
Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(942 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.949 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(149 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(410 prodotti)
- Recettore dell'endotelina(75 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(32 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(166 prodotti)
- Proteina Hedgehog/Smoothened(45 prodotti)
- Recettore dell'istamina(359 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(298 prodotti)
- PAFR(11 prodotti)
- PKA(49 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
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Trovati 5378 prodotti di "Proteina G/GPCR"
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Ozanimod hydrochloride
CAS:Ozanimod (RPC-1063) HCl is a selective S1P1/S1P5 modulator with high affinity, used in relapsing MS research.Formula:C23H25ClN4O3Purezza:99.81%Colore e forma:SolidPeso molecolare:440.92Levocetirizine Dihydrochloride
CAS:<p>Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.</p>Formula:C21H27Cl3N2O3Purezza:99.89%Colore e forma:White Or Off-White Crystalline PowderPeso molecolare:461.81Nebentan potassium
CAS:<p>Nebentan potassium (YM598) is an ETA receptor antagonist that inhibits pulmonary arterial hypertension and is used in the study of neurologic diseases.</p>Formula:C24H20KN5O5SPurezza:99.05%Colore e forma:SolidPeso molecolare:529.61Atipamezole
CAS:Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.Formula:C14H16N2Purezza:99.88%Colore e forma:Off-White To Light Yellow Crystal PowderPeso molecolare:212.29GRK6-IN-2
CAS:<p>GRK6-IN-2 is a potent G protein-coupled receptor kinase 6 (GRK6) inhibitor with potential antitumor activity.GRK6-IN-2 has been studied in multiple myeloma.</p>Formula:C21H21FN6Purezza:98.94%Colore e forma:SolidPeso molecolare:376.43Renzapride
CAS:Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.Formula:C16H22ClN3O2Purezza:98.97% - 99.09%Colore e forma:SolidPeso molecolare:323.82BMS-986278
CAS:<p>BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb values of 6.9 nM and 4.0 nM for human and mouse LPA1,</p>Formula:C22H31N5O5Purezza:99.86%Colore e forma:SolidPeso molecolare:445.51Poly-D-lysine hydrobromide (MW 30000-70000)
CAS:Poly-D-lysine hydrobromide (MW 30000-70000) (Poly-D-lysine HBr) is a peptide CaSR agonist that removes proteinase K-resistant PrP from SN56 neuroblastoma cells.Formula:(C6H14N2O2)x·xHBrColore e forma:SolidPeso molecolare:227.102Setiptiline
CAS:Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.Formula:C19H19NPurezza:98.05% - 98.07%Colore e forma:SolidPeso molecolare:261.36AF-710B
CAS:<p>AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.</p>Formula:C20H27N3OSPurezza:98.62% - 99.89%Colore e forma:SolidPeso molecolare:357.51Trazpiroben
CAS:Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.Formula:C31H39N3O4Purezza:99.41% - >99.99%Colore e forma:SolidPeso molecolare:517.66Alfuzosin
CAS:<p>Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and urethral dysfunction.</p>Formula:C19H27N5O4Purezza:99.64%Colore e forma:White Crystaline PowderPeso molecolare:389.45(R)-Mirtazapine
CAS:<p>(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.</p>Formula:C17H19N3Purezza:99.75%Colore e forma:SolidPeso molecolare:265.35KB-5492 free base
CAS:<p>KB-5492 free base is an antiulcer agent that inhibits sigma receptors and can be used to study gastric lesions and gastric secretion.</p>Formula:C23H30N2O6Purezza:97.10% - 97.94%Colore e forma:SolidPeso molecolare:430.49Dexpramipexole
