CymitQuimica logo
Proteasi/Proteasoma

Proteasi/Proteasoma

Gli inibitori delle proteasi e del proteasoma sono composti che bloccano l'attività delle proteasi e del proteasoma, che sono coinvolti nella degradazione e nel turnover delle proteine. Questi inibitori sono fondamentali per studiare la regolazione dell'omeostasi proteica, il controllo del ciclo cellulare e l'apoptosi. Gli inibitori delle proteasi e del proteasoma vengono anche utilizzati nel trattamento di malattie come il cancro, dove la degradazione anomala delle proteine svolge un ruolo nella progressione della malattia. Inibendo le proteasi o il proteasoma, questi composti possono indurre la morte cellulare nelle cellule tumorali e sono strumenti critici sia per la ricerca di base che per lo sviluppo terapeutico. Presso CymitQuimica, offriamo una vasta gamma di inibitori delle proteasi e del proteasoma di alta qualità per supportare la tua ricerca in biochimica, biologia cellulare e sviluppo di farmaci.

Sottocategorie di "Proteasi/Proteasoma"

Mostrare 3 più sottocategorie

Trovati 1092 prodotti di "Proteasi/Proteasoma"

Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
prodotti per pagina.
  • Inogatran
    Targetmol
    + Info

    Inogatran

    CAS:
    Inogatran is a synthetic thrombin inhibitor, developed for the possible treatment and prophylaxis of venous and arterial thrombotic diseases.
    Formula:C21H38N6O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:438.56

    Ref: TM-T11659

  • LY52
    Targetmol
    + Info

    LY52

    CAS:
    LY52 is a matrix metalloproteinase-2 inhibitor. It acts by suppressing tumor invasion and metastasis.
    Formula:C22H24N4O6
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:440.45

    Ref: TM-T25765

  • KCC009
    Targetmol
    + Info

    KCC009

    CAS:
    KCC009 is a potent and selective Transglutaminase 2 Inhibitor.
    Formula:C21H22BrN3O5
    Colore e forma:Solid
    Peso molecolare:476.32

    Ref: TM-T27717

  • JTK-853
    Targetmol
    + Info

    JTK-853

    CAS:
    JTK-853: novel non-nucleoside HCV polymerase inhibitor with strong antiviral activity (EC50: 0.38 μM genotype 1a, 0.035 μM 1b).
    Formula:C28H23F7N6O4S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:704.64

    Ref: TM-T15631

  • PTC725
    Targetmol
    + Info

    PTC725

    CAS:
    PTC725 is a selective HCV 1b replicons inhibitor. It has been shown to target the nonstructural protein 4B.
    Formula:C23H18F4N6O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:518.49

    Ref: TM-T24682

  • NCI-B16
    Targetmol
    + Info

    NCI-B16

    CAS:
    NCI-B16 is a small-molecule RNA binder that inhibits HCV (hepatitis C virus) replication [1].
    Formula:C27H26N8O4
    Colore e forma:Solid
    Peso molecolare:526.55

    Ref: TM-T81694

  • DS-1040 Tosylate
    Targetmol
    + Info

    DS-1040 Tosylate

    CAS:
    DS-1040 Tosylate is a thrombin-activated fibrinolysis inhibitor (TAFI) inhibitor and a fibrinolysis enhancer, used for researching thromboembolic diseases.
    Formula:C23H35N3O5S
    Colore e forma:Solid
    Peso molecolare:465.61

    Ref: TM-T11100

  • MK-3281
    Targetmol
    + Info

    MK-3281

    CAS:
    MK-3281: Oral, potent HCV NS5B inhibitor with promising properties and efficacy in replication trials, suitable for clinical use.
    Formula:C29H37N3O3
    Colore e forma:Solid
    Peso molecolare:475.62

    Ref: TM-T33432

  • Cipemastat
    Targetmol
    + Info

    Cipemastat

    CAS:
    Cipemastat is a competitive inhibitor of human collagenases 1, 2, and 3 (Kis: 3.0, 4.4, and 3.4 nM).
    Formula:C22H36N4O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:436.55

