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Proteasi/Proteasoma

Proteasi/Proteasoma

Gli inibitori delle proteasi e del proteasoma sono composti che bloccano l'attività delle proteasi e del proteasoma, che sono coinvolti nella degradazione e nel turnover delle proteine. Questi inibitori sono fondamentali per studiare la regolazione dell'omeostasi proteica, il controllo del ciclo cellulare e l'apoptosi. Gli inibitori delle proteasi e del proteasoma vengono anche utilizzati nel trattamento di malattie come il cancro, dove la degradazione anomala delle proteine svolge un ruolo nella progressione della malattia. Inibendo le proteasi o il proteasoma, questi composti possono indurre la morte cellulare nelle cellule tumorali e sono strumenti critici sia per la ricerca di base che per lo sviluppo terapeutico. Presso CymitQuimica, offriamo una vasta gamma di inibitori delle proteasi e del proteasoma di alta qualità per supportare la tua ricerca in biochimica, biologia cellulare e sviluppo di farmaci.

Sottocategorie di "Proteasi/Proteasoma"

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Trovati 1094 prodotti di "Proteasi/Proteasoma"

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  • Calpain-2-IN-1
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    Calpain-2-IN-1

    CAS:
    Calpain-2-IN-1 is a selective calpain-2 inhibitor with Ki values of 181 nM for calpain-1 and 7.8 nM for calpain-2, applicable for neurodegenerative diseases a.
    Formula:C28H37N3O7
    Colore e forma:Solid
    Peso molecolare:527.61

    Ref: TM-T63708

  • Tyrosinase-IN-10
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    Tyrosinase-IN-10

    CAS:
    Tyrosinase-IN-10 serves as a partially competitive inhibitor of tyrosinase, demonstrating an inhibition concentration (IC50) value of 1.6 μM against the enzyme'
    Formula:C16H12O4
    Colore e forma:Solid
    Peso molecolare:268.26

    Ref: TM-T72720

  • TAPI-0
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    TAPI-0

    CAS:
    TAPI-0 is a matrix metalloprotease (MMP) and TACE inhibitor.
    Formula:C24H32N4O5
    Colore e forma:Solid
    Peso molecolare:456.53

    Ref: TM-T70664

  • NAAA-IN-2
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    NAAA-IN-2

    CAS:
    <p>NAAA-IN-2, a selective inhibitor with 50 nM IC50, targets NAAA, an enzyme hydrolyzing PEA/OEA, and may aid inflammation and pain studies.</p>
    Formula:C11H13N3O2S
    Colore e forma:Solid
    Peso molecolare:251.3

    Ref: TM-T60378

  • Garvagliptin
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    Garvagliptin

    CAS:
    Garvagliptin has antidiabetic activity.
    Formula:C18H23F2N3O3S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:399.46

    Ref: TM-T27402

  • MMP-1-IN-1
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    MMP-1-IN-1

    MMP-1-IN-1 is a highly potent MMP-1 inhibitor with an IC 50 of 0.034 μM .
    Formula:C14H17ClN2O3
    Colore e forma:Solid
    Peso molecolare:296.75

    Ref: TM-T73175

  • (3S,4S)-A2-32-01
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    (3S,4S)-A2-32-01

    (3S,4S)-A2-32-01, a less active (S,S)-enantiomer of A2-32-01. A2-32-01 is a potent caseinolytic protein proteases (ClpP) inhibitor .
    Formula:C19H27NO2
    Colore e forma:Solid
    Peso molecolare:301.42

    Ref: TM-T72657

  • Azo-Resveratrol
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    Azo-Resveratrol

    CAS:
    Azo-Resveratrol is an analog of Resveratrol used as a potent tyrosinase inhibitor.
    Formula:C12H10N2O3
    Colore e forma:Solid
    Peso molecolare:230.22

    Ref: TM-T70783

  • HCV-IN-34
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    HCV-IN-34

    CAS:
    HCV-IN-35, an oral HCV blocker, has an EC50 of 0.010 μM and a CC50 of 7.5 μM, indicating strong antiviral effects.
    Formula:C31H36ClN5
    Colore e forma:Solid
    Peso molecolare:514.1

    Ref: TM-T63567

  • Tyrosinase-IN-7
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    Tyrosinase-IN-7

    CAS:
    Tyrosinase-IN-7 is a small-molecule tyrosinase inhibitor (IC50 1.57 μM) that suppresses melanin activity and cell growth with low cytotoxicity.
    Formula:C15H10O5
    Purezza:99%
    Colore e forma:Solid
    Peso molecolare:270.24

    Ref: TM-T72786

  • EI-1
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    EI-1

    CAS:
    EI-1 is an inhibitor of Hepatitis C virus entry.
    Formula:C16H19F3N6O3
    Colore e forma:Solid
    Peso molecolare:400.36

    Ref: TM-T71871

  • BC-05
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    BC-05

    CAS:
    BC-05, an orally active inhibitor targeting CD13 and the proteasome, displays potent inhibition with IC50 values of 0.13 μM against human CD13 and 1.39 μM for
    Formula:C21H29BN2O9
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:464.27

    Ref: TM-T78847

  • RID-F
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    RID-F

    CAS:
    RID-F is an inhibitor of the nonpeptidic proteasome.
    Formula:C38H50N2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:566.82

    Ref: TM-T26082

  • AL-9
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    AL-9

    CAS:
    AL-9 is a GT-1b and GT-2a replication inhibitor.
    Formula:C23H22N4O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:402.45

    Ref: TM-T25020

  • PMPA sodium
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    PMPA sodium

    CAS:
    PMPA sodium is a potent and selective glutamate carboxypeptidase 2 (GCP II/N-acetylated a-linked dipeptidase/NAALADase) inhibitor.
    Formula:C6H11Na4O7P
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:318.08

    Ref: TM-T25968

  • TNIK-IN-4
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    TNIK-IN-4

    CAS:
    TNIK-IN-4: strong TNIK inhibitor, IC50 of 0.61 μM, suppresses HCT116 colorectal cancer cells.
    Formula:C20H16FN3O3
    Colore e forma:Solid
    Peso molecolare:365.36

    Ref: TM-T61396

  • PF-00356231 hydrochloride
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    PF-00356231 hydrochloride

    CAS:
    PF-00356231 hydrochloride is an inhibitor of matrix metalloproteinase MMP-12 with IC50 of 1.4 μM.
    Formula:C25H21ClN2O3S
    Purezza:98.39%
    Colore e forma:Solid
    Peso molecolare:464.96

    Ref: TM-T12414

  • Tyrosinase-IN-11
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    Tyrosinase-IN-11

    CAS:
    Tyrosinase-IN-11: potent inhibitor, IC50 - 50nM/64nM (L-tyrosinase/L-dopa), antioxidant, low toxicity, for hyperpigmentation study.
    Formula:C15H14O5
    Colore e forma:Solid
    Peso molecolare:274.27

    Ref: TM-T72703

  • Kallikrein 5-IN-2
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    Kallikrein 5-IN-2

    CAS:
    Kallikrein 5-IN-2 inhibits KLK5 (pIC50=7.1); may normalize skin shedding, lessen inflammation & itching.
    Formula:C23H22N6O
    Colore e forma:Solid
    Peso molecolare:398.46

    Ref: TM-T72624

  • VA4 TG2 inhibitor
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    VA4 TG2 inhibitor

    CAS:
    VA4 is a novel irreversible TG2 transamidase site-specific inhibitor.
    Formula:C33H41N5O6S
    Colore e forma:Solid
    Peso molecolare:635.77

    Ref: TM-T69933