Proteasi/Proteasoma
Gli inibitori delle proteasi e del proteasoma sono composti che bloccano l'attività delle proteasi e del proteasoma, che sono coinvolti nella degradazione e nel turnover delle proteine. Questi inibitori sono fondamentali per studiare la regolazione dell'omeostasi proteica, il controllo del ciclo cellulare e l'apoptosi. Gli inibitori delle proteasi e del proteasoma vengono anche utilizzati nel trattamento di malattie come il cancro, dove la degradazione anomala delle proteine svolge un ruolo nella progressione della malattia. Inibendo le proteasi o il proteasoma, questi composti possono indurre la morte cellulare nelle cellule tumorali e sono strumenti critici sia per la ricerca di base che per lo sviluppo terapeutico. Presso CymitQuimica, offriamo una vasta gamma di inibitori delle proteasi e del proteasoma di alta qualità per supportare la tua ricerca in biochimica, biologia cellulare e sviluppo di farmaci.
Sottocategorie di "Proteasi/Proteasoma"
- Acetil-CoA carbossilasi(36 prodotti)
- Cisteina proteasi(110 prodotti)
- DPP-4(20 prodotti)
- Glutaminasi(45 prodotti)
- Proteasi HIV(506 prodotti)
- PAI-1(26 prodotti)
- Inibitori della proteasi(50 prodotti)
- Ricettore attivato dalla proteasi(54 prodotti)
- Proteasoma(95 prodotti)
- Proteasi serina(55 prodotti)
- p97(15 prodotti)
Mostrare 3 più sottocategorie
Trovati 1095 prodotti di "Proteasi/Proteasoma"
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GM 1489
CAS:GM 1489 is an MMP inhibitor, effective against MMP-1, -2, -3, -8, -9, reduces cancer cell invasion, and prevents ear thickening in mice.Formula:C27H33N3O4Colore e forma:SolidPeso molecolare:463.57GSK2793660 free base
CAS:GSK-2793660, a cathepsin C inhibitor, may treat cystic fibrosis and related lung conditions.Formula:C22H31N3O3Colore e forma:SolidPeso molecolare:385.5THDP-17
CAS:THDP-17 is a inhibitor of glutaminase. THDP-17 shows a partial uncompetitive inhibition in vitro.Formula:C12H16N2SPurezza:98%Colore e forma:SolidPeso molecolare:220.33Garvagliptin
CAS:Garvagliptin has antidiabetic activity.Formula:C18H23F2N3O3SPurezza:98%Colore e forma:SolidPeso molecolare:399.46Cysteine protease inhibitor-2
CAS:Cysteine protease inhibitor from US20070032499A1; halts DCT116 at 6.5μM, PC3 at 4.4μM.Formula:C13H5N5OPurezza:98%Colore e forma:SolidPeso molecolare:247.21ZD8321
CAS:<p>ZD8321 is an effective inhibitor of human Neutrophil elastase (Ki: 13±1.7 nM).</p>Formula:C18H28F3N3O5Purezza:98%Colore e forma:SolidPeso molecolare:423.43Proteasome-IN-1
CAS:Proteasome-IN-1 is an inhibitor of proteasome.Formula:C42H35N5O3Purezza:98%Colore e forma:SolidPeso molecolare:657.76TAPI-1
CAS:TAPI1 (TAPI) , an ADAM17/TACE inhibitor, inhibits shedding of cytokine receptors.Formula:C26H37N5O5Purezza:≥95%Colore e forma:SolidPeso molecolare:499.6GS-9256
CAS:GS-9256 is a selective inhibitor of the HCV NS3 protease, exhibiting favorable pharmacokinetic properties and antiviral activity [1].Formula:C46H56ClF2N6O8PSPurezza:98%Colore e forma:SolidPeso molecolare:957.46Z-LLF-CHO
