Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(1.025 prodotti)
- Recettore dell'adenosina(249 prodotti)
- Recettore adrenergico(3.030 prodotti)
- Recettore della bombesina(35 prodotti)
- Recettore della bradichinina(61 prodotti)
- CXCR(159 prodotti)
- CaSR(34 prodotti)
- Recettore dei cannabinoidi(217 prodotti)
- Colecistochinina(1 prodotti)
- Recettore della dopamina(444 prodotti)
- Recettore dell'endotelina(86 prodotti)
- Recettore GNRH(84 prodotti)
- GPCR19(33 prodotti)
- GRK(33 prodotti)
- GTPase(22 prodotti)
- Recettore del glucagone(196 prodotti)
- Proteina Hedgehog/Smoothened(49 prodotti)
- Recettore dell'istamina(385 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(26 prodotti)
- Recettore OX(42 prodotti)
- Recettore degli oppioidi(325 prodotti)
- PAFR(14 prodotti)
- PKA(55 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(31 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 19 più sottocategorie
Trovati 5984 prodotti di "Proteina G/GPCR"
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Adenosine receptor antagonist 2
CAS:Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.Formula:C23H21FN8OColore e forma:SolidPeso molecolare:444.46JNJ-17156516
CAS:JNJ-17156516 is a potent, and selective cholecystokinin 1 receptor antagonist.Formula:C26H22Cl2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:481.37Bag-1
CAS:Bag-1 is a novel potent, non-peptidic bombesin receptor subtype-3 (BRS-3) agonist.Formula:C22H27N3Colore e forma:SolidPeso molecolare:333.47ABT-546
CAS:ABT-546 is a potent, selective endothelin ETA receptor antagonist, Ki 0.46 nM for [125I]ET-1 binding.Formula:C30H48N2O6Purezza:98%Colore e forma:SolidPeso molecolare:532.71SDZ 205-557 hydrochloride
CAS:5-HT3/5-HT4 receptor antagonistFormula:C14H22Cl2N2O3Purezza:98%Colore e forma:SolidPeso molecolare:337.24Benafentrine dimaleate
CAS:Benafentrine dimaleate is a platelet activating factor receptor (PAFR) antagonists and phosphodiesterase (PDE) 3/4 inhibitors.Formula:C31H35N3O11Purezza:98%Colore e forma:SolidPeso molecolare:625.63Bremazocine
CAS:Bremazocineis a potent opiate kappa-agonist and centrally acting analgesic.Formula:C20H29NO2Purezza:98%Colore e forma:SolidPeso molecolare:315.45L 11204
CAS:L 11204 is an antifertility in vivo. It is an inhibitor of prostaglandin synthesis.Formula:C18H17N3OPurezza:98%Colore e forma:SolidPeso molecolare:291.35Altanserin hydrochloride
CAS:Altanserin hydrochloride is a 5-HT2A receptor antagonist.Formula:C22H23ClFN3O2SPurezza:98%Colore e forma:SolidPeso molecolare:447.95LBP-1
CAS:LBP-1 is a cannabinoid receptor type 1 (CB1) agonist.Formula:C23H29ClN6O3Colore e forma:SolidPeso molecolare:472.97Seproxetine HCl
CAS:Seproxetine HCl, a more active enantiomer of N-desmethyl metabolite fluoxetine, works by selectively inhibiting the serotonin uptake carrier.Formula:C16H17ClF3NOPurezza:98%Colore e forma:SolidPeso molecolare:331.76MRS2395
CAS:MRS2395, a dipivaloyl P2Y12 receptor blocker, inhibits ADP-induced platelet activation with a Ki of 3.6 μM and boosts TRAP-6-triggered dense granule release.Formula:C20H30ClN5O4Colore e forma:SolidPeso molecolare:439.94LP 20 hydrochloride
