Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(1.003 prodotti)
- Recettore dell'adenosina(247 prodotti)
- Recettore adrenergico(3.010 prodotti)
- Recettore della bombesina(33 prodotti)
- Recettore della bradichinina(60 prodotti)
- CXCR(153 prodotti)
- CaSR(33 prodotti)
- Recettore dei cannabinoidi(215 prodotti)
- Colecistochinina(1 prodotti)
- Recettore della dopamina(435 prodotti)
- Recettore dell'endotelina(83 prodotti)
- Recettore GNRH(82 prodotti)
- GPCR19(33 prodotti)
- GRK(32 prodotti)
- GTPase(22 prodotti)
- Recettore del glucagone(190 prodotti)
- Proteina Hedgehog/Smoothened(48 prodotti)
- Recettore dell'istamina(381 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(26 prodotti)
- Recettore OX(41 prodotti)
- Recettore degli oppioidi(321 prodotti)
- PAFR(13 prodotti)
- PKA(51 prodotti)
- Recettore S1P(18 prodotti)
- SGLT(31 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 19 più sottocategorie
Trovati 5838 prodotti di "Proteina G/GPCR"
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SLF1081851
CAS:<p>SLF1081851 is a Spns2 inhibitor. SLF1081851 inhibits S1P release with IC50 of 1.93 μM.</p>Formula:C21H33N3OPurezza:99.26%Colore e forma:SolidPeso molecolare:343.51Viloxazine
CAS:<p>Viloxazine (Viloxazin) (Viloxazin) is a dual-action compound that functions as a norepinephrine reuptake inhibitor and exhibits potent agonistic activity</p>Formula:C13H19NO3Purezza:99.67%Colore e forma:SolidPeso molecolare:237.29N-[(4-Aminophenyl)methyl]adenosine
CAS:N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).Formula:C17H20N6O4Purezza:98.75%Colore e forma:SolidPeso molecolare:372.38Fipamezole
CAS:Fipamezole is a potent alpha2 adrenergic receptor antagonist that may be useful for studying autonomic dysfunction in Parkinson's disease.Formula:C14H15FN2Purezza:99.32% - 99.97%Colore e forma:SolidPeso molecolare:230.28Dimethindene
CAS:Dimethindene (Dimetindeno) is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits antihistamine and anticholinergic effects.Formula:C20H24N2Purezza:98.3% - 98.99%Colore e forma:SolidPeso molecolare:292.42Bedoradrine sulfate
CAS:<p>Bedoradrine sulfate (MN-221 sulfate) is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.</p>Formula:C24H32N2O5H2O4SPurezza:99.31%Colore e forma:SolidPeso molecolare:477.56GR 46611
CAS:GR 46611 is a selective 5-HT1B and 5-HT1D receptor agonist and can be used in studies about the treatment of epilepsy.Formula:C23H27N3O2Purezza:99.75%Colore e forma:SolidPeso molecolare:377.48Ticalopride
CAS:Ticalopride: 5-HT3 agonist for digestive, orofacial, ENT disorders, and bulimia, GERD, IBS research.Formula:C14H20ClN3O3Purezza:99.51%Colore e forma:SolidPeso molecolare:313.78N 0861
CAS:N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled hypotension in rats.Formula:C13H17N5Purezza:98.78%Colore e forma:SolidPeso molecolare:243.31Ronacaleret HCl
CAS:Ronacaleret HCl (SB-751689) is a small molecule CaSR antagonist for the treatment of endocrine and metabolic diseases, skin and musculoskeletal disorders.Formula:C25H32ClF2NO4Purezza:99.97%Colore e forma:SolidPeso molecolare:483.98Regrelor disodium
