Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(939 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.945 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(148 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(407 prodotti)
- Recettore dell'endotelina(76 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(31 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(165 prodotti)
- Proteina Hedgehog/Smoothened(44 prodotti)
- Recettore dell'istamina(358 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(297 prodotti)
- PAFR(11 prodotti)
- PKA(48 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5352 prodotti di "Proteina G/GPCR"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Sumatriptan hydrochloride
CAS:<p>Sumatriptan hydrochloride (GR 43175), an oral 5-HT1 receptor agonist, treats migraines; Ki: 5-HT1D - 17 nM, 5-HT1B - 27 nM, 5-HT1A - 100 nM.</p>Formula:C14H22ClN3O2SColore e forma:SolidPeso molecolare:331.86Dioxopromethazine
CAS:<p>Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.</p>Formula:C17H20N2O2SPurezza:98%Colore e forma:SolidPeso molecolare:316.42Men 10376 TFA(135306-85-3,free)
<p>Men 10376 TFA(135306-85-3,free) (Neurokinin-2 receptor antagonist TFA) is an effective and selective tachykinin nk-2 receptor antagonist with a K I value of 4.4</p>Formula:C59H69F3N12O12Purezza:99.22%Colore e forma:SolidPeso molecolare:1195.25Temanogrel
CAS:<p>Temanogrel (APD791) is a highly selective antagonist of the 5-HT2A receptor (Ki: 4.9 nM).</p>Formula:C24H28N4O4Purezza:99.24%Colore e forma:SolidPeso molecolare:436.5Vercirnon sodium
CAS:<p>Vercirnon (GSK1605786A) sodium: oral CCR9 antagonist, inhibits Ca2+ mobilization/chemotaxis, IC50 = 2.6-5.4 nM, selective for CCR9 vs. CCR1-12/CX3CR1-7.</p>Formula:C22H21ClN2NaO4SColore e forma:SolidPeso molecolare:467.92AdipoRon hydrochloride
CAS:<p>AdipoRon hydrochloride is a specific, orally active AdipoR agonist, capable of binding AdipoR1 (Kd: 1.8 μM) and AdipoR2 (Kd: 3.1 μM).</p>Formula:C27H29ClN2O3Colore e forma:SolidPeso molecolare:464.99Risperidone hydrochloride
CAS:<p>Risperidone hydrochloride blocks 5-HT2, inhibits P-glycoprotein, and antagonizes D2 receptors (Ki: 5-HT2A - 4.8 nM, D2 - 5.9 nM).</p>Formula:C23H28ClFN4O2Colore e forma:SolidPeso molecolare:446.95Cinanserin
CAS:<p>Cinanserin is a serotonin 5-HT2 antagonist.</p>Formula:C20H24N2OSColore e forma:SolidPeso molecolare:340.48GSK2018682
CAS:<p>GSK2018682 is an agonist of sphingosine-1-phosphate receptor (s1p1) and (s1p5) agonist(pEC50s of 7.7 and 7.2,respectively).</p>Formula:C22H21ClN4O4Purezza:99.04%Colore e forma:SolidPeso molecolare:440.88Spiperone hydrochloride
CAS:<p>5-HT2A serotonin and selective D2-like dopamine receptor antagonist</p>Formula:C23H27ClFN3O2Purezza:98%Colore e forma:SolidPeso molecolare:431.93THIQ
CAS:<p>THIQ is a selective melanocortin-4 receptor (MC4R) agonist (hMC4R and rMC4R with IC50 of 1.2 nM and 0.6 nM , respectively).</p>Formula:C33H41ClN6O2Purezza:98.93%Colore e forma:SolidPeso molecolare:589.17Betazole
CAS:<p>Betazole, an oral H2 receptor agonist, stimulates gastric acid and raises bile duct pressure, used for gastric secretory testing.</p>Formula:C5H9N3Colore e forma:SolidPeso molecolare:111.15Nuciferine
CAS:<p>Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.</p>Formula:C19H21NO2Purezza:98.76% - 99.79%Colore e forma:SolidPeso molecolare:295.38Lys-Bradykinin acetate(342-10-9 free base)
CAS:<p>Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.</p>Formula:C58H89N17O14Purezza:99.86%Colore e forma:SolidPeso molecolare:1248.43SLF1081851 TFA
