Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(942 prodotti)
- Recettore dell'adenosina(242 prodotti)
- Recettore adrenergico(2.949 prodotti)
- Recettore della bombesina(30 prodotti)
- Recettore della bradichinina(59 prodotti)
- CXCR(149 prodotti)
- CaSR(32 prodotti)
- Recettore dei cannabinoidi(195 prodotti)
- Recettore della dopamina(410 prodotti)
- Recettore dell'endotelina(75 prodotti)
- Recettore GNRH(73 prodotti)
- GPCR19(31 prodotti)
- GRK(32 prodotti)
- GTPase(21 prodotti)
- Recettore del glucagone(166 prodotti)
- Proteina Hedgehog/Smoothened(45 prodotti)
- Recettore dell'istamina(359 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(24 prodotti)
- Recettore OX(40 prodotti)
- Recettore degli oppioidi(298 prodotti)
- PAFR(11 prodotti)
- PKA(49 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(30 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 18 più sottocategorie
Trovati 5378 prodotti di "Proteina G/GPCR"
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MF266-1
CAS:<p>MF266-1, a selective E prostanoid receptor 4 antagonist, relieves joint inflammation and pain in rodent models of osteoarthritis and rheumatoid.</p>Formula:C24H17ClF3NO3SColore e forma:SolidPeso molecolare:491.91SKF 81297
CAS:<p>SKF 81297 is a selective and potent agonist for the dopamine D1 receptor [1].</p>Formula:C16H16ClNO2Purezza:98%Colore e forma:SolidPeso molecolare:289.765-HT2 agonist-1
CAS:<p>Compound 24, a 5-HT2 agonist-1, selectively activates 5-HT2A, 5-HT2B, and 5-HT2C receptors with IC50 values of 10 nM, 8.3 nM, and 1.6 nM, respectively.</p>Formula:C19H23ClN2O2Purezza:98%Colore e forma:SolidPeso molecolare:346.85mPGES1-IN-3
CAS:<p>mPGES1-IN-3 is a potent and selective inhibitor of microsomal prostaglandin E2 synthase-1 (mPGES-1) .</p>Formula:C24H16ClF5N4O3Purezza:98%Colore e forma:SolidPeso molecolare:538.85JTE-952
CAS:<p>JTE-952: oral, selective Type II CSF-1R inhibitor, IC50 = 13 nM for CSF1R, 261 nM for TrkA, effective in mouse arthritis model.</p>Formula:C30H34N2O6Purezza:98%Colore e forma:SolidPeso molecolare:518.6RP-001 hydrochloride
CAS:<p>RP-001 hydrochloride: S1P1 agonist, EC50 9 pM; low activity on S1P2-4, moderate S1P5 affinity.</p>Formula:C24H25ClN4O4Purezza:98%Colore e forma:SolidPeso molecolare:468.93MF498
CAS:MF498 is a novel and selective E prostanoid receptor 4 (EP4 receptor) antagonist, displayed a strong binding affinity for the EP4 receptor (Ki: 0.7 nM).Formula:C32H33N3O7SPurezza:98%Colore e forma:SolidPeso molecolare:603.694-Amino-PPHT Hydrobromide
CAS:<p>4-Amino-PPHT Hydrobromide is a precursor for fluorescent labeled Dopamine D2 receptors agonist.</p>Formula:C21H28N2OPurezza:98%Colore e forma:SolidPeso molecolare:324.46L-644,698
CAS:<p>L-644,698 is a selective agonist of human prostanoid DP receptor.</p>Formula:C21H31NO4SPurezza:98%Colore e forma:SolidPeso molecolare:393.545-HT3-In-1
CAS:5-HT3-In-1 (compound example 8) exhabits with 5-HT3 inhibition activity.Formula:C16H21ClN4O3Purezza:98%Colore e forma:SolidPeso molecolare:352.82TRAP-6-IN-1
