Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(1.025 prodotti)
- Recettore dell'adenosina(249 prodotti)
- Recettore adrenergico(3.030 prodotti)
- Recettore della bombesina(35 prodotti)
- Recettore della bradichinina(61 prodotti)
- CXCR(159 prodotti)
- CaSR(34 prodotti)
- Recettore dei cannabinoidi(217 prodotti)
- Colecistochinina(1 prodotti)
- Recettore della dopamina(444 prodotti)
- Recettore dell'endotelina(86 prodotti)
- Recettore GNRH(84 prodotti)
- GPCR19(33 prodotti)
- GRK(33 prodotti)
- GTPase(22 prodotti)
- Recettore del glucagone(196 prodotti)
- Proteina Hedgehog/Smoothened(49 prodotti)
- Recettore dell'istamina(385 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(26 prodotti)
- Recettore OX(42 prodotti)
- Recettore degli oppioidi(325 prodotti)
- PAFR(14 prodotti)
- PKA(55 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(31 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 19 più sottocategorie
Trovati 5984 prodotti di "Proteina G/GPCR"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
NF-56-EJ40 hydrochloride
CAS:NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 nM; low rat SUCNR1 activity, Ki = 17.4 nM.Formula:C27H31Cl2N3O3Purezza:99.33%Colore e forma:SoildPeso molecolare:516.46Naftopidil
CAS:Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as a selective α1-adrenergic receptor antagonist or α-Formula:C24H28N2O3Purezza:99.60% - 99.97%Colore e forma:White Crystalline PowderPeso molecolare:392.49Apelin-13
CAS:Apelin-13 is a 13-amino acid peptide sequence found in the central and peripheral nervous system that is an endogenous ligand for the G protein-coupled receptorFormula:C69H111N23O16SPurezza:96.81%Colore e forma:SolidPeso molecolare:1550.83Bromopride
CAS:Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.Formula:C14H22BrN3O2Purezza:99.95%Colore e forma:SolidPeso molecolare:344.25Ref: TM-T1175
2mg39,00€5mg58,00€10mg93,00€25mg167,00€50mg260,00€100mg409,00€200mg595,00€1mL*10mM (DMSO)64,00€2',5'-Dideoxyadenosine
CAS:2',5'-Dideoxyadenosine is a potent and non-competitive adenylyl cyclase inhibitor via binding the P-site (IC50: 3 μM).Formula:C10H13N5O2Purezza:99.55%Colore e forma:White SolidPeso molecolare:235.24Ref: TM-T10066
1mg39,00€5mg84,00€10mg119,00€25mg210,00€50mg354,00€100mg562,00€500mg1.225,00€1mL*10mM (DMSO)92,00€Luzindole
CAS:Luzindole (N-0774) is a selective melatonin receptor antagonist.Formula:C19H20N2OPurezza:98.53%Colore e forma:Off-White Amorphous SolidPeso molecolare:292.37Ref: TM-T15795
1mg49,00€2mg66,00€5mg92,00€10mg138,00€25mg245,00€50mg349,00€100mg512,00€200mg730,00€1mL*10mM (DMSO)147,00€Doxofylline
CAS:Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.Formula:C11H14N4O4Purezza:99.958% - >99.99%Colore e forma:SolidPeso molecolare:266.25LCKLSL hydrochloride
LCKLSL hydrochloride is an AnxA2 inhibitor with potential anti-angiogenic activity and inhibits the development of EAE.Formula:C30H58ClN7O8SPurezza:98.02% - 99.31%Colore e forma:SolidPeso molecolare:712.34Midodrine hydrochloride
CAS:<p>Midodrine, metabolized to desglymidodrine, activates alpha-1 receptors, raising blood pressure without CNS effects. It's a prodrug in hydrochloride form.</p>Formula:C12H19ClN2O4Purezza:99.79% - >99.99%Colore e forma:Crystalline SolidPeso molecolare:290.74Droperidol
CAS:Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.Formula:C22H22FN3O2Purezza:97.16% - 98%Colore e forma:SolidPeso molecolare:379.43Triprolidine hydrochloride monohydrate