CAS:ligand of the 5-HT7 receptorFormula:C17H21ClN2OPurezza:98%Colore e forma:SolidPeso molecolare:304.81LY 25648
CAS:LY 25648 is an antagonist of leukotriene B4.Formula:C19H27NO2SColore e forma:SolidPeso molecolare:333.49Asperlicin D
CAS:Asperlicin D is a cholecystokinin antagonist agent.Formula:C25H18N4O2Purezza:98%Colore e forma:SolidPeso molecolare:406.44JTH-601 free base
CAS:JTH-601 free base is an antagonist of alpha 1 adrenergic receptor.Formula:C24H35NO4Purezza:98%Colore e forma:SolidPeso molecolare:401.54Ro 04-6790 dihydrochloride
CAS:Ro 04-6790 dihydrochloride is an effective and selective antagonist of the serotonin 5-HT6 receptor.Formula:C12H18Cl2N6O2SPurezza:98%Colore e forma:SolidPeso molecolare:381.28H-9 dihydrochloride
CAS:H-9 dihydrochloride: Strong PKA inhibitor, curbs 5-HT response and EGF signaling, affects pharyngeal function.Formula:C11H15Cl2N3O2SPurezza:97.3%Colore e forma:SolidPeso molecolare:324.23Felcisetrag
CAS:<p>Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi 9.4) for h5-HT4(c) receptors.</p>Formula:C25H37N5O3Purezza:99.99%Colore e forma:SolidPeso molecolare:455.59FK-453
CAS:FK-453 is a potent antagonist of non-xanthine adenosine A1 receptor with diuretic and renal vasodilatory activity.Formula:C23H25N3O2Purezza:99.44%Colore e forma:SolidPeso molecolare:375.46NGD 94-1
CAS:NGD 94-1 is a D4 receptor antagonist that can be used to study psychiatric disorders such as cognitive impairment.Formula:C18H20N6Purezza:99.61%Colore e forma:SolidPeso molecolare:320.395-HT1A modulator 1
CAS:5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).Formula:C21H25N3O2SPurezza:99.68%Colore e forma:SolidPeso molecolare:383.51LY266097 hydrochloride
CAS:<p>LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.</p>Formula:C21H24Cl2N2O2Purezza:98.58%Colore e forma:SolidPeso molecolare:407.33BMS-470539 dihydrochloride
CAS:BMS-470539 dihydrochloride is a MC-1 R agonist with anti-inflammatory activity.Formula:C32H43Cl2N5O4Purezza:>99.99%Colore e forma:SolidPeso molecolare:632.62Opigolix
CAS:Opigolix is a Gonadotropin-releasing hormone receptor antagonist.Formula:C25H19F3N4O5SPurezza:98.60% - 98.97%Colore e forma:SolidPeso molecolare:544.5cis-Urocanic acid
CAS:cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).Formula:C6H6N2O2Purezza:99.81%Colore e forma:SolidPeso molecolare:138.12L-693,403 maleate
CAS:L-693,403 maleate has analgesic activity.Formula:C24H27NO4Purezza:99.88%Colore e forma:SolidPeso molecolare:393.48Ref: TM-T22899
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€Torbafylline
CAS:Torbafylline is a xanthine-based PDE inhibitor reducing protein breakdown via PDE4/cAMP/EPAC/PI3K/Akt in rats with burns, cancer, or sepsis.Formula:C16H26N4O4Purezza:99.96% - 99.97%Colore e forma:SoildPeso molecolare:338.4Ref: TM-T67965
1mg81,00€5mg172,00€10mg259,00€25mg424,00€50mg583,00€100mg800,00€1mL*10mM (DMSO)178,00€SB-215505
CAS:SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, 5-HT2A - 6.77).Formula:C19H16ClN3OPurezza:98.33%Colore e forma:SolidPeso molecolare:337.8Abt-288
CAS:ABT-288 is a selective and potent H3 antagonist for the treatment of mild to moderate Alzheimer's dementia.Formula:C23H24N4OPurezza:98.17% - 98.49%Colore e forma:SolidPeso molecolare:372.46BMS CCR2 22