CAS:Z-LLF-CHO (Z-Leu-Leu-Phe-CHO) effectively inhibits the chymotrypsin-like activity of the pituitary multicatalytic proteinase complex with a Ki value of 460 nM.Formula:C29H39N3O5Purezza:98%Colore e forma:SolidPeso molecolare:509.64MMP13-IN-4
CAS:MMP13-IN-4 (compound 13) is a potent, selective MMP-13 inhibitor with an IC50 of 14.6 μM, implicated in the pathology of osteoarthritis (OA) [1].Formula:C21H17BrN4O5Purezza:98%Colore e forma:SolidPeso molecolare:485.29ND-322 HCl
CAS:ND-322 HCl (ND 322 Hydrochloride) is a selective inhibitor of MT1-MMP and MMP2 and reduces in vitro melanoma cell growth, migration and invasion.Formula:C15H16ClNO3S2Purezza:99.49%Colore e forma:SolidPeso molecolare:357.88Ref: TM-T28145
1mg160,00€5mg354,00€10mg518,00€25mg822,00€50mg1.103,00€100mg1.491,00€1mL*10mM (DMSO)369,00€(S)-BI-1001
CAS:(S)-BI-1001 is an active S-enantiomer of BI-1001. (S)-BI-1001 has antiviral potency against HIV-1 integrase (IC50: 28 nM, and EC50: 450 nM and a Kd: 4.7 μM).Formula:C19H15BrClNO3Purezza:98%Colore e forma:SolidPeso molecolare:420.68PF-00356231 hydrochloride
CAS:PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.Formula:C25H21ClN2O3SPurezza:98.39%Colore e forma:SolidPeso molecolare:464.96Ref: TM-T12414
1mg71,00€5mg187,00€10mg300,00€25mg490,00€50mg678,00€100mg900,00€500mgPrezzo su richiestaNNGH
CAS:NNGH is a matrix metalloproteinase 3 (MMP-3) inhibitor with anticancer activity that counteracts the inhibitory effects of E2 and DHT on RANKL membrane-binding.Formula:C13H20N2O5SPurezza:98.41%Colore e forma:SolidPeso molecolare:316.37Navuridine
CAS:Navuridine (AZdU) is an oral active inhibitor of HIV reverse transcriptase with a relatively short half-life.Formula:C9H11N5O4Purezza:99.83%Colore e forma:SolidPeso molecolare:253.22Ref: TM-T21474
5mg48,00€10mg71,00€25mg131,00€50mg188,00€100mg298,00€500mg1.216,00€1mL*10mM (DMSO)52,00€ZM223 hydrochloride (2031177-48-5 free base)
ZM223 hydrochloride is an orally active, potent non-covalent inhibitor of NEDD8 activating enzyme (NAE), and with excellent anticancer activity.Formula:C23H18ClF3N4O2S2Purezza:98%Colore e forma:SolidPeso molecolare:538.99Flovagatran
CAS:Flovagatran (TGN 255) is a potent, and selective inhibitor of thrombin and parenteral direct factor II.Flovagatran is used to study venous thromboembolism.Formula:C27H36BN3O7Purezza:99.56%Colore e forma:SolidPeso molecolare:525.4RO-9187
CAS:RO-9187 is an effective HCV virus replication inhibitor(IC50: 171 nM).Formula:C9H12N6O5Purezza:98%Colore e forma:SolidPeso molecolare:284.232-MPPA
CAS:2-MPPA (GPI-5693) is a GCP II inhibitor and NAALADase inhibitor, used in research on neurodegenerative diseases.Formula:C8H14O4SPurezza:99.81%Colore e forma:SolidPeso molecolare:206.26Ref: TM-T22497
1mg49,00€5mg104,00€10mg169,00€25mg378,00€50mg655,00€100mg1.169,00€200mg1.586,00€1mL*10mM (DMSO)115,00€Cofrogliptin
CAS:Cofrogliptin (HSK7653) is a DPP-4 inhibitor with hypoglycemic effects, which can be used to study type 2 diabetes (T2D).Formula:C18H19F5N4O3SColore e forma:SolidPeso molecolare:466.43Gosogliptin
CAS:Gosogliptin is a potent, orally active, highly selective, reversible and competitive inhibitor of DPP-4, increasing the level of intestinal GLP-1 and GIP.Formula:C17H24F2N6OPurezza:99.74%Colore e forma:SolidPeso molecolare:366.41Efegatran sulfate
