Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(939 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.945 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(148 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(407 prodotti)
- Recettore dell'endotelina(76 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(31 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(165 prodotti)
- Proteina Hedgehog/Smoothened(44 prodotti)
- Recettore dell'istamina(358 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(297 prodotti)
- PAFR(11 prodotti)
- PKA(48 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5352 prodotti di "Proteina G/GPCR"
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GRK5-IN-2
CAS:<p>GRK5-IN-2, a pyridine-based bicyclic compound, is a potent G-protein-coupled receptor kinase 5 (GRK5) inhibitor.</p>Formula:C20H20N4O4Purezza:99.92%Colore e forma:SolidPeso molecolare:380.4Afamelanotide acetate
CAS:<p>Afamelanotide acetate is a synthetic α-melanocyte stimulating hormone analogue and first-in-class melanocortin-1 receptor agonist.</p>Formula:C80H115N21O21Purezza:98% - 99.494%Colore e forma:SolidPeso molecolare:1706.9Dobutamine tartrate
CAS:<p>Dobutamine tartrate is a cardiotonic.</p>Formula:C22H29NO9Colore e forma:SolidPeso molecolare:451.472SB-200646
CAS:<p>SB-200646 is a selective and potent antagonist of 5-HT2B/5-HT2C receptor</p>Formula:C15H14N4OPurezza:99.61%Colore e forma:SolidPeso molecolare:266.3Nifenalol
CAS:<p>Nifenalol is an adrenergic beta-blocker with good antiarrhythmic properties. It tends to lower blood pressure and provide protection against angina.</p>Formula:C11H16N2O3Purezza:98%Colore e forma:SolidPeso molecolare:224.26Chlorpheniramine
CAS:<p>Chlorpheniramine is an H1 anti-histamine agent for IgE-mediated inflammation that is commonly used for allergic diseases.</p>Formula:C16H19ClN2Colore e forma:SolidPeso molecolare:274.79Ralmitaront
CAS:<p>Ralmitaront (RO6889450) is a potent, orally active partial agonist of the trace amine-associated receptor 1 (TAAR1).</p>Formula:C17H22N4O2Purezza:99.71% - 99.79%Colore e forma:SolidPeso molecolare:314.38AdipoRon
CAS:<p>AdipoRon (SC-396658) is an orally bioavailable adiponectin receptor agonist. It can combine with AdipoR1/2 (KD: 1.8/3.1 μM).</p>Formula:C27H28N2O3Purezza:97.90% - 99.86%Colore e forma:SolidPeso molecolare:428.52Bupranolol
CAS:<p>Bupranolol blocks β2-adrenergic receptor; treats angina, hypertension, glaucoma, arrhythmia, and prevents clots.</p>Formula:C14H22ClNO2Purezza:97.63%Colore e forma:SolidPeso molecolare:271.78Droxidopa
CAS:<p>Droxidopa (L-DOPS), an oral prodrug, treats symptomatic orthostatic hypotension from neurogenic autonomic failure.</p>Formula:C9H11NO5Purezza:97.27% - 99.88%Colore e forma:SolidPeso molecolare:213.19Ocaperidone
CAS:<p>Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.</p>Formula:C24H25FN4O2Purezza:99.33%Colore e forma:SolidPeso molecolare:420.48Neuropeptide Y (29-64), amide, human acetate
<p>Neuropeptide Y (29-64), amide, human acetate is involved in Alzheimer's disease (AD) and protects rat cortical neurons against β-Amyloid toxicity.</p>Purezza:98.42%Colore e forma:LiquidPeso molecolare:N/AVeralipride