CAS:BMS CCR2 22 is a potent and selective antagonist of CCR2 with calcium flux IC50 of 18 nM, chemotaxis IC50 of 1 nM, and binding IC50 of 5.1 nM.Formula:C28H34F3N5O4SPurezza:99.65%Colore e forma:SolidPeso molecolare:593.66Ref: TM-T14688
1mg58,00€5mg116,00€10mg183,00€25mg368,00€50mg562,00€100mg758,00€200mg1.017,00€1mL*10mM (DMSO)156,00€Viloxazine
CAS:Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activityFormula:C13H19NO3Purezza:99.65%Colore e forma:SolidPeso molecolare:237.29Amosulalol
CAS:Amosulalol is a combined alpha and beta adrenoceptor antagonist.Formula:C18H24N2O5SPurezza:99.5%Colore e forma:SolidPeso molecolare:380.46Ref: TM-T30027
1mg185,00€2mg279,00€5mg425,00€10mg625,00€25mg938,00€50mg1.311,00€100mg1.795,00€1mL*10mM (DMSO)454,00€Thonzylamine hydrochloride
CAS:Thonzylamine hydrochloride (Resistab) is an anticholinergic and antihistamine used as an antipruritic.Formula:C16H23ClN4OPurezza:99.67%Colore e forma:White Crystalline PowderPeso molecolare:322.83Upacicalcet
CAS:Upacicalcet (AJT-240) is a calcium mimetic for SHPT in dialysis, reducing PTH by targeting parathyroid receptors.Formula:C11H14ClN3O6SPurezza:99.88%Colore e forma:SolidPeso molecolare:351.76RLX-33
CAS:<p>RLX-33 blocks RXFP3 and relaxin 3 effects, controls food intake in rats, and may help study metabolic syndrome.</p>Formula:C24H19ClN4O4Purezza:99.89%Colore e forma:SolidPeso molecolare:462.89CYM5181
CAS:<p>CYM5181 is related to the body's immune system and can be used to study multiple sclerosis, transplant rejection, and adult respiratory distress syndrome.</p>Formula:C17H17N3O3Purezza:99.51%Colore e forma:SolidPeso molecolare:311.34NCGC00135472
CAS:NCGC00135472: DRV1 agonist with pro-catabolic effects, activates DRV1/GPR32, EC50: 0.37 uM (beta-blocker), 0.05 uM (cAMP), enhances phagocytosis.Formula:C20H14F2N4OPurezza:99.41% - 99.48%Colore e forma:SolidPeso molecolare:364.35Ref: TM-T33613
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€Halopemide
CAS:Halopemide is a potent inhibitor of PLD (IC50 = 220 and 310 nM for human PLD1 and PLD2).Formula:C21H22ClFN4O2Purezza:96.57%Colore e forma:SolidPeso molecolare:416.88Anpirtoline hydrochloride
CAS:Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.Formula:C10H14Cl2N2SPurezza:>99.99% - >99.99%Colore e forma:SolidPeso molecolare:265.20Ancriviroc
CAS:Ancriviroc (SCH-351125) is an orally bioavailable small molecule chemokine receptor CCR5 antagonist.Cost-effective and quality-assured.Formula:C28H37BrN4O3Purezza:99.76% - 99.82%Colore e forma:SolidPeso molecolare:557.533SDZ-62-434
CAS:SDZ-62-434 is a platelet-activating factor inhibitor with antitumor activity and may be used in the study of leukemia.Formula:C23H27Cl2N3Purezza:98.38%Colore e forma:SolidPeso molecolare:416.39GW438014A
CAS:GW438014A 是一种有效且具有选择性的 NPY-Y5 受体拮抗剂。GW438014A 对食物摄入并减少肥胖啮齿动物的体重增加具有抑制作用。Formula:C23H23N3O4SPurezza:99.94%Colore e forma:SolidPeso molecolare:437.51Rilapine
CAS:Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.Formula:C22H20ClN3Purezza:97.76% - 99.20%Colore e forma:SolidPeso molecolare:361.87SCH-336
