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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

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Trovati 5378 prodotti di "Proteina G/GPCR"

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  • Ozanimod hydrochloride

    CAS:
    Ozanimod (RPC-1063) HCl is a selective S1P1/S1P5 modulator with high affinity, used in relapsing MS research.
    Formula:C23H25ClN4O3
    Purezza:99.81%
    Colore e forma:Solid
    Peso molecolare:440.92
  • Levocetirizine Dihydrochloride

    CAS:
    <p>Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.</p>
    Formula:C21H27Cl3N2O3
    Purezza:99.89%
    Colore e forma:White Or Off-White Crystalline Powder
    Peso molecolare:461.81
  • Nebentan potassium

    CAS:
    <p>Nebentan potassium (YM598) is an ETA receptor antagonist that inhibits pulmonary arterial hypertension and is used in the study of neurologic diseases.</p>
    Formula:C24H20KN5O5S
    Purezza:99.05%
    Colore e forma:Solid
    Peso molecolare:529.61
  • Atipamezole

    CAS:
    Atipamezole (Antisedan) is a synthetic α2 adrenergic receptor antagonist. It has also been researched in humans as a potential anti-Parkinsonian drug.
    Formula:C14H16N2
    Purezza:99.88%
    Colore e forma:Off-White To Light Yellow Crystal Powder
    Peso molecolare:212.29
  • GRK6-IN-2

    CAS:
    <p>GRK6-IN-2 is a potent G protein-coupled receptor kinase 6 (GRK6) inhibitor with potential antitumor activity.GRK6-IN-2 has been studied in multiple myeloma.</p>
    Formula:C21H21FN6
    Purezza:98.94%
    Colore e forma:Solid
    Peso molecolare:376.43
  • Renzapride

    CAS:
    Renzapride (BRL 24924) is a mixed 5-hydroxytryptamine type 4 (5-HT4) agonist and 5-HT3 receptor antagonist used in the study of irritable bowel syndrome.
    Formula:C16H22ClN3O2
    Purezza:98.97% - 99.09%
    Colore e forma:Solid
    Peso molecolare:323.82
  • BMS-986278

    CAS:
    <p>BMS-986278 is an orally active and potent hemophosphatidic acid receptor 1 (LPA1) antagonist with Kb values of 6.9 nM and 4.0 nM for human and mouse LPA1,</p>
    Formula:C22H31N5O5
    Purezza:99.86%
    Colore e forma:Solid
    Peso molecolare:445.51
  • Poly-D-lysine hydrobromide (MW 30000-70000)

    CAS:
    Poly-D-lysine hydrobromide (MW 30000-70000) (Poly-D-lysine HBr) is a peptide CaSR agonist that removes proteinase K-resistant PrP from SN56 neuroblastoma cells.
    Formula:(C6H14N2O2)x·xHBr
    Colore e forma:Solid
    Peso molecolare:227.102
  • Setiptiline

    CAS:
    Setiptiline (Org-8282) is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist with antidepressant activity.
    Formula:C19H19N
    Purezza:98.05% - 98.07%
    Colore e forma:Solid
    Peso molecolare:261.36
  • AF-710B

    CAS:
    <p>AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.</p>
    Formula:C20H27N3OS
    Purezza:98.62% - 99.89%
    Colore e forma:Solid
    Peso molecolare:357.51
  • Trazpiroben

    CAS:
    Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.
    Formula:C31H39N3O4
    Purezza:99.41% - >99.99%
    Colore e forma:Solid
    Peso molecolare:517.66
  • Alfuzosin

    CAS:
    <p>Alfuzosin (SL 77499) is an alpha-1 adrenergic antagonist used to treat benign prostatic hypertrophy and urethral dysfunction.</p>
    Formula:C19H27N5O4
    Purezza:99.64%
    Colore e forma:White Crystaline Powder
    Peso molecolare:389.45
  • (R)-Mirtazapine

    CAS:
    <p>(R)-Mirtazapine ((R)-Org3770) is a 5-HT3 receptor antagonist, a potential analgesic with anti-injury perception properties.</p>
    Formula:C17H19N3
    Purezza:99.75%
    Colore e forma:Solid
    Peso molecolare:265.35
  • KB-5492 free base