CAS:<p>Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.</p>Formula:C17H25N3O5SPurezza:99.65%Colore e forma:SolidPeso molecolare:383.46Adenosine amine congener
CAS:<p>Adenosine amine congener (ADAC) (ADAC) is an agonist of selective A1 adenosine receptor,.</p>Formula:C28H32N8O6Purezza:97.86%Colore e forma:SolidPeso molecolare:576.6Amezinium methylsulfate
CAS:<p>Amezinium methylsulfate (Lu-1631) has multiple mechanisms, including stimulation of α and β-1 receptors and inhibition of noradrenaline and tyramine uptake.</p>Formula:C12H15N3O5SPurezza:99.64%Colore e forma:SolidPeso molecolare:313.33Canagliflozin
CAS:<p>Canagliflozin (JNJ 28431754AAA) is a selective SGLT2 inhibitor. Canagliflozin is used to treat type II diabetes mellitus. Cost-effective and quality-assured.</p>Formula:C24H25FO5SPurezza:98.01% - >99.99%Colore e forma:SolidPeso molecolare:444.52Tripelennamine
CAS:<p>Tripelennamine: ethylenediamine derivative, H1-receptor blocker, reduces allergic reactions, treats rhinitis and conjunctivitis.</p>Formula:C16H21N3Colore e forma:SolidPeso molecolare:255.36GW627368
CAS:<p>GW627368 (GW 627368X)X is a novel, potent and selective antagonist of prostanoid EP4 receptor.</p>Formula:C30H28N2O6SPurezza:99.75% - 99.92%Colore e forma:SolidPeso molecolare:544.62Syk Inhibitor II dihydrochloride
CAS:<p>Syk inhibitor II selectively blocks Syk (IC50 = 41 nM), impacting platelet function and inflammation, with lower potency against other kinases.</p>Formula:C14H17Cl2F3N6OPurezza:98.53%Colore e forma:SolidPeso molecolare:413.22AVN-101
CAS:<p>AVN-101 is a very potent 5-HT7 receptor antagonist.Cost-effective and quality-assured.</p>Formula:C21H25ClN2Purezza:99.61%Colore e forma:SolidPeso molecolare:340.89Diquafosol tetrasodium
CAS:<p>Diquafosol Tetrasodium is a P2Y2 receptor agonist that stimulates the secretion of mucins from ocular tissues Diquafosol tetrasodium (INS365) improves tear film</p>Formula:C18H22N4Na4O23P4Purezza:98.25% - 99.97%Colore e forma:SolidPeso molecolare:878.23(+)-PD 128907 hydrochloride
CAS:<p>(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .</p>Formula:C14H20ClNO3Purezza:97.76%Colore e forma:SolidPeso molecolare:285.77Exendin-4
CAS:<p>Exenatide: GLP-1 receptor agonist, 39-amino acid, longer half-life (2.4 hrs), IC50 of 3.22 nM.</p>Formula:C184H282N50O60SPurezza:97.71% - 99.78%Colore e forma:SolidPeso molecolare:4186.57Conopressin S acetate(111317-90-9 free base)
<p>Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b</p>Formula:C43H77N17O12S2Purezza:99.79%Colore e forma:SolidPeso molecolare:1088.32BD1063 dhydrochloride
CAS:<p>BD1063 dhydrochloride is a potent and selective sigma 1(σ1) receptor antagonist(Ki = 9 nM).</p>Formula:C13H20Cl4N2Purezza:99.52% - ≥95%Colore e forma:SolidPeso molecolare:346.12Vilanterol trifenatate
CAS:<p>Vilanterol trifenatate is a long-acting agonist of β2-adrenoceptor (β2-AR) with inherent 24-hour activity(β2-AR, β1-AR and β3-AR pEC50s of 10.37, 6.98 and 7.36, respectively)</p>Formula:C44H49Cl2NO7Purezza:99.51% - >99.99%Colore e forma:SolidPeso molecolare:774.77S 14506 HCl