CAS:<p>SLF1081851 (TFA) inhibits Spns2, IC50 at 1.93 μM for S1P release, crucial for development and immunity.</p>Formula:C23H34F3N3O3Colore e forma:SolidPeso molecolare:457.538Haloperidol hydrochloride
CAS:<p>Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist which is a potent antipsychotic agent.</p>Formula:C21H24Cl2FNO2Colore e forma:SolidPeso molecolare:412.335-Hydroxy-1-methylhydantoin
CAS:<p>5-Hydroxy-1-methylhydantoin (HD-003) is an antioxidant potentially for the treatment of renal failure.</p>Formula:C4H6N2O3Purezza:99.99%Colore e forma:SolidPeso molecolare:130.1TCS-OX2-29
CAS:<p>TCS-OX2-29 is a potent and selective OX2 receptor antagonist (IC50: 40 nM). It displays >250-fold selectivity for OX2 over OX1.</p>Formula:C23H31N3O3Purezza:99.81%Colore e forma:SolidPeso molecolare:397.51Netupitant
CAS:<p>Netupitant (CID 6451149) is a specific neurokinin 1 (NK1) receptor antagonist (Ki: 0.95 nM).</p>Formula:C30H32F6N4OPurezza:99.43%Colore e forma:SolidPeso molecolare:578.59Zuclopenthixol
CAS:<p>Zuclopenthixol (cis-Clopenthixol) is a thioxanthene with therapeutic actions similar to the phenothiazine antipsychotics.</p>Formula:C22H25ClN2OSPurezza:98.9% - 99.82%Colore e forma:SolidPeso molecolare:400.96RS-127445
CAS:<p>RS-127445 (MT500) is a selective 5-HT2B receptor antagonist with pKi of 9.5 and pIC50 of 10.4, exhibits >1000-fold selectivity against other 5-HT receptors.</p>Formula:C17H16FN3Purezza:99.32%Colore e forma:SolidPeso molecolare:281.33H2L 5765834
CAS:<p>H2L 5765834 is a lysophosphatidic acid receptors antagonist</p>Formula:C21H12N2O7Purezza:98.25% - 99.47%Colore e forma:SolidPeso molecolare:404.33Paltusotine
CAS:<p>Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.</p>Formula:C27H22F2N4OPurezza:99.91%Colore e forma:SolidPeso molecolare:456.49ELA-14(human) acetate
<p>ELA-14(human) acetate, a fragment of ELA, targets APJ, activates Gαi1 and β-arrestin-2, and prompts receptor internalization like its parent peptide.</p>Formula:C77H123N25O19S2Purezza:97.2%Colore e forma:SolidPeso molecolare:1767.09Dasotraline hydrochloride
CAS:<p>Dasotraline hydrochloride, a dopamine, norepinephrine, and serotonin reuptake inhibitor with IC50s: 4, 6, 11 nM.</p>Formula:C16H16Cl3NPurezza:98.92% - 99.6%Colore e forma:SolidPeso molecolare:328.66SB399885
CAS:<p>SB399885 is a potent, brain-penetrant, oral SR-6 antagonist with 200-fold selectivity for SR-6 receptors.</p>Formula:C18H21Cl2N3O4SPurezza:98.94%Colore e forma:SolidPeso molecolare:446.35HTMT dimaleate
CAS:<p>HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.</p>Formula:C27H33F3N4O9Purezza:99.51%Colore e forma:SolidPeso molecolare:614.57Pardoprunox hydrochloride
CAS:<p>Pardoprunox hydrochloride (SLV-308 hydrochloride) is a novel partial dopamine D2 and D3 receptor agonist and serotonin 5-HT1A receptor agonist, D2 (pKi = 8.1)</p>Formula:C12H16ClN3O2Purezza:98.95% - 99.13%Colore e forma:SolidPeso molecolare:269.73BAY 41-8543
CAS:<p>BAY 41-8543 is a nitric oxide (NO)-independent stimulator of soluble guanylyl cyclase (sGC).</p>Formula:C21H21FN8OPurezza:99.86%Colore e forma:SolidPeso molecolare:420.44RO1138452
CAS:<p>RO1138452 (CAY10441) blocks prostacyclin receptor; orally active, high affinity (Ki: 1.5 nM), analgesic in rats (2-20 mg/kg).</p>Formula:C19H23N3OPurezza:97.01% - 99.34%Colore e forma:SolidPeso molecolare:309.41Carcinine ditrifluoroacetate Acetate