CAS:<p>SCH-336: potent, selective CB2 agonist (Ki=1.8 nM, EC50=2 nM), orally active, 100x CB2 vs. CB1 preference, reduces leukocyte migration and eosinophilia.</p>Formula:C23H25NO8S3Purezza:95.01%Colore e forma:SolidPeso molecolare:539.64Itriglumide
CAS:Itriglumide, a CCK2 receptor antagonist, is used potentially for the treatment of peptic ulcers, dyspepsia, and gastroesophageal reflux disease (GERD).Formula:C33H38N2O4Purezza:99.95%Colore e forma:SolidPeso molecolare:526.67GR 46611
CAS:GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in studies about the treatment of epilepsy.Formula:C23H27N3O2Purezza:99.75%Colore e forma:SolidPeso molecolare:377.48JZP-361
CAS:JZP-361: selective MAGL inhibitor (IC50 = 46 nM); weaker on FAAH, hABHD6; anti-histamine; for asthma research.Formula:C22H20ClN5OPurezza:99.82%Colore e forma:SolidPeso molecolare:405.88A-437203
CAS:A-437203 (Lu201640), selective D3 antagonist with Ki: D2-71nM, D3-1.6nM, D4-6220nM; based on 1H-pyrimidin-2-one scaffold.Formula:C20H27F3N6OSPurezza:98.80%Colore e forma:SolidPeso molecolare:456.53Ref: TM-T10213
1mg94,00€5mg188,00€10mg264,00€25mg411,00€50mg532,00€100mg740,00€200mg982,00€1mL*10mM (DMSO)215,00€JP1302
CAS:JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, renal issues.Formula:C24H24N4Purezza:99.96%Colore e forma:SolidPeso molecolare:368.47GBR 12783 dihydrochloride
CAS:<p>GBR 12783 dihydrochloride inhibits dopamine uptake in rats/mice; IC50s: 1.8/1.2 nM. Enhances memory, boosts hippocampal acetylcholine.</p>Formula:C28H34Cl2N2OPurezza:98.08%Colore e forma:SolidPeso molecolare:485.49ATC 0175 hydrochloride
CAS:ATC 0175 hydrochloride is an orally active melanocyte concentrating hormone 1 receptor antagonist that is potent and selective.Formula:C23H26ClF2N5OPurezza:99.98%Colore e forma:SolidPeso molecolare:461.93PNU-282987 free base
CAS:<p>PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for nervous system research.</p>Formula:C14H17ClN2OPurezza:99.64%Colore e forma:SolidPeso molecolare:264.75Lecozotan HCl
CAS:<p>Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) tolerance.</p>Formula:C28H30ClN5O3Purezza:99.04%Colore e forma:SolidPeso molecolare:520.02Femoxetine hydrochloride
CAS:Femoxetine hydrochloride is a selective 5-hydroxytryptamine reuptake inhibitor used in the study of migraine, depression and eating disorders.Formula:C20H26ClNO2Purezza:99.63%Colore e forma:SolidPeso molecolare:347.88Terbogrel
CAS:Terbogrel is an antiplatelet drug, blocking thromboxane A2 receptor/synthase. Helps prevent clots.Formula:C23H27N5O2Purezza:98.95%Colore e forma:SolidPeso molecolare:405.49MRS1220
CAS:MRS1220, a selective and potent antagonist for the human A3 adenosine receptor (hA3AR) with a dissociation constant (Ki) of 0.59 nM, exhibits therapeuticFormula:C21H14ClN5O2Purezza:98.43%Colore e forma:SolidPeso molecolare:403.82Ref: TM-T23016
1mg50,00€5mg110,00€10mg168,00€25mg288,00€50mg414,00€100mg583,00€500mgPrezzo su richiestaCYM50374
CAS:CYM50374 inhibits Sphingosine-1-phosphate receptor 4 (S1P4 ) with an IC50 of µM.Formula:C19H19NO3SPurezza:98.35% - 98.96%Colore e forma:SolidPeso molecolare:341.42Ref: TM-T27106