CAS:Regrelor disodium (INS 50589) is a p2y12 receptor antagonist that prevents thrombosis, effectively inhibits vascular smooth muscle cell contraction, inhibitsFormula:C22H23N6Na2O8PPurezza:99.89%Colore e forma:SolidPeso molecolare:576.41Ensaculin
CAS:<p>Ensaculin, a benzopyrone-piperazine compound, enhances memory, protects neurons, and may treat dementia.</p>Formula:C26H32N2O5Purezza:99.17% - 99.67%Colore e forma:SolidPeso molecolare:452.54cis-Urocanic acid
CAS:cis-Urocanic acid ((E)-Urocanic acid) is a 5-HT2A receptor agonist (Kd: 4.6 nM).Formula:C6H6N2O2Purezza:99.81%Colore e forma:SolidPeso molecolare:138.12UNC0006
CAS:<p>UNC0006 is a β-arrestin-biased dopamine D2 ligand.</p>Formula:C24H29Cl2N3O2Purezza:99.35% - 99.97%Colore e forma:SolidPeso molecolare:462.41SK609 HCl
CAS:<p>SK609 HCl is a selective dopamine D3 receptor agonist. It also has atypical signaling properties.</p>Formula:C10H15Cl2NPurezza:99.02%Colore e forma:SolidPeso molecolare:220.14Cyamemazine
CAS:Cyamemazine is an antipsychotic compound with sedative and anxiolytic activity.Cyamemazine is a 5-HT3, 5-HT2A, and 5-HT2C receptor antagonist.Formula:C19H21N3SPurezza:97.01%Colore e forma:SolidPeso molecolare:323.46AS-35
CAS:AS-35, an oral selective leukotriene antagonist, counters ileum contractions with IC50: 8 nM (LTC4), 4 nM (LTD4), 3 nM (LTE4); shows antiallergic effects.Formula:C21H20N6O4Purezza:96.69%Colore e forma:SolidPeso molecolare:420.42LY 272015 hydrochloride
CAS:LY 272015 hydrochloride is a 5-HT2B receptor antagonist.Formula:C21H25ClN2O2Purezza:99.47%Colore e forma:SolidPeso molecolare:372.89Runcaciguat
CAS:Runcaciguat, a soluble guanylate cyclase stimulator, aids in cardiovascular and renal research.Formula:C23H22Cl2F3NO3Purezza:99.17%Colore e forma:SolidPeso molecolare:488.33CCR2 antagonist 5
CAS:JNJ-41443532: oral hCCR2 antagonist, IC50=37 nM, anti-chemotaxis, treats inflammation & diabetes.Formula:C22H25F3N4O3SPurezza:99.98%Colore e forma:SolidPeso molecolare:482.52PSB-16133 sodium
CAS:<p>PSB-16133 sodium is a selective P2Y purine receptor variant antagonist with an IC of 233 nM.</p>Formula:C28H21N2NaO5S2Purezza:98.03% - 98.93%Colore e forma:SolidPeso molecolare:552.60Sarizotan HCl
CAS:Sarizotan HCl (EMD 128130 HCl) is a 5-HT1A receptor and dopamine receptor agonist and an hERG channel inhibitor used in Parkinson;s disease research.Formula:C22H22ClFN2OPurezza:96%Colore e forma:SolidPeso molecolare:384.87Ex26
CAS:<p>Ex26 (S1P1-IN-Ex26) is an S1P1 antagonist used in experimental autoimmune encephalomyelitis, atherosclerosis, and gastric cancer.</p>Formula:C28H28ClFN2O3Purezza:99.62%Colore e forma:SolidPeso molecolare:494.99Pavinetant
CAS:Pavinetant (MLE-4901) is an orally available neurokinin-3 receptor (NK3R) antagonist used to improve menopausal symptoms.Formula:C26H25N3O3SPurezza:99.8%Colore e forma:SolidPeso molecolare:459.56CP 316311
CAS:CP 316311 is a specific CRF1 receptor antagonist with potential antidepressant activity and may be used in the study of depression.Formula:C21H29NO2Purezza:99.71% - >99.99%Colore e forma:SolidPeso molecolare:327.46Rilapine
CAS:<p>Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can be used to study neurological disorders.</p>Formula:C22H20ClN3Purezza:97.76% - 99.20%Colore e forma:SolidPeso molecolare:361.87Anpirtoline hydrochloride