    CAS:
    <p>KB-5492 free base is an antiulcer agent that inhibits sigma receptors and can be used to study gastric lesions and gastric secretion.</p>
    Formula:C23H30N2O6
    Purezza:97.10% - 97.94%
    Colore e forma:Solid
    Peso molecolare:430.49
  • Dexpramipexole

    CAS:
    Dexpramipexole ((R)-Pramipexole) is a mitochondrial protective agent that maintains mitochondrial function and energy production.
    Formula:C10H17N3S
    Purezza:99.78%
    Colore e forma:Solid
    Peso molecolare:211.33
  • Syk Inhibitor II

    CAS:
    <p>Syk inhibitor II, a cell-permeable, ATP-competitive, pyrimidine-carboxamide compound, selectively and reversibly inhibits Syk (IC50 = 41 nM).</p>
    Formula:C14H15F3N6O
    Purezza:97.63%
    Colore e forma:Solid
    Peso molecolare:340.3
  • L-745870

    CAS:
    <p>L-745870 is a D4 receptor antagonist that also inhibits D2 receptors, 5-HT2 receptors, and α-adrenergic receptors.</p>
    Formula:C18H19ClN4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:326.82
  • R 59-022

    CAS:
    <p>R 59-022 (DKGI-I) is a DGK inhibitor and a 5-HT Receptor antagonist that blocks filovirus internalization in host cells.</p>
    Formula:C27H26FN3OS
    Purezza:98.55%
    Colore e forma:Solid
    Peso molecolare:459.58
  • Ropinirole

    CAS:
    <p>Ropinirole, D2-like agonist, no D1 affinity, Ki 29 nM for D2, treats Parkinson's.</p>
    Formula:C16H24N2O
    Purezza:99.68%
    Colore e forma:Solid
    Peso molecolare:260.38
  • SR59230A hydrochloride

    CAS:
    <p>SR59230A hydrochloride (SR59230A HCl) is a beta3-adrenergic receptor antagonist that inhibits ultradian brown adipose tissue thermogenesis.</p>
    Formula:C21H28ClNO2
    Purezza:99.49%
    Colore e forma:Solid
    Peso molecolare:361.91
  • PACAP (1-38), human, ovine, rat

    CAS:
    PACAP (1-38), human, ovine, rat (Pituitary Adenylate Cyclase Activating Polypeptide 38) is a neuropeptide with 38 amino acid residues.
    Formula:C203H331N63O53S
    Purezza:96.93% - 98.16%
    Colore e forma:Solid
    Peso molecolare:4534.26
  • Cyproheptadine hydrochloride

    CAS:
    <p>Cyproheptadine hydrochloride (Periactin hydrochloride) is a hydrochloride salt form of cyproheptadine which is a histamine receptor antagonist.</p>
    Formula:C21H21N·HCl
    Purezza:99.88% - 99.97%
    Colore e forma:Solid
    Peso molecolare:323.86
  • Travoprost

    CAS:
    <p>Travoprost (Fluprostenol isopropyl ester) is used to treat glaucoma and ocular hypertension,is a potent and selective FP prostaglandin receptor agonist.</p>
    Formula:C26H35F3O6
    Purezza:97.39% - 99.58%
    Colore e forma:Colorless Oil
    Peso molecolare:500.55
  • Tulobuterol

    CAS:
    <p>Tulobuterol is mainly used for the prevention and treatment of bronchial asthma, asthmatic bronchitis and chronic bronchitis. Research shows that it could inhibit rhinovirus infection in primary cultures of human tracheal epithelial cells.</p>
    Formula:C12H18ClNO
    Colore e forma:Crystalline Solid
    Peso molecolare:227.73
  • Eptinezumab

    CAS:
    <p>Eptinezumab is a humanised monoclonal antibody targeting CGRP (calcitonin gene-related peptide), which prevents CGRP binding to its receptor, migraine.</p>
    Purezza:95% - 95%
    Colore e forma:Liquid
  • Escitalopram