CAS:Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.Formula:C19H25ClN2OPurezza:99.68% - 99.81%Colore e forma:White Crystalline PowderPeso molecolare:332.87Pizotifen Malate
CAS:Pizotifen Malate (BC-105 malate), a highly selective 5-HT receptor blocking agent, is a drug based on benzocycloheptane.Formula:C19H21NS·C4H6O5Purezza:99.96% - >99.99%Colore e forma:SolidPeso molecolare:429.53Olanzapine
CAS:Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.Formula:C17H20N4SPurezza:99.86% - ≥95%Colore e forma:Yellowish Crystalline PowderPeso molecolare:312.43Labetalol
CAS:Labetalol: mixed alpha/beta blocker for hypertension, oral or IV; affected by CYP2C19 genetics.Formula:C19H24N2O3Purezza:99.87% - 99.89%Colore e forma:SolidPeso molecolare:328.41Lamotrigine
CAS:Lamotrigine (BW430C) is an Anti-epileptic Agent and Mood Stabilizer.Formula:C9H7Cl2N5Purezza:99.76% - 99.95%Colore e forma:White To Pale Cream-Colored Powder Crystals From Isopropanol SolidPeso molecolare:256.09Astemizole
CAS:Astemizole (Laridal) is a long-acting antihistamine for allergies like rhinitis and asthma, with fewer anticholinergic effects.Formula:C28H31FN4OPurezza:98.24% - 99.67%Colore e forma:White Crystals SolidPeso molecolare:458.57GANT 58
CAS:GANT 58 (NSC-75503) is a potent antagonist of Gli. Which inhibits GLI1-induced transcription (IC50: 5 μM).Formula:C24H16N4SPurezza:99.53%Colore e forma:SolidPeso molecolare:392.48SR59230A
CAS:SR59230A is a potent, selective antagonist of β3-adrenergic receptor(β3, β1, and β2 receptors with IC50s of 40, 408, and 648 nM , respectively).Formula:C23H29NO6Purezza:98.84%Colore e forma:SolidPeso molecolare:415.48Ref: TM-T13016
1mg52,00€2mg77,00€5mg107,00€10mg172,00€25mg343,00€50mg510,00€100mg737,00€1mL*10mM (DMSO)125,00€Terbutaline
CAS:Terbutaline is a short-acting agonist of β2-adrenergic receptor (β2-AR) . It is an active metabolite of bambuterolFormula:C12H19NO3Purezza:99.12%Colore e forma:SolidPeso molecolare:225.3Pheniramine maleate
CAS:Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 receptors.Formula:C16H20N2·C4H4O4Purezza:99.85%Colore e forma:Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°CPeso molecolare:356.42Quetiapine hemifumarate
CAS:Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.Formula:C46H54N6O8S2Purezza:99.32% - >99.99%Colore e forma:White Crystalline SolidPeso molecolare:883.09Evatanepag
CAS:<p>Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting fracture healing in rats.</p>Formula:C25H28N2O5SPurezza:97.09%Colore e forma:SolidPeso molecolare:468.57Tropanserin
CAS:Tropanserin (MDL 72422) is a 5-hydroxytryptamine receptor antagonist with anxiolytic activity that is used to treat depression and cognitive impairment.Formula:C17H23NO2Purezza:99.74%Colore e forma:SolidPeso molecolare:273.37Fezolinetant
CAS:Fezolinetant (ESN-364) is a neurokinin-3 receptor antagonist that is being investigated for menopausal hot flashes.Cost-effective and quality-assured.Formula:C16H15FN6OSPurezza:98.62% - 99.7%Colore e forma:SolidPeso molecolare:358.39Ref: TM-T15278
1mg75,00€5mg141,00€10mg219,00€25mg439,00€50mg708,00€100mg1.063,00€1mL*10mM (DMSO)156,00€Sarizotan 2HCl
CAS:Sarizotan 2HCl is an hERG channel inhibitor and 5-hydroxytryptamine 5-HT1A receptor agonist with potential antidepressant effects for the study of Parkinsonian movement disorders.Formula:C22H23Cl2FN2OPurezza:98.83%Colore e forma:SoildPeso molecolare:421.34Orphenadrine hydrochloride