CAS:<p>TRAP-6-IN-1 inhibits collagen/TRAP-6, IC50: 17.12/11.88 μM, blocks platelet aggregation.</p>Formula:C18H20O3Colore e forma:SolidPeso molecolare:284.35Bunazosin Hydrochloride
CAS:<p>Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an ocular hypotensive drug.</p>Formula:C19H28ClN5O3Purezza:99.12%Colore e forma:SolidPeso molecolare:409.91Prostaglandin E2 serinol amide
CAS:<p>Prostaglandin E2 Serinol Amide acts as a weak inhibitor against the hydrolysis of [3H]2-oleoylglycerol, but it is non-hydrolyzable and cannot produce PGE2. Consequently, it is unable to inhibit leukotriene B4 biosynthesis, superoxide production, migration, and the release of antimicrobial peptides [1].</p>Formula:C23H39NO6Colore e forma:SolidPeso molecolare:425.566Orvepitant maleate
CAS:<p>Orvepitant maleate, a selective NK-1 receptor antagonist (pKi 10.2), may treat depression and CRC; crosses the blood-brain barrier.</p>Formula:C35H39F7N4O6Purezza:98%Colore e forma:SolidPeso molecolare:744.7Phentolamine Analogue 1
CAS:<p>Phentolamine Analogue 1 is an analogue of phentolamine. Phentolamine is a nonselective antagonist of α-adrenergic.</p>Formula:C17H19N3OPurezza:99.96%Colore e forma:SolidPeso molecolare:281.35MK 0893
CAS:MK 0893 is a potent and selective Glucagon Receptor (GR) antagonist competitive, reversible cAMP activity, which attenuates blood glucose elevation.Formula:C32H27Cl2N3O4Purezza:98.79%Colore e forma:SolidPeso molecolare:588.48SB 258719
CAS:<p>SB 258719 is a selective antagonist of 5-HT7 receptor with pKi of 7.5.</p>Formula:C18H30N2O2SPurezza:99.73%Colore e forma:SolidPeso molecolare:338.51Gestonorone Capronate
CAS:<p>Gestonorone Capronate is a progesterone used in benign prostatic hyperplasia and endometrial cancer studies.</p>Formula:C26H38O4Purezza:99.19%Colore e forma:SolidPeso molecolare:414.58JNJ-19567470
CAS:<p>JNJ-19567470 is a selective, non-peptide CRF receptor 1 antagonist.</p>Formula:C22H27BrN4OColore e forma:SolidPeso molecolare:443.38LY-368975
CAS:<p>LY-368975 is a potent and selective inhibitor of the norepinephrine (NE) reuptake site. LY-368975 reduces food consumption in rodents.</p>Formula:C17H21NOSColore e forma:SolidPeso molecolare:287.42Ubrogepant
CAS:Ubrogepant (MK-1602) is an antagonist of calcitonin gene-related peptide receptor that can be used in the acute treatment of migraine studies.Formula:C29H26F3N5O3Purezza:99.452% - 99.78%Colore e forma:SolidPeso molecolare:549.54SQ 26655
CAS:<p>SQ 26655 is an antagonist of thromboxane A2/prostaglandin H2.</p>Formula:C21H34O4Purezza:98%Colore e forma:SolidPeso molecolare:350.49AH13205
CAS:<p>AH13205 is an agonist of EP2 prostanoid receptor.</p>Formula:C24H36O4Purezza:98%Colore e forma:SolidPeso molecolare:388.54(+)-Fluprostenol
CAS:<p>(+)-Fluprostenol (AL-5848), an analogue of prostaglandin F2 alpha, is a prostaglandin F2α receptor PTGFR agonist and decreases the expression of Oviductal</p>Formula:C23H29F3O6Purezza:97.35%Colore e forma:SolidPeso molecolare:458.47GR 127935 hydrochloride
