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Proteasi/Proteasoma

Proteasi/Proteasoma

Gli inibitori delle proteasi e del proteasoma sono composti che bloccano l'attività delle proteasi e del proteasoma, che sono coinvolti nella degradazione e nel turnover delle proteine. Questi inibitori sono fondamentali per studiare la regolazione dell'omeostasi proteica, il controllo del ciclo cellulare e l'apoptosi. Gli inibitori delle proteasi e del proteasoma vengono anche utilizzati nel trattamento di malattie come il cancro, dove la degradazione anomala delle proteine svolge un ruolo nella progressione della malattia. Inibendo le proteasi o il proteasoma, questi composti possono indurre la morte cellulare nelle cellule tumorali e sono strumenti critici sia per la ricerca di base che per lo sviluppo terapeutico. Presso CymitQuimica, offriamo una vasta gamma di inibitori delle proteasi e del proteasoma di alta qualità per supportare la tua ricerca in biochimica, biologia cellulare e sviluppo di farmaci.

Sottocategorie di "Proteasi/Proteasoma"

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Trovati 1092 prodotti di "Proteasi/Proteasoma"

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  • 7-Methoxy obtusifolin
    Targetmol
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    7-Methoxy obtusifolin

    CAS:
    7-Methoxy obtusifolin (Compound 4) is a chemical compound that acts as a competitive inhibitor of the enzyme tyrosinase, displaying an inhibitory concentration
    Formula:C17H14O6
    Colore e forma:Solid
    Peso molecolare:314.29

    Ref: TM-T75613

  • RXP470
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    RXP470

    CAS:
    RXP470 is a potent and selective MMP-12 inhibitor (Ki 0.24 nM).
    Formula:C35H35BrClN4O10P
    Colore e forma:Solid
    Peso molecolare:818

    Ref: TM-T28633

  • NVP-DPP728 dihydrochloride
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    NVP-DPP728 dihydrochloride

    CAS:
    <p>NVP-DPP728 dihydrochloride is a potent, selective DPP-IV inhibitor with a Ki of 11 nM, useful in diabetes research.</p>
    Formula:C15H20Cl2N6O
    Colore e forma:Solid
    Peso molecolare:371.27

    Ref: TM-T39481

  • Pseudostellarin G
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    Pseudostellarin G

    CAS:
    Pseudostellarin G, a naturally occurring cyclo-octapeptide, exhibits inhibitory activity against tyrosinase and suppresses melanin production.
    Formula:C42H56N8O9
    Colore e forma:Solid
    Peso molecolare:816.94

    Ref: TM-TP2861

  • Logo CymitQuimica
    Targetmol
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    RJS308

    <p>RJS308 is a PROTAC degrader of cyclosporin A (cyclosporin A) with a DC50 of 284 nM. It exhibits antiviral activity by inhibiting the replication of HIV-1 and HCV. (Pink: ligand for target protein CypA ligand-2; Black: linker; Blue: ligand for E3 ligase VHL (S,R,S)-AHPC-Me)</p>
    Formula:C63H75N13O11S
    Colore e forma:Solid
    Peso molecolare:1222.42

    Ref: TM-T205591

  • Logo CymitQuimica
    Targetmol
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    Ellipyrone A

    Ellipyrone A: γ-pyrone macrocycle, inhibits DPP-4 (IC50=0.35mM), α-glucosidase (IC50=0.74mM), α-amylase (IC50=0.59mM).
    Formula:C25H34O8
    Colore e forma:Solid
    Peso molecolare:462.53

    Ref: TM-T75492

  • Sofosbuvir impurity H
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    Sofosbuvir impurity H

    Sofosbuvir impurity H, an diastereoisomer of Sofosbuvir, is the impurity of Sofosbuvir.
    Formula:C29H33FN3O10P
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:633.56

    Ref: TM-T12963

  • GSK2336805
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    GSK2336805

    CAS:
    <p>GSK-2336805, an HCV NS5A inhibitor, is effective against genotypes 1, 4, 5, and some of 6.</p>
    Formula:C42H52N8O8
    Colore e forma:Solid
    Peso molecolare:796.91

