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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

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Trovati 5378 prodotti di "Proteina G/GPCR"

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  • Flestolol sulfate

    CAS:
    <p>Flestolol sulfate is an anti-adrenergic beta-receptor.</p>
    Formula:C15H24FN3O8S
    Colore e forma:Solid
    Peso molecolare:425.43
  • Phenindamine Tartrate

    CAS:
    <p>Phenindamine Tartrate, an antihistamine and anticholinergic, treats colds and allergies like sneezing and rashes.</p>
    Formula:C23H25NO6
    Colore e forma:Solid
    Peso molecolare:411.454
  • LY 163443

    CAS:
    <p>LY 163443 is an dual receptor antagonist of LTD4 and LTE4.</p>
    Formula:C20H22N4O3
    Colore e forma:Solid
    Peso molecolare:366.41
  • NPEC-caged-dopamine

    CAS:
    <p>Dopamine receptor agonist</p>
    Formula:C17H18N2O6
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:346.33
  • NPS ALX Compound 4a dihydrochloride

    CAS:
    <p>NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)</p>
    Formula:C25H27Cl2N3O2S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:504.47
  • WAY 163909

    CAS:
    WAY 163909 is an effective and selective agonist of the 5-HT(2C) receptor (Ki: 10.5±1.1 nM).
    Formula:C14H18N2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:214.31
  • ZD-1611

    CAS:
    <p>ZD-1611 is an effective and selective ETA receptor antagonist. It is used for the research of ischemic stroke.</p>
    Formula:C22H24N4O5S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:456.51
  • ROS 234 dioxalate

    CAS:
    <p>ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)</p>
    Formula:C17H19N5O8
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:421.37
  • AZ-GHS-22

    CAS:
    <p>AZ-GHS-22, an inverse agonist for GHS-R1a (ghrelin receptor), binds with 0.77 nM IC50, cutting mice food intake by 54% at 100 mg/kg.</p>
    Formula:C27H33ClN6O5S2
    Colore e forma:Solid
    Peso molecolare:621.17
  • N-Methyldopamine hydrochloride

    CAS:
    <p>N-Methyldopamine hydrochloride (Ephinine hydrochloride) is an α and β agonist, with indirect sympathomimetic effects similar to dopamine.</p>
    Formula:C9H14ClNO2
    Colore e forma:Solid
    Peso molecolare:203.67
  • BPIPP

    CAS:
    <p>guanylyl cyclase (GC) and adenylyl cyclase (AC) inhibitor</p>
    Formula:C22H16BrN3O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:450.28
  • MLN3126

    CAS:
    <p>MLN3126: Oral CCR9 blocker, hinders CCL25-triggered chemotaxis/thymocyte calcium influx, IC50 of 6.3 nM.</p>
    Formula:C21H19ClN2O5S
    Colore e forma:Solid
    Peso molecolare:446.9
  • KSCM-1

    CAS:
    <p>KSCM-1 is a selective sigma-1 receptor ligand.</p>
    Formula:C26H32N2O4
    Colore e forma:Solid
    Peso molecolare:436.54
  • GR-55562 dihydrobromide

    CAS:
    <p>GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.</p>
    Formula:C23H26ClN3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:411.93
  • Quinelorane dihydrochloride

    CAS:
    <p>Dopamine D2 and D3 receptor agonist</p>
    Formula:C14H23ClN4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:282.81
  • ATC0065 HCl

    CAS:
    <p>ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.</p>
    Formula:C25H31BrCl2F3N5O
    Colore e forma:Solid
    Peso molecolare:625.35
  • CL-184005

    CAS:
    <p>CL-184005 is a PAF inhibitor that blocks tumor necrosis factor synthesis and reduces spleen-associated TNF protein.</p>
    Formula:C33H46NO7PS
    Colore e forma:Solid
    Peso molecolare:631.76
  • Dapiprazole

    CAS:
    <p>Dapiprazole, an alpha blocker, is used to reverse mydriasis after eye examination.</p>
    Formula:C19H27N5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:325.45
  • COR 170