CAS:Dexpramipexole ((R)-Pramipexole) is a mitochondrial protective agent that maintains mitochondrial function and energy production.Formula:C10H17N3SPurezza:99.78%Colore e forma:SolidPeso molecolare:211.33Syk Inhibitor II
CAS:<p>Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).</p>Formula:C14H15F3N6OPurezza:97.63%Colore e forma:SolidPeso molecolare:340.3L-745870
CAS:<p>L-745870 is a D4 receptor antagonist that also inhibits D2 receptors, 5-HT2 receptors, and α-adrenergic receptors.</p>Formula:C18H19ClN4Purezza:98%Colore e forma:SolidPeso molecolare:326.82R 59-022
CAS:<p>R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.</p>Formula:C27H26FN3OSPurezza:98.55%Colore e forma:SolidPeso molecolare:459.58Ropinirole
CAS:<p>Ropinirole, D2-like agonist, no D1 affinity, Ki 29 nM for D2, treats Parkinson's.</p>Formula:C16H24N2OPurezza:99.68%Colore e forma:SolidPeso molecolare:260.38SR59230A hydrochloride
CAS:<p>SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue thermogenesis.</p>Formula:C21H28ClNO2Purezza:99.49%Colore e forma:SolidPeso molecolare:361.91PACAP (1-38), human, ovine, rat
CAS:PACAP (1-38), human, ovine, rat (Pituitary Adenylate Cyclase Activating Polypeptide 38) is a neuropeptide with 38 amino acid residues.Formula:C203H331N63O53SPurezza:96.93% - 98.16%Colore e forma:SolidPeso molecolare:4534.26Cyproheptadine hydrochloride
CAS:<p>Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.</p>Formula:C21H21N·HClPurezza:99.88% - 99.97%Colore e forma:SolidPeso molecolare:323.86Travoprost
CAS:<p>Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.</p>Formula:C26H35F3O6Purezza:97.39% - 99.58%Colore e forma:Colorless OilPeso molecolare:500.55Tulobuterol
CAS:<p>Tulobuterol is mainly used for the prevention and treatment of bronchial asthma, asthmatic bronchitis and chronic bronchitis. Research shows that it could inhibit rhinovirus infection in primary cultures of human tracheal epithelial cells.</p>Formula:C12H18ClNOColore e forma:Crystalline SolidPeso molecolare:227.73Eptinezumab
CAS:<p>Eptinezumab is a humanised monoclonal antibody targeting CGRP (calcitonin gene-related peptide), which prevents CGRP binding to its receptor, migraine.</p>Purezza:95% - 95%Colore e forma:LiquidEscitalopram
CAS:<p>Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.</p>Formula:C20H21FN2OPurezza:99.82%Colore e forma:White Or White Crystalline PowderPeso molecolare:324.39Methaphenilene hydrochloride
CAS:<p>Methaphenilene hydrochloride is an H1 receptor antagonist with antihistaminic and anticholinergic activity, in allergic inflammation and autonomic research.</p>Formula:C15H21ClN2SPurezza:99.84%Colore e forma:SolidPeso molecolare:296.86Arazasetron HCl
CAS:<p>Arazasetron is an antiemetic which acts as a 5-HT3 receptor antagonist, pKi = 9.27.</p>Formula:C17H20ClN3O3Purezza:98%Colore e forma:SolidPeso molecolare:349.81Carlumab
CAS:<p>Carlumab is a high-affinity human monoclonal antibody that targets CCL2, suppressing the recruitment of monocytes/macrophages in the tumour microenvironment.</p>Purezza:95%Colore e forma:LiquidFremanezumab
CAS:<p>Fremanezumab (TEV-48125) is a humanised monoclonal antibody targeting CGRP, capable of neutralising human, mouse and rat CGRP, migraine.</p>Purezza:95% - 95%Colore e forma:LiquidOlopatadine