CAS:Orphenadrine hydrochloride (Mephenamin) is a muscarinic antagonist used to treat drug-induced parkinsonism and to relieve pain from muscle spasm.Formula:C18H23NO·HClPurezza:99.88%Colore e forma:Liquid About 5 5 Bitter Numbing Taste (Ntp 1992)Peso molecolare:305.85Tabernanthalog fumarate
CAS:Tabernanthalog fumarate is a 5-HT2A agonist that promotes neuronal growth and reduces alcohol consumption in mice, producing antidepressant-like effects.Formula:C18H22N2O5Purezza:99.83%Colore e forma:SoildPeso molecolare:346.38Enrasentan
CAS:Enrasentan (sb-217242) is a mixed antagonist of ET(A) and ET(B) receptors that reduces blood pressure and protects myocardial function.Formula:C29H30O8Purezza:97.9% - 98.39%Colore e forma:SolidPeso molecolare:506.54Quetiapine
CAS:<p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>Formula:C21H25N3O2SPurezza:99.14% - 99.63%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:383.51Xylometazoline hydrochloride
CAS:Xylometazoline hydrochloride (Xylometazoline HCl) is an α-adrenoceptor agonist usually used as nasal decongestant.Formula:C16H24N2·HClPurezza:99.77% - 99.87%Colore e forma:White To Off-White Crystalline PowderPeso molecolare:280.84Promethazine hydrochloride
CAS:Promethazine HCl: First-gen antihistamine, H1 and mACh blocker, affects 5-HT2A/C, D2, α1 receptors.Formula:C17H20N2S·HClPurezza:99.85%Colore e forma:Crystals In Water Has A Ph Of 3 5-5 0 (Ntp 1992)Peso molecolare:320.88Degarelix acetate(214766-78-6 free base)
CAS:Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .Formula:C84H107ClN18O18Purezza:98.66%Colore e forma:SolidPeso molecolare:1692.34Dynarrestin
CAS:Dynarrestin inhibits cytoplasmic dynein 1/2, preventing microtubule sliding without affecting ATP hydrolysis or ciliogenesis.Formula:C22H23F2N3O2SPurezza:99.64%Colore e forma:SolidPeso molecolare:431.5SEP-363856 hydrochloride
CAS:<p>SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.</p>Formula:C9H14ClNOSPurezza:99.86% - 99.99%Colore e forma:SolidPeso molecolare:219.73Ref: TM-T12899L
1mg70,00€2mg92,00€5mg154,00€10mg243,00€25mg425,00€50mg628,00€100mg938,00€500mg1.882,00€Chlorpheniramine maleate
CAS:Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, urticaria, and asthma.Formula:C20H23ClN2O4Purezza:99.64% - 99.98%Colore e forma:Odorless White Crystalline Solid Or White Powder With A Bitter TastePeso molecolare:390.87PF-04995274
CAS:PF-04995274: potent, selective partial 5-HT4R agonist; EC50 0.26-0.47 nM; brain penetrant; may treat Alzheimer's cognitive issues.Formula:C23H32N2O6Purezza:99.52%Colore e forma:SolidPeso molecolare:432.51INCB-9471
CAS:INCB-9471 is a CCR5 antagonist with anti-HIV activity and inhibits the interaction between HIV-1 gp120.Formula:C30H40F3N5O2Purezza:98.80%Colore e forma:SolidPeso molecolare:559.666Ezlopitant
CAS:Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and pain.Formula:C31H38N2OPurezza:97.49%Colore e forma:SolidPeso molecolare:454.65Methoxamine hydrochloride
CAS:Methoxamine hydrochloride (Methoxamine HCl) is an alpha-1 adrenergic agonist that causes prolonged peripheral VASOCONSTRICTION.Formula:C11H18ClNO3Purezza:99.84% - >99.99%Colore e forma:Colorless Or White Plate-Like Crystals Or White Crystalline Powder SolidPeso molecolare:247.719Glycerol phenylbutyrate
CAS:Glycerol phenylbutyrate (HPN-100) (GPB) is a new generation ammonia scavenger drug and it also is a sigma-2 (σ2) receptor ligand (pKi: 8.02).Formula:C33H38O6Purezza:98.54% - 99.74%Colore e forma:SolidPeso molecolare:530.65Phentolamine mesylate