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€BP14979
CAS:BP14979 is D3R-selective partial agonist.Formula:C23H34N4O2Purezza:98.29% - 99.73%Colore e forma:SolidPeso molecolare:398.54Crinecerfont
CAS:Crinecerfont (SSR-125543) is a CRF1 antagonist, useful in congenital adrenal hyperplasia research.Formula:C27H28ClFN2OSPurezza:97.79% - 98.55%Colore e forma:SolidPeso molecolare:483.04Bedoradrine
CAS:Bedoradrine (MN-221) free base is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.Formula:C24H32N2O5Purezza:>99.99%Colore e forma:SolidPeso molecolare:428.52YIL 781
CAS:YIL 781 is a selective ghrelin receptor antagonist (GHS-R1a) (Ki = 17 nM), showing a weak affinity for kinesin receptors (K = 6 μM).Formula:C24H28FN3O2Purezza:98.8%Colore e forma:SolidPeso molecolare:409.5PD 168568 dihydrochloride
CAS:PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).Formula:C22H29Cl2N3OPurezza:99.71%Colore e forma:SolidPeso molecolare:422.39Ref: TM-T12383
5mg48,00€10mg58,00€25mg117,00€50mg170,00€100mg248,00€200mg348,00€1mL*10mM (DMSO)60,00€GS-9667
CAS:GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective therapy for Type 2 diabetes (T2DM) and dyslipidemia viaFormula:C21H24FN5O4SPurezza:99.77% - 99.96%Colore e forma:SolidPeso molecolare:461.51U 99194 maleate
CAS:U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice.Formula:C21H31NO6Purezza:99.45%Colore e forma:SolidPeso molecolare:393.47Edonentan
CAS:Edonentan is A potent endothelin A (ETA) receptor antagonist that can be used to study heart failure.Formula:C28H32N4O5SPurezza:98.07% - 99.6%Colore e forma:SolidPeso molecolare:536.64Besipirdine
CAS:Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic activity and cardiovascular activity.Formula:C16H17N3Purezza:97.15% - 98.85%Colore e forma:SolidPeso molecolare:251.33Butofilolol
CAS:Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.Formula:C17H26FNO3Purezza:98.96% - >99.99%Colore e forma:SolidPeso molecolare:311.392CCG 203769
CAS:CCG 203769 (Thiadiazolidinone (TDZD) deriv. 6) is a selective inhibitor of RGS4 with an IC50 of 17 nM for the RGS4-Gαo protein-protein interaction.Formula:C8H14N2O2SPurezza:99.88%Colore e forma:SolidPeso molecolare:202.27Ref: TM-T10705
1mg88,00€5mg187,00€10mg264,00€25mg469,00€50mg657,00€100mg944,00€500mg1.882,00€1mL*10mM (DMSO)207,00€48740 RP
CAS:48740 RP (RP 55779) is an antagonist of platelet-activating factor.Formula:C12H11N3OSPurezza:99.79%Colore e forma:SolidPeso molecolare:245.3Ref: TM-T10159
1mg356,00€5mg567,00€10mg907,00€25mg1.339,00€50mg1.815,00€100mg2.432,00€1mL*10mM (DMSO)567,00€TC LPA5 4
CAS:TC LPA5 4 is a LPA5 receptor antagonist.Formula:C23H23ClN2O3Purezza:99.93%Colore e forma:SolidPeso molecolare:410.89Ref: TM-T23438
1mg49,00€5mg98,00€10mg157,00€25mg324,00€50mg485,00€100mg713,00€200mg982,00€1mL*10mM (DMSO)107,00€KI-7
CAS:KI-7 is an adenosine A2B receptor positive allosteric modulator.Formula:C23H18N2O2Purezza:98.33%Colore e forma:SolidPeso molecolare:354.4Ref: TM-T9238
2mg35,00€5mg55,00€10mg95,00€25mg172,00€50mg264,00€100mg399,00€200mg560,00€1mL*10mM (DMSO)62,00€GSK299115A