    CAS:
    <p>inverse agonist of CB2 receptors</p>
    Formula:C31H36N2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:468.63
  • Pronethalol hydrochloride

    CAS:
    <p>β-adrenergic antagonist</p>
    Formula:C15H20ClNO
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:265.78
  • Naminterol

    CAS:
    <p>Naminterol is a phenethanolamine derivative is an agonist of β2 adrenoceptor with bronchodilatory properties, and used for treatment of asthma.</p>
    Formula:C19H26N2O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:330.42
  • Ro 19-1400

    CAS:
    <p>Ro 19-1400, a platelet-activating factor antagonist, directly inhibits immunoglobulin E-dependent mediator release.</p>
    Formula:C31H56N2O8S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:616.85
  • (Rac)-E1R

    CAS:
    <p>(Rac)-E1R is the racemate of E1R. (Rac)-E1R is a sigma-1 receptor positive allosteric (Sig1R PAM) modulator of for the treatment of cognition/memory disorders.</p>
    Formula:C13H16N2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:232.28
  • GSK 189254 HCl

    CAS:
    <p>GSK 189254A: histamine H3 antagonist, treats narcolepsy, may improve cognition and help with dementia, neuropathic pain.</p>
    Formula:C21H26ClN3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:387.9
  • (-)-S-Timolol

    CAS:
    <p>(-)-S-Timolol is an antagonist of the beta-Adrenergic .</p>
    Formula:C13H26N4O4S
    Colore e forma:Solid
    Peso molecolare:334.44
  • Inupadenant

    CAS:
    <p>Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].</p>
    Formula:C25H26F2N8O4S2
    Colore e forma:Solid
    Peso molecolare:604.65
  • A3AR antagonist 1

    CAS:
    <p>A3AR antagonist 1 is a potent and selective human A3adenosine receptor (AR) antagonist (Ki: 4.63) and has no affinity for the rat A3AR.</p>
    Formula:C32H24N4O4S
    Colore e forma:Solid
    Peso molecolare:560.62
  • L-902688

    CAS:
    <p>L-902688 is an orally active EP4 receptor agonist (Ki: 0.38 nM; EC50: 0.6 nM).</p>
    Formula:C21H27F2N5O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:419.47
  • Alaproclate

    CAS:
    <p>Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.</p>
    Formula:C13H18ClNO2
    Purezza:98.29% - 98.64%
    Colore e forma:Solid
    Peso molecolare:255.74
  • Immepip

    CAS:
    <p>Immepip, a H3 agonist, has been shown to attenuate cortical histamine release and is utilized in the research of neurological diseases.</p>
    Formula:C9H15N3
    Colore e forma:Solid
    Peso molecolare:165.24
  • Phenyltoloxamine

    CAS:
    <p>Phenyltoloxamine (Bistrimin): antihistamine with sedative, analgesic properties, and Sigma-1 receptor affinity (Ki=160 nM).</p>
    Formula:C17H21NO
    Colore e forma:Solid
    Peso molecolare:255.35
  • CP 93129 dihydrochloride

    CAS:
    <p>5-HT1B agonist, potent and highly selective</p>
    Formula:C12H14ClN3O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:251.71
  • CCG-2046

    CAS:
    <p>CCG-2046 is a chemical inhibitor targeting RGS4, demonstrating an inhibition concentration (IC50) of 4.3 μM for the interaction between RGS4 and Gαo signal.</p>
    Formula:C11H10N4
    Colore e forma:Solid
    Peso molecolare:198.22
  • Mizolastine dihydrochloride

    CAS:
    <p>Mizolastine dihydrochloride is a histamine H1-receptor antagonist (IC50: 47 nM).</p>
    Formula:C24H27Cl2FN6O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:505.42
  • VPC 23019

    CAS:
    <p>VPC 23019 is a competitive antagonist at the S1P1 and S1P3 receptors (pKi= 7.86 and 5.93, respectively).</p>
    Formula:C17H29N2O5P
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:372.4
  • CH 141