CAS:Phentolamine mesylate: nonselective alpha-blocker for hypertension, pheochromocytoma, Raynaud's, frostbite, impotence, and vascular issues.Formula:C17H19N3O·CH4O3SPurezza:99.87% - >99.99%Colore e forma:By The Metabolic Processes Of Bacillus Subtilis And LicheniformisPeso molecolare:377.46Adenosine A1 receptor activator T62
CAS:Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and alsoFormula:C15H14ClNOSPurezza:97.83%Colore e forma:SolidPeso molecolare:291.8Ref: TM-T14127
1mg67,00€5mg133,00€10mg190,00€25mg306,00€50mg419,00€100mg567,00€200mg752,00€1mL*10mM (DMSO)197,00€Levocetirizine
CAS:Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a Histamine H1 Receptor Antagonist.Formula:C21H25ClN2O3Purezza:98% - 99.94%Colore e forma:White PowderPeso molecolare:388.89Amisulpride
CAS:Amisulpride (Solian/Deniban), a dopamine antagonist antipsychotic, treats psychosis and schizophrenia in Europe/Australia, not in the US.Formula:C17H27N3O4SPurezza:99.97% - 99.99%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:369.486-Iodopravadoline
CAS:6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity more than CB1 receptors.Formula:C23H25IN2O3Purezza:99.29%Colore e forma:Off-White SolidPeso molecolare:504.36Ref: TM-T14204
1mg38,00€2mg52,00€5mg70,00€10mg90,00€25mg198,00€50mg326,00€100mg520,00€1mL*10mM (DMSO)99,00€[Leu15]-Gastrin I, human
CAS:[Leu15]-Gastrin I, human is a variant of Gastrin I, modulating the binding of cholecystokinin to mucosal membranes.Formula:C98H126N20O31Purezza:98.02% - 98.84%Colore e forma:SolidPeso molecolare:2080.16Mifentidine
CAS:Mifentidine (DA 4577) is an orally available H2 receptor antagonist for the study of gastric emptying and experimental gastric and duodenal ulcers.Formula:C13H16N4Purezza:98.34% - 99.73%Colore e forma:SolidPeso molecolare:228.29Carbinoxamine Maleate Salt
CAS:Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and sedative properties.Formula:C20H23ClN2O5Purezza:99.97%Colore e forma:Off-White SolidPeso molecolare:406.86Alosetron hydrochloride
CAS:Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin at 5-HT3 sites in the peripheral nervous system.Formula:C17H19ClN4OPurezza:99.90%Colore e forma:Off-White PowderPeso molecolare:330.81Sergliflozin A
CAS:Sergliflozin A is a selective SGLT2 inhibitor that induces diabetes in a dose-dependent manner. It reduces hyperglycemia.Formula:C20H24O7Purezza:99.71%Colore e forma:SolidPeso molecolare:376.4ALLO-2
CAS:ALLO-2 is a Inhibitor of Drug-Resistant Smo Mutant.It inhibits Smo agonist Hh-Ag1.5-induced luciferase expression in TM3-Gli-Luc cells with IC50 of 6 nM.Formula:C18H12F3N5OPurezza:99.19%Colore e forma:SolidPeso molecolare:371.32Ref: TM-T14188
1mg64,00€5mg140,00€10mg212,00€25mg353,00€50mg500,00€100mg658,00€200mg905,00€1mL*10mM (DMSO)156,00€Desvenlafaxine
CAS:Desvenlafaxine, a venlafaxine metabolite, is an SNRI used as an antidepressant.Formula:C16H25NO2Purezza:99.46% - 99.81%Colore e forma:White Crystalline PowderPeso molecolare:263.38ML-109
CAS:<p>ML-109 is a potent agonist of thyroid stimulating hormone receptor (TSHR) (EC50 of 40 nM)</p>Formula:C31H29N3O5Purezza:98.63%Colore e forma:SolidPeso molecolare:523.58Carbazochrome sodium sulfonate
CAS:Carbazochrome sodium sulfonate (AC-17) (AC-17) is an antihemorrhagic for the treatment of hemorrhoids.Formula:C10H11N4NaO5SPurezza:99.63%Colore e forma:Orange Yellow Crystalline PowderPeso molecolare:322.03Vibozilimod
CAS:Vibozilimod (SCD-044) is S1P receptor-1 (S1PR1) agonist .Formula:C29H36ClN3O5Purezza:99.97%Colore e forma:SolidPeso molecolare:542.07Mirabegron