CAS:5-HT1B/1D receptor antagonistFormula:C29H32ClN5O3Purezza:98%Colore e forma:SolidPeso molecolare:534.05CY 208-243
CAS:CY 208-243 is a selective dopamine D1 receptor agonist with anti-Parkinson disease activity.Formula:C19H18N2Purezza:98%Colore e forma:SolidPeso molecolare:274.36AGN 210676
CAS:AGN 210676 is a selective agonist of prostaglandin EP2(EC50 : 5 nM).Formula:C23H29NO5SPurezza:98%Colore e forma:SolidPeso molecolare:431.55GSK494581A
CAS:GSK494581A is a GPR55 agonist and glycine transporter subtype 1 inhibitor.Formula:C27H28F2N2O4SPurezza:98%Colore e forma:SolidPeso molecolare:514.58FR-181877
CAS:<p>FR-181877: nonprostanoid PGI2 agonist, ADP-induced platelet aggregation inhibitor (IC50=0.081μM), orally bioavailable (56%), long half-life (4.3h) in rats.</p>Formula:C30H28N2O4Purezza:98%Colore e forma:SolidPeso molecolare:480.55PF 514273
CAS:<p>PF 514273 is a CB1 receptor antagonist.</p>Formula:C21H17Cl2F2N3O2Purezza:98%Colore e forma:SolidPeso molecolare:452.28RU-SKI 43
CAS:<p>RU-SKI 43: Potent, selective Hhat inhibitor, IC50 850 nM. Anticancer; potential lung adenocarcinoma treatment. Inhibits Gli-1, Akt, mTOR pathways.</p>Formula:C22H30N2O2SPurezza:99.85%Colore e forma:SolidPeso molecolare:386.55Domesticine, (-)-
CAS:<p>Domesticine, (-)- is an antagonist of alpha-1D-adrenoceptor.</p>Formula:C19H19NO4Purezza:98%Colore e forma:SolidPeso molecolare:325.36OMDM-5
CAS:<p>OMDM-5 is a potent vanilloid receptor type 1 (TRPV1, EC50 = 75 nM) agonist, showing weak ligand activity at cannabinoid type 1 receptor (CB1, Ki=4.9 μM).</p>Formula:C26H44N2O3Purezza:99.73%Colore e forma:SolidPeso molecolare:432.64IIIM-8
CAS:<p>IIIM-8 is a melanogenesis inhibitor that suppresses pigment production in both in vitro and in vivo settings, exhibiting no cytotoxic effects on Human Adult</p>Formula:C14H17NO4Purezza:98%Colore e forma:SolidPeso molecolare:263.29GSK-1004723
CAS:<p>GSK-1004723 is a novel antagonist of histamine H(1) and H(3) receptor. It represents a potential novel therapy for allergic rhinitis.</p>Formula:C39H49ClN4O2Colore e forma:SolidPeso molecolare:641.284-hydroxy Nebivolol hydrochloride
CAS:<p>4-Hydroxy Nebivolol, a primary metabolite of Nebivolol, results from the enzymatic hydroxylation of Nebivolol by the cytochrome P450 (CYP) isoform CYP2D6.</p>Formula:C22H25F2NO5HClColore e forma:SolidPeso molecolare:457.9RXFP1 receptor agonist-2
CAS:<p>RXFP1 Receptor Agonist-2 (Example 124), an EC50 value of 1 nM [1].</p>Formula:C33H32F7N3O5Colore e forma:SolidPeso molecolare:683.61NGD9002
CAS:<p>NGD9002 is a novel generation, topology 2 selective corticotropin releasing factor-1 (CRF-1) receptor antagonist agent.</p>Formula:C20H31N5OPurezza:98%Colore e forma:SolidPeso molecolare:357.49NNC 26-9100
CAS:<p>Somatostatin sst4 receptor agonist</p>Formula:C22H25BrCl2N6SPurezza:98%Colore e forma:SolidPeso molecolare:556.35Isopropyl dodec-11-enylfluorophosphonate