CAS:Efegatran sulfate (LY294468 sulfate) is a potent thrombin inhibitor used in the treatment of thrombotic disorders.Formula:C21H34N6O7SPurezza:≥98% - ≥98%Colore e forma:SolidPeso molecolare:514.6ZD-0892
CAS:<p>ZD-0892: potent, selective neutrophil elastase inhibitor; Ki 6.7 nM (human), 200 nM (porcine).</p>Formula:C24H32F3N3O5Purezza:95% - 99.53%Colore e forma:SolidPeso molecolare:499.52Calpain Inhibitor XII
CAS:<p>Calpain Inhibitor XII (Z-L-Nva-CONH-CH2-2-Py) is a calpain I inhibitor that inhibits calpain II and cathepsin B.</p>Formula:C26H34N4O5Colore e forma:SolidPeso molecolare:482.57MMP2-IN-2
CAS:MMP2-IN-2 is an MMP-2 inhibitor that inhibits MMP-13, MMP-9, and MMP-8, and can be used in the study of cancer and immune diseases.Formula:C13H8N4O4Purezza:98.09%Colore e forma:SolidPeso molecolare:284.23TS-021
CAS:TS-021 is a selective dipeptidyl peptidase 4 (DPP-4) inhibitor with antidiabetic activity for the study of type 2 diabetes.Formula:C17H24FN3O5SPurezza:>99.99% - >99.99%Colore e forma:SolidPeso molecolare:401.45Cathepsin X-IN-1
CAS:<p>Cathepsin X-IN-1 (compound 25) reduces the migration of PC-3 cell with low cytotoxic that is a potent inhibitor of Cathepsin X (IC 50 = 7.13 μM) [1].</p>Formula:C15H13N3O3SPurezza:99.34%Colore e forma:SolidPeso molecolare:315.35CPA inhibitor
CAS:CPA inhibitor (Carboxypeptidase inhibitor) is a potent carboxypeptidase A (CPA) inhibitor with a Ki of 0.32 μM.Formula:C18H19NO4Purezza:99.94%Colore e forma:SolidPeso molecolare:313.35Ref: TM-T10876
1mg57,00€5mg125,00€10mg163,00€25mg278,00€50mg405,00€100mgPrezzo su richiesta1mL*10mM (DMSO)138,00€TY-51469
CAS:TY-51469 is an inhibitor of chymase (IC50s for simian and human chymases: 0.4 and 7.0 nM, respectively).Formula:C20H15FN2O6S4Purezza:99.65%Colore e forma:SolidPeso molecolare:526.6P32/98 hemifumarate
CAS:P32/98 hemifumarate is a DPP4 inhibitor with hypoglycemic properties and is used in the study of type 2 diabetes.Formula:C22H40N4O6S2Purezza:99.46%Colore e forma:SolidPeso molecolare:520.71Isatoribine
CAS:Isatoribine(ANA245) free base is a potent TLR7 receptor agonist with anti-hepatitis C virus infection activity for the study of HCV infection.Formula:C10H12N4O6SPurezza:98.99% - 99.75%Colore e forma:SolidPeso molecolare:316.29Uprifosbuvir
CAS:Uprifosbuvir is an inhibitor of uridine nucleotide analog HCV NS5B polymerase.Formula:C22H29ClN3O9PPurezza:99.73% - >99.99%Colore e forma:SolidPeso molecolare:545.91TG2-IN-3h
CAS:TG2-IN-3h is a highly selective, potent, cell-permeable fluorescent irreversible tissue transglutaminase (tg2) inhibitorFormula:C21H26N4O4SPurezza:99.34% - 99.76%Colore e forma:SolidPeso molecolare:430.52TG-2-IN-1
CAS:TG-2-IN-1 (Compound D003) is a transglutaminase-2 ( TGM-2 ) inhibitor. TG-2-IN-1 can be used in myopia research[1].Formula:C8H13ClN2OSPurezza:98.43%Colore e forma:SolidPeso molecolare:220.72GSK-364735
CAS:GSK-364735 is an HIV-1 IN inhibitor.Formula:C19H18FN3O4Purezza:97.73%Colore e forma:SolidPeso molecolare:371.36(2RS)-FPMPA