    CAS:
    <p>Escitalopram (Seroplex), a serotonin inhibitor for depression, curbs alcohol intake and is favored over tricyclics for tardive dyskinesia.</p>
    Formula:C20H21FN2O
    Purezza:99.82%
    Colore e forma:White Or White Crystalline Powder
    Peso molecolare:324.39
  • Methaphenilene hydrochloride

    CAS:
    <p>Methaphenilene hydrochloride is an H1 receptor antagonist with antihistaminic and anticholinergic activity, in allergic inflammation and autonomic research.</p>
    Formula:C15H21ClN2S
    Purezza:99.84%
    Colore e forma:Solid
    Peso molecolare:296.86
  • Arazasetron HCl

    CAS:
    <p>Arazasetron is an antiemetic which acts as a 5-HT3 receptor antagonist, pKi = 9.27.</p>
    Formula:C17H20ClN3O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:349.81
  • Carlumab

    CAS:
    <p>Carlumab is a high-affinity human monoclonal antibody that targets CCL2, suppressing the recruitment of monocytes/macrophages in the tumour microenvironment.</p>
    Purezza:95%
    Colore e forma:Liquid
  • Fremanezumab

    CAS:
    <p>Fremanezumab (TEV-48125) is a humanised monoclonal antibody targeting CGRP, capable of neutralising human, mouse and rat CGRP, migraine.</p>
    Purezza:95% - 95%
    Colore e forma:Liquid
  • Olopatadine

    CAS:
    <p>Olopatadine is an antihistamine and anti-allergy medication for itchy eyes, also possibly treats red skin syndrome.</p>
    Formula:C21H23NO3
    Purezza:98%
    Colore e forma:White Or Off-White Crystalline Powder
    Peso molecolare:337.41
  • 17-phenyl trinor Prostaglandin F2α isopropyl ester

    CAS:
    <p>17-phenyl trinor PGF2α N-ethyl amide is an F-series prostaglandin analog which has been approved for use as an ocular hypotensive drug, sold under the Allergan</p>
    Formula:C26H38O5
    Colore e forma:Solid
    Peso molecolare:430.58
  • Buflomedil

    CAS:
    <p>Buflomedil is a vasoactive compound. Buflomedil has been used for peripheral arterial diseases.</p>
    Formula:C17H25NO4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:307.38
  • Meticillin

    CAS:
    <p>Methicillin: Narrow-spectrum beta-lactam, penicillin-type antibiotic for certain gram-positive bacterial infections.</p>
    Formula:C17H20N2O6S
    Colore e forma:Solid
    Peso molecolare:380.42
  • N-Methyl amisulpride

    CAS:
    <p>N-Methyl amisulpride (Amisulpride impurity H) is a 5-HT7 receptor, D2 receptor, and D3 receptor antagonist used in the study of acute schizophrenia.</p>
    Formula:C18H29N3O4S
    Colore e forma:Solid
    Peso molecolare:383.51
  • Keto Ziprasidone

    CAS:
    <p>Ziprasidone, an antipsychotic agent, functions as a dual antagonist of 5-HT (serotonin) and dopamine receptors.</p>
    Formula:C21H19ClN4O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:426.92
  • Metoxibutropate

    CAS:
    <p>Metoxibutropate is a biochemical.</p>
    Formula:C20H24O3
    Colore e forma:Solid
    Peso molecolare:312.4
  • PF-610355

    CAS:
    <p>PF-610355 is a long-acting and potent β2-adrenergic receptor agonist (EC50: 0.26 nM).PF-610355 can be used to study asthma and COPD.</p>
    Formula:C34H39N3O6S
    Purezza:99.73%
    Colore e forma:Solid
    Peso molecolare:617.76
  • Triflupromazine

    CAS:
    <p>Triflupromazine is a dopamine receptor D1/D2 antagonist and LHDA inhibitor that suppresses dopamine activity in (CNS)mental disorders, sedation, and antiemesis.</p>
    Formula:C18H19F3N2S
    Colore e forma:Solid
    Peso molecolare:352.42
  • DL-Phenylephrine HCl

    CAS:
    DL-Phenylephrine HCl is a selective agonist of the alpha1-adrenergic receptor.
    Formula:C9H14ClNO2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:203.67
  • GPR183-IN-1