CAS:Mirabegron (YM178) is a beta-3 adrenergic agonist that is used for treatment of overactive bladder syndrome.Formula:C21H24N4O2SPurezza:99.64%Colore e forma:Light Yellow To Yellow SolidPeso molecolare:396.51EMPA
CAS:EMPA is a selective, high-affinity and reversible antagonist of orexin OX2 receptor(human and rat OX2-HEK293 membranes with KD values of 1.1 and 1.4 nMFormula:C23H26N4O4SPurezza:99.11%Colore e forma:SolidPeso molecolare:454.54Ref: TM-T11186
1mg49,00€2mg69,00€5mg92,00€10mg142,00€25mg250,00€50mg375,00€100mg563,00€200mg795,00€1mL*10mM (DMSO)104,00€Erenumab
CAS:Erenumab: human antibody blocking CGRP receptors to prevent migraines.Purezza:99.43% (SEC-HPLC) - > 95%Colore e forma:LiquidPeso molecolare:146.2 kDaN6-Ethyladenosine
CAS:N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).Formula:C12H17N5O4Purezza:99.96%Colore e forma:SolidPeso molecolare:295.29Fluphenazine dihydrochloride
CAS:Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used to probe effects and metabolic process.Formula:C22H28Cl2F3N3OSPurezza:99.23%Colore e forma:Off-White SolidPeso molecolare:510.44Labetalol hydrochloride
CAS:Labetalol hydrochloride (Sch-15719W), a salicylamide derivative, is a non-cardioselective blocker of β-adrenergic receptors and α1-adrenergic receptors.Formula:C19H25ClN2O3Purezza:99.54% - 99.85%Colore e forma:SolidPeso molecolare:364.87Ethamsylate
CAS:Ethamsylate (Dicynene) 通常用作止血药，增加毛细血管内皮阻力和血小板粘附，抑制前列腺素的生物合成和作用。Formula:C10H17NO5SPurezza:98.55%Colore e forma:White Crystals Or Crystalline PowderPeso molecolare:263.31Urapidil hydrochloride
CAS:Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.Formula:C20H29N5O3·HClPurezza:99.58%Colore e forma:White Or Off-White Crystalline PowderPeso molecolare:423.94Orforglipron
CAS:Orforglipron (LY3502970; GLP-1 receptor agonist 1) is an orally available glucagon-like peptide (GLP-1) receptor agonist for the study of obesity and type 1Formula:C48H48F2N10O5Purezza:99.47% - 99.8%Colore e forma:SolidPeso molecolare:882.96Ref: TM-T11408
1mg57,00€5mg120,00€10mg187,00€25mg354,00€50mg494,00€100mg692,00€200mg1.026,00€1mL*10mM (DMSO)47,00€Fosopamine(HCl)
CAS:Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.Formula:C9H15ClNO5PPurezza:99.84%Colore e forma:SolidPeso molecolare:283.65Iloperidone
CAS:Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.Formula:C24H27FN2O4Purezza:99.42%Colore e forma:SolidPeso molecolare:426.48(S)-(-)-Atenolol
CAS:(S)-(-)-Atenolol has beta-adrenergic blocking effects.Formula:C14H22N2O3Purezza:99.31% - 99.81%Colore e forma:SolidPeso molecolare:266.34Avexitide acetate
CAS:Avexitide acetate (exendin 9-39) is a potent glucagon-like peptide 1 receptor (GLP-1R) antagonist for the study of post-obesity hypoglycemia.Formula:C155H246N40O53SPurezza:96.64% - 98.65%Colore e forma:SolidPeso molecolare:3549.91Ranitidine Hydrochloride
CAS:Ranitidine Hydrochloride (AH19065) is a competitive and reversible inhibitor of histamine H2-receptor antagonists with antacid activity.Formula:C13H23ClN4O3SPurezza:99.30% - 99.49%Colore e forma:SolidPeso molecolare:350.86Aripiprazole Lauroxil
CAS:Aripiprazole lauroxil, the N-acyloxymethyl prodrug form of aripiprazole, a long-acting injectable (LAI) antipsychotic.Formula:C36H51Cl2N3O4Purezza:99.64%Colore e forma:SolidPeso molecolare:660.71Ref: TM-T14319
10mg48,00€25mg72,00€50mg96,00€100mg130,00€200mg188,00€500mg318,00€1mL*10mM (DMSO)49,00€CB1 antagonist 2
