shedding, lessen inflammation & itching.Formula:C23H22N6OColore e forma:SolidPeso molecolare:398.46VA4 TG2 inhibitor
CAS:VA4 is a novel irreversible TG2 transamidase site-specific inhibitor.Formula:C33H41N5O6SColore e forma:SolidPeso molecolare:635.77AZD5248
CAS:AZD-5248 is a potent, selective, first generation, oral inhibitor of dipeptidyl peptidase 1 (DPP1).Formula:C22H22N4O2Colore e forma:SolidPeso molecolare:374.44Cysteine Protease inhibitor hydrochloride
CAS:Cysteine Protease inhibitor hydrochloride is a cysteine protease inhibitor.Formula:C18H15ClN4OPurezza:98%Colore e forma:SolidPeso molecolare:338.79Tec-IN-21
CAS:Tec-IN-21 is an inhibitor of Tec kinase, it also blocks unconventional secretion of fibroblast growth factor 2 (FGF2).Formula:C16H15ClN4O2SPurezza:98%Colore e forma:SolidPeso molecolare:362.83Sheng Gelieting
CAS:CGT-8012 inhibits DP-IV enzyme, aiding type II diabetes research, with an IC50 of 87 nM.Formula:C17H16F6N4OColore e forma:SolidPeso molecolare:406.33CP-471474
CAS:MMP inhibitor with IC50: MMP-2 (0.7 nM), MMP-13 (0.9 nM), MMP-9 (13 nM), MMP-3 (16 nM), MMP-1 (1170 nM); reduces heart dilation post-infarct.Formula:C16H17FN2O5SPurezza:98%Colore e forma:SolidPeso molecolare:368.38BMS-363131
CAS:BMS-363131 (BMS363131) is a potent and selective trypsin inhibitor with an IC50 value of <1.7 nM.Formula:C28H40N6O5Purezza:97.99%Colore e forma:SolidPeso molecolare:540.65α-Glucosidase-IN-5
CAS:α-Glucosidase-IN-5 (compound 8) is isolated from a twig extract of Polyalthia cinnamomea which is a potent α-glucosidase inhibitor with an IC50 of 57.9 µM.Formula:C15H13NO3Colore e forma:SolidPeso molecolare:255.27SAP2-IN-1
CAS:SAP2-IN-1 inhibits secreted aspartate protease 2 (IC50: 0.92 μM), doesn't work in vitro, and helps research infections.Formula:C34H29NO7Colore e forma:SolidPeso molecolare:563.6Glutaminase-IN-4
CAS:Glutaminase-IN-4 (compound 2a) is a glutaminase (GLS) inhibitor (IC50: 2.3 μM).Formula:C23H22N6O2S2Colore e forma:SolidPeso molecolare:478.59L 658758
CAS:L 658758 is an inhibitor of serine proteinase.Formula:C16H20N2O9SColore e forma:SolidPeso molecolare:416.4SJA6017
CAS:SJA6017: inhibits calpain-1/2, cathepsins B/L; prevents apoptosis, protects spinal cord, boosts function. IC50s: 7.5-78 nM.Formula:C17H25FN2O4SPurezza:98%Colore e forma:SolidPeso molecolare:372.45SQ 32602
CAS:SQ 32602 is a cathepsin E inhibitor.Formula:C32H52N3O7PColore e forma:SolidPeso molecolare:621.74Tyrosinase-IN-8
Tyrosinase-IN-8, a potent inhibitor of tyrosinase, demonstrates an inhibitory concentration (IC 50) value of 1.6 µM and exhibits low cytotoxicity whileFormula:C16H12O4Colore e forma:SolidPeso molecolare:268.26DPP-4-IN-2
CAS:DPP-4-IN-2, analog of Alogliptin with 79 nM IC50, is a research tool for diabetes.Formula:C18H18N6OColore e forma:SolidPeso molecolare:334.38Alvelestat tosylate
CAS:Alvelestat can inhibit neutrophil elastase (NE), which acts an important role in NET formation.Formula:C32H30F3N5O7S2Purezza:98%Colore e forma:SolidPeso molecolare:717.73Thrombin Inhibitor 2
CAS:Thrombin Inhibitor 2 is a small molecule direct thrombin inhibitor. Thrombin Inhibitor 2 has antithrombotic activity.Formula:C19H16ClF3N6O2Purezza:98%Colore e forma:SolidPeso molecolare:452.82PSI-7409 tetrasodium
CAS:PSI-7409 tetrasodium, a sofosbuvir metabolite, inhibits GT 1b, 2a, 3a, 4a NS5B polymerases with IC50s of 1.6, 2.8, 0.7, 2.6 μM.Formula:C10H16FN2Na4O14P3Purezza:98%Colore e forma:SolidPeso molecolare:592.117Evogliptin HCl
CAS:Evogliptin (DA-1229), a DPP4 inhibitor, enhances insulin sensitivity and delays diabetes onset.Formula:C19H27ClF3N3O3Colore e forma:SolidPeso molecolare:437.88LY 806303
CAS:LY 806303 is a highly selective thrombin inhibitor.Formula:C16H14O5SPurezza:98%Colore e forma:SolidPeso molecolare:318.34Nucleoside-Analog-2
CAS:Nucleoside-Analog-2 is a 4'-Azidocytidine analogue, used to against Hepatitis C virus (HCV) replication.Formula:C9H11N5O6Purezza:98%Colore e forma:SolidPeso molecolare:285.21GLS1 Inhibitor