<p>Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.</p>Formula:C14H20F6N4O7Purezza:98.18%Colore e forma:SolidPeso molecolare:470.32Hemokinin 1 (mouse) acetate(208041-90-1 free base)
<p>Mouse Hemokinin-1 acetate: NK1 receptor agonist, Ki=0.175 nM; NK2 Ki=560 nM.</p>Formula:C63H104N22O17SPurezza:98.33%Colore e forma:SolidPeso molecolare:1473.72MHP
CAS:<p>MHP (Methyl caprooyl tyrosinate) is an activator of sphingosine kinase (SPHK1), and significantly stimulates CAMP mRNA and protein production in KC.</p>Formula:C16H23NO4Purezza:98.58%Colore e forma:SolidPeso molecolare:293.36Vericiguat
CAS:<p>Vericiguat (BAY1021189) is a potent and orally available guanylate cyclase stimulator.</p>Formula:C19H16F2N8O2Purezza:98.86% - 99.93%Colore e forma:SolidPeso molecolare:426.38Sarpogrelate hydrochloride
CAS:<p>Sarpogrelate hydrochloride (MCI-9042), a 5-HT2 antagonist with high affinity (Ki=8.39nM), is used as an anti-platelet for PAD, improving vascular function.</p>Formula:C24H32ClNO6Purezza:99.73%Colore e forma:Colorless LiquidPeso molecolare:465.97Cinitapride
CAS:<p>Cinitapride (Blaston) treats acid reflux and gastric issues, targeting 5-HT2, 5-HT1, and 5-HT4 receptors.</p>Formula:C21H30N4O4Purezza:99.52%Colore e forma:SolidPeso molecolare:402.49LY2828360
CAS:<p>LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and >100 μM.</p>Formula:C22H27ClN6OPurezza:98.45% - 99.51%Colore e forma:SolidPeso molecolare:426.94Thozalinone
CAS:<p>Thozalinone is a psychostimulant agent inducing the release of norepinephrine and dopamine.</p>Formula:C11H12N2O2Purezza:99.68%Colore e forma:SolidPeso molecolare:204.23Fabomotizole
CAS:<p>Fabomotizole (Obenoxazine) is an anxiolytic drug; produces anxiolytic and neuroprotective effects without any sedative or muscle relaxant actions.</p>Formula:C15H21N3O2SPurezza:99.4%Colore e forma:SolidPeso molecolare:307.41BI-6015
CAS:<p>BI 6015 is an antagonist of HNF4α. HNF4α is a nuclear receptor that regulates gene expression in the intestine cells, liver cells, and pancreas-β cells.</p>Formula:C15H13N3O4SPurezza:99.81%Colore e forma:SolidPeso molecolare:331.35ACTH (1-39) human
CAS:<p>Adrenocorticotropic Hormone (ACTH) (1-39), human (ACTH (1-39), human) is an agonist of melanocortin receptor.</p>Formula:C207H308N56O58SPurezza:99.6%Colore e forma:White Lyophilised SolidPeso molecolare:4541.14Solabegron HCl
CAS:<p>Solabegron is a β3 adrenergic receptor agonist that also promotes visceral pain relief by releasing somatostatin.</p>Formula:C23H24Cl2N2O3Colore e forma:SolidPeso molecolare:447.35Tiaramide hydrochloride
CAS:<p>Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.</p>Formula:C15H19Cl2N3O3SPurezza:98.48%Colore e forma:SolidPeso molecolare:392.3Acitazanolast
CAS:<p>Acitazanolast (WP-871) is an anti-allergic drug candidate.</p>Formula:C9H7N5O3Purezza:98.25%Colore e forma:SolidPeso molecolare:233.18Emorfazone
CAS:<p>Emorfazone (PH011085) has an anti-nociceptive effect.</p>Formula:C11H17N3O3Purezza:99.89%Colore e forma:SolidPeso molecolare:239.27Darbufelone mesylate
CAS:<p>Darbufelone mesylate blocks PGF2α, LTB4, PGHS-2 (IC50: 0.19 μM), and PGHS-1 (IC50: 20 μM).</p>Formula:C19H28N2O5S2Purezza:96.81% - 99.92%Colore e forma:SolidPeso molecolare:428.57Cloprostenol sodium salt
CAS:<p>Cloprostenol sodium salt (ICI 80996 sodium salt) is a synthetic prostaglandin analogue, an agonist at the PGF2α receptor, with luteolytic properties.</p>Formula:C22H28ClNaO6Purezza:97.17% - 98.47%Colore e forma:White To Almost White Hygroscopic PowderPeso molecolare:446.9Tianeptine