    CAS:
    <p>GPR183-IN-1 (compound 15) is an effective orally active inhibitor of GPR183. It inhibits Ca2+ mobilization with an IC50 value of 39.97 nM. GPR183-IN-1 holds potential for research in cancer, autoimmune diseases, pain, and osteoporosis.</p>
    Formula:C16H19BrN2O2
    Colore e forma:Solid
    Peso molecolare:351.24
  • Blontuvetmab

    CAS:
    <p>Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].</p>
    Colore e forma:Liquid
  • P2Y14R antagonist 1

    CAS:
    <p>P2Y14R antagonist 1 (compound I-17) is a selective oral that inhibits inflammatory response in acute gouty arthritis the NLRP3/GSDMD y and cellular pyroptosis.</p>
    Formula:C15H12BrN3O2
    Purezza:98.88%
    Colore e forma:Solid
    Peso molecolare:346.18
  • Risperidone Mesylate

    CAS:
    <p>Risperidone Mesylate is a selective serotonin 5-HT2 receptor and dopamine D2 receptor blocker.</p>
    Formula:C24H31FN4O5S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:506.59
  • Mibavademab

    CAS:
    <p>Mibavademab is a humanized anti-leptin receptor (LEPR) mAb under investigation for treating congenital leptin deficiency.</p>
    Purezza:95%
    Colore e forma:Liquid
  • Uliledlimab

    CAS:
    <p>Uliledlimab, a humanized monoclonal antibody against CD73, reduces extracellular adenosine production and modulates immunosuppressive pathways.</p>
    Purezza:95% - 95%
    Colore e forma:Liquid
  • Dapagliflozin-d5

    CAS:
    Dapagliflozin D5 (BMS-512148 D5) is deuterated Dapagliflozin. Dapagliflozin is a competitive SGLT2 inhibitor.
    Formula:C21H25ClO6
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:413.9
  • Cinnarizine D8

    CAS:
    <p>Cinnarizine D8 is a deuterium-labeled Cinnarizine which is an antihistamine and a calcium channel blocker.</p>
    Formula:C26H28N2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:376.573
  • 15-keto Prostaglandin F2α

    CAS:
    <p>15-keto Prostaglandin F2α is a metabolite of Prostaglandin F2α that lowers intraocular pressure in rabbits.</p>
    Formula:C20H32O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:352.47
  • Amitriptyline-d6 Hydrochloride

    CAS:
    <p>Amitriptyline-d6 Hydrochloride is a deuterated compound of Amitriptyline Hydrochloride. Amitriptyline Hydrochloride has a CAS number of 549-18-8. Amitriptyline Hydrochloride is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and antinociceptive activities.</p>
    Formula:C20H18D6ClN
    Colore e forma:Solid
    Peso molecolare:319.90
  • Mirtazapine D3

    CAS:
    Mirtazapine D3 is a deuterium labeled Mirtazapine. Mirtazapine is an inhibitor of 5-HT receptor .
    Formula:C17H19N3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:268.37
  • Brexpiprazole-d8

    CAS:
    <p>Brexpiprazole D8 is a deuterium-modified partial agonist of 5-HT1A and dopamine receptors, with Ki values of 0.12 nM and 0.3 nM respectively.</p>
    Formula:C25H27N3O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:441.62
  • R-138727

    CAS:
    <p>R-138727 is a novel P2Y12 receptor inhibitor.</p>
    Formula:C18H20FNO3S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:349.42
  • MK-447

    CAS:
    <p>MK-447 is a nonsteroidal antiinflammatory agent.</p>
    Formula:C11H16INO
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:305.16
  • Ketanserinol

    CAS:
    <p>Ketanserinol is a metabolite of the antihypertensive drug ketanserin, which blocks 5-HT2 receptors to treat protamine-induced pulmonary hypertension.</p>
    Formula:C22H24FN3O3
    Colore e forma:Solid
    Peso molecolare:397.44
  • Penbutolol sulfate

    CAS:
    <p>Penbutolol sulfate ((-)-Terbuclomine) is able to bind to both β2-adrenergic receptor and β1-adrenergic receptor, thus making it a non-selective β blocker.</p>
    Formula:C18H29NO2H2O4S
    Purezza:98.55%
    Colore e forma:Solid
    Peso molecolare:340.47
  • Vanoxerine