CAS:<p>S 14506 HCl: Strong 5-HT1A agonist; pKi - 9.0 (5-HT1A), 6.6 (5-HT1B/C), <6.0 (5-HT3).</p>Formula:C24H26FN3O2Colore e forma:SolidPeso molecolare:407.48Etrasimod
CAS:<p>Etrasimod (APD334) is a specific and orally available antagonist of the sphingosine-1-phosphate-1 (S1P1) receptor (IC50: 1.88 nM in CHO cells).</p>Formula:C26H26F3NO3Purezza:98.52% - 99.73%Colore e forma:SolidPeso molecolare:457.48Fluparoxan HCl
CAS:<p>Fluparoxan is a potent α2-adrenergic receptor antagonist (pKB = 7.9) with excellent α2/α1 selectivity (2630 fold).</p>Formula:C10H11ClFNO2Colore e forma:SolidPeso molecolare:231.65CP 376395
CAS:<p>CP 376395 (CP-316311) is an effective and specific Corticotropin-releasing factor 1 (CRF1) receptor antagonist.</p>Formula:C21H30N2OPurezza:99.86% - 99.94%Colore e forma:SolidPeso molecolare:326.48T-1095
CAS:<p>T-1095 is an inhibitor of renal glucose reabsorption and the expression of Na+-glucose cotransporters (SGLTs) and facilitative glucose transporter 2 (GLUT2).</p>Formula:C26H28O11Purezza:99.78%Colore e forma:SolidPeso molecolare:516.49Dasotraline
CAS:<p>Dasotraline: a triple reuptake inhibitor targeting DA, NE, and 5-HT with IC50 values of 4, 6, 11 nM. Possible new antidepressant class.</p>Formula:C16H15Cl2NColore e forma:SolidPeso molecolare:292.2Nelotanserin
CAS:<p>Nelotanserin (APD125): strong 5-HT2A inverse agonist (IC50: 1.7 nM), moderate 5-HT2C (79 nM), weak 5-HT2B (791 nM).</p>Formula:C18H15BrF2N4O2Purezza:98.42% - 99.88%Colore e forma:SolidPeso molecolare:437.24Pancreatic Polypeptide (human) acetate
<p>Pancreatic Polypeptide (human) acetate is a C-terminally amidated 36 amino acid peptide, which acts as a neuropeptide Y (NPY) Y4/Y5 receptor agonist.</p>Purezza:97.26%Colore e forma:LiquidPeso molecolare:N/AClobenpropit 2HBr
CAS:<p>Clobenpropit 2HBr is a histamine H3 receptor antagonist. It has neuroprotective effects via stimulation of GABA release in the brain.</p>Formula:C14H17ClN4SColore e forma:SolidPeso molecolare:308.83TNCA
CAS:<p>TNCA (Lycoperodine-1) is a high-affinity CaSR ligand (CaSRL) with co-agonist activity.</p>Formula:C12H12N2O2Purezza:97.33% - 97.73%Colore e forma:SolidPeso molecolare:216.24Velneperit
CAS:<p>Velneperit (S2367) is potent and selective neuropeptide Y (NPY) Y5 receptor under evaluating for treatment of obesity.</p>Formula:C17H24F3N3O3SPurezza:99.70%Colore e forma:SolidPeso molecolare:407.45Mecamylamine
CAS:<p>Mecamylamine: oral, noncompetitive nAChR blocker, crosses blood-brain barrier, for neuropsychiatric and hypertension research.</p>Formula:C11H21NColore e forma:SolidPeso molecolare:167.29Midaglizole
CAS:<p>Midaglizole, an α2-adrenoceptor blocker, raises blood pressure and lowers glucose.</p>Formula:C16H17N3Colore e forma:SolidPeso molecolare:251.33SCH442416
CAS:<p>SCH442416: selective A2A adenosine receptor antagonist; Ki: 0.048 nM (human), 0.5 nM (rat).</p>Formula:C20H19N7O2Purezza:99.58%Colore e forma:SolidPeso molecolare:389.41CHEMBL241987
CAS:<p>CHEMBL241987 targets the Adenosine receptor A3 (human)</p>Formula:C16H11N3OPurezza:99.81%Colore e forma:SolidPeso molecolare:261.28Ritanserin