CAS:<p>Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in the study of dyskinesia.</p>Formula:C10H14Cl2N2SPurezza:>99.99% - >99.99%Colore e forma:SolidPeso molecolare:265.20(S)-(+)-Niguldipine hydrochloride
CAS:(S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.Formula:C36H40ClN3O6Purezza:98.27%Colore e forma:SolidPeso molecolare:646.17PD 168568 dihydrochloride
CAS:<p>PD 168568 dihydrochloride (PD 168568 (dihydrochloride)) is an orally active and selective antagonist of D4 dopamine receptor(Ki of 8.8 nM).</p>Formula:C22H29Cl2N3OPurezza:99.71%Colore e forma:SolidPeso molecolare:422.39Ancriviroc
CAS:Ancriviroc (SCH-351125) is an orally bioavailable small molecule chemokine receptor CCR5 antagonist.Cost-effective and quality-assured.Formula:C28H37BrN4O3Purezza:99.76% - 99.82%Colore e forma:SolidPeso molecolare:557.533Tedatioxetine
CAS:Tedatioxetine (Lu AA24530) is a serotonin-norepinephrine-dopamine reuptake inhibitor (SNDRI) with antidepressant properties.Formula:C18H21NSPurezza:99.76% - >99.99%Colore e forma:SolidPeso molecolare:283.43SR144528
CAS:<p>SR144528 is an antagonist of the CB2 receptor (Ki = 0.6 nM) and inhibits microsomal ACAT activity (IC50 = 3.6 μM).</p>Formula:C29H34ClN3OPurezza:99.63%Colore e forma:SolidPeso molecolare:476.05GSK2239633A
CAS:GSK2239633A is an allosteric antagonist of CC-chemokine receptor 4 (CCR4) with a pIC50 of 7.96 for the binding of [125I]-TARC to human CCR4.Formula:C24H25ClN4O5S2Purezza:99.82%Colore e forma:SolidPeso molecolare:549.06ReN-1869
CAS:ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity for the study of neurological diseasesFormula:C24H27NO2Purezza:99.83% - 99.98%Colore e forma:SolidPeso molecolare:361.48CGRP antagonist 1
CAS:CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for theFormula:C29H26N4O4Purezza:99.55%Colore e forma:SolidPeso molecolare:494.54Bedoradrine
CAS:Bedoradrine (MN-221) free base is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.Formula:C24H32N2O5Purezza:>99.99%Colore e forma:SolidPeso molecolare:428.52BMS-470539 dihydrochloride
CAS:BMS-470539 dihydrochloride is a MC-1 R agonist with anti-inflammatory activity.Formula:C32H43Cl2N5O4Purezza:>99.99%Colore e forma:SolidPeso molecolare:632.62Thonzylamine hydrochloride
CAS:Thonzylamine hydrochloride (Resistab) is an anticholinergic and antihistamine used as an antipruritic.Formula:C16H23ClN4OPurezza:99.67%Colore e forma:White Crystalline PowderPeso molecolare:322.83Opigolix
CAS:Opigolix is a Gonadotropin-releasing hormone receptor antagonist.Formula:C25H19F3N4O5SPurezza:98.60% - 98.97%Colore e forma:SolidPeso molecolare:544.5Butofilolol
CAS:<p>Butofilolol is a novel beta-blocker with antihypertensive activity and can be used to study hypertension.</p>Formula:C17H26FNO3Purezza:98.96% - >99.99%Colore e forma:SolidPeso molecolare:311.392Perphenazine dihydrochloride
CAS:Perphenazine dihydrochloride: Oral dopamine, histamine-1 antagonist; targets D2, D3, 5-HT2A, Alpha-1A; may treat psychiatric disorders, cancer.Formula:C21H28Cl3N3OSPurezza:99.67%Colore e forma:SolidPeso molecolare:476.89Ecastolol