CAS:GLS1 inhibitor blocks glutaminase 1 (IC50=0.021 μM), hinders NCI H1703 NSCLC cell growth in vitro (GI50=0.011 μM), and suppresses tumors in mice.Formula:C19H21N7O2SColore e forma:SolidPeso molecolare:411.48BC-23
CAS:BC-23 (NSC 45382) is a proteasome inhibitor with antitumor and antimicrobial activity for the study of leukemia and small cell lung cancer.Formula:C21H14ClN3O4SPurezza:98%Colore e forma:SolidPeso molecolare:439.87NVP DPP 728 dihydrochloride
CAS:NVP-DPP728 is a reversible DPP-IV inhibitor with a K i of 11 nM, enhancing insulin release by preventing GLP-1 degradation, used for diabetes research.Formula:C15H18N6OColore e forma:SolidPeso molecolare:298.34Diprotin B
CAS:Diprotin B is a dipeptidyl peptidase IV inhibitor.Formula:C16H29N3O4Purezza:98%Colore e forma:White Lyophilized PowderPeso molecolare:327.42Bz-D-Arg-pNA hydrochloride
CAS:Bz-D-Arg-pNA hydrochloride is a competitive trypsin inhibitor.Formula:C19H23ClN6O4Colore e forma:SolidPeso molecolare:434.88ND-336
CAS:ND-336 selectively inhibits MMP-2, MMP-9, MMP-14, boosts diabetic wound healing, reduces inflammation, and promotes angiogenesis and skin repair.Formula:C16H18ClNO3S2Colore e forma:SolidPeso molecolare:371.9YM-53601
CAS:YM-53601 is an SQS inhibitor that inhibits adipogenic biosynthesis and lipid secretion in rodents.YM-53601 is a cholesterol-lowering agent that inhibits FDFT1.Formula:C21H22ClFN2OPurezza:99.65%Colore e forma:SolidPeso molecolare:372.86Nucleoside-Analog-1
CAS:Nucleoside-Analog-1 is a 4′-Azidocytidine analogue, used to against Hepatitis C virus replication.Formula:C9H9N5O5Purezza:98%Colore e forma:SolidPeso molecolare:267.2WAY-151693
CAS:WAY-151693 is an inhibitor of human collagenase-3 (MMP-13).Formula:C21H22ClN3O5SColore e forma:SolidPeso molecolare:463.93Epostatin
CAS:Epostatin is a new dipeptidyl peptidase II (DPP-II, EC 3.4.14.2) inhibitor.Formula:C23H33N3O5Purezza:98%Colore e forma:SolidPeso molecolare:431.53GSK-2793660
CAS:GSK-2793660, an oral, irreversible CTSC inhibitor, aids bronchiectasis research.Formula:C20H27N3O3Purezza:98%Colore e forma:SolidPeso molecolare:357.45TNK2-IN-1
CAS:TNK2-IN-1 is a TNK2 inhibitor (IC50: 224 nM) that can be used in cancer research.Formula:C23H24N6O2Colore e forma:SolidPeso molecolare:416.48AGLME
CAS:AGLME is used in a direct enzymatic assay for activated Hageman factor measuring the ability of Hageman factor to hydrolyze the cpd.Formula:C11H21N3O4Colore e forma:SolidPeso molecolare:259.3K 579
CAS:K 579 is a dipeptidyl peptidase IV inhibitor.Formula:C17H24N6OPurezza:98%Colore e forma:SolidPeso molecolare:328.41PTIQ
CAS:MMP-3 expression inhibitorFormula:C13H17NO3Purezza:98%Colore e forma:SolidPeso molecolare:235.28BAY-678 racemate
CAS:BAY-678 racemate: orally active, selective cell-permeable HNE inhibitor with IC50 of 20 nM.Formula:C20H15F3N4O2Purezza:98%Colore e forma:SolidPeso molecolare:400.35WNK-IN-7
CAS:WNK-IN-7 is a potent and selective WNK1 kinase inhibitor.Formula:C26H29N3OPurezza:98%Colore e forma:SolidPeso molecolare:399.53BR351 precursor
CAS:BR351 precursor is a precursor of BR351. BR351 is a brain penetrant MMP inhibitor (IC50s: 4, 2, 11, 50 nM for MMP2, MMP8, MMP9 and MMP13).Formula:C27H32N2O8S2Purezza:98%Colore e forma:SolidPeso molecolare:576.68RS-104966
CAS:RS-104966 is an inhibitor of collagenase that acts by inducing the conformational change in the side-chains of the S1 pocket of MMP-1.Formula:C19H21NO6SPurezza:98%Colore e forma:SolidPeso molecolare:391.44Ono-3307 mesylate
CAS:no-3307 mesylate is a protease inhibitor that inhibits a variety of proteases and may be used to study pancreatitis.Formula:C15H18N4O7S2Purezza:97.60% - 98.16%Colore e forma:SolidPeso molecolare:430.46Thrombin inhibitor 6
CAS:Thrombin Inhibitor 6, with an IC 50 of 1 nM, acts as a potent anticoagulant by inhibiting thrombin.Formula:C18H19ClN4O2SColore e forma:SolidPeso molecolare:390.89BI-L 45XX
CAS:BI-L 45XX, an anti-inflammatory benzimidazole derivative, has inhibitory effects on neutrophil function.Formula:C10H9F3N2O2SColore e forma:SolidPeso molecolare:278.25
