
Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(942 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.949 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(149 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(410 prodotti)
- Recettore dell'endotelina(75 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(32 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(166 prodotti)
- Proteina Hedgehog/Smoothened(45 prodotti)
- Recettore dell'istamina(359 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(298 prodotti)
- PAFR(11 prodotti)
- PKA(49 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5378 prodotti di "Proteina G/GPCR"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Flestolol sulfate
CAS:<p>Flestolol sulfate is an anti-adrenergic beta-receptor.</p>Formula:C15H24FN3O8SColore e forma:SolidPeso molecolare:425.43Phenindamine Tartrate
CAS:<p>Phenindamine Tartrate, an antihistamine and anticholinergic, treats colds and allergies like sneezing and rashes.</p>Formula:C23H25NO6Colore e forma:SolidPeso molecolare:411.454LY 163443
CAS:<p>LY 163443 is an dual receptor antagonist of LTD4 and LTE4.</p>Formula:C20H22N4O3Colore e forma:SolidPeso molecolare:366.41NPEC-caged-dopamine
CAS:<p>Dopamine receptor agonist</p>Formula:C17H18N2O6Purezza:98%Colore e forma:SolidPeso molecolare:346.33NPS ALX Compound 4a dihydrochloride
CAS:<p>NPS ALX Compound 4a dihydrochloride is a potent and selective antagonist of 5-HT6 receptor (IC50 of 7.2 nM)</p>Formula:C25H27Cl2N3O2SPurezza:98%Colore e forma:SolidPeso molecolare:504.47WAY 163909
CAS:WAY 163909 is an effective and selective agonist of the 5-HT(2C) receptor (Ki: 10.5±1.1 nM).Formula:C14H18N2Purezza:98%Colore e forma:SolidPeso molecolare:214.31ZD-1611
CAS:<p>ZD-1611 is an effective and selective ETA receptor antagonist. It is used for the research of ischemic stroke.</p>Formula:C22H24N4O5SPurezza:98%Colore e forma:SolidPeso molecolare:456.51ROS 234 dioxalate
CAS:<p>ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)</p>Formula:C17H19N5O8Purezza:98%Colore e forma:SolidPeso molecolare:421.37AZ-GHS-22
CAS:<p>AZ-GHS-22, an inverse agonist for GHS-R1a (ghrelin receptor), binds with 0.77 nM IC50, cutting mice food intake by 54% at 100 mg/kg.</p>Formula:C27H33ClN6O5S2Colore e forma:SolidPeso molecolare:621.17N-Methyldopamine hydrochloride
CAS:<p>N-Methyldopamine hydrochloride (Ephinine hydrochloride) is an α and β agonist, with indirect sympathomimetic effects similar to dopamine.</p>Formula:C9H14ClNO2Colore e forma:SolidPeso molecolare:203.67BPIPP
CAS:<p>guanylyl cyclase (GC) and adenylyl cyclase (AC) inhibitor</p>Formula:C22H16BrN3O3Purezza:98%Colore e forma:SolidPeso molecolare:450.28MLN3126
CAS:<p>MLN3126: Oral CCR9 blocker, hinders CCL25-triggered chemotaxis/thymocyte calcium influx, IC50 of 6.3 nM.</p>Formula:C21H19ClN2O5SColore e forma:SolidPeso molecolare:446.9KSCM-1
CAS:<p>KSCM-1 is a selective sigma-1 receptor ligand.</p>Formula:C26H32N2O4Colore e forma:SolidPeso molecolare:436.54GR-55562 dihydrobromide
CAS:<p>GR-55562 dihydrobromide is a antagonist of 5-HT1B/5-HT1D serotonin receptor.</p>Formula:C23H26ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:411.93Quinelorane dihydrochloride
CAS:<p>Dopamine D2 and D3 receptor agonist</p>Formula:C14H23ClN4Purezza:98%Colore e forma:SolidPeso molecolare:282.81ATC0065 HCl