CAS:Ecastolol has anti-angina activity and is an adrenergic receptor antagonist.Formula:C26H33N3O6Purezza:99.89%Colore e forma:SolidPeso molecolare:483.56Bavisant
CAS:Bavisant (JNJ-31001074) is a selective and orally active Human H3 receptor antagonist.Formula:C19H27N3O2Purezza:99.21% - 99.65%Colore e forma:SolidPeso molecolare:329.44SCH-336
CAS:<p>SCH-336: potent, selective CB2 agonist (Ki=1.8 nM, EC50=2 nM), orally active, 100x CB2 vs. CB1 preference, reduces leukocyte migration and eosinophilia.</p>Formula:C23H25NO8S3Purezza:95.01%Colore e forma:SolidPeso molecolare:539.64Nexopamil
CAS:<p>Nexopamil (LU-49938) is a dual calcium channel and 5-HT2A receptor antagonist that inhibits cell contraction and growth.</p>Formula:C24H40N2O3Purezza:97.87% - >99.99%Colore e forma:SolidPeso molecolare:404.59SB-277011
CAS:<p>SB-277011A: dopamine D3 antagonist, pKi 8.0 (D3), 6.0 (D2), 5.0 (5-HT1D), <5.2 (5-HT1B).</p>Formula:C28H30N4OPurezza:99.39%Colore e forma:SolidPeso molecolare:438.56N6-(2-Phenylethyl)adenosine
CAS:<p>N6-(2-Phenylethyl)adenosine (N6-Phenethyladenosine) is an adenosine derivative and an agonist of adenosine receptors with Ki values of 11.8 nM and 30.1 nM for</p>Formula:C18H21N5O4Purezza:99.83%Colore e forma:SolidPeso molecolare:371.39GW-493838
CAS:GW-493838 is a potent adenosine A1A receptor agonist for the treatment of dyslipidemia and neuropathic pain, with analgesic effects on post-herpetic neuralgiaFormula:C21H21ClFN7O4Purezza:99.11% - 99.58%Colore e forma:SolidPeso molecolare:489.89Liafensine
CAS:Liafensine(BMS-820836): Selective inhibitor for serotonin, norepinephrine, dopamine reuptake; targets major depression, CNS disorders.Formula:C24H22N4Purezza:99.91%Colore e forma:SolidPeso molecolare:366.46Antalarmin hydrochloride
CAS:Antalarmin hydrochloride, a CRF1 antagonist, offers anti-inflammatory benefits and prevents stress ulcers in IBS.Formula:C24H35ClN4Purezza:99.84% - 99.85%Colore e forma:SolidPeso molecolare:415.02Besipirdine
CAS:Besipirdine (HP 749 free base) is a non-receptor-dependent cholinomimetic compound with alpha-adrenergic activity and cardiovascular activity.Formula:C16H17N3Purezza:97.15% - 98.85%Colore e forma:SolidPeso molecolare:251.33U 99194 maleate
CAS:U 99194 maleate (U-99194A maleate) is a D3 antagonist and increases social behaviors of isolation-induced aggressive male mice.Formula:C21H31NO6Purezza:99.45%Colore e forma:SolidPeso molecolare:393.47KI-7
CAS:KI-7 is an adenosine A2B receptor positive allosteric modulator.Formula:C23H18N2O2Purezza:98.33%Colore e forma:SolidPeso molecolare:354.4LY266097 hydrochloride
CAS:<p>LY266097 hydrochloride is a 5-HT2 antagonist with pKi of 7.7/9.8/7.6 for 5-HT2A/B/C, used in depression research.</p>Formula:C21H24Cl2N2O2Purezza:98.58%Colore e forma:SolidPeso molecolare:407.33Thiethylperazine dimaleate
CAS:<p>Thiethylperazine dimaleate (Thiethylperazine maleate) is an antagonist of the D2 receptor and H1 receptor.</p>Formula:C30H37N3O8S2Purezza:99.07%Colore e forma:SolidPeso molecolare:631.76L-168049
CAS:<p>L-168049: Human glucagon receptor antagonist, IC50 - 3.7 nM human, 63 nM murine, 60 nM canine.</p>Formula:C24H20BrClN2OPurezza:>99.99%Colore e forma:SolidPeso molecolare:467.79SB-209670