CAS:<p>Isopropyl dodec-11-enylfluorophosphonate (IDEFP) is an organophosphorus ester functioning as a central cannabinoid receptor (CB1) antagonist and exhibits</p>Formula:C15H30FO2PPurezza:98%Colore e forma:SolidPeso molecolare:292.37Naxagolide free base
CAS:Naxagolide is a sustained release formulation. It is a dopamine agonist.Formula:C15H21NO2Purezza:98%Colore e forma:SolidPeso molecolare:247.33TXNIP-IN-1
CAS:<p>TXNIP-IN-1: TXNIP-TRX complex inhibitor, targets diabetes, cardiovascular, and inflammatory diseases.</p>Formula:C12H12N2O4Purezza:99.11%Colore e forma:SolidPeso molecolare:248.23Setipafant
CAS:<p>Setipafant is an antagonist of the platelet-activating factor.</p>Formula:C26H23ClN6O2SPurezza:98%Colore e forma:SolidPeso molecolare:519.02Fosnetupitant chloride monohydrochloride
CAS:<p>Fosnetupitant chloride monohydrochloride (Pro-netupitant chloride monohydrochloride) is a selective NK1 antagonist exhibiting high affinity for the human NK1</p>Formula:C31H37Cl2F6N4O5PPurezza:98%Colore e forma:SolidPeso molecolare:761.52Ritodrine
CAS:<p>Ritodrine (DU21220) is a β-adrenergic agonist as well as an effective uterine relaxant that can be used in arrest premature labor research[1] [2].</p>Formula:C17H21NO3Colore e forma:SolidPeso molecolare:287.355-HT2C agonist-3 free base
CAS:<p>5-HT2C agonist-3 ((+)-19) free base, a selective 5-HT2C agonist (EC50: 24 nM, Ki: 78 nM), exhibits antipsychotic drug-like activity and inhibits Amphetamine-</p>Formula:C19H22FNO2Purezza:98%Colore e forma:SolidPeso molecolare:315.38LGD-6972 sodium
CAS:<p>LGD-6972 sodium is a glucagon receptor antagonist.</p>Formula:C43H46N2NaO5SPurezza:98%Colore e forma:SolidPeso molecolare:725.95-HT2 agonist-1 free base
CAS:<p>Compound 24 (5-HT2 agonist-1 free base) is a potent agonist for 5-HT2A, 5-HT2B, and 5-HT2C receptors, exhibiting IC50 values of 10 nM, 8.3 nM, and 1.6 nM,</p>Formula:C19H22N2O2Purezza:98%Colore e forma:SolidPeso molecolare:310.39Mesembrine
CAS:<p>Mesembrine is an alkaloid, a 5-HT transporter inhibitor (K i 1.4 nM), and inhibits PDE4B (IC50 7.8 μM).</p>Formula:C17H23NO3Colore e forma:SolidPeso molecolare:289.37GSK1842799
CAS:GSK1842799 is a selective S1P1 receptor agonist with good oral bioavailability.Formula:C24H30F9N3O6SColore e forma:SolidPeso molecolare:659.56N-5984
CAS:<p>N-5984, a β3-adrenergic receptor agonist, is used potentially for the treatment of obesity, overactive bladder and type 2 diabetes.</p>Formula:C20H22ClNO5Purezza:98%Colore e forma:SolidPeso molecolare:391.85ASP6432
CAS:ASP6432 is an antagonist of type 1 lysophosphatidic acid receptor (LPA1). For human LPA1 and rat LPA1, the IC50s are 11 nM and 30 nM , respectively.Formula:C26H32KN4O6S2Colore e forma:SolidPeso molecolare:599.78BMS-639623
CAS:<p>BMS-639623 is a CCR3 antagonist with a picomolar inhibitory effect on eosinophilic chemotaxis and can be used in the treatment of asthma.</p>Formula:C25H32FN7O2Colore e forma:SolidPeso molecolare:481.57PF-04634817
CAS:<p>PF-0463481: safe, well-tolerated, dual CCR2/CCR5 antagonist for diabetic nephropathy