CAS:<p>ATC0065 dihydrochloride is a novel nonpeptidic and potent melanin-concentrating hormone receptor 1 (MCHR1) selective antagonist.</p>Formula:C25H31BrCl2F3N5OColore e forma:SolidPeso molecolare:625.35CL-184005
CAS:<p>CL-184005 is a PAF inhibitor that blocks tumor necrosis factor synthesis and reduces spleen-associated TNF protein.</p>Formula:C33H46NO7PSColore e forma:SolidPeso molecolare:631.76Dapiprazole
CAS:<p>Dapiprazole, an alpha blocker, is used to reverse mydriasis after eye examination.</p>Formula:C19H27N5Purezza:98%Colore e forma:SolidPeso molecolare:325.45COR 170
CAS:<p>inverse agonist of CB2 receptors</p>Formula:C31H36N2O2Purezza:98%Colore e forma:SolidPeso molecolare:468.63Pronethalol hydrochloride
CAS:<p>β-adrenergic antagonist</p>Formula:C15H20ClNOPurezza:98%Colore e forma:SolidPeso molecolare:265.78Naminterol
CAS:<p>Naminterol is a phenethanolamine derivative is an agonist of β2 adrenoceptor with bronchodilatory properties, and used for treatment of asthma.</p>Formula:C19H26N2O3Purezza:98%Colore e forma:SolidPeso molecolare:330.42Ro 19-1400
CAS:<p>Ro 19-1400, a platelet-activating factor antagonist, directly inhibits immunoglobulin E-dependent mediator release.</p>Formula:C31H56N2O8SPurezza:98%Colore e forma:SolidPeso molecolare:616.85(Rac)-E1R
CAS:<p>(Rac)-E1R is the racemate of E1R. (Rac)-E1R is a sigma-1 receptor positive allosteric (Sig1R PAM) modulator of for the treatment of cognition/memory disorders.</p>Formula:C13H16N2O2Purezza:98%Colore e forma:SolidPeso molecolare:232.28GSK 189254 HCl
CAS:<p>GSK 189254A: histamine H3 antagonist, treats narcolepsy, may improve cognition and help with dementia, neuropathic pain.</p>Formula:C21H26ClN3O2Purezza:98%Colore e forma:SolidPeso molecolare:387.9(-)-S-Timolol
CAS:<p>(-)-S-Timolol is an antagonist of the beta-Adrenergic .</p>Formula:C13H26N4O4SColore e forma:SolidPeso molecolare:334.44Inupadenant
CAS:<p>Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].</p>Formula:C25H26F2N8O4S2Colore e forma:SolidPeso molecolare:604.65A3AR antagonist 1
CAS:<p>A3AR antagonist 1 is a potent and selective human A3adenosine receptor (AR) antagonist (Ki: 4.63) and has no affinity for the rat A3AR.</p>Formula:C32H24N4O4SColore e forma:SolidPeso molecolare:560.62L-902688
CAS:<p>L-902688 is an orally active EP4 receptor agonist (Ki: 0.38 nM; EC50: 0.6 nM).</p>Formula:C21H27F2N5O2Purezza:98%Colore e forma:SolidPeso molecolare:419.47Alaproclate
CAS:<p>Alaproclate is a non-competitive NMDA receptor antagonist and a new selective 5-HT uptake inhibitor for the study of depression and dementia.</p>Formula:C13H18ClNO2Purezza:98.29% - 98.64%Colore e forma:SolidPeso molecolare:255.74Immepip
CAS:<p>Immepip, a H3 agonist, has been shown to attenuate cortical histamine release and is utilized in the research of neurological diseases.</p>Formula:C9H15N3Colore e forma:SolidPeso molecolare:165.24Phenyltoloxamine
CAS:<p>Phenyltoloxamine (Bistrimin): antihistamine with sedative, analgesic properties, and Sigma-1 receptor affinity (Ki=160 nM).</p>Formula:C17H21NOColore e forma:SolidPeso molecolare:255.35CP 93129 dihydrochloride
CAS:<p>5-HT1B agonist, potent and highly selective</p>Formula:C12H14ClN3OPurezza:98%Colore e forma:SolidPeso molecolare:251.71CCG-2046