CAS:<p>Olopatadine is an antihistamine and anti-allergy medication for itchy eyes, also possibly treats red skin syndrome.</p>Formula:C21H23NO3Purezza:98%Colore e forma:White Or Off-White Crystalline PowderPeso molecolare:337.4117-phenyl trinor Prostaglandin F2α isopropyl ester
CAS:<p>17-phenyl trinor PGF2α N-ethyl amide is an F-series prostaglandin analog which has been approved for use as an ocular hypotensive drug, sold under the Allergan</p>Formula:C26H38O5Colore e forma:SolidPeso molecolare:430.58Buflomedil
CAS:<p>Buflomedil is a vasoactive compound. Buflomedil has been used for peripheral arterial diseases.</p>Formula:C17H25NO4Purezza:98%Colore e forma:SolidPeso molecolare:307.38Meticillin
CAS:<p>Methicillin: Narrow-spectrum beta-lactam, penicillin-type antibiotic for certain gram-positive bacterial infections.</p>Formula:C17H20N2O6SColore e forma:SolidPeso molecolare:380.42N-Methyl amisulpride
CAS:<p>N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.</p>Formula:C18H29N3O4SColore e forma:SolidPeso molecolare:383.51Keto Ziprasidone
CAS:<p>Ziprasidone, an antipsychotic agent, functions as a dual antagonist of 5-HT (serotonin) and dopamine receptors.</p>Formula:C21H19ClN4O2SPurezza:98%Colore e forma:SolidPeso molecolare:426.92Metoxibutropate
CAS:<p>Metoxibutropate is a biochemical.</p>Formula:C20H24O3Colore e forma:SolidPeso molecolare:312.4PF-610355
CAS:<p>PF-610355 is a long-acting and potent β2-adrenergic receptor agonist (EC50: 0.26 nM).PF-610355 can be used to study asthma and COPD.</p>Formula:C34H39N3O6SPurezza:99.73%Colore e forma:SolidPeso molecolare:617.76Triflupromazine
CAS:<p>Triflupromazine is a dopamine receptor D1/D2 antagonist and LHDA inhibitor that suppresses dopamine activity in (CNS)mental disorders, sedation, and antiemesis.</p>Formula:C18H19F3N2SColore e forma:SolidPeso molecolare:352.42DL-Phenylephrine HCl
CAS:DL-Phenylephrine HCl is a selective agonist of the alpha1-adrenergic receptor.Formula:C9H14ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:203.67GPR183-IN-1
CAS:<p>GPR183-IN-1 (compound 15) is an effective orally active inhibitor of GPR183. It inhibits Ca2+ mobilization with an IC50 value of 39.97 nM. GPR183-IN-1 holds potential for research in cancer, autoimmune diseases, pain, and osteoporosis.</p>Formula:C16H19BrN2O2Colore e forma:SolidPeso molecolare:351.24Blontuvetmab
CAS:<p>Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].</p>Colore e forma:LiquidP2Y14R antagonist 1
CAS:<p>P2Y14R antagonist 1 (compound I-17) is a selective oral that inhibits inflammatory response in acute gouty arthritis the NLRP3/GSDMD y and cellular pyroptosis.</p>Formula:C15H12BrN3O2Purezza:98.88%Colore e forma:SolidPeso molecolare:346.18Risperidone Mesylate
CAS:<p>Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.</p>Formula:C24H31FN4O5SPurezza:98%Colore e forma:SolidPeso molecolare:506.59Mibavademab
CAS:<p>Mibavademab is a humanized anti-leptin receptor (LEPR) mAb under investigation for treating congenital leptin deficiency.</p>Purezza:95%Colore e forma:LiquidUliledlimab
CAS:<p>Uliledlimab, a humanized monoclonal antibody against CD73, reduces extracellular adenosine production and modulates immunosuppressive pathways.</p>Purezza:95% - 95%Colore e forma:LiquidDapagliflozin-d5
CAS:Dapagliflozin D5 (BMS-512148 D5) is deuterated Dapagliflozin. Dapagliflozin is a competitive SGLT2 inhibitor.Formula:C21H25ClO6Purezza:98%Colore e forma:SolidPeso molecolare:413.9Cinnarizine D8