    CAS:
    <p>Vanoxerine is an antagonist of dopamine transporter (Ki: 16.9nM).</p>
    Formula:C28H32F2N2O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:450.56
  • Amidephrine hydrochloride

    CAS:
    <p>Amidephrine hydrochloride is a biochemical.</p>
    Formula:C10H17ClN2O3S
    Colore e forma:Solid
    Peso molecolare:280.77
  • Dehydroabiethylamine

    CAS:
    <p>Dehydroabiethylamine (NSC-2955) boosts liver CYP2B, blocks PDKs &amp; cholesterol transport, and has anti-tumor effects.</p>
    Formula:C20H31N
    Purezza:98.79%
    Colore e forma:Pale Yellow Viscous Liquid /Technical Grade/ Viscous Colorless To Amber Liquid
    Peso molecolare:285.47
  • Isoproterenol sulfate anhydrous

    CAS:
    <p>Isoproterenol sulfate anhydrous is a useful alkaloid. It is used for biological research.</p>
    Formula:C22H36N2O10S
    Purezza:98%
    Colore e forma:Coa
    Peso molecolare:520.59
  • Tivumecirnon

    CAS:
    <p>Tivumecirnon (FLX475) is a selective and oral CCR4 antagonist inhibits the infiltration and migration of Treg into the tumour microenvironment, antitumour</p>
    Formula:C24H27Cl2F3N6O
    Purezza:99.88%
    Colore e forma:Solid
    Peso molecolare:543.41
  • Amidephrine

    CAS:
    <p>Amidephrine is an adrenergic agent.</p>
    Formula:C10H16N2O3S
    Colore e forma:Solid
    Peso molecolare:244.31
  • Amthamine

    CAS:
    <p>Compound AMTHAMINE DIHYDROBROMIDE is a useful organic compound for research related to life sciences.</p>
    Formula:C6H11N3S
    Colore e forma:Soild
    Peso molecolare:157.24
  • S 25585

    CAS:
    <p>S 25585 is a neuropeptide Y (NPY) Y5 receptor antagonist.</p>
    Formula:C22H23F3N4O6S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:528.5
  • Diclofensine

    CAS:
    <p>Diclofensine (Ro 8-4650) inhibits the uptake of serotonin, noradrenaline and dopamine.</p>
    Formula:C17H17Cl2NO
    Purezza:97.01% - 98.13%
    Colore e forma:Solid
    Peso molecolare:322.23
  • Ciproxifan

    CAS:
    <p>Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).</p>
    Formula:C16H18N2O2
    Purezza:98.00%
    Colore e forma:Solid
    Peso molecolare:270.33
  • Litorin

    CAS:
    <p>Litorin suppresses appetite and stimulates smooth muscle, gastrin, gastric acid, and pancreatic secretion.</p>
    Formula:C51H68N14O11S
    Colore e forma:White Powder
    Peso molecolare:1085.24
  • 7-Desmethyl-3-hydroxyagomelatine

    CAS:
    <p>7-Desmethyl-3-hydroxyagomelatine, less active than parent drug Agomelatine, is a melatonergic agonist and 5-HT2C antagonist.</p>
    Formula:C14H15NO3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:245.27
  • 5-Methyltryptamine hydrochloride

    CAS:
    <p>5-Methyltryptamine hydrochloride is a high-affinity 5-HT1C receptor ligand and a partial agonist of 5-HT. 5-Methyltryptamine hydrochloride protects mice subjected to burn, tourniquet and endotoxin shock.</p>
    Formula:C11H15ClN2
    Purezza:99.45%
    Colore e forma:Solid
    Peso molecolare:210.703
  • Roxatidine acetate

    CAS:
    <p>Roxatidine acetate: anti-ulcer, blocks histamine, reduces acid. Safer at lower doses.</p>
    Formula:C19H28N2O4
    Purezza:98%
    Colore e forma:White Or Off-White Powder
    Peso molecolare:348.44
  • 7-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene

    CAS:
    <p>7-[4-(2-Piperidinyl)ethoxy]benzoyl Raloxifene is a liver receptor homolog-1 (LRH-1) antagonist (IC50: 3.1 μM).</p>
    Formula:C42H44N2O6S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:704.87
  • Pardoprunox