CAS:<p>CCG-2046 is a chemical inhibitor targeting RGS4, demonstrating an inhibition concentration (IC50) of 4.3 μM for the interaction between RGS4 and Gαo signal.</p>Formula:C11H10N4Colore e forma:SolidPeso molecolare:198.22Mizolastine dihydrochloride
CAS:<p>Mizolastine dihydrochloride is a histamine H1-receptor antagonist (IC50: 47 nM).</p>Formula:C24H27Cl2FN6OPurezza:98%Colore e forma:SolidPeso molecolare:505.42VPC 23019
CAS:<p>VPC 23019 is a competitive antagonist at the S1P1 and S1P3 receptors (pKi= 7.86 and 5.93, respectively).</p>Formula:C17H29N2O5PPurezza:98%Colore e forma:SolidPeso molecolare:372.4CH 141
CAS:<p>CH 141 is a new type of peripheral vasodilator.</p>Formula:C19H21N3OColore e forma:SolidPeso molecolare:307.39ABT-546
CAS:<p>ABT-546 is a potent, selective endothelin ETA receptor antagonist, Ki 0.46 nM for [125I]ET-1 binding.</p>Formula:C30H48N2O6Purezza:98%Colore e forma:SolidPeso molecolare:532.71Bag-1
CAS:<p>Bag-1 is a novel potent, non-peptidic bombesin receptor subtype-3 (BRS-3) agonist.</p>Formula:C22H27N3Colore e forma:SolidPeso molecolare:333.47JNJ-17156516
CAS:<p>JNJ-17156516 is a potent, and selective cholecystokinin 1 receptor antagonist.</p>Formula:C26H22Cl2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:481.37Adenosine receptor antagonist 2
CAS:<p>Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.</p>Formula:C23H21FN8OColore e forma:SolidPeso molecolare:444.46Mianserin
CAS:<p>Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.</p>Formula:C18H20N2Purezza:99.85%Colore e forma:SolidPeso molecolare:264.36GCGR antagonist 2
CAS:<p>Orally active GCGR antagonist 2, a furan-2-carbohydrazide, binds hGluR at 2.3 nM. Blocks glucagon, inhibits rat receptor at 0.43 nM.</p>Formula:C28H26N4O2Colore e forma:SolidPeso molecolare:450.53Ko-3290
CAS:<p>Ko-3290 is a cardioselective antagonist of β-adrenoceptors known for its antilipolytic effects in animals.</p>Formula:C19H25N3O3Purezza:98%Colore e forma:SolidPeso molecolare:343.42Sequifenadine
CAS:<p>Sequifenadine has the potential in researching of inflammatory eye disease with allergic symptoms that is a H1-antihistamine [1] [2].</p>Formula:C22H27NOColore e forma:SolidPeso molecolare:321.46CCG-271423
CAS:<p>CCG-271423: potent GRK5 inhibitor (IC50: 0.0021 μM), less on GRK2 (IC50: 44 μM); lowers Ca2+ events and heart cell contractility.</p>Formula:C28H26N4O3Colore e forma:SolidPeso molecolare:466.532-ThioUTP tetrasodium salt
CAS:<p>2-ThioUTP tetrasodium salt is a P2Y2 agonist.</p>Formula:C9H15N2O14P3SPurezza:98%Colore e forma:SolidPeso molecolare:500.21O-2093
CAS:<p>anandamide uptake inhibitor</p>Formula:C34H43Cl2NO3Purezza:98%Colore e forma:SolidPeso molecolare:584.62ATC0065
CAS:<p>ATC0065 is a melanin-concentrating hormone receptor 1 antagonist with oral activity.</p>Formula:C25H29BrF3N5OColore e forma:SolidPeso molecolare:552.43Acetylaszonalenin
CAS:<p>Acetylaszonalenin, from A. flavipes, is an NK1 receptor antagonist with a Ki of 170 μM, blocking substance P.</p>Formula:C25H25N3O3Colore e forma:SolidPeso molecolare:415.48SKF 77434 hydrobromide
CAS:<p>SKF 77434 hydrobromide is a dopamine D1-like receptor partial agonist.</p>Formula:C19H22BrNO2Purezza:98%Colore e forma:SolidPeso molecolare:376.29CP 96345
CAS:<p>CP 96345 is a NK1 receptor antagonist.</p>Formula:C28H32N2OPurezza:98%Colore e forma:SolidPeso molecolare:412.573-epi-Vitamin D3
CAS:<p>3-epi-Vitamin D3 (Epicholecalciferol), an analogue of Vitamin D3, serves as a Hedgehog pathway inhibitor, exhibiting potency with an IC50 value of 39.2 μM in</p>Formula:C27H44OColore e forma:SolidPeso molecolare:384.64Fenmetozole Tosylate
CAS:<p>Fenmetozole Tosylate , acts as an antidepressant drug. is an antagonist of the actions of ethanol, also antagonizes α2-adrenergic receptor,</p>Formula:C17H18Cl2N2O4SPurezza:98%Colore e forma:SolidPeso molecolare:417.31RUSKI-201
CAS:<p>RUSKI-201 is the first selective Hedgehog acyltransferase (Hhat) chemical probe in cells.</p>Formula:C20H27N3OSColore e forma:SolidPeso molecolare:357.51MRS2179
CAS:<p>MRS2179: P2Y1 antagonist, Kb=100 nM, inactive on P2Y2/4/6 (to 30µM), inhibits ADP-induced platelet changes, prolongs bleeding in rodents.</p>Formula:C11H17N5O9P2Colore e forma:SolidPeso molecolare:425.23CI 1020
CAS:<p>endothelin-A receptor (ETA) antagonist</p>Formula:C28H26O9Purezza:98%Colore e forma:SolidPeso molecolare:506.5Lidanserin
CAS:<p>Lidanserin is an antagonist of the 5-HT2A and α1-adrenergic receptor.</p>Formula:C26H31FN2O4Purezza:98%Colore e forma:SolidPeso molecolare:454.53Atigliflozin
CAS:<p>Atigliflozin is an antihyperglycaemic drug candidate.</p>Formula:C18H22O7SColore e forma:SolidPeso molecolare:382.43Ro 363 hydrochloride
CAS:<p>Ro 363 hydrochloride: selective β1-adrenoceptor agonist, boosts heart contraction, lowers diastolic pressure.</p>Formula:C19H26ClNO6Colore e forma:SolidPeso molecolare:399.87Rolapitant
CAS:<p>Rolapitant Hydrochloride is an oral NK1-receptor blocker that prevents nausea and has a fast onset and long half-life.</p>Formula:C25H26F6N2O2Purezza:99.86%Colore e forma:SolidPeso molecolare:500.48FG-5893
CAS:<p>FG-5893 is a 5-HT1A agonist and 5-HT2 antagonist with potential anxiolytic activity.</p>Formula:C27H29F2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:465.53CCR8 antagonist 2
CAS:<p>CCR8 antagonist 2 blocks CCR8 activity, mainly on Treg and Th2 cells, for treating related diseases. See WO2022000443A1, compound 220.</p>Formula:C23H30ClN3O3SColore e forma:SolidPeso molecolare:464.02Methyldopate hydrochloride
CAS:<p>Methyldopate HCl is an agent of antihypertensive.</p>Formula:C12H18ClNO4Colore e forma:SolidPeso molecolare:275.73CP-195543
CAS:<p>CP-195543 is an effective leukotriene B4 antagonist for the treatment of inflammatory diseases.</p>Formula:C24H19F3O4Colore e forma:SolidPeso molecolare:428.4Guanethidine
CAS:<p>Guanethidine sulphate, made in 1959, lowers blood pressure by disrupting neurotransmitters in sympathetic nerves.</p>Formula:C10H22N4Colore e forma:SolidPeso molecolare:198.31EP4 receptor antagonist 4
CAS:<p>EP4 receptor antagonist 4 is an agonist of EP4 receptor (human pEC 50 = 6.3) [1].</p>Formula:C19H14N2OSColore e forma:SolidPeso molecolare:318.39SKF-75670 Hydrobromide
CAS:<p>SKF-75670 hydrobromide is an atypical D1DR (dopamine receptor) agonist. It displays agonist activity in vivo and antagonist activity in vitro.</p>Formula:C17H20BrNO2Colore e forma:SolidPeso molecolare:350.25Zicronapine
CAS:<p>Zicronapine (LU 31-130), an atypical antipsychotic with monoaminergic action, targets dopamine D1/D2 and serotonin 5HT2A.</p>Formula:C22H27ClN2Colore e forma:SolidPeso molecolare:354.92WB403
CAS:<p>WB403 activates TGR5, lowers fasting/postprandial glucose and HbA1c, enhances glucose tolerance, and normalizes pancreatic α/β-cells in diabetic mice.</p>Formula:C19H19BrN2OSPurezza:98%Colore e forma:SolidPeso molecolare:403.34LY 219057
CAS:LY 219057 is a potent, competitive, and specific antagonist of CCK receptor on the exocrine pancreas.Formula:C23H17ClF3N3OSColore e forma:SolidPeso molecolare:475.91S-777469
CAS:<p>S-777469: Selective CB2 agonist, oral, inhibits itching in mice (Ki: 36 nM). Anti-pruritic.</p>Formula:C23H27FN2O4Colore e forma:SolidPeso molecolare:414.47CB2 receptor agonist 3
CAS:<p>GP 2A is a selective agonist of CB2 receptor.</p>Formula:C24H23Cl2N3OColore e forma:SolidPeso molecolare:440.36ATL-801
CAS:<p>ATL-801 is anselective antagonist of A2B receptor with herapeutic activity for colitis.</p>Formula:C24H25N7O3Colore e forma:SolidPeso molecolare:459.5Remogliflozin
CAS:<p>Remogliflozin is an effective sodium-glucose transporter 2 inhibitor (Kis = 12.4 and 26 nM for human and rat SGLT2, respectively).</p>Formula:C23H34N2O7Colore e forma:SolidPeso molecolare:450.53Medroxalol
CAS:<p>Medroxalol (RMI81968), an oral α- & β-adrenergic blocker, has antihypertensive and vasodilatory effects.</p>Formula:C20H24N2O5Colore e forma:SolidPeso molecolare:372.42LY377604
CAS:<p>LY377604 is a human β3-adrenergic receptor agonist (EC50: 2.4 nM) and β1/2-adrenergic receptor antagonist for the study of obesity.</p>Formula:C31H32N4O4Purezza:99.72% - >99.99%Colore e forma:SolidPeso molecolare:524.61Adenosine receptor A1 antagonist 5
CAS:<p>1,3-Dipropyl-8-phenylxanthine is an adenosine antagonist, oxypurine, insecticide, and reduces high blood pressure.</p>Formula:C17H20N4O2Purezza:99.97%Colore e forma:SolidPeso molecolare:312.37Ampreloxetine
CAS:<p>Ampreloxetine (TD-9855) is a norepinephrine reuptake inhibitor used to study neurological diseases.</p>Formula:C18H18F3NOPurezza:98%Colore e forma:SolidPeso molecolare:321.34EMD 56551
CAS:<p>EMD 56551 is a selective small molecule 5-HT1A receptor agonist with anxiolytic activity for the study of anxiety disorders.</p>Formula:C24H31N3O2Purezza:95.64% - 99.39%Colore e forma:SolidPeso molecolare:393.522(S)-(-)-Propranolol hydrochloride
CAS:<p>(S)-(-)-Propranolol hydrochloride 是一种有效的肾上腺素能受体 (β-adrenergic receptor) 拮抗剂,具有抗高血压活性和潜在的抗癌活性,对β1,β2,和β3受体有抑制作用。(S)-(-)-Propranolol hydrochloride 可改善严重烧伤患者的预后,可用于研究酒精症。</p>Formula:C16H22ClNO2Purezza:99.02% - 99.91%Colore e forma:SolidPeso molecolare:295.8Befetupitant
CAS:<p>Befupupitant(Ro67-5930) is a potent and selective tachykinin 1 receptor (NK1R) antagonist for the study of corneal neovascularization.</p>Formula:C29H29F6N3O2Purezza:98.72%Colore e forma:SolidPeso molecolare:565.55CB1R Allosteric modulator 3
CAS:<p>CB1R Allosteric modulator 3 is a CB1R modulator.CB1R Allosteric modulator 3 inhibits cAMP, and can be used for the study of obesity and nicotine addiction.</p>Formula:C22H17ClN2O2Purezza:98.18%Colore e forma:SolidPeso molecolare:376.84(R)-SLV 319
CAS:<p>(R)-SLV 319: potent CB1 antagonist, K i of 894 nM, dextrorotatory isomer.</p>Formula:C23H20Cl2N4O2SColore e forma:SolidPeso molecolare:487.4WS 009A
CAS:<p>WS 009A is an antagonist of the endothelin receptor.</p>Formula:C24H25NO10SPurezza:98%Colore e forma:SolidPeso molecolare:519.52ST1936