CAS:<p>Cinnarizine D8 is a deuterium-labeled Cinnarizine which is an antihistamine and a calcium channel blocker.</p>Formula:C26H28N2Purezza:98%Colore e forma:SolidPeso molecolare:376.57315-keto Prostaglandin F2α
CAS:<p>15-keto Prostaglandin F2α is a metabolite of Prostaglandin F2α that lowers intraocular pressure in rabbits.</p>Formula:C20H32O5Purezza:98%Colore e forma:SolidPeso molecolare:352.47Amitriptyline-d6 Hydrochloride
CAS:<p>Amitriptyline-d6 Hydrochloride is a deuterated compound of Amitriptyline Hydrochloride. Amitriptyline Hydrochloride has a CAS number of 549-18-8. Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.</p>Formula:C20H18D6ClNColore e forma:SolidPeso molecolare:319.90Mirtazapine D3
CAS:Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .Formula:C17H19N3Purezza:98%Colore e forma:SolidPeso molecolare:268.37Brexpiprazole-d8
CAS:<p>Brexpiprazole D8 is a deuterium-modified partial agonist of 5-HT1A and dopamine receptors, with Ki values of 0.12 nM and 0.3 nM respectively.</p>Formula:C25H27N3O2SPurezza:98%Colore e forma:SolidPeso molecolare:441.62R-138727
CAS:<p>R-138727 is a novel P2Y12 receptor inhibitor.</p>Formula:C18H20FNO3SPurezza:98%Colore e forma:SolidPeso molecolare:349.42MK-447
CAS:<p>MK-447 is a nonsteroidal antiinflammatory agent.</p>Formula:C11H16INOPurezza:98%Colore e forma:SolidPeso molecolare:305.16Ketanserinol
CAS:<p>Ketanserinol is a metabolite of the antihypertensive drug ketanserin, which blocks 5-HT2 receptors to treat protamine-induced pulmonary hypertension.</p>Formula:C22H24FN3O3Colore e forma:SolidPeso molecolare:397.44Penbutolol sulfate
CAS:<p>Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.</p>Formula:C18H29NO2H2O4SPurezza:98.55%Colore e forma:SolidPeso molecolare:340.47Vanoxerine
CAS:<p>Vanoxerine is an antagonist of dopamine transporter (Ki: 16.9nM).</p>Formula:C28H32F2N2OPurezza:98%Colore e forma:SolidPeso molecolare:450.56Amidephrine hydrochloride
CAS:<p>Amidephrine hydrochloride is a biochemical.</p>Formula:C10H17ClN2O3SColore e forma:SolidPeso molecolare:280.77Dehydroabiethylamine
CAS:<p>Dehydroabiethylamine (NSC-2955) boosts liver CYP2B, blocks PDKs & cholesterol transport, and has anti-tumor effects.</p>Formula:C20H31NPurezza:98.79%Colore e forma:Pale Yellow Viscous Liquid /Technical Grade/ Viscous Colorless To Amber LiquidPeso molecolare:285.47Isoproterenol sulfate anhydrous
CAS:<p>Isoproterenol sulfate anhydrous is a useful alkaloid. It is used for biological research.</p>Formula:C22H36N2O10SPurezza:98%Colore e forma:CoaPeso molecolare:520.59Tivumecirnon
CAS:<p>Tivumecirnon (FLX475) is a selective and oral CCR4 antagonist inhibits the infiltration and migration of Treg into the tumour microenvironment, antitumour</p>Formula:C24H27Cl2F3N6OPurezza:99.88%Colore e forma:SolidPeso molecolare:543.41Amidephrine
CAS:<p>Amidephrine is an adrenergic agent.</p>Formula:C10H16N2O3SColore e forma:SolidPeso molecolare:244.31Amthamine
CAS:<p>Compound AMTHAMINE DIHYDROBROMIDE is a useful organic compound for research related to life sciences.</p>Formula:C6H11N3SColore e forma:SoildPeso molecolare:157.24S 25585
CAS:<p>S 25585 is a neuropeptide Y (NPY) Y5 receptor antagonist.</p>Formula:C22H23F3N4O6SPurezza:98%Colore e forma:SolidPeso molecolare:528.5Diclofensine
CAS:<p>Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.</p>Formula:C17H17Cl2NOPurezza:97.01% - 98.13%Colore e forma:SolidPeso molecolare:322.23Ciproxifan
CAS:<p>Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).</p>Formula:C16H18N2O2Purezza:98.00%Colore e forma:SolidPeso molecolare:270.33Litorin