    CAS:
    <p>Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.</p>
    Formula:C12H15N3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:233.27
  • Itopride free base

    CAS:
    <p>Itopride HCl combats dyspepsia and GERD, inhibiting AChE and blocking D2 receptors.</p>
    Formula:C20H26N2O4
    Colore e forma:White
    Peso molecolare:358.43
  • (RS)-ICI-118551 Hydrochloride

    CAS:
    ICI-118551 Hydrochloride (ICI-118,551) is a highly selective β2-adrenergic receptor antagonist with Ki values of 0.7, 49.5 and 611 nM for β2, β1 and β3
    Formula:C17H27NO2·HCl
    Purezza:98.02%
    Colore e forma:Solid
    Peso molecolare:313.86
  • Atenolol Hydrochloride

    CAS:
    <p>Atenolol Hydrochloride is a selective antagonist of ß1 receptor.</p>
    Formula:C14H23ClN2O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:302.80
  • Hydroxy ziprasidone

    CAS:
    <p>Hydroxy ziprasidone is an impurity of Ziprasidone. Ziprasidone, an antipsychotic agent, is a 5-HT and dopamine receptor antagonist.</p>
    Formula:C21H21ClN4O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:428.94
  • Caerulein, desulfated

    CAS:
    Caerulein, desulfated (FI-6934, desulfated) is a desulfated compound formed after caerulein hydrolysis, a neuropeptide with lower smooth muscle activity.
    Formula:C58H73N13O18S
    Purezza:99.46%
    Colore e forma:Solid
    Peso molecolare:1272.34
  • SB 271046 hydrochloride

    CAS:
    <p>SB 271046 hydrochloride (SB 271046A) is selective, orally active 5-HT6 antagonist and is &gt; 200-fold selective over 55 other receptors, enzymes and ion channels.</p>
    Formula:C20H22ClN3O3S2·HCl
    Purezza:99.77%
    Colore e forma:Solid
    Peso molecolare:488.45
  • Ridazolol HCl

    CAS:
    <p>Ridazolol HCl (CAS 413) is a novel β-adrenoceptor (β-AR) blocker with α-adrenerolytic activity.</p>
    Formula:C15H19Cl3N4O3
    Purezza:99.48%
    Colore e forma:Soild
    Peso molecolare:409.7
  • Ticlopidine

    CAS:
    <p>Ticlopidine (PCR 5332) is an antiplatelet drug in the thienopyridine family which is an adenosine diphosphate (ADP) receptor inhibitor.</p>
    Formula:C14H14ClNS
    Purezza:99.67%
    Colore e forma:Solid
    Peso molecolare:263.79
  • Norreticuline

    CAS:
    <p>Norreticuline is a potential adrenoceptor-α/β agonist and CYP2D6 and D2 receptor inhibitor for the study of neurodegenerative diseases.</p>
    Formula:C18H21NO4
    Colore e forma:Solid
    Peso molecolare:315.36
  • Dolasetron Mesylate

    CAS:
    <p>Dolasetron Mesylate (MDL-73147EF) is an antagonist of the 5-HT3 receptor and can be used in research on the treatment of vomiting and nausea following</p>
    Formula:C20H24N2O6S
    Purezza:99.05%
    Colore e forma:White Powder
    Peso molecolare:420.48
  • LY 344864

    CAS:
    <p>LY 344864, a specifc receptor agonist, is an affinity of 6 nM (Ki) at the recently cloned 5-HT1F receptor.</p>
    Formula:C21H22FN3O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:351.42
  • Guacetisal

    CAS:
    <p>Guacetisal, from acetylsalicylic acid and guaiacol, may treat chronic bronchitis.</p>
    Formula:C16H14O5
    Purezza:99.18%
    Colore e forma:Solid
    Peso molecolare:286.28
  • Lodoxamide tromethamine

    CAS:
    <p>Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergic</p>
    Formula:C19H28ClN5O12
    Purezza:98.8%
    Colore e forma:Solid
    Peso molecolare:553.91
  • Paroxetine hydrochloride hemihydrate