CAS:(2RS)-FPMPA（FPMPA） has antiviral activity with an IC50 value of 1.85 μM measured in human MT12 cells infected with SHIV (DH4R).Formula:C9H13FN5O4PPurezza:99.9% - >99.99%Colore e forma:SolidPeso molecolare:305.2CZL55
CAS:CZL55 is a potent caspase-1 inhibitor with an IC50 value of 0.024 μM.CZL55 has low cytotoxicity and can be used in the study of febrile seizures (FS).Formula:C20H22N2O6Purezza:98.19%Colore e forma:SolidPeso molecolare:386.4Lenacapavir
CAS:Lenacapavir (GS-6207) is the first HIV-1 capsid inhibitor approved by the U.S. Food and Drug Administration, the European Medicines Agency, and Health Canada for the treatment of MDR HIV-1 infection.Cost-effective and quality-assured.Formula:C39H32ClF10N7O5S2Purezza:99.61% - 99.87%Colore e forma:SolidPeso molecolare:968.28Ref: TM-T11465
1mg187,00€5mg376,00€10mg565,00€25mg998,00€50mg1.388,00€100mg1.882,00€200mg2.622,00€1mL*10mM (DMSO)615,00€Atevirdine
CAS:<p>Atevirdine is an HIV-1 reverse transcriptase inhibitor with antiviral activity for the study of the AIDS dementia complex (ADC).</p>Formula:C21H25N5O2Purezza:98.20%Colore e forma:SolidPeso molecolare:379.46VRK-IN-1
CAS:VRK-IN-1 is a potent and selective inhibitor of cowpox-associated kinase 1 (VRK1), which can be used in the study of neurological disorders.Formula:C18H11F4NO2Purezza:99.18% - 99.25%Colore e forma:SolidPeso molecolare:349.28Ref: TM-T35863
1mg103,00€5mg236,00€10mg379,00€25mg750,00€50mg1.130,00€100mg1.510,00€200mg2.062,00€1mL*10mM (DMSO)259,00€BMS-929075
CAS:BMS-929075 is an orally active HCV NS5B replicase (HCV NS5B replicase) palm site variant inhibitor with potency, high oral bioavailability and pharmacokineticFormula:C31H24F2N4O3Purezza:99.81% - 99.94%Colore e forma:SolidPeso molecolare:538.54Ref: TM-T26863
1mg180,00€5mg457,00€10mg652,00€25mg1.026,00€50mg1.406,00€100mg1.890,00€500mg3.725,00€1mL*10mM (DMSO)568,00€CP-544439
CAS:CP-544439 is an inhibitor of matrix metalloproteinase-13, which has an effect on adipose tissue development.Formula:C18H19FN2O6SPurezza:95.02% - 98.66%Colore e forma:SolidPeso molecolare:410.4220S Proteasome activator 1
CAS:20S Proteasome activator 1: IC50—0.3 μM (trypsin), 0.7 μM (chymotrypsin), 1.8 μM (caspase); reduces alpha-synuclein A53T, aids neurodegenerative studies.Formula:C27H19ClF2N2OSPurezza:99.82%Colore e forma:SolidPeso molecolare:492.97L 756423
CAS:L756423 is a potent, selective HIV protease inhibitor (Ki=0.049 nM), effective against HIV spread in MT25 lymphocytes at 0.1-0.5 nM, useful for AIDS research.Formula:C39H48N4O5Purezza:99.34% - 99.88%Colore e forma:SolidPeso molecolare:652.82DB04760
CAS:DB04760: selective MMP-13 inhibitor, non-zinc-chelating, IC50=8nM, reduces paclitaxel neurotoxicity, anticancer.Formula:C22H20F2N4O2Purezza:99.93% - 99.99%Colore e forma:SolidPeso molecolare:410.42Ref: TM-T15055
1mg88,00€5mg216,00€10mg325,00€25mg550,00€50mg787,00€100mg1.093,00€500mg2.167,00€1mL*10mM (DMSO)188,00€Sirpiglenastat
CAS:Sirpiglenastat (DRP-104) is a glutamine antagonist, a prodrug of DON, with antitumor activity that acts by suppressing the adaptive immune system.Formula:C22H27N5O5Purezza:98.01% - 98.37%Colore e forma:SolidPeso molecolare:441.48MMP2-IN-3