CAS:<p>Litorin suppresses appetite and stimulates smooth muscle, gastrin, gastric acid, and pancreatic secretion.</p>Formula:C51H68N14O11SColore e forma:White PowderPeso molecolare:1085.247-Desmethyl-3-hydroxyagomelatine
CAS:<p>7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.</p>Formula:C14H15NO3Purezza:98%Colore e forma:SolidPeso molecolare:245.275-Methyltryptamine hydrochloride
CAS:<p>5-Methyltryptamine hydrochloride is a high-affinity 5-HT1C receptor ligand and a partial agonist of 5-HT. 5-Methyltryptamine hydrochloride protects mice subjected to burn, tourniquet and endotoxin shock.</p>Formula:C11H15ClN2Purezza:99.45%Colore e forma:SolidPeso molecolare:210.703Roxatidine acetate
CAS:<p>Roxatidine acetate: anti-ulcer, blocks histamine, reduces acid. Safer at lower doses.</p>Formula:C19H28N2O4Purezza:98%Colore e forma:White Or Off-White PowderPeso molecolare:348.447-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene
CAS:<p>7-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene is a liver receptor homolog-1 (LRH-1) antagonist (IC50: 3.1 μM).</p>Formula:C42H44N2O6SPurezza:98%Colore e forma:SolidPeso molecolare:704.87Pardoprunox
CAS:<p>Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.</p>Formula:C12H15N3O2Purezza:98%Colore e forma:SolidPeso molecolare:233.27Itopride free base
CAS:<p>Itopride HCl combats dyspepsia and GERD, inhibiting AChE and blocking D2 receptors.</p>Formula:C20H26N2O4Colore e forma:WhitePeso molecolare:358.43(RS)-ICI-118551 Hydrochloride
CAS:ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3Formula:C17H27NO2·HClPurezza:98.02%Colore e forma:SolidPeso molecolare:313.86Atenolol Hydrochloride
CAS:<p>Atenolol Hydrochloride is a selective antagonist of ß1 receptor.</p>Formula:C14H23ClN2O3Purezza:98%Colore e forma:SolidPeso molecolare:302.80Hydroxy ziprasidone
CAS:<p>Hydroxy ziprasidone is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a 5-HT and dopamine receptor antagonist.</p>Formula:C21H21ClN4O2SPurezza:98%Colore e forma:SolidPeso molecolare:428.94Caerulein, desulfated
CAS:Caerulein, desulfated (FI-6934, desulfated) is a desulfated compound formed after caerulein hydrolysis, a neuropeptide with lower smooth muscle activity.Formula:C58H73N13O18SPurezza:99.46%Colore e forma:SolidPeso molecolare:1272.34SB 271046 hydrochloride
CAS:<p>SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is > 200-fold selective over 55 other receptors, enzymes and ion channels.</p>Formula:C20H22ClN3O3S2·HClPurezza:99.77%Colore e forma:SolidPeso molecolare:488.45Ridazolol HCl
CAS:<p>Ridazolol HCl (CAS 413) is a novel β-adrenoceptor (β-AR) blocker with α-adrenerolytic activity.</p>Formula:C15H19Cl3N4O3Purezza:99.48%Colore e forma:SoildPeso molecolare:409.7Ticlopidine
CAS:<p>Ticlopidine (PCR 5332) is an antiplatelet drug in the thienopyridine family which is an adenosine diphosphate (ADP) receptor inhibitor.</p>Formula:C14H14ClNSPurezza:99.67%Colore e forma:SolidPeso molecolare:263.79Norreticuline
CAS:<p>Norreticuline is a potential adrenoceptor-α/β agonist and CYP2D6 and D2 receptor inhibitor for the study of neurodegenerative diseases.</p>Formula:C18H21NO4Colore e forma:SolidPeso molecolare:315.36Dolasetron Mesylate
CAS:<p>Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea following</p>Formula:C20H24N2O6SPurezza:99.05%Colore e forma:White PowderPeso molecolare:420.48LY 344864