    CAS:
    <p>CH 141 is a new type of peripheral vasodilator.</p>
    Formula:C19H21N3O
    Colore e forma:Solid
    Peso molecolare:307.39
  • ABT-546

    CAS:
    <p>ABT-546 is a potent, selective endothelin ETA receptor antagonist, Ki 0.46 nM for [125I]ET-1 binding.</p>
    Formula:C30H48N2O6
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:532.71
  • Bag-1

    CAS:
    <p>Bag-1 is a novel potent, non-peptidic bombesin receptor subtype-3 (BRS-3) agonist.</p>
    Formula:C22H27N3
    Colore e forma:Solid
    Peso molecolare:333.47
  • JNJ-17156516

    CAS:
    <p>JNJ-17156516 is a potent, and selective cholecystokinin 1 receptor antagonist.</p>
    Formula:C26H22Cl2N2O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:481.37
  • Adenosine receptor antagonist 2

    CAS:
    <p>Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.</p>
    Formula:C23H21FN8O
    Colore e forma:Solid
    Peso molecolare:444.46
  • Mianserin

    CAS:
    <p>Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.</p>
    Formula:C18H20N2
    Purezza:99.85%
    Colore e forma:Solid
    Peso molecolare:264.36
  • GCGR antagonist 2

    CAS:
    <p>Orally active GCGR antagonist 2, a furan-2-carbohydrazide, binds hGluR at 2.3 nM. Blocks glucagon, inhibits rat receptor at 0.43 nM.</p>
    Formula:C28H26N4O2
    Colore e forma:Solid
    Peso molecolare:450.53
  • Ko-3290

    CAS:
    <p>Ko-3290 is a cardioselective antagonist of β-adrenoceptors known for its antilipolytic effects in animals.</p>
    Formula:C19H25N3O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:343.42
  • Sequifenadine

    CAS:
    <p>Sequifenadine has the potential in researching of inflammatory eye disease with allergic symptoms that is a H1-antihistamine [1] [2].</p>
    Formula:C22H27NO
    Colore e forma:Solid
    Peso molecolare:321.46
  • CCG-271423

    CAS:
    <p>CCG-271423: potent GRK5 inhibitor (IC50: 0.0021 μM), less on GRK2 (IC50: 44 μM); lowers Ca2+ events and heart cell contractility.</p>
    Formula:C28H26N4O3
    Colore e forma:Solid
    Peso molecolare:466.53
  • 2-ThioUTP tetrasodium salt

    CAS:
    <p>2-ThioUTP tetrasodium salt is a P2Y2 agonist.</p>
    Formula:C9H15N2O14P3S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:500.21
  • O-2093

    CAS:
    <p>anandamide uptake inhibitor</p>
    Formula:C34H43Cl2NO3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:584.62
  • ATC0065

    CAS:
    <p>ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.</p>
    Formula:C25H29BrF3N5O
    Colore e forma:Solid
    Peso molecolare:552.43
  • Acetylaszonalenin

    CAS:
    <p>Acetylaszonalenin, from A. flavipes, is an NK1 receptor antagonist with a Ki of 170 μM, blocking substance P.</p>
    Formula:C25H25N3O3
    Colore e forma:Solid
    Peso molecolare:415.48
  • SKF 77434 hydrobromide

    CAS:
    <p>SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.</p>
    Formula:C19H22BrNO2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:376.29
  • CP 96345

    CAS:
    <p>CP 96345 is a NK1 receptor antagonist.</p>
    Formula:C28H32N2O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:412.57
  • 3-epi-Vitamin D3

    CAS:
    <p>3-epi-Vitamin D3 (Epicholecalciferol), an analogue of Vitamin D3, serves as a Hedgehog pathway inhibitor, exhibiting potency with an IC50 value of 39.2 μM in</p>
    Formula:C27H44O
    Colore e forma:Solid
    Peso molecolare:384.64
  • Fenmetozole Tosylate