CAS:SB-209670 is a selective endothelin receptor antagonist that inhibits the activity of ET(B) receptors in rat vascular endothelium and vascular smooth muscle.Formula:C29H28O9Purezza:98.29% - 99.40%Colore e forma:SolidPeso molecolare:520.53Felcisetrag
CAS:<p>Felcisetrag (TD-8954), an oral 5-HT4 agonist with GI prokinetic effects, has a high affinity (pKi 9.4) for h5-HT4(c) receptors.</p>Formula:C25H37N5O3Purezza:99.99%Colore e forma:SolidPeso molecolare:455.59ANR 94
CAS:ANR94 is a potent hAA2AR antagonist (Ki 46 nM) with potential for Parkinson's research.Formula:C9H13N5OPurezza:98.9%Colore e forma:SolidPeso molecolare:207.23KSK94
CAS:KSK94 is an H3 receptor antagonist that inhibits sigma-2 receptors , with a Ki value of 75.2 nM, and can be used to study injurious pain.Formula:C25H26N4OPurezza:99.60%Colore e forma:SolidPeso molecolare:398.55-HT1A modulator 1
CAS:<p>5-HT1A modulator 1 displays very high affinities for the 5-HT1A, α1-adrenergic receptor, and D2 receptor (IC50s = 2 nM, 10 nM, and 40 nM).</p>Formula:C21H25N3O2SPurezza:99.68%Colore e forma:SolidPeso molecolare:383.51Oxyfedrine L-form HCl
CAS:<p>Oxyfedrine L-form HCl (Ildamen) is a partial agonist at beta-adrenergic receptors and acts as a coronary vasodilator and cardiotonic agent.</p>Formula:C19H24ClNO3Purezza:99.5% - 99.57%Colore e forma:SolidPeso molecolare:349.85Neldazosin
CAS:Neldazosin is used as a potent α1-adrenoceptor antagonist.Formula:C18H25N5O4Purezza:99.76% - 99.97%Colore e forma:SolidPeso molecolare:375.42SPD-473 citrate
CAS:<p>SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.</p>Formula:C23H31Cl2NO8SPurezza:99.37%Colore e forma:SolidPeso molecolare:552.47Camonagrel
CAS:<p>Camonagrel is a compound that has inhibitory effects on Prostaglandin E2.</p>Formula:C15H16N2O3Purezza:98.71% - 99.25%Colore e forma:SolidPeso molecolare:272.3Adenosine antagonist-1
CAS:<p>Adenosine antagonist-1 acts as an adenosine A3 receptor (AA3R) antagonist.</p>Formula:C18H13N7SPurezza:99.28% - 99.95%Colore e forma:SolidPeso molecolare:359.41Masilukast
CAS:Masilukast(MCC-847) is an oral leukotriene D4 (LTD4) receptor antagonist for the study of diseases associated with inflammation.Formula:C31H32F3N3O5SPurezza:99.23% - 99.62%Colore e forma:SolidPeso molecolare:615.66ST-1535
CAS:<p>ST 1535: potent, oral A2A adenosine receptor antagonist with antiparkinsonian and antitremor effects, promising for Parkinson's research.</p>Formula:C12H16N8Purezza:99.64% - 99.69%Colore e forma:SolidPeso molecolare:272.31BMY-14802 hydrochloride
CAS:BMY-14802 hydrochloride (BMS 181100 hydrochloride) is a selective antagonist of σ receptor (IC50 = 112 nM) with antipsychotic effects.Formula:C18H23ClF2N4OPurezza:99.97%Colore e forma:SolidPeso molecolare:384.85O-1602
CAS:O-1602 is a novel GPR55 agonist, an atypical cannabinoid associated with the central nervous system and obesity, and is a candidate compound for the treatmentFormula:C17H22O2Purezza:99.85%Colore e forma:SolidPeso molecolare:258.36Pentiapine
CAS:Pentiapine (CGS 10746) is a novel inhibitor of dopamine release.Formula:C15H17N5SPurezza:99.35%Colore e forma:SolidPeso molecolare:299.39LTB4 antagonist 3