CAS:<p>LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.</p>Formula:C21H22FN3OPurezza:98%Colore e forma:SolidPeso molecolare:351.42Guacetisal
CAS:<p>Guacetisal, from acetylsalicylic acid and guaiacol, may treat chronic bronchitis.</p>Formula:C16H14O5Purezza:99.18%Colore e forma:SolidPeso molecolare:286.28Lodoxamide tromethamine
CAS:<p>Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergic</p>Formula:C19H28ClN5O12Purezza:98.8%Colore e forma:SolidPeso molecolare:553.91Paroxetine hydrochloride hemihydrate
CAS:<p>Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).</p>Formula:C38H44Cl2F2N2O7Purezza:99.949%Colore e forma:SolidPeso molecolare:749.67MK-5046
CAS:MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).Formula:C20H18F6N4OPurezza:98.56%Colore e forma:SolidPeso molecolare:444.37A 63162
CAS:<p>A 63162 is an inhibitor of 5-lipoxygenase.</p>Formula:C17H19NO3Purezza:98%Colore e forma:SolidPeso molecolare:285.34HSK0935
CAS:<p>HSK0935 is a highly selective and orally available SGLT2 inhibitor (IC50: 1.3 nM). It has antihyperglycemic activities.</p>Formula:C22H25ClO7Purezza:98%Colore e forma:SolidPeso molecolare:436.88Ipsapirone
CAS:<p>Ipsapirone is a partial agonist of 5-HT1A receptor and produces an inhibitory effect on 5-HT2 and the α1-adrenergic function at high doses.</p>Formula:C19H23N5O3SPurezza:99.51%Colore e forma:SolidPeso molecolare:401.48N,N-Dimethylsphingosine
CAS:<p>N,N-Dimethylsphingosine,is a potent competitive SphK phosphorylation inhibitor.DMS is elevated in models of neuropathic pain by increasing IL-1β and MCP-1.</p>Formula:C20H41NO2Purezza:98%Colore e forma:Clear Colorless To Faint Yellow Liquid/White To Off-White PowderPeso molecolare:327.55L 640033
CAS:<p>L 640033 is a beta-agonist.</p>Formula:C18H25N3OPurezza:98%Colore e forma:SolidPeso molecolare:299.41RUSKI-201 dihydrochloride
CAS:<p>RUSKI-201 dihydrochloride: potent Hhat inhibitor (IC50: 0.20 μM), blocks Hh signaling, and inhibits Hh palmitoylation.</p>Formula:C20H29Cl2N3OSColore e forma:SolidPeso molecolare:430.43Sigma-LIGAND-1
CAS:<p>Sigma-LIGAND-1 is a selective Sigma Receptor ligand with an IC50s of 16 nM, 19 nM at the DTG site and the PPP site, respectively.</p>Formula:C27H33NO4Purezza:99.89%Colore e forma:SolidPeso molecolare:435.56Isamoltane hemifumarate
CAS:<p>5-HT1B antagonist</p>Formula:C16H22N202C4H404Purezza:98%Colore e forma:SolidPeso molecolare:332.45-HT3 antagonist 3
CAS:<p>5-HT3 antagonist 3 (Compound 15b) is a high-affinity 5-HT3 receptor antagonist. It binds to 5-HT3 receptors in rat brain cortical membranes (Ki: 0.25 nM).</p>Formula:C20H21N3OPurezza:99.9%Colore e forma:SolidPeso molecolare:319.42-Methylthioadenosine diphosphate trisodium
CAS:<p>2-Methylthioadenosine diphosphate trisodium(2-MeS-ADP) is a purinergic P2Y receptor agonist that agonizes P2Y13 and P2Y12, induces platelet aggregation.</p>Formula:C11H14N5Na3O10P2SColore e forma:SolidPeso molecolare:539.24SCH-23390 maleate
CAS:<p>SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,</p>Formula:C21H22ClNO5Purezza:98%Colore e forma:SolidPeso molecolare:403.865-HT3 antagonist 2
CAS:<p>5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.</p>Formula:C18H21N3OPurezza:98%Colore e forma:SolidPeso molecolare:295.38Afurolol Hydrochloride
CAS:<p>Afurolol Hydrochloride (DL 071-IT) is a non-selective β-adrenergic receptor antagonist. DL 071 IT exhibits intrinsic sympathomimetic activity.</p>Formula:C15H22ClNO4Purezza:98.86%Colore e forma:SolidPeso molecolare:315.79