CAS:<p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>Formula:C27H25F2N3OSPurezza:99.77% - 99.89%Colore e forma:SolidPeso molecolare:477.57Neuropeptide SF(mouse,rat) acetate
<p>Neuropeptide SF (mouse,rat) acetate is a NPFF receptor agonist with Ki of 48.4 nM (NPFF1) & 12.1 nM (NPFF2), enhancing ASIC3 current.</p>Formula:C42H69N13O12Purezza:98.37%Colore e forma:SolidPeso molecolare:948.08Eltoprazine hydrochloride
CAS:<p>Eltoprazine hydrochloride (DU 28853 hydrochloride) is a partial agonist at serotonin 5-HT1A, 5-HT1B, and 5-HT2B receptors (Ki value of 40, 52, and 81 nM,</p>Formula:C12H17ClN2O2Purezza:99.35%Colore e forma:SolidPeso molecolare:256.73Guanfacine hydrochloride
CAS:<p>Guanfacine hydrochloride (Intuniv) is a centrally acting antihypertensive agent with specificity towards ADRENERGIC ALPHA-2 RECEPTORS.</p>Formula:C9H10Cl3N3OPurezza:99.89% - 99.91%Colore e forma:SolidPeso molecolare:282.55TY-52156
CAS:<p>TY-52156 is an effective and selective S1P3 receptor antagonist (Ki: 110 nM).</p>Formula:C18H19Cl2N3OPurezza:99.91% - 99.91%Colore e forma:SolidPeso molecolare:364.27Nemifitide acetate(173240-15-8 free base)
<p>Nemifitide acetate, synthetic 5-amino acid antidepressant, has quick effect, mimics MIF.</p>Formula:C35H47FN10O8Purezza:97.97%Colore e forma:SolidPeso molecolare:754.85Paltusotine
CAS:<p>Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.</p>Formula:C27H22F2N4OPurezza:99.91%Colore e forma:SolidPeso molecolare:456.49Carazolol
CAS:<p>Carazolol (Suacron) is a high-affinity antagonist/partial inverse agonist (also referred to as a beta blocker) of the β-adrenergic receptor.</p>Formula:C18H22N2O2Purezza:99% - 99.53%Colore e forma:Yellowish SolidPeso molecolare:298.38PD-168077 maleate
CAS:<p>PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)</p>Formula:C24H26N4O5Purezza:99.13%Colore e forma:SolidPeso molecolare:450.49ANP(1-28) Acetate (human, porcine)
CAS:<p>Carperitide acetate: 28-amino acid hormone from human heart, counters cardiac injury/stretch, reduces endothelin-1.</p>Formula:C129H207N45O41S3Purezza:98.24%Colore e forma:SolidPeso molecolare:3140.5Verucerfont
CAS:<p>Verucerfont (NBI77860) is an antagonist of corticotropin-releasing factor receptor 1 (CRF1) .</p>Formula:C22H26N6O2Purezza:99.90%Colore e forma:SolidPeso molecolare:406.48Opaganib
CAS:<p>Opaganib (ABC294640) is an orally active and specific sphingosine kinase-2 (SphK2) inhibitor (IC50: 60 μM).</p>Formula:C23H25ClN2OPurezza:98.86% - 99.85%Colore e forma:SolidPeso molecolare:380.91Dimemorfan phosphate
CAS:<p>Dimemorfan phosphate (3,17-dimethylmorphinan) is a sigma 1 receptor agonist. Dimemorfan phosphate is used as a potent antitussive.</p>Formula:C18H25N·H3O4PPurezza:99.65%Colore e forma:SolidPeso molecolare:353.4Phenelzine
CAS:Phenelzine is a MAOI antidepressant, boosting brain catecholamines, effective for endogenous depression.Formula:C8H12N2Purezza:98%Colore e forma:LiquidPeso molecolare:136.19MK-1064
CAS:<p>MK-1064 (Urokinase inhibitor 1) is a selective orexin 2 receptor antagonist (2-SORA).</p>Formula:C24H20ClN5O3Purezza:99.19% - 99.82%Colore e forma:SolidPeso molecolare:461.9Melatonin