    CAS:
    <p>Fenmetozole Tosylate , acts as an antidepressant drug. is an antagonist of the actions of ethanol, also antagonizes α2-adrenergic receptor,</p>
    Formula:C17H18Cl2N2O4S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:417.31
  • RUSKI-201

    CAS:
    <p>RUSKI-201 is the first selective Hedgehog acyltransferase (Hhat) chemical probe in cells.</p>
    Formula:C20H27N3OS
    Colore e forma:Solid
    Peso molecolare:357.51
  • MRS2179

    CAS:
    <p>MRS2179: P2Y1 antagonist, Kb=100 nM, inactive on P2Y2/4/6 (to 30µM), inhibits ADP-induced platelet changes, prolongs bleeding in rodents.</p>
    Formula:C11H17N5O9P2
    Colore e forma:Solid
    Peso molecolare:425.23
  • CI 1020

    CAS:
    <p>endothelin-A receptor (ETA) antagonist</p>
    Formula:C28H26O9
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:506.5
  • Lidanserin

    CAS:
    <p>Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.</p>
    Formula:C26H31FN2O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:454.53
  • Atigliflozin

    CAS:
    <p>Atigliflozin is an antihyperglycaemic drug candidate.</p>
    Formula:C18H22O7S
    Colore e forma:Solid
    Peso molecolare:382.43
  • Ro 363 hydrochloride

    CAS:
    <p>Ro 363 hydrochloride: selective β1-adrenoceptor agonist, boosts heart contraction, lowers diastolic pressure.</p>
    Formula:C19H26ClNO6
    Colore e forma:Solid
    Peso molecolare:399.87
  • Rolapitant

    CAS:
    <p>Rolapitant Hydrochloride is an oral NK1-receptor blocker that prevents nausea and has a fast onset and long half-life.</p>
    Formula:C25H26F6N2O2
    Purezza:99.86%
    Colore e forma:Solid
    Peso molecolare:500.48
  • FG-5893

    CAS:
    <p>FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.</p>
    Formula:C27H29F2N3O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:465.53
  • CCR8 antagonist 2

    CAS:
    <p>CCR8 antagonist 2 blocks CCR8 activity, mainly on Treg and Th2 cells, for treating related diseases. See WO2022000443A1, compound 220.</p>
    Formula:C23H30ClN3O3S
    Colore e forma:Solid
    Peso molecolare:464.02
  • Methyldopate hydrochloride

    CAS:
    <p>Methyldopate HCl is an agent of antihypertensive.</p>
    Formula:C12H18ClNO4
    Colore e forma:Solid
    Peso molecolare:275.73
  • CP-195543

    CAS:
    <p>CP-195543 is an effective leukotriene B4 antagonist for the treatment of inflammatory diseases.</p>
    Formula:C24H19F3O4
    Colore e forma:Solid
    Peso molecolare:428.4
  • Guanethidine

    CAS:
    <p>Guanethidine sulphate, made in 1959, lowers blood pressure by disrupting neurotransmitters in sympathetic nerves.</p>
    Formula:C10H22N4
    Colore e forma:Solid
    Peso molecolare:198.31
  • EP4 receptor antagonist 4

    CAS:
    <p>EP4 receptor antagonist 4 is an agonist of EP4 receptor (human pEC 50 = 6.3) [1].</p>
    Formula:C19H14N2OS
    Colore e forma:Solid
    Peso molecolare:318.39
  • SKF-75670 Hydrobromide

    CAS:
    <p>SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.</p>
    Formula:C17H20BrNO2
    Colore e forma:Solid
    Peso molecolare:350.25
  • Zicronapine

    CAS:
    <p>Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.</p>
    Formula:C22H27ClN2
    Colore e forma:Solid
    Peso molecolare:354.92
  • WB403

    CAS:
    <p>WB403 activates TGR5, lowers fasting/postprandial glucose and HbA1c, enhances glucose tolerance, and normalizes pancreatic α/β-cells in diabetic mice.</p>
    Formula:C19H19BrN2OS
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:403.34
  • LY 219057