    Ref: TM-T10817

  • Collagen proline hydroxylase inhibitor
    Targetmol
    + Info

    Collagen proline hydroxylase inhibitor

    CAS:
    <p>Collagen proline hydroxylase inhibitor is an inhibitor collagen proline hydroxylase and useful for antifibrotic proliferative agents.</p>
    Formula:C18H18N4O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:354.36

    Ref: TM-T10862

  • Z-PDLDA-NHOH
    Targetmol
    + Info

    Z-PDLDA-NHOH

    CAS:
    Z-PDLDA-NHOH is a potent, specific vertebrate collagenase inhibitor [1].
    Formula:C22H32N4O6
    Colore e forma:Solid
    Peso molecolare:448.51

    Ref: TM-T80719

  • MMP13-IN-3
    Targetmol
    + Info

    MMP13-IN-3

    CAS:
    MMP13-IN-3 is an oral, selective MMP-13 inhibitor with IC50 of 1 nM, >1000x selective, for osteoarthritis treatment.
    Formula:C24H22N4O5
    Purezza:99.76%
    Colore e forma:Solid
    Peso molecolare:446.46

    Ref: TM-T16124

  • GSK-2485852
    Targetmol
    + Info

    GSK-2485852

    CAS:
    GSK-2485852, a NS5B inhibitor, is used potentially for treatment of HCV infection.
    Formula:C27H25BF2N2O6S
    Colore e forma:Solid
    Peso molecolare:554.37

    Ref: TM-T27463

  • XL-784 free base
    Targetmol
    + Info

    XL-784 free base

    CAS:
    XL-784 free base selectively inhibits MMPs with IC50: MMP-1 (1.9µM), MMP-2 (0.81nM), MMP-3 (120nM), MMP-8 (10.8nM), MMP-9 (18nM), MMP-13 (0.56nM).
    Formula:C21H22ClF2N3O8S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:549.93

    Ref: TM-T13357

  • MDL-101146, (R)-
    Targetmol
    + Info

    MDL-101146, (R)-

    CAS:
    MDL-101146, (R)- is an effective orally active inhibitor of human neutrophil elastase.
    Formula:C29H37F5N4O6
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:632.62

    Ref: TM-T25784

  • SSR 69071
    Targetmol
    + Info

    SSR 69071

    CAS:
    SSR69071: selective neutrophil elastase inhibitor, stronger for humans (Ki=0.0168 nM), may treat COPD, asthma, and reduce heart injury.
    Formula:C27H32N4O7S
    Colore e forma:Solid
    Peso molecolare:556.63

    Ref: TM-T21989

  • MMP-7-IN-3
    Targetmol
    + Info

    MMP-7-IN-3

    CAS:
    MMP-7-IN-3 (compound 15) is a potent and selective MMP-7 inhibitor, inhibiting renal fibrosis in a unilateral ureteral obstruction mouse model.
    Formula:C34H43ClF3N7O9S
    Purezza:99.915%
    Colore e forma:Solid
    Peso molecolare:818.26

    Ref: TM-T81778

  • Phe-Pro-Ala-pNA
    Targetmol
    + Info

    Phe-Pro-Ala-pNA

    CAS:
    Phe-Pro-Ala-pNA is a chromogenic substrate utilized for assessing tripeptidyl peptidase activity.
    Formula:C23H27N5O5
    Colore e forma:Solid
    Peso molecolare:453.49

    Ref: TM-T84840

  • MDL 27324
    Targetmol
    + Info

    MDL 27324

    CAS:
    MDL 27324 is an inhibitor of human neutrophil elastase.
    Formula:C29H38F3N5O6S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:641.7

    Ref: TM-T25782

  • BAY-678
    Targetmol
    + Info

    BAY-678

    CAS:
    BAY-678: Oral selective human neutrophil elastase inhibitor; IC50: 20 nM; SGC-approved chemical probe.
    Formula:C20H15F3N4O2
    Purezza:99.36%
    Colore e forma:Solid
    Peso molecolare:400.35

    Ref: TM-T10473