CAS:MMP2-IN-3 is a potent inhibitor of matrix metalloproteinases (MMP-2) (IC50: 31 μM).Formula:C23H21N3OPurezza:99.38%Colore e forma:SolidPeso molecolare:355.43Ref: TM-T61271
1mg67,00€5mg139,00€10mg205,00€25mg334,00€50mg462,00€100mg622,00€200mg837,00€1mL*10mM (DMSO)148,00€JNJ-10311795
CAS:JNJ-10311795 (RWJ-355871) is an inhibitor of neutrophil elastase G and mast cell chymase, demonstrating significant anti-inflammatory effects.Formula:C40H35N2O6PPurezza:97.43%Colore e forma:SolidPeso molecolare:670.69Opaviraline
CAS:<p>Opaviraline (GW-420867X) is a potent reverse transcriptase inhibitor that inhibits Human immunodeficiency virus 1 and has the potential to treat HIV infection.</p>Formula:C14H17FN2O3Purezza:99.94%Colore e forma:SolidPeso molecolare:280.29Melagatran
CAS:<p>Melagatran is an orally available, direct synthetic thrombin inhibitor that does not require endogenous cofactors other than thrombin.Cost-effective and quality-assured.</p>Formula:C22H31N5O4Purezza:98.29% - >99.99%Colore e forma:SolidPeso molecolare:429.51PG-116800
CAS:PG-116800 (PG-530742) is a matrix metalloproteinase (MMP) inhibitor. PG-116800 can be used in studies about the treatment of osteoarthritis.Formula:C24H27N3O7SPurezza:98.03% - 99.66%Colore e forma:SolidPeso molecolare:501.55BDCRB
BDCRB disrupts HCMV DNA maturation by altering terminase cleavage, extending packaging 30 kb until second site.Formula:C12H11BrCl2N2O4Purezza:99.41% - 99.85%Colore e forma:SoildPeso molecolare:398.04Sovaprevir
CAS:Sovaprevir is a non-structural 3 (NS3) protease inhibitor with antiviral activity for the treatment of HCV infection.Formula:C43H53N5O8SPurezza:99.89%Colore e forma:SolidPeso molecolare:799.97Ref: TM-T28830
1mg266,00€5mg655,00€10mg934,00€25mg1.388,00€50mg1.872,00€100mg2.517,00€1mL*10mM (DMSO)1.035,00€Setrobuvir
CAS:Setrobuvir (ANA-598) is an orally active non-nucleoside HCV NS5B polymerase inhibitor with inhibitory effects on de novo RNA synthesis and primer extension withFormula:C25H25FN4O6S2Purezza:99.95% - 99.97%Colore e forma:SolidPeso molecolare:560.62Ref: TM-T28762
1mg229,00€5mg570,00€10mg812,00€25mg1.216,00€50mg1.663,00€100mg2.242,00€500mg4.494,00€1mL*10mM (DMSO)737,00€BMS-488043
CAS:BMS-488043 is a novel and unique oral small molecule HIV fusion inhibitor that inhibits the attachment of Human Immunodeficiency Virus type 1 (HIV-1) to CD4(+)Formula:C22H22N4O5Purezza:99.95%Colore e forma:SolidPeso molecolare:422.43UPGL00004
CAS:UPGL00004: potent GAC inhibitor, IC50=29 nM, Kd=27 nM, suppresses triple-negative breast cancer cell growth.Formula:C25H26N8O2S2Purezza:97.93%Colore e forma:SolidPeso molecolare:534.66BAY-43-9695
CAS:BAY-43-9695 is a non-nucleoside compound with anti-human cytomegalovirus (HCMV) activity. It is the major metabolite of BAY-38-4766.Formula:C22H25N3O4SPurezza:99.50% - 99.98%Colore e forma:SolidPeso molecolare:427.52MK-8325
CAS:MK-8325 is a potent and orally available HCV NS5A inhibitor with replicative activity against a wide range of genotypes.MK-8325 has demonstrated bioavailabilityFormula:C43H54Cl2F2N8O6SiPurezza:99.61%Colore e forma:SolidPeso molecolare:915.93BILB-1941