CAS:<p>Melatonin (Melatonine) is a natural hormone that activates melatonin receptors. Melatonin regulates the biological clock. Cost-effective and quality-assured.</p>Formula:C13H16N2O2Purezza:98% - 99.89%Colore e forma:Pale Yellow Leaflets From Benzene SolidPeso molecolare:232.28Exo-1
CAS:<p>Exo-1 (Methyl 3-(4-fluorobenzoyl)-6-methyl-2-pyridinecarboxylate) is a synthetic compound that has been shown to affect the metabolism of various nutrients, as</p>Formula:C15H12FNO3Purezza:99.45%Colore e forma:SolidPeso molecolare:273.26Vortioxetine hydrobromide
CAS:<p>Vortioxetine hydrobromide (Lu AA21004 hydrobromide) is a serotonin (5-HT) modulator and stimulator (SMS), inhibits 5-HT1A/1B/3A/7 receptor and SERT (IC50: 15/33</p>Formula:C18H22N2S·HBrPurezza:98.85% - 99.98%Colore e forma:SolidPeso molecolare:379.36Niaprazine
CAS:<p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>Formula:C20H25FN4OPurezza:99.56%Colore e forma:SolidPeso molecolare:356.44Olcegepant
CAS:<p>Olcegepant (BIBN-4096) is an effective and selective non-peptide calcitonin gene-related peptide 1 (CGRP1) receptor antagonist (IC50 of 0.03 nM and Ki of 14.4</p>Formula:C38H47Br2N9O5Purezza:96.08% - 97.24%Colore e forma:SolidPeso molecolare:869.65NPS ALX Compound 4a
CAS:<p>NPS ALX Compound 4a is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)</p>Formula:C25H25N3O2SPurezza:98%Colore e forma:SolidPeso molecolare:431.55Lodoxamide
CAS:<p>Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.</p>Formula:C11H6ClN3O6Purezza:99.13% - 99.81%Colore e forma:SolidPeso molecolare:311.63CRT0273750
CAS:<p>CRT0273750 regulates plasma LPA levels and is suitable for in vivo studies. CRT0273750 is an autotaxin (ATX) inhibitor with IC50 of 0.014 μM.</p>Formula:C25H22ClF3N4O2Purezza:99.91%Colore e forma:SolidPeso molecolare:502.92Ondansetron
CAS:<p>Ondansetron (GR 38032) is a serotonin 5-HT3 receptor antagonist used mainly as an antiemetic.</p>Formula:C18H19N3OPurezza:99.92%Colore e forma:White To Yellow CrystalsPeso molecolare:293.36Mequitazine
CAS:<p>Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.</p>Formula:C20H22N2SPurezza:99.98%Colore e forma:SolidPeso molecolare:322.47MCL0020
CAS:<p>MCL0020 is a potent and selective melanocortin MC4 receptor antagonist, reverses stress-induced anorexia but has no effect on food intake in free-feeding rats.</p>Formula:C34H39N7O4Purezza:99.18%Colore e forma:SolidPeso molecolare:609.72S1p receptor agonist 1
CAS:<p>S1p receptor agonist 1 (S1p-receptor-agonist-1) is an S1P receptor agonist.</p>Formula:C23H24FN3O3Purezza:99.07% - 99.9%Colore e forma:SolidPeso molecolare:409.45F-15599
CAS:<p>F-15599 is a highly selective G-protein biased 5-HT1A receptor agonist(Ki : 3.4 nM).</p>Formula:C19H21ClF2N4OPurezza:98.72%Colore e forma:SolidPeso molecolare:394.85N-Acetylhistamine acetate
<p>N-Acetylhistamine acetate is a histamine metabolite. It can be used as a potential biomarker of histidine metabolism for anaphylactoid reactions.</p>Formula:C9H15N3O3Purezza:98%Colore e forma:SolidPeso molecolare:213.23Pentagastrin