    CAS:
    <p>Paroxetine hydrochloride hemihydrate (Paxil) is an effective and selective serotonin reuptake inhibitor (SSRI).</p>
    Formula:C38H44Cl2F2N2O7
    Purezza:99.949%
    Colore e forma:Solid
    Peso molecolare:749.67
  • MK-5046

    CAS:
    MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = 1.6 nM, human Ki = 25 nM).
    Formula:C20H18F6N4O
    Purezza:98.56%
    Colore e forma:Solid
    Peso molecolare:444.37
  • A 63162

    CAS:
    <p>A 63162 is an inhibitor of 5-lipoxygenase.</p>
    Formula:C17H19NO3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:285.34
  • HSK0935

    CAS:
    <p>HSK0935 is a highly selective and orally available SGLT2 inhibitor (IC50: 1.3 nM). It has antihyperglycemic activities.</p>
    Formula:C22H25ClO7
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:436.88
  • Ipsapirone

    CAS:
    <p>Ipsapirone is a partial agonist of 5-HT1A receptor and produces an inhibitory effect on 5-HT2 and the α1-adrenergic function at high doses.</p>
    Formula:C19H23N5O3S
    Purezza:99.51%
    Colore e forma:Solid
    Peso molecolare:401.48
  • N,N-Dimethylsphingosine

    CAS:
    <p>N,N-Dimethylsphingosine,is a potent competitive SphK phosphorylation inhibitor.DMS is elevated in models of neuropathic pain by increasing IL-1β and MCP-1.</p>
    Formula:C20H41NO2
    Purezza:98%
    Colore e forma:Clear Colorless To Faint Yellow Liquid/White To Off-White Powder
    Peso molecolare:327.55
  • L 640033

    CAS:
    <p>L 640033 is a beta-agonist.</p>
    Formula:C18H25N3O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:299.41
  • RUSKI-201 dihydrochloride

    CAS:
    <p>RUSKI-201 dihydrochloride: potent Hhat inhibitor (IC50: 0.20 μM), blocks Hh signaling, and inhibits Hh palmitoylation.</p>
    Formula:C20H29Cl2N3OS
    Colore e forma:Solid
    Peso molecolare:430.43
  • Sigma-LIGAND-1

    CAS:
    <p>Sigma-LIGAND-1 is a selective Sigma Receptor ligand with an IC50s of 16 nM, 19 nM at the DTG site and the PPP site, respectively.</p>
    Formula:C27H33NO4
    Purezza:99.89%
    Colore e forma:Solid
    Peso molecolare:435.56
  • Isamoltane hemifumarate

    CAS:
    <p>5-HT1B antagonist</p>
    Formula:C16H22N202C4H404
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:332.4
  • 5-HT3 antagonist 3

    CAS:
    <p>5-HT3 antagonist 3 (Compound 15b) is a high-affinity 5-HT3 receptor antagonist. It binds to 5-HT3 receptors in rat brain cortical membranes (Ki: 0.25 nM).</p>
    Formula:C20H21N3O
    Purezza:99.9%
    Colore e forma:Solid
    Peso molecolare:319.4
  • 2-Methylthioadenosine diphosphate trisodium

    CAS:
    <p>2-Methylthioadenosine diphosphate trisodium(2-MeS-ADP) is a purinergic P2Y receptor agonist that agonizes P2Y13 and P2Y12, induces platelet aggregation.</p>
    Formula:C11H14N5Na3O10P2S
    Colore e forma:Solid
    Peso molecolare:539.24
  • SCH-23390 maleate

    CAS:
    <p>SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,</p>
    Formula:C21H22ClNO5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:403.86
  • 5-HT3 antagonist 2

    CAS:
    <p>5-HT3 antagonist 2 is an antagonist of 5-HT3 receptor.</p>
    Formula:C18H21N3O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:295.38
  • Afurolol Hydrochloride

    CAS:
    <p>Afurolol Hydrochloride (DL 071-IT) is a non-selective β-adrenergic receptor antagonist. DL 071 IT exhibits intrinsic sympathomimetic activity.</p>
    Formula:C15H22ClNO4
    Purezza:98.86%
    Colore e forma:Solid
    Peso molecolare:315.79