CAS:BILB-1941 (BILB-1941ZW) is an inhibitor of HCV NS5B polymerase and can be used in studies about HCV infection.Formula:C34H34N4O4Purezza:99.51% - 99.65%Colore e forma:SolidPeso molecolare:562.66Ref: TM-T26815
1mg313,00€5mg758,00€10mg1.035,00€25mg1.568,00€50mg2.118,00€100mg2.783,00€1mL*10mM (DMSO)1.103,00€NP-313
CAS:NP-313 (NSC-4264) is a potent antithrombotic that blocks platelet aggregation via thromboxane A2 synthesis inhibition and targets SOCC-mediated Ca2+ efflux.Formula:C12H8ClNO3Purezza:99.92%Colore e forma:SolidPeso molecolare:249.652'-C-Methyladenosine
CAS:<p>2'-C-Methyladenosine from C. renalis inhibits HCV, NS5B RNA synthesis (IC50: 0.3, 1.9µM), and LRV1 in L. guyanensis, L. braziliensis.</p>Formula:C11H15N5O4Purezza:99.85%Colore e forma:SolidPeso molecolare:281.27KM-023
CAS:KM-023 is a new second-generation non-nucleoside reverse transcriptase inhibitor for the study of human immunodeficiency virus (HIV) type 1 infection.Formula:C18H19N3O3Purezza:99.03% - 99.47%Colore e forma:SolidPeso molecolare:325.36Ref: TM-T67804
1mg150,00€5mg361,00€10mg542,00€25mg870,00€50mg1.188,00€100mg1.596,00€500mg3.202,00€1mL*10mM (DMSO)359,00€MMP-2/MMP-9 Inhibitor I
CAS:<p>MMP-2/MMP-9-IN-1: oral IV collagenase inhibitor; IC50: 0.24 μM (MMP-9), 0.31 μM (MMP-2); targets cancer.</p>Formula:C21H19NO4SPurezza:99.74%Colore e forma:SolidPeso molecolare:381.44Tyrosinase-IN-2
CAS:Tyrosinase-IN-2, a potent tyrosinase inhibitor, may help in skin lightening and food preservation research.Formula:C8H8N4O2SPurezza:99.78%Colore e forma:SolidPeso molecolare:224.24Ref: TM-T60278
5mg48,00€10mg71,00€25mg135,00€50mg212,00€100mg340,00€200mg467,00€1mL*10mM (DMSO)49,00€Gemigliptin
CAS:Gemigliptin (LC15-0444) is a potent dipeptidyl peptidase-4 (DPP-4) inhibitor(KD : 7.25 nM.)Formula:C18H19F8N5O2Purezza:99.72%Colore e forma:SolidPeso molecolare:489.36Ref: TM-T7369
2mg40,00€5mg60,00€10mg87,00€25mg157,00€50mg259,00€100mg406,00€500mg920,00€1mL*10mM (DMSO)88,00€Etarotene
CAS:Etarotene (Arotinoid ethyl sulphone) is an ethylsulfonyl derivative of aloe acid with differentiation-inducing and potentially antitumor activity.Etarotene is aFormula:C25H32O2SPurezza:99.58% - 99.98%Colore e forma:SolidPeso molecolare:396.59HIV-1 integrase inhibitor 8
CAS:<p>HIV-1 integrase inhibitor 8 is an inhibitor of HIV-1 integrase. Integration is a required step in HIV replication [1].</p>Formula:C21H24O2Purezza:98.91%Colore e forma:SolidPeso molecolare:308.41AGPS-IN-2i
CAS:AGPS-IN-2i inhibits alkylglycerol phosphate synthase, affecting ether lipid metabolism and reducing cancer cell migration and proliferation.Formula:C18H17F2N3O2Purezza:98.92%Colore e forma:SolidPeso molecolare:345.34Ref: TM-T69685
1mg74,00€5mg188,00€10mg311,00€25mg525,00€50mg747,00€100mg1.017,00€1mL*10mM (DMSO)154,00€UK-396082
CAS:UK-396082 is a TAFI inhibitor that inhibits Carboxypeptidase B and can be used in the study of thrombosis, atherosclerosis, cancer and fibrotic conditions.Formula:C12H21N3O2Purezza:99.89%Colore e forma:SolidPeso molecolare:239.31Emivirine