CAS:<p>Pentagastrin (ICI-50123) is a synthetic polypeptide that has effects like gastrin when given parenterally, which can cause the secretion and synthesis of</p>Formula:C37H49N7O9SPurezza:96.98% - 99.49%Colore e forma:Fine Colorless Needle-Shaped Crystals From 2-Ethoxyethanol + Water SolidPeso molecolare:767.89Ciproxifan maleate
CAS:<p>Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity</p>Formula:C20H22N2O6Purezza:99.39%Colore e forma:SolidPeso molecolare:386.4Brimonidine Tartrate
CAS:<p>Brimonidine Tartrate (AGN190342 tartrate) is a quinoxaline derivative and adrenergic α-2 receptor agonist (EC50: 0.45 nM).</p>Formula:C15H16BrN5O6Purezza:99.95%Colore e forma:Off-White Crystalline SolidPeso molecolare:442.22Loxapine hydrochloride
CAS:<p>Loxapine hydrochloride, an oral anti-psychotic, inhibits dopamine and blocks 5-HT receptors.</p>Formula:C18H19Cl2N3OColore e forma:SolidPeso molecolare:364.27Samelisant dihydrochloride
CAS:<p>SUVN-G3031: H3 receptor antagonist; may treat cognitive issues, ADHD, epilepsy, sleep, obesity, schizophrenia, eating disorders, pain.</p>Formula:C21H33Cl2N3O3Colore e forma:SolidPeso molecolare:446.41Betahistine EP Impurity C
CAS:<p>Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.</p>Formula:C15H19N3Purezza:≥95%Colore e forma:SolidPeso molecolare:241.33AM095
CAS:<p>AM095 is a potent LPA1 receptor antagonist with IC50 values of 0.98 and 0.73 μM for recombinant human or mouse LPA1 respectively.</p>Formula:C27H23N2NaO5Purezza:98.87%Colore e forma:SolidPeso molecolare:478.47Pizuglanstat
CAS:<p>Pizuglanstat is a hematopoietic prostaglandin synthase inhibitor.</p>Formula:C27H36N6O4Purezza:99.62%Colore e forma:SolidPeso molecolare:508.61Naratriptan
CAS:<p>Naratriptan is a selective agonist of 5-HT1 receptor and is is used for the treatment of migraine headaches.</p>Formula:C17H25N3O2SPurezza:99.08%Colore e forma:SolidPeso molecolare:335.47ELA-14(human) acetate
<p>ELA-14(human) acetate, a fragment of ELA, targets APJ, activates Gαi1 and β-arrestin-2, and prompts receptor internalization like its parent peptide.</p>Formula:C77H123N25O19S2Purezza:97.2%Colore e forma:SolidPeso molecolare:1767.09Amylin, amide, rat acetate(124447-81-0,free base)
<p>Amylin, amide, rat acetate is a potent and high affinity ligand of AMY1 and AMY3 receptors and variably of AMY2 receptors.</p>Formula:C169H276N52O55S2Purezza:98.93%Colore e forma:SolidPeso molecolare:3980.45Scyliorhinin II acetate
<p>Scyliorhinin II acetate is a selective agonist of the neurokinin-3 (NK3) receptor (Ki = 2.5 nM) in rat cerebral cortex.</p>Formula:C79H123N21O28S3Purezza:99.06%Colore e forma:SolidPeso molecolare:1911.14Triprolidine hydrochloride
CAS:<p>Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.</p>Formula:C19H23ClN2Colore e forma:SolidPeso molecolare:314.852RS 100329
CAS:<p>RS 100329 HCl is a selective α1A-adrenoceptor antagonist (pKi = 9.6 for human cloned α1A receptors).</p>Formula:C20H25F3N4O3Colore e forma:SolidPeso molecolare:426.43Phenylephrine
CAS:<p>Phenylephrine ((R)-(-)-Phenylephrine) is a selective α1-adrenoceptor agonist ( pKi: 5.86, 4.87 and 4.70 for α1D, α1B, and α1A receptors respectively).</p>Formula:C9H13NO2Purezza:99.5% - 99.89%Colore e forma:SolidPeso molecolare:167.21Tandospirone citrate