CAS:<p>Tianeptine (Tianeptine sodium) 是一种选择性5-HT 摄取促进剂，具有抗抑郁、抗焦虑和神经保护作用，可用于缓解疼痛的研究。</p>Formula:C21H25ClN2O4SPurezza:99.04%Colore e forma:SolidPeso molecolare:436.95ML-097
CAS:<p>ML-097 (CID-2160985) is a pan activator of Ras-related GTPases</p>Formula:C14H11BrO3Purezza:99.12%Colore e forma:SolidPeso molecolare:307.139Atipamezole hydrochloride
CAS:<p>Atipamezole is a synthetic α2 adrenergic receptor antagonist.</p>Formula:C14H16N2·HClPurezza:99.74%Colore e forma:SolidPeso molecolare:248.75AM281
CAS:<p>AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.</p>Formula:C21H19Cl2IN4O2Purezza:98.6% - >99.99%Colore e forma:White To Off-White SolidPeso molecolare:557.21Prazosin
CAS:<p>Prazosin (Prazosine), an α1-blocker, acts as an inverse agonist at alpha-1 adrenergic receptors and is used to treat hypertension.</p>Formula:C19H21N5O4Purezza:99.86%Colore e forma:White To Tan Powder SolidPeso molecolare:383.4MK-571 sodium
CAS:<p>MK-571 sodium, a CysLT1 antagonist and MRP2 inhibitor, obstructs drug efflux and hampers enterocyte phase-2 conjugation of flavonoids.</p>Formula:C26H27ClN2O3S2·NaPurezza:97.86% - 99.58%Colore e forma:SolidPeso molecolare:537.07E7046
CAS:<p>E7046 is a specific, orally bioavailable EP4 antagonist (IC50: 13.5 nM, Ki: 23.14 nM), exhibiting anti-tumor activities.</p>Formula:C22H18F5N3O4Purezza:99.86%Colore e forma:SolidPeso molecolare:483.4Phenylephrine
CAS:<p>Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).</p>Formula:C9H13NO2Purezza:99.5% - 99.89%Colore e forma:SolidPeso molecolare:167.21Isocorynoxeine
CAS:<p>Isocorynoxeine reduces blood pressure, dilates vessels, and guards neurons against ischemia and glutamate toxicity.</p>Formula:C22H26N2O4Purezza:98% - 99.9%Colore e forma:SolidPeso molecolare:382.45Etelcalcetide hydrochloride
CAS:<p>Etelcalcetide HCl, a synthetic peptide modulator of CaSR, lowers PTH in dialysis patients with secondary hyperparathyroidism.</p>Formula:C38H73N21O10S2HClPurezza:>99.99%Colore e forma:SolidPeso molecolare:1353.33Betahistine EP Impurity C
CAS:<p>Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.</p>Formula:C15H19N3Purezza:≥95%Colore e forma:SolidPeso molecolare:241.33Methiothepin mesylate
CAS:<p>Methiothepin mesylate (Metitepine mesylate) is a potent and non-selective 5-HT2 receptor antagonist, used as an antipsychotic.</p>Formula:C21H28N2O3S3Purezza:98% - 99.92%Colore e forma:SolidPeso molecolare:452.65Praliciguat
CAS:<p>Praliciguat (IW-1973) is an orally active sGC stimulator with a 197 nM EC50 in HEK-293 cells, enhances NO signaling, and is a vasodilator.</p>Formula:C21H14F8N6O2Purezza:98.82%Colore e forma:SolidPeso molecolare:534.365-Benzyloxygramine
CAS:<p>5-Benzyloxygramine blocks the Dopamin receptors and antagonizes the effects of 5-HT on the rat uterus and the rabbit ear.</p>Formula:C18H20N2OPurezza:99.13%Colore e forma:SolidPeso molecolare:280.36S1p receptor agonist 1
CAS:<p>S1p receptor agonist 1 (S1p-receptor-agonist-1) is an S1P receptor agonist.</p>Formula:C23H24FN3O3Purezza:99.07% - 99.9%Colore e forma:SolidPeso molecolare:409.45[Pyr1]-Apelin-13
CAS:<p>[Pyr1]-Apelin-13 ([pGlu1]-Apelin-13) is a potent and selective endogenous Apelin receptor (APJ) agonist.</p>Formula:C69H108N22O16SPurezza:99.71%Colore e forma:SolidPeso molecolare:1533.8VPC171
CAS:<p>VPC171 is a novel adenosine A1 receptor positive allosteric modulator (PAM).</p>Formula:C18H12F3NOSPurezza:99.78%Colore e forma:SolidPeso molecolare:347.35BAY-545