    CAS:
    LY 219057 is a potent, competitive, and specific antagonist of CCK receptor on the exocrine pancreas.
    Formula:C23H17ClF3N3OS
    Colore e forma:Solid
    Peso molecolare:475.91
  • S-777469

    CAS:
    <p>S-777469: Selective CB2 agonist, oral, inhibits itching in mice (Ki: 36 nM). Anti-pruritic.</p>
    Formula:C23H27FN2O4
    Colore e forma:Solid
    Peso molecolare:414.47
  • CB2 receptor agonist 3

    CAS:
    <p>GP 2A is a selective agonist of CB2 receptor.</p>
    Formula:C24H23Cl2N3O
    Colore e forma:Solid
    Peso molecolare:440.36
  • ATL-801

    CAS:
    <p>ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.</p>
    Formula:C24H25N7O3
    Colore e forma:Solid
    Peso molecolare:459.5
  • Remogliflozin

    CAS:
    <p>Remogliflozin is an effective sodium-glucose transporter 2 inhibitor (Kis = 12.4 and 26 nM for human and rat SGLT2, respectively).</p>
    Formula:C23H34N2O7
    Colore e forma:Solid
    Peso molecolare:450.53
  • Medroxalol

    CAS:
    <p>Medroxalol (RMI81968), an oral α- &amp; β-adrenergic blocker, has antihypertensive and vasodilatory effects.</p>
    Formula:C20H24N2O5
    Colore e forma:Solid
    Peso molecolare:372.42
  • LY377604

    CAS:
    <p>LY377604 is a human β3-adrenergic receptor agonist (EC50: 2.4 nM) and β1/2-adrenergic receptor antagonist for the study of obesity.</p>
    Formula:C31H32N4O4
    Purezza:99.72% - >99.99%
    Colore e forma:Solid
    Peso molecolare:524.61
  • Adenosine receptor A1 antagonist 5

    CAS:
    <p>1,3-Dipropyl-8-phenylxanthine is an adenosine antagonist, oxypurine, insecticide, and reduces high blood pressure.</p>
    Formula:C17H20N4O2
    Purezza:99.97%
    Colore e forma:Solid
    Peso molecolare:312.37
  • Ampreloxetine

    CAS:
    <p>Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.</p>
    Formula:C18H18F3NO
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:321.34
  • EMD 56551

    CAS:
    <p>EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.</p>
    Formula:C24H31N3O2
    Purezza:95.64% - 99.39%
    Colore e forma:Solid
    Peso molecolare:393.522
  • (S)-(-)-Propranolol hydrochloride

    CAS:
    <p>(S)-(-)-Propranolol hydrochloride 是一种有效的肾上腺素能受体 (β-adrenergic receptor) 拮抗剂,具有抗高血压活性和潜在的抗癌活性,对β1,β2,和β3受体有抑制作用。(S)-(-)-Propranolol hydrochloride 可改善严重烧伤患者的预后,可用于研究酒精症。</p>
    Formula:C16H22ClNO2
    Purezza:99.02% - 99.91%
    Colore e forma:Solid
    Peso molecolare:295.8
  • Befetupitant

    CAS:
    <p>Befupupitant(Ro67-5930) is a potent and selective tachykinin 1 receptor (NK1R) antagonist for the study of corneal neovascularization.</p>
    Formula:C29H29F6N3O2
    Purezza:98.72%
    Colore e forma:Solid
    Peso molecolare:565.55
  • CB1R Allosteric modulator 3

    CAS:
    <p>CB1R Allosteric modulator 3 is a CB1R modulator.CB1R Allosteric modulator 3 inhibits cAMP, and can be used for the study of obesity and nicotine addiction.</p>
    Formula:C22H17ClN2O2
    Purezza:98.18%
    Colore e forma:Solid
    Peso molecolare:376.84
  • (R)-SLV 319