CAS:Compound 24e, a leukotriene B4 (LTB4) antagonist, exhibits an inhibitory concentration 50 (IC50) of 477 nM and demonstrates anti-inflammatory activity [1].Formula:C29H27NO6Purezza:98%Colore e forma:SolidPeso molecolare:485.53TM-N1324
CAS:<p>TM-N1324 is a GPR39 agonist; 280 nM potency without Zn2+, 9 nM with; similar effects on murine GPR39 (EC50s: 180 nM/5 nM).</p>Formula:C18H13ClFN7OPurezza:99.88%Colore e forma:SolidPeso molecolare:397.79CCR4 antagonist 4
CAS:CCR4 Antagonist 4 (Compound 22) is a potent and selective antagonist of the CC chemokine receptor-4 (CCR4), displaying an IC50 value of 0.02 μM. It also inhibits MDC-mediated chemotaxis and Ca2+ mobilization, with IC50 values of 0.007 μM and 0.003 μM, respectively. This compound is utilized in research on allergic inflammation [1].Formula:C24H27Cl2N7OColore e forma:SolidPeso molecolare:500.42Gentisein
CAS:Gentisein (NSC-329491), a primary metabolite of Mangiferin, exhibits significant inhibition of serotonin uptake, demonstrating potency with an IC50 value of 4.7Formula:C13H8O5Purezza:96.89%Colore e forma:SolidPeso molecolare:244.2RBC10
CAS:RBC10 inhibits the binding of Ral to its effector RALBP1, as well as inhibiting Ral-mediated cell spreading of murine embryonic fibroblasts and anchorage-Formula:C24H25ClN2O2Purezza:99.71%Colore e forma:SolidPeso molecolare:408.92Cenerimod
CAS:Cenerimod (ACT-334441) is an S1P1 agonist used in the study of murine experimental autoimmune encephalomyelitis (EAE) and murine scleroderma.Formula:C25H31N3O5Purezza:97.43% - 99.97%Colore e forma:SolidPeso molecolare:453.53CCR2 antagonist 4
CAS:<p>CCR2 antagonist 4 (Teijin compound 1) is a potent and specific antagonist of CCR2(IC50s of 180 nM), and potently inhibits MCP-1-induced chemotaxis(IC50 of 24 nM</p>Formula:C21H21ClF3N3O2Purezza:99.86%Colore e forma:SolidPeso molecolare:439.86LX-1031
CAS:LX-1031 is an effective inhibitor of tryptophan 5-hydroxylase. LX-1031 decreases serotonin (5-HT) synthesis peripherally.Formula:C28H25F3N4O4Purezza:97.123% - 98.97%Colore e forma:SolidPeso molecolare:538.52Hh-Ag1.5
CAS:Hh-Ag1.5 is a dual Hedgehog/Smo agonist (EC50/Ki: 0.5-2.3 nM), reprograms hepatic stem cells, and differentiates hiPSCs into neural/skin cells.Formula:C28H26ClF2N3OSPurezza:99.8%Colore e forma:SolidPeso molecolare:526.04Casopitant mesylate
CAS:Casopitant mesylate (GW679769B): Selective, brain-permeable NK1 receptor blocker, oral antiemetic.Formula:C31H39F7N4O5SPurezza:98%Colore e forma:SolidPeso molecolare:712.72Sulmazole
CAS:<p>Sulmazole (AR-L 115-BS) is a small molecule Sulmazole is a small molecule cGMP-PDE inhibitor.Sulmazole is a competitive inhibitor of A1 adenosine receptors.</p>Formula:C14H13N3O2SPurezza:99.94%Colore e forma:SolidPeso molecolare:287.34PF-04634817
CAS:PF-0463481: safe, well-tolerated, dual CCR2/CCR5 antagonist for diabetic nephropathy; similar human/rodent CCR2 potency, less rodent CCR5 effect.Formula:C25H36F3N5O3Purezza:98%Colore e forma:SolidPeso molecolare:511.58RU-SKI 43
CAS:RU-SKI 43: Potent, selective Hhat inhibitor, IC50 850 nM. Anticancer; potential lung adenocarcinoma treatment. Inhibits Gli-1, Akt, mTOR pathways.Formula:C22H30N2O2SPurezza:99.85%Colore e forma:SolidPeso molecolare:386.55Fiduxosin