CAS:<p>BAY-545 is an antagonist of A2B adenosine receptor(IC50 : 59 nM).</p>Formula:C18H22F3N3O4SPurezza:98.05%Colore e forma:SolidPeso molecolare:433.45Lixisenatide acetate (320367-13-3 free base)
CAS:<p>Lixisenatide acetate is a receptor agonist similar to glucagon-like peptide-1 (glp-1) for the treatment of type 2 diabetes mellitus (T2DM).</p>Formula:C215H347N61O65S·6C2H4O2Purezza:98% - 99.9%Colore e forma:SolidPeso molecolare:5218.88MF-766
CAS:<p>MF-766: potent, selective oral EP4 antagonist, Ki=0.23 nM, IC50=1.4 nM; shifts to 1.8 nM with 10% HS. Useful in cancer, inflammation studies.</p>Formula:C27H21F3N2O3Purezza:99.54% - 99.59%Colore e forma:SolidPeso molecolare:478.46Regadenoson
CAS:<p>Regadenoson (CVT-3146) is a selective A2A receptor agonist that increases coronary blood flow with a longer half-life than adenosine.</p>Formula:C15H18N8O5Purezza:99.57% - 99.81%Colore e forma:Off-White SolidPeso molecolare:390.35Ciproxifan maleate
CAS:<p>Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity</p>Formula:C20H22N2O6Purezza:99.39%Colore e forma:SolidPeso molecolare:386.4BWX 46 Acetate
<p>BWX 46 Acetate is a potent, highly selective neuropeptide Y (NPY) receptor agonist with IC50 of 0.5 nM.</p>Formula:C118H190N36O30S2Purezza:96.86%Colore e forma:SolidPeso molecolare:2657.12ACEPROMAZINE MALEATE
CAS:<p>ACEPROMAZINE MALEATE is a dopamine receptor antagonist</p>Formula:C23H26N2O5SPurezza:98.87% - 99.51%Colore e forma:Off White Or Yellow Crystalline PowderPeso molecolare:442.53CGP71683 hydrochloride
CAS:<p>CGP71683 hydrochloride: NPY5 receptor antagonist, Ki=1.3 nM; inactive at Y1 (Ki >4000 nM) and Y2 (Ki=200 nM).</p>Formula:C26H30ClN5O2SPurezza:99.92%Colore e forma:SolidPeso molecolare:512.07Perospirone
CAS:<p>Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.</p>Formula:C23H30N4O2SPurezza:99.23%Colore e forma:White PowderPeso molecolare:426.57DAPTA
CAS:<p>DAPTA (Adaptavir) is an inhibitor of CCR5, shows potent anti-HIV activities.</p>Formula:C35H56N10O15Purezza:>99.99%Colore e forma:SolidPeso molecolare:856.88Bevantolol hydrochloride
CAS:<p>Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.</p>Formula:C20H28ClNO4Purezza:99.49%Colore e forma:SolidPeso molecolare:381.9Pimozide
CAS:<p>Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.</p>Formula:C28H29F2N3OPurezza:99.63% - >99.99%Colore e forma:SolidPeso molecolare:461.55N-Desmethylclozapine
CAS:<p>N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.</p>Formula:C17H17ClN4Purezza:97.25% - 99.83%Colore e forma:Yellow Crystalline SolidPeso molecolare:312.8OXOMEMAZINE
CAS:<p>Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.</p>Formula:C18H22N2O2SPurezza:99.58%Colore e forma:SolidPeso molecolare:330.44Clemizole
CAS:<p>Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.</p>Formula:C19H20ClN3Purezza:98% - 99.65%Colore e forma:SolidPeso molecolare:325.84Taladegib
CAS:<p>Taladegib (LY2940680), an oral Smo receptor antagonist, targets Hedgehog signaling for cancer treatment.</p>Formula:C26H24F4N6OPurezza:98.75% - >99.99%Colore e forma:SolidPeso molecolare:512.5Sevoflurane
CAS:<p>Sevoflurane (Fluoromethyl), a noncompetitive inhibitor of 5-HT3 receptor, acts as a low-soluble inhalation anesthetics.</p>Formula:C4H3F7OPurezza:98%Colore e forma:Less Oil Colorless OilPeso molecolare:200.05ML-SI3
CAS:<p>CCG-143140 is a GLP-1 receptor inverse agonists.</p>Formula:C23H31N3O3SPurezza:99.75%Colore e forma:SolidPeso molecolare:429.58PF-4136309