CAS:GSK299115A (GSK-299115A) is a selective ROCK1 Inhibitor. GSK299115A exhibits IC50 of 8nM, 620nM, 560nM for ROCK1, RSK1, p70S6K, respectively.Formula:C20H16Cl2N4O2Purezza:99.81%Colore e forma:SolidPeso molecolare:415.27Ref: TM-T27471
1mg319,00€5mg772,00€10mg1.074,00€25mg1.596,00€50mg2.147,00€100mg2.822,00€1mL*10mM (DMSO)945,00€BMS 182874
CAS:BMS 182874: Oral ETA antagonist, IC50=0.150 μM, Ki=0.055 μM, lowers hypertension in rats.Formula:C17H19N3O3SPurezza:99.73%Colore e forma:SolidPeso molecolare:345.42Adoprazine
CAS:<p>Adoprazine (SLV313) is a potential atypical antipsychotic bearing potent D2 receptor antagonist and 5-HT1A receptor agonist properties.</p>Formula:C24H24FN3O2Purezza:99.83%Colore e forma:SolidPeso molecolare:405.46Rocepafant
CAS:Rocepafant (LAU8080), a PAF antagonist, reduces neonatal rat brain damage and inhibits TNF-α toxicity in L929 cells.Formula:C26H23ClN6OS2Purezza:97.31% - 98.95%Colore e forma:SolidPeso molecolare:535.08PSB-16133 sodium
CAS:PSB-16133 sodium is a selective P2Y purine receptor variant antagonist with an IC of 233 nM.Formula:C28H21N2NaO5S2Purezza:98.03% - 98.93%Colore e forma:SolidPeso molecolare:552.60Spizofurone
CAS:Spizofurone (Espizofurona) has anti-ulcer activity, protective effect on the gastric mucosa of rats and can increase alkaline secretion.Formula:C12H10O3Purezza:>99.99%Colore e forma:SolidPeso molecolare:202.212'-MeCCPA
CAS:2'-MeCCPA is an A1AR agonist that inhibits trichothecene-stimulated adenylate cyclase activity and has analgesic activity for the study of HCV.Formula:C16H22ClN5O4Purezza:99.93%Colore e forma:SolidPeso molecolare:383.83Midaglizole hydrochloride
CAS:Midaglizole hydrochloride (DG5128) is an α2-adrenoceptor antagonist with 7.4x more affinity than α1-adrenoceptors (pKi=6.28).Formula:C16H19Cl2N3Purezza:99.39% - 99.82%Colore e forma:SolidPeso molecolare:324.25Ref: TM-T11015
1mg57,00€5mg126,00€10mg198,00€25mg324,00€50mg439,00€100mg562,00€200mg743,00€1mL*10mM (DMSO)160,00€Antalarmin hydrochloride
CAS:Antalarmin hydrochloride, a CRF1 antagonist, offers anti-inflammatory benefits and prevents stress ulcers in IBS.Formula:C24H35ClN4Purezza:99.84% - 99.85%Colore e forma:SolidPeso molecolare:415.02KSK68
CAS:KSK68 is a sigma-1 and histamine H3 receptor antagonist with analgesic activity, inhibits H3 receptors and can be used to study pain.Formula:C23H28N2O2Purezza:99.11%Colore e forma:SolidPeso molecolare:364.48SB-209670
CAS:SB-209670 is a selective endothelin receptor antagonist that inhibits the activity of ET(B) receptors in rat vascular endothelium and vascular smooth muscle.Formula:C29H28O9Purezza:98.29% - 99.40%Colore e forma:SolidPeso molecolare:520.53Ref: TM-T34541
1mg333,00€5mg787,00€10mg1.074,00€25mg1.510,00€50mg1.882,00€100mg2.375,00€500mg4.655,00€1mL*10mM (DMSO)797,00€(S)-(+)-Niguldipine hydrochloride
CAS:(S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.Formula:C36H40ClN3O6Purezza:98.27%Colore e forma:SolidPeso molecolare:646.17TASP0390325
CAS:<p>TASP0390325, a potent and orally active V1B receptor antagonist, has antidepressant and anxiolytic activities in rodents.</p>Formula:C25H30Cl2FN5O4Purezza:98.62%Colore e forma:SolidPeso molecolare:554.44RS 67333 hydrochloride