CAS:Emivirine (MKC-442) is a potent and selective nonnucleoside reverse transcriptase inhibitor of human immunodeficiency virus type 1.Formula:C17H22N2O3Purezza:99.8%Colore e forma:SolidPeso molecolare:302.37Z-DEVD-CMK
CAS:Z-DEVD-CMK irreversibly inhibits various cathepsins in vitro [1].Formula:C27H35ClN4O12Colore e forma:SolidPeso molecolare:643.04AZD-9819
CAS:AZD-9819 is a neutrophil elastase (HNE) inhibitor applicable for research into chronic obstructive pulmonary disease (COPD).Formula:C25H19F3N6O2Purezza:100% - 99.18%Colore e forma:SolidPeso molecolare:492.45H-Gly-Pro-Hyp-OH acetate
CAS:H-Gly-Pro-Hyp-OH, a peptide dipeptidyl peptidase 4 (DPP-4) inhibitor with an inhibition concentration (IC50) of 2.51 mM, effectively hinders the activity of the DPP-4 enzyme.Formula:C12H19N3O5C2H4O2Colore e forma:SolidPeso molecolare:345.35(Rac)-Neurodegenerative Disorder-Targeting Compound 1
CAS:(Rac)-Neurodegenerative Disorder-Targeting Compound 1 is a calpain inhibitor.Formula:C28H28N4O4Colore e forma:SolidPeso molecolare:484.55Ro 31-9790
CAS:Ro 31-9790 is a synthetic inhibitor of metalloproteinase (MMP).Formula:C15H29N3O4Purezza:98%Colore e forma:SolidPeso molecolare:315.41Thrombin inhibitor 1
CAS:<p>Thrombin inhibitor 1 is a potent inhibitor of thrombin (Ki: 0.66 nM, 2xaPTT=0.43 μM).</p>Formula:C22H20Cl2F2N4O3Purezza:98%Colore e forma:SolidPeso molecolare:497.32AA74-1
CAS:AA74-1 is a potent, selective APEH inhibitor that significantly enhances T-cell proliferation by inhibiting APEH activity [1].Formula:C16H28N4O2Purezza:98%Colore e forma:SolidPeso molecolare:308.42JW 480
CAS:JW480 is a potent and selective inhibitor of KIAA1363, a serine hydrolase enzyme.Formula:C22H23NO2Purezza:99.72%Colore e forma:SolidPeso molecolare:333.42Ref: TM-T22883
2mg38,00€5mg51,00€10mg84,00€25mg169,00€50mg273,00€100mg439,00€200mg620,00€1mL*10mM (DMSO)60,00€Flovagatran sodium
CAS:Flovagatran sodium, a thrombin inhibitor, is used potentially for the treatment of thrombosis.Formula:C27H36BN3NaO7Purezza:98%Colore e forma:SolidPeso molecolare:548.4BAY-320
CAS:BAY-320 is a Bub1 inhibitor. With an IC50 of 680 nM for human Bub1 in the presence of 2 mM ATP.Formula:C26H26F2N6O2Purezza:98%Colore e forma:SolidPeso molecolare:492.52SQ 32056
CAS:SQ 32056 is a cathepsin E inhibitor.Formula:C37H56N4O5Purezza:98%Colore e forma:SolidPeso molecolare:636.86BMS-189664 HCl
CAS:BMS-189664 HCl is a selective and orally active thrombin active site inhibitor.Formula:C22H35ClN6O4SPurezza:98%Colore e forma:SolidPeso molecolare:515.07Tyropeptin A-4
CAS:Tyropeptin A-4 is used as a proteasome inhibitor.Formula:C31H41N3O6Purezza:98%Colore e forma:SolidPeso molecolare:551.67LM-030
CAS:LM-030, also known as BPR277, is a novel inhibitor of kallikrein-related peptidase 7 (KLK7) and epidermal elastase 2 (ELA2).Formula:C46H72N8O12Colore e forma:SolidPeso molecolare:929.11M190S
CAS:M109S is a novel small molecule that shields cells from mitochondria-dependent apoptosis, demonstrating effectiveness both in vitro and in vivo.Formula:C21H21N5O2Purezza:98%Colore e forma:SolidPeso molecolare:375.42NS5A-IN-3