CAS:CB1 antagonist 2 (AM4113) is caimabinoid 1 (CB1) antagonist which inhibits CB1 in vivo with an IC50 of 25.5 nM.Formula:C17H12Cl3N3OPurezza:99.75%Colore e forma:SolidPeso molecolare:380.66BIBO3304 TFA
CAS:BIBO3304 TFA: Oral, selective NPY Y1 receptor blocker; IC50: 0.38 nM (human), 0.72 nM (rat).Formula:C31H36F3N7O5Purezza:99.5%Colore e forma:SolidPeso molecolare:643.66Ref: TM-T10539
1mg63,00€5mg137,00€10mg243,00€25mg550,00€50mg757,00€100mg1.018,00€1mL*10mM (DMSO)187,00€Evocalcet
CAS:Evocalcet (KHK7580) has an activating effect on the calcium-sensing receptor (CaSR).Formula:C24H26N2O2Purezza:98.88% - 99.68%Colore e forma:SolidPeso molecolare:374.48Atomoxetine hydrochloride
CAS:Atomoxetine HCl (LY 139603) is a selective non-stimulant ADHD drug that blocks norepinephrine reuptake, enhancing focus and reducing impulsivity.Formula:C17H22ClNOPurezza:99.86%Colore e forma:White SolidPeso molecolare:291.82Cericlamine
CAS:Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.Formula:C12H17Cl2NOPurezza:99.06%Colore e forma:SolidPeso molecolare:262.18Itopride hydrochloride
CAS:Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.Formula:C20H27ClN2O4Purezza:99.59%Colore e forma:White Or Pale Brownish CrystalPeso molecolare:394.9Dipivefrin hydrochloride
CAS:Dipivefrin hydrochloride (Dipivefrin HCl) that is available as an ophthalmic solution is a prodrug of adrenaline, which is used to treat glaucoma.Formula:C19H27NO5·HClPurezza:99.22% - 99.92%Colore e forma:Less Gas With A Sweet Odor Colorless Gas With A Sweet OdorPeso molecolare:387.9Mirtazapine
CAS:Mirtazapine is a unique tetracyclic antidepressant, may cause temporary liver enzyme elevation, and is linked to rare liver injury.Formula:C17H19N3Purezza:99.98%Colore e forma:SolidPeso molecolare:265.35DF-1012 FA
DF-1012 FA is a structural analog of DF-1012, a neuropeptide inhibitor used in the study of asthma and cough.Formula:C17H22N4O3Purezza:99.15% - 99.97%Colore e forma:SolidPeso molecolare:330.382L-741626
CAS:L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3Formula:C20H21ClN2OPurezza:98.57%Colore e forma:SolidPeso molecolare:340.85Azasetron hydrochloride
CAS:Azasetron hydrochloride (Y-25130 HCl) is a 5-HT3 receptor antagonist which is used as an anti-emetic.Formula:C17H20ClN3O3·HClPurezza:99.50%Colore e forma:SolidPeso molecolare:386.27Ebalzotan
CAS:NAE-086 is a high-affinity and selective 5-HT(1A) receptor ligand with a K(i) value of 4.5 nM in membranes from rat hippocampus.Formula:C19H30N2O2Purezza:98.09% - 99.41%Colore e forma:SolidPeso molecolare:318.45Buflomedil hydrochloride
CAS:Buflomedil hydrochloride (Fonzylane), a vasodilator, is used in therapy of claudication or the symptoms of the peripheral arterial disease.Formula:C17H26ClNO4Purezza:99.7% - 99.91%Colore e forma:White Or Off-White Crystalline PowderPeso molecolare:343.85Bufotenidine hydrochloride(487-91-2 Free base)
CAS:Bufotenidine hydrochloride(487-91-2 Free base) is a natural product for research related to life sciences.Formula:C13H19ClN2OPurezza:99.88%Colore e forma:SolidPeso molecolare:254.76Ciliobrevin D
CAS:Ciliobrevin D is a AAA+ ATPase motor cytoplasmic dynein inhibitor.Formula:C17H8Cl3N3O2Purezza:98.09%Colore e forma:SolidPeso molecolare:392.62Ref: TM-T14965
1mg60,00€2mg87,00€5mg133,00€10mg203,00€25mg401,00€50mg592,00€100mg827,00€1mL*10mM (DMSO)148,00€Bambuterol hydrochloride
CAS:Bambuterol hydrochloride (KWD-2183 hydrochloride) , a long-acting beta-adrenoceptor agonist, is utilized for the treating of asthma.Formula:C18H30ClN3O5Purezza:99.53% - 99.61%Colore e forma:White SolidPeso molecolare:403.91Solabegron