CAS:RS 67333 hydrochloride is a selective 5-HT4R partial agonist (pKi=8.7) with neuroprotective properties for Alzheimer's research.Formula:C19H30Cl2N2O2Purezza:98.78%Colore e forma:SolidPeso molecolare:389.36CB1 agonist 1
CAS:CB1 agonist 1 is a potent CB1 agonist with a pIC50 value of 5.7 for CB1 receptors.CB1 agonist 1 can be used to study brain disorders, pain, and inflammation.Formula:C24H24N2O5SPurezza:98.56%Colore e forma:SolidPeso molecolare:452.52AZ-1355
CAS:AZ-1355 is a novel dibenzoxepine derivative with lipid-lowering properties.Formula:C17H17NO4Purezza:99.81%Colore e forma:SolidPeso molecolare:299.32Ref: TM-T13563
1mg78,00€5mg170,00€10mg224,00€25mg338,00€50mg460,00€100mg600,00€200mg820,00€1mL*10mM (DMSO)156,00€Seridopidine
CAS:Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy for schizophrenia, Parkinson's disease, and Tourette's syndrome.Formula:C14H20FNO2SPurezza:99.77%Colore e forma:SolidPeso molecolare:285.38Pitolisant
CAS:Pitolisant is a potent and selective nonimidazole inverse agonist that acts on the recombinant human histamine H3 receptor with Ki of 0.16 nM.Formula:C17H26ClNOPurezza:99.84%Colore e forma:SolidPeso molecolare:295.85Ref: TM-T60636
5mg48,00€10mg70,00€25mg120,00€50mg188,00€100mg311,00€500mg747,00€1mL*10mM (DMSO)52,00€5-HT2 antagonist 1
CAS:5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.Formula:C22H29FN4O2Purezza:99.76%Colore e forma:SolidPeso molecolare:400.49Ref: TM-T12597
1mg678,00€5mg1.359,00€10mg1.833,00€25mg2.727,00€50mg3.676,00€100mg4.969,00€1mL*10mM (DMSO)1.605,00€CP 316311
CAS:CP 316311 is a specific CRF1 receptor antagonist with potential antidepressant activity and may be used in the study of depression.Formula:C21H29NO2Purezza:99.71% - >99.99%Colore e forma:SolidPeso molecolare:327.46Imiloxan
CAS:Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive disorder.Formula:C14H16N2O2Purezza:98.13% - 99.8%Colore e forma:SolidPeso molecolare:244.29CCR1 antagonist 6
CAS:<p>CCR1 antagonist 6 is a CCR1 antagonist (IC50: 3 nM).</p>Formula:C21H23ClN4O3SPurezza:99.02% - 99.15%Colore e forma:SolidPeso molecolare:446.95SMO-IN-2
CAS:SMO-IN-2 is a SMO inhibitor with antiproliferative activity and anticancer activity and inhibits Hh signaling.SMO-IN-2 can be used in the study of cancer.Formula:C25H25F4N5O2Purezza:98.64%Colore e forma:SolidPeso molecolare:503.49Ticolubant
CAS:Ticolubant: Oral LTB4 antagonist, Ki=0.78 nM; blocks Ca2+ migration, IC50=6.6 nM; anti-inflammatory in mice.Formula:C23H19Cl2NO3SPurezza:99.5%Colore e forma:SolidPeso molecolare:460.37MK-0686
CAS:MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.Formula:C22H19ClF4N2O4Purezza:99.88%Colore e forma:SolidPeso molecolare:486.84Linetastine
CAS:Linetastine (TMK-688) inhibits 5-LOX, blocks leukotrienes, counters histamine; researched for asthma, atherosclerosis, ulcers.Formula:C35H40N2O6Purezza:99.99%Colore e forma:SolidPeso molecolare:584.7Ordopidine
CAS:<p>Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during inactivity.</p>Formula:C14H20FNO2SPurezza:99.39%Colore e forma:SolidPeso molecolare:285.38L 651896
CAS:L 651896 is an inhibitor of 5-lipoxygenase.Formula:C18H18O3Purezza:96.06% - 99.85%Colore e forma:SolidPeso molecolare:282.33