CAS:NS5A-IN-3 is a potent NS5A inhibitor with high efficacy against HCV 1b, good activity on 3a, and strong metabolic stability; superior to daclatasvir.Formula:C44H44N6O8Purezza:98%Colore e forma:SolidPeso molecolare:784.86Azt-pmap
CAS:AZT-PMPA, an aryl phosphate derivative of AZT and a nucleoside analogue, demonstrates anti-HIV activity[1].Formula:C20H25N6O8PPurezza:98%Colore e forma:SolidPeso molecolare:508.42HIV-1 protease-IN-11
CAS:HIV-1 protease-IN-11 (compound 34a), an HIV-1 protease inhibitor, demonstrates potent inhibition with an IC50 of 0.41 nM and maintains substantial efficacyFormula:C26H37N3O5SPurezza:98%Colore e forma:SolidPeso molecolare:503.65HIV-1 protease-IN-8
CAS:HIV-1 protease-IN-8 (compound 34b) is a potent inhibitor of the HIV-1 protease enzyme, exhibiting an IC50 of 0.32 nM.Formula:C25H35N3O5SPurezza:98%Colore e forma:SolidPeso molecolare:489.63HIV-1 protease-IN-7
CAS:HIV-1 protease-IN-7 (compound 16) is an orally active inhibitor of HIV-1 protease, exhibiting an IC50 of 3.52 nM and an EC50 of 37 nM [1].Formula:C68H104N10O12SPurezza:98%Colore e forma:SolidPeso molecolare:1285.68HIV-1 protease-IN-12
CAS:HIV-1 protease-IN-12 (compound 35b) serves as a potent inhibitor of HIV-1 protease, exhibiting an IC50 value of 0.51 nM, and demonstrates efficacy against drug-Formula:C25H35N3O5SPurezza:98%Colore e forma:SolidPeso molecolare:489.63NS5A-IN-2
CAS:NS5A-IN-2, a potent inhibitor, is highly effective against HCV 1b and shows increased activity for GT 3a with good metabolic stability.Formula:C46H45N7O7Purezza:98%Colore e forma:SolidPeso molecolare:807.89NCI-B16
CAS:NCI-B16 is a small-molecule RNA binder that inhibits HCV (hepatitis C virus) replication [1].Formula:C27H26N8O4Colore e forma:SolidPeso molecolare:526.55HIV-1 protease-IN-9
CAS:HIV-1 protease-IN-9 (compound 5b), a potent HIV-1 protease inhibitor, exhibits strong antiviral efficacy with a dissociation constant (K_i) of 0.028 nM and aFormula:C37H41N7O4SPurezza:98%Colore e forma:SolidPeso molecolare:679.83TP0556351
CAS:TP0556351: potent MMP2 inhibitor with 0.2 nM IC50, reduces collagen in pulmonary fibrosis mice.Formula:C50H70N10O16Purezza:98%Colore e forma:SolidPeso molecolare:1067.15HCV-IN-44
CAS:HCV-IN-44 (compound 28) is an inhibitor of the HCV NS5B protein, efficacious in suppressing HCV virus replication and useful for researching HCV infection [1].Formula:C24H26FN3O5SColore e forma:SolidPeso molecolare:487.54(1R,4S)-Yimitasvir diphosphate
CAS:Yimitasvir diphosphate, also known as Emitasvir, is an orally-administered inhibitor of the hepatitis C virus (HCV) nonstructural protein 5A (NS5A).Formula:C49H64N8O14P2Colore e forma:SolidPeso molecolare:1051.03MeOSuc-AAPV-CMK
CAS:MeOSuc-AAPV-CMK (Elastase Inhibitor III) serves as an inhibitor of elastase, as well as cathepsin G and proteinase 3, and impedes leukocyte elastase-mediatedFormula:C22H35ClN4O7Colore e forma:SolidPeso molecolare:502.99Ecallantide
CAS:Ecallantide (DX-88) is a recombinant inhibitor specifically targeting plasma kallikrein, which serves to impede the synthesis of bradykinin.Formula:C305H448N88O91S8Colore e forma:SolidPeso molecolare:7059.88