CAS:<p>Tandospirone citrate (SM-3997 citrate) is a potent and selective 5-HT1A receptor partial agonist (Ki : 27 nM)</p>Formula:C27H37N5O9Purezza:97.84% - 99.90%Colore e forma:SolidPeso molecolare:575.61MEN 10207 acetate
<p>MEN 10207 acetate is a selective antagonist for NK-2 tachykinin receptor.</p>Formula:C59H72N14O12Purezza:99.18%Colore e forma:SolidPeso molecolare:1169.29[Lys5,MeLeu9,Nle10]-NKA(4-10)
CAS:<p>Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).</p>Formula:C39H65N9O9Purezza:>99.99%Colore e forma:SolidPeso molecolare:803.99idalopirdine
CAS:<p>Idalopirdine (Lu AE58054), a selective 5-HT6 receptor antagonist( Ki : 0.83 nM),as a treatment for Alzheimer's disease.</p>Formula:C20H19F5N2OPurezza:99.73%Colore e forma:SolidPeso molecolare:398.37Piboserod
CAS:<p>Piboserod (SB-207266) (SB 207266) is a selective 5-HT(4) receptor antagonist.</p>Formula:C22H31N3O2Purezza:97.21% - 99.49%Colore e forma:SolidPeso molecolare:369.5FSLLRY-NH2 TFA(245329-02-6 free base)
<p>FSLLRY-NH2 TFA inhibits PAR2, reverses taxol-induced pain, and reduces itch in mice; blocks ERK and collagen in fibroblasts.</p>Formula:C41H61F3N10O10Purezza:99.32%Colore e forma:SolidPeso molecolare:910.99MK-571 sodium
CAS:<p>MK-571 sodium, a CysLT1 antagonist and MRP2 inhibitor, obstructs drug efflux and hampers enterocyte phase-2 conjugation of flavonoids.</p>Formula:C26H27ClN2O3S2·NaPurezza:97.86% - 99.58%Colore e forma:SolidPeso molecolare:537.07ICI 89406
CAS:<p>ICI 89406 (1-[2-[[3-(2-cyanophenoxy)-2-hydroxypropyl]amino]ethyl]-3-phenylurea) is a β-adrenergic antagonist.</p>Formula:C19H22N4O3Purezza:99.92%Colore e forma:SolidPeso molecolare:354.4Pirenperone
CAS:<p>Pirenperone is a putative 5-HT2 receptor antagonist with the central antiserotonergic and antidopaminergic action.</p>Formula:C23H24FN3O2Purezza:99.2%Colore e forma:SolidPeso molecolare:393.45Alizapride hydrochloride
CAS:<p>Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.</p>Formula:C16H21N5O2·HClPurezza:99.35% - 99.48%Colore e forma:CoaPeso molecolare:351.834i
CAS:<p>4i (CHEMBL1269981) is a 5-HT3 receptor antagonist,It modulates the serotonergic system.</p>Formula:C16H12ClN3OPurezza:99.49%Colore e forma:SolidPeso molecolare:297.74Guanabenz hydrochloride
CAS:<p>Guanabenz hydrochloride (NE56490) is an orally active α2-adrenoceptor agonist with hypotensive effects.</p>Formula:C8H9Cl3N4Purezza:99.45%Colore e forma:SolidPeso molecolare:267.54Decloxizine
CAS:<p>Decloxizine is a H1 receptor antagonist</p>Formula:C21H28N2O2Purezza:99.53%Colore e forma:White Or Similar To White PowderPeso molecolare:340.46CPI-444
CAS:<p>CPI-444 (V81444) is an antagonist of the adenosine A2A receptor.It reduces tumor area in mouse model of murine Her2/neu-expressing breast cancer.</p>Formula:C20H21N7O3Purezza:98.78%Colore e forma:SolidPeso molecolare:407.43GLP-1(7-36), amide
CAS:<p>GLP-1 secretion by human enteroendocrine NCI-H716 cells is augmented in a dose-dependent manner by the addition of CPE.Cost-effective and quality-assured.</p>Formula:C149H226N40O45Purezza:99.85%Colore e forma:White PowderPeso molecolare:3297.63
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