CAS:<p>PF-4136309 (INCB8761) is a specific, effective, and orally bioavailable CCR2 antagonist.</p>Formula:C29H31F3N6O3Purezza:98.85% - 99.47%Colore e forma:SolidPeso molecolare:568.59HhAntag
CAS:<p>HhAntag is a small molecule inhibitor of GLI1-mediated transcription, an essential down-stream element of the Hedgehog (Hh) pathway with the anti-tumor activity</p>Formula:C24H23ClN4O3Purezza:95.73%Colore e forma:SolidPeso molecolare:450.92SAG
CAS:<p>SAG (Smoothened Agonist) is a Smo receptor agonist (EC50=3 nM) that is cell-permeable and selective.</p>Formula:C28H28ClN3OSPurezza:97.37% - 98.88%Colore e forma:SolidPeso molecolare:490.06Ciliobrevin A
CAS:<p>Ciliobrevin A (HPI-4) is an inhibitor of hedgehog signaling pathway with an IC50 <10 μM.</p>Formula:C17H9Cl2N3O2Purezza:98.54% - 99.57%Colore e forma:SolidPeso molecolare:358.18SANT-1
CAS:<p>SANT-1 directly binds to Smoothened (Smo) receptor (Kd: 1.2 nM) and inhibits Smo agonist effects (IC50: 20 nM).</p>Formula:C23H27N5Purezza:99.98% - >99.99%Colore e forma:SolidPeso molecolare:373.49Felypressin
CAS:<p>Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.</p>Formula:C46H65N13O11S2Purezza:99.65%Colore e forma:SolidPeso molecolare:1040.22VUF10460
CAS:<p>VUF10460 is a non-imidazole histamine H4 receptor agonist.</p>Formula:C15H19N5Purezza:99.44% - 99.57%Colore e forma:SolidPeso molecolare:269.34Ansofaxine hydrochloride
CAS:<p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>Formula:C24H32ClNO3Purezza:99.57% - 99.77%Colore e forma:SolidPeso molecolare:417.97Nelotanserin
CAS:<p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>Formula:C18H15BrF2N4O2Purezza:98.42% - 99.88%Colore e forma:SolidPeso molecolare:437.24I-191
CAS:<p>I-191 is a potent antagonist of protease-activated receptor 2 (PAR2), inhibits multiple signaling functions in human cancer cells.</p>Formula:C23H26FN5O2Purezza:99.8%Colore e forma:SolidPeso molecolare:423.48AR-M 1896 Acetate
<p>AR-M 1896 Acetate is the selective agonist of GalR2.</p>Formula:C56H85N13O16Purezza:99.76%Colore e forma:SolidPeso molecolare:1196.35AM966
CAS:<p>AM966, a excellent affinity, specific, oral LPA1(IC50=17 nM) antagonist, suppresses LPA-stimulated intracellular calcium release.</p>Formula:C27H23ClN2O5Purezza:98.06% - 99.79%Colore e forma:SolidPeso molecolare:490.93Lurasidone hydrochloride
CAS:<p>Lurasidone HCl: Atypical antipsychotic, treats schizophrenia & bipolar, affects dopamine, serotonin & adrenergic receptors.</p>Formula:C28H36N4O2S·HClPurezza:99.51%Colore e forma:SolidPeso molecolare:529.14GBR 12935 dihydrochloride
CAS:<p>GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.</p>Formula:C28H36Cl2N2OPurezza:99.09% - ≥95%Colore e forma:SolidPeso molecolare:487.5GLP-1(7-36), amide
CAS:<p>GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.</p>Formula:C149H226N40O45Purezza:99.85%Colore e forma:White PowderPeso molecolare:3297.63FSLLRY-NH2 TFA(245329-02-6 free base)
<p>FSLLRY-NH2 TFA inhibits PAR2, reverses taxol-induced pain, and reduces itch in mice; blocks ERK and collagen in fibroblasts.</p>Formula:C41H61F3N10O10Purezza:99.32%Colore e forma:SolidPeso molecolare:910.99Brexpiprazole
CAS:<p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>Formula:C25H27N3O2SPurezza:99.06% - 99.96%Colore e forma:SolidPeso molecolare:433.57Brimonidine Tartrate
CAS:<p>Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM).</p>Formula:C15H16BrN5O6Purezza:99.95%Colore e forma:Off-White Crystalline SolidPeso molecolare:442.22
![[Pyr1]-Apelin-13](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1260.webp&w=3840&q=75)