    Ref: TM-T27461

  • BMS-767778
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    BMS-767778

    CAS:
    BMS-767778, a DPP-4 inhibitor, is used potentially for the treatment of type 2 diabetes.
    Formula:C19H20Cl2N4O2
    Colore e forma:Solid
    Peso molecolare:407.29

    Ref: TM-T26857

  • Dutogliptin tartrate
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    Dutogliptin tartrate

    CAS:
    Dutogliptin tartrate is an effective and selective oral dipeptide-peptide-4 (DPP4) inhibitor for the treatment of type 2 diabetes mellitus.
    Formula:C14H26BN3O9
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:391.18

    Ref: TM-T11127

  • JC-10
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    JC-10

    CAS:
    JC-10 is a potent inhibitor of metalloproteinases and is often used as a probe.
    Formula:C25H29Cl2IN4
    Purezza:95%
    Colore e forma:Solid
    Peso molecolare:583.34

    Ref: TM-TD0056

  • Linagliptin Methyldimer
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    Linagliptin Methyldimer

    CAS:
    Linagliptin Methyldimer is a potent dipeptidyl peptidase IV inhibitor, IC50=6 pM.
    Formula:C50H56N16O4
    Purezza:99.91%
    Colore e forma:Solid
    Peso molecolare:945.08

    Ref: TM-T67852

  • NS5A-IN-4
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    NS5A-IN-4

    CAS:
    NS5A-IN-4 (Compound 1.12) is a hepatitis C inhibitor effective against multiple genotypes, with IC50 values ranging from 1.2 to 2296 pM.
    Formula:C47H48N8O6
    Colore e forma:Solid
    Peso molecolare:820.93

    Ref: TM-T74495

  • PSI-7409
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    PSI-7409

    CAS:
    <p>PSI-7409 is the active 5'-triphosphate metabolite of Sofosbuvir (PSI-7977).</p>
    Formula:C10H16FN2O14P3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:500.16

    Ref: TM-T12572

  • Logo CymitQuimica
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    α 1 Antichymotrypsin, Human Plasma

    CAS:
    Alpha 1 Antichymotrypsin, Human Plasma is an inhibitor of serine proteases. This compound is present in amyloid lesions associated with Alzheimer's disease and can be utilized in Alzheimer's research.
    Colore e forma:Solid

    Ref: TM-TP3129

  • MK-6169
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    MK-6169

    CAS:
    MK-6169 is an effective Pan-Genotype Hepatitis C Virus NS5A inhibitor. It also has Optimized Activity against Common Resistance-Associated Substitutions.
    Formula:C54H62FN9O8S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1016.2

    Ref: TM-T24476

  • Logo CymitQuimica
    Targetmol
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    Nostosin G

    Nostosin G, a linear peptide with Hpla, Hty, and argininal, inhibits trypsin effectively (IC50 = 0.1 μM).
    Formula:C25H33N5O6
    Colore e forma:Solid
    Peso molecolare:499.56

    Ref: TM-T75647

  • 5-epi-Arvestonate A
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    5-epi-Arvestonate A

    CAS:
    <p>5-epi-Arvestonate A, a sesquiterpenoid from Seriphidium transiliense, stimulates melanogenesis and suppresses IFN-γ-chemokine in HaCaT cells.</p>
    Formula:C16H26O5
    Colore e forma:Solid
    Peso molecolare:298.37

    Ref: TM-T75535

  • Elastatinal
    Targetmol
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    Elastatinal

    CAS:
    Elastatinal is an elastase inhibitor. It is found in culture filtrates of various species of actinomyces.
    Formula:C21H36N8O7
    Colore e forma:Yellowish Solid
    Peso molecolare:512.56

    Ref: TM-T20130

  • Sofosbuvir impurity M
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    Sofosbuvir impurity M

    CAS:
    Sofosbuvir impurity M is an diastereoisomer of Sofosbuvir.Sofosbuvir is an HCV RNA replication inhibitor, with potent anti-hepatitis C virus activity.
    Formula:C22H30N3O10P
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:527.467

    Ref: TM-T12968