CAS:Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and α1d-adrenoceptor, with KiFormula:C30H29N5O4SPurezza:99.73%Colore e forma:SolidPeso molecolare:555.65Wf-516
CAS:Wf-516 is a 5-HT reuptake inhibitor (Kis: 5 nM and 40 nM for 5-HT1A receptor and 5-HT2A receptor in humans, respectively), and with potent antidepressantFormula:C25H25Cl2N3O4Purezza:98%Colore e forma:SolidPeso molecolare:502.39AM841
CAS:AM841, a high-affinity electrophilic ligand, covalently interacts with a cysteine residue in helix six, thus activating the CB1 cannabinoid receptor.Formula:C26H39NO3SPurezza:98%Colore e forma:SolidPeso molecolare:445.66Phentolamine Analogue 1
CAS:Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.Formula:C17H19N3OPurezza:99.96%Colore e forma:SolidPeso molecolare:281.35Bunazosin Hydrochloride
CAS:Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.Formula:C19H28ClN5O3Purezza:99.12%Colore e forma:SolidPeso molecolare:409.91YM348
CAS:YM348 is an effective and orally active 5-HT2C receptor agonist. YM348 also shows a high affinity for the cloned human 5-HT2C receptor (Ki: 0.89 nM).Formula:C14H17N3OPurezza:98%Colore e forma:SolidPeso molecolare:243.3NTNCB hydrochloride
CAS:<p>NTNCB hydrochloride is an antagonist of neuropeptide Y (NPY) Y5 receptor.</p>Formula:C25H34ClN3O4SPurezza:98.38%Colore e forma:SolidPeso molecolare:508.07ASP6432
CAS:ASP6432 is an antagonist of type 1 lysophosphatidic acid receptor (LPA1). For human LPA1 and rat LPA1, the IC50s are 11 nM and 30 nM , respectively.Formula:C26H32KN4O6S2Colore e forma:SolidPeso molecolare:599.78Tedalinab
CAS:<p>Tedalinab is an effective and selective cannabinoid receptor 2 agonist.</p>Formula:C19H21F2N3OPurezza:98%Colore e forma:SolidPeso molecolare:345.39FK788
CAS:FK788 is a diphenylcarbamate derivative that functions as a highly potent and selective IP agonist.Formula:C26H25NO6Colore e forma:SolidPeso molecolare:447.48Veldoreotide TFA
CAS:<p>Veldoreotide (DG3173) TFA, a somatostatin analogue, effectively binds to and activates somatostatin receptors (SSTR) 2, 4, and 5. This compound demonstrates a higher efficacy in inhibiting growth hormone (GH) secretion in adenomas than Octreotide, showcasing its potential as a pain modulating agent [1].</p>Formula:C62H75F3N12O12Colore e forma:SolidPeso molecolare:1237.33NAS-181 free base
CAS:NAS-181 free base is a 5-HT(1B) receptor antagonist.Formula:C19H26N2O4Colore e forma:SolidPeso molecolare:346.42Flesinoxan HCl
CAS:Flesinoxan HCl is the salt form of Flesinoxan, which is a selective 5-HT1A receptor agonist.Formula:C22H27ClFN3O4Colore e forma:SolidPeso molecolare:451.92SGC agonist 1
CAS:SGC agonist 1 is a potent soluble guanylate cyclase (SGC) agonist. SGC agonist 1 is able to increase solubility and has high cell permeability.Formula:C22H19F2N7OColore e forma:SolidPeso molecolare:435.43BMS-870145
CAS:BMS-870145 is a potent and selective P2Y1 purinergic receptor antagonist..Formula:C30H24ClF4N3O3Colore e forma:SolidPeso molecolare:585.98SDZ-216525
CAS:SDZ-216525, a 5-HT1A receptor antagonist, inhibits the tracheal contractions induced both by NKA (10 nM-3 microM) and 5-HT (10 nM-10 microM) (n=4-10).Formula:C25H28N4O5SColore e forma:SolidPeso molecolare:496.58
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