    CAS:
    <p>(R)-SLV 319: potent CB1 antagonist, K i of 894 nM, dextrorotatory isomer.</p>
    Formula:C23H20Cl2N4O2S
    Colore e forma:Solid
    Peso molecolare:487.4
  • WS 009A

    CAS:
    <p>WS 009A is an antagonist of the endothelin receptor.</p>
    Formula:C24H25NO10S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:519.52
  • ST1936

    CAS:
    <p>ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.</p>
    Formula:C13H17ClN2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:236.74
  • CJ 033466

    CAS:
    <p>CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.</p>
    Formula:C19H28ClN5O
    Purezza:99.72%
    Colore e forma:Solid
    Peso molecolare:377.91
  • Eplivanserin

    CAS:
    Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.
    Formula:C19H21FN2O2
    Purezza:97.04%
    Colore e forma:Solid
    Peso molecolare:328.38
  • DOV-216,303 Free Base

    CAS:
    <p>DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.</p>
    Formula:C11H11Cl2N
    Purezza:96.7%
    Colore e forma:Solid
    Peso molecolare:228.12
  • Chlorazanil

    CAS:
    <p>Chlorazanil is a triazine-based, orally active diuretic that blocks Na+ and Cl– reabsorption in distal tubules, increases renal prostaglandin.</p>
    Formula:C9H8ClN5
    Purezza:98.89%
    Colore e forma:Solid
    Peso molecolare:221.65
  • Nedocromil

    CAS:
    <p>Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).</p>
    Formula:C19H17NO7
    Purezza:95% - 97.34%
    Colore e forma:Solid
    Peso molecolare:371.34
  • Quinpirole Hydrochloride

    CAS:
    <p>Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and mice</p>
    Formula:C13H22ClN3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:255.79
  • AM6545

    CAS:
    <p>AM6545 is a CB1 receptor antagonist used in the study of obesity and diabetes.</p>
    Formula:C26H23Cl2N5O3S
    Purezza:97.03%
    Colore e forma:Solid
    Peso molecolare:556.46
  • Adatanserin

    CAS:
    <p>Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C receptor antagonist.</p>
    Formula:C21H31N5O
    Purezza:99.33%
    Colore e forma:Solid
    Peso molecolare:369.5
  • Aligeron

    CAS:
    <p>Aligeron is a non-selective prostaglandin (PG) antagonist that inhibits PGF2α- and PGE2-induced decreases in blood pressure in cats, and can be used to inhibit</p>
    Formula:C20H24N2
    Purezza:99.09% - >99.99%
    Colore e forma:Solid
    Peso molecolare:292.42
  • Vapitadine dihydrochloride

    CAS:
    <p>Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.</p>
    Formula:C17H22Cl2N4O
    Purezza:98.28% - 99.30%
    Colore e forma:Solid
    Peso molecolare:369.29
  • ML179

    CAS:
    <p>ML179 is a potent and selective inverse agonist of liver receptor homolog-1 (LRH1, NR5A2) with IC50 of 320 nM.</p>
    Formula:C21H25F3N4O2
    Purezza:99.77%
    Colore e forma:Solid
    Peso molecolare:422.44
  • TIK-301

    CAS:
    <p>TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM</p>
    Formula:C14H17ClN2O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:280.75
  • Amgen-23

    CAS:
    <p>Amgen-23 is a selective and highly potent sphingosine kinase 1 (SPHK1) inhibitor that inhibits SPHK2 and can be used in anticancer research.</p>
    Formula:C23H25Cl2N3O2S
    Purezza:97.31%
    Colore e forma:Solid
    Peso molecolare:478.44
  • SDZ 205-557 hydrochloride

    CAS:
    <p>5-HT3/5-HT4 receptor antagonist</p>
    Formula:C14H22Cl2N2O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:337.24
  • RS 15385-197

    CAS:
    <p>RS 15385-197 is a selective alpha 2-adrenoceptor antagonist.</p>
    Formula:C18H26N2O3S
    Colore e forma:Solid
    Peso molecolare:350.48