CAS:<p>ST1936 (ST 1936 oxalate) is a 5-HT6 receptor agonist that stimulates cAMP, Ca2+, ERK1/2, and Fyn kinases by fully activating cloned human 5-HT6 receptors.</p>Formula:C13H17ClN2Purezza:98%Colore e forma:SolidPeso molecolare:236.74CJ 033466
CAS:<p>CJ 033466 is a selective partial agonist of 5-HT4 receptor (EC50 = 9 nM) with gastroprokinetic effect.</p>Formula:C19H28ClN5OPurezza:99.72%Colore e forma:SolidPeso molecolare:377.91Eplivanserin
CAS:Eplivanserin (SR-46349) is an effective and selective antagonist of 5-HT2A receptor with a Kd of 1.14 nM and an IC50 value of 5.8 nM in rat cortical membrane.Formula:C19H21FN2O2Purezza:97.04%Colore e forma:SolidPeso molecolare:328.38DOV-216,303 Free Base
CAS:<p>DOV-216,303 inhibits serotonin, norepinephrine, dopamine reuptake (IC50s: 14, 20, 78 nM) with antidepressant properties.</p>Formula:C11H11Cl2NPurezza:96.7%Colore e forma:SolidPeso molecolare:228.12Chlorazanil
CAS:<p>Chlorazanil is a triazine-based, orally active diuretic that blocks Na+ and Cl– reabsorption in distal tubules, increases renal prostaglandin.</p>Formula:C9H8ClN5Purezza:98.89%Colore e forma:SolidPeso molecolare:221.65Nedocromil
CAS:<p>Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).</p>Formula:C19H17NO7Purezza:95% - 97.34%Colore e forma:SolidPeso molecolare:371.34Quinpirole Hydrochloride
CAS:<p>Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and mice</p>Formula:C13H22ClN3Purezza:98%Colore e forma:SolidPeso molecolare:255.79AM6545
CAS:<p>AM6545 is a CB1 receptor antagonist used in the study of obesity and diabetes.</p>Formula:C26H23Cl2N5O3SPurezza:97.03%Colore e forma:SolidPeso molecolare:556.46Adatanserin
CAS:<p>Adatanserin (WY 50324) is a mixed 5-HT1A receptor partial agonist and a 5-HT2A and 5-HT2C receptor antagonist.</p>Formula:C21H31N5OPurezza:99.33%Colore e forma:SolidPeso molecolare:369.5Aligeron
CAS:<p>Aligeron is a non-selective prostaglandin (PG) antagonist that inhibits PGF2α- and PGE2-induced decreases in blood pressure in cats, and can be used to inhibit</p>Formula:C20H24N2Purezza:99.09% - >99.99%Colore e forma:SolidPeso molecolare:292.42Vapitadine dihydrochloride
CAS:<p>Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.</p>Formula:C17H22Cl2N4OPurezza:98.28% - 99.30%Colore e forma:SolidPeso molecolare:369.29ML179
CAS:<p>ML179 is a potent and selective inverse agonist of liver receptor homolog-1 (LRH1, NR5A2) with IC50 of 320 nM.</p>Formula:C21H25F3N4O2Purezza:99.77%Colore e forma:SolidPeso molecolare:422.44TIK-301
CAS:<p>TIK-301 is a chlorinated melatonin derivative and a potent, high-affinity, and orally active melatonin MT1 and MT2 receptors agonist (Kis: 0.081 nM and 0.042 nM</p>Formula:C14H17ClN2O2Purezza:98%Colore e forma:SolidPeso molecolare:280.75Amgen-23
CAS:<p>Amgen-23 is a selective and highly potent sphingosine kinase 1 (SPHK1) inhibitor that inhibits SPHK2 and can be used in anticancer research.</p>Formula:C23H25Cl2N3O2SPurezza:97.31%Colore e forma:SolidPeso molecolare:478.44SDZ 205-557 hydrochloride
CAS:<p>5-HT3/5-HT4 receptor antagonist</p>Formula:C14H22Cl2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:337.24RS 15385-197
CAS:<p>RS 15385-197 is a selective alpha 2-adrenoceptor antagonist.</p>Formula:C18H26N2O3SColore e forma:SolidPeso molecolare:350.48