CAS:Solabegron (GW 427353) is a selective agonist of β3-adrenergic receptor, stimulating cAMP accumulation in Chinese hamster ovary cells expressing the human β3-ARFormula:C23H23ClN2O3Purezza:97.89%Colore e forma:SolidPeso molecolare:410.89Ref: TM-T12970
1mg58,00€5mg164,00€10mg259,00€25mg472,00€50mg638,00€100mg848,00€200mg1.121,00€1mL*10mM (DMSO)170,00€Loratadine
CAS:<p>Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of allergic rhinitis and urticaria.</p>Formula:C22H23ClN2O2Purezza:99.71% - 99.98%Colore e forma:White PowderPeso molecolare:382.88Isoxsuprine hydrochloride
CAS:Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular smooth muscle.Formula:C18H24ClNO3Purezza:99.38%Colore e forma:Crystals From Water SolidPeso molecolare:337.84Clopidogrel
CAS:Clopidogrel (SR-25990C), a P2Y12 receptor antagonist, decreases platelet aggregation.Formula:C16H16ClNO2SPurezza:98.23% - 98.83%Colore e forma:White PowderPeso molecolare:321.82Retatrutide sodium salt
Retatrutide sodium salt is a glucagon receptor and glucagon-like peptide-1 receptor agonist for the study of type 2 diabetes mellitus.Purezza:99.97%Colore e forma:SoildGLP-1(28-36)amide acetate
GLP-1(28-36)amide acetate inhibits mitochondrial permeability transition with antioxidant, anti-diabetic and cardioprotection activities.Formula:C56H89N15O11Purezza:99.9500%Colore e forma:SolidPeso molecolare:1148.4Ref: TM-T37890L
1mg127,00€5mg249,00€10mg419,00€25mg692,00€50mg938,00€100mg1.320,00€500mg2.642,00€1mL*10mM (DMSO)Prezzo su richiesta2-Furoyl-LIGRLO-amide
CAS:2-Furoyl-LIGRLO-amide TFA is a peptide that acts as a proteinase-activated receptor-2 (PAR2) agonist, and contains a furoyl group addition at its N-terminal.Formula:C36H63N11O8Purezza:98%Colore e forma:SolidPeso molecolare:777.95Glucagon-like peptide 1 (1-37), human TFA
Human Glucagon-like peptide 1 (1-37) TFA is a potent GLP-1 receptor agonist derived from proglucagon.Formula:C188H276N51F3O61Purezza:98%Colore e forma:SolidPeso molecolare:4283.5Secretoneurin, rat
CAS:Secretoneurin, rat, a 33-amino acid polypeptide, is generated by proteolytic processing of secretogranin II (SgII).Formula:C159H252N40O58Purezza:98%Colore e forma:SolidPeso molecolare:3651.95SAG dihydrochloride
CAS:<p>SAG dihydrochloride: potent Smo agonist, activates Hedgehog pathway, counters Cyclopamine. EC50=3 nM, Kd=59 nM.</p>Formula:C28H30Cl3N3OSPurezza:>99.99%Colore e forma:SoildPeso molecolare:562.98L-796,778
CAS:L-796,778 is an SST3 agonist and a selective ligand of SST3, which can increase the level of cAMP in the body.Formula:C29H40N6O7Purezza:99.24%Colore e forma:SolidPeso molecolare:584.66Ref: TM-T32511
1mg175,00€5mg404,00€10mg592,00€25mg888,00€50mg1.243,00€100mg1.701,00€500mg3.402,00€1mL*10mM (DMSO)522,00€p-MPPF
CAS:p-MPPF is a 5-HT antagonist that can be used to study neurological diseases.Formula:C25H27FN4O2Purezza:99.92%Colore e forma:SolidPeso molecolare:434.51Olcegepant hydrochloride
CAS:Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a selective calcitonin gene-related peptide 1 (CGRP1) receptor antagonist.Formula:C38H48Br2ClN9O5Purezza:99.69%Colore e forma:SolidPeso molecolare:906.11Prosaptide TX14(A)
CAS:GPR37L1/GPR37 agonist with EC50 of 5/7 nM, activates G proteins, enhances ERK, myelin synthesis, neuro/glioprotection.Formula:C69H110N16O26Purezza:98%Colore e forma:SolidPeso molecolare:1579.72
![[Leu15]-Gastrin I, human](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT8761.webp&w=3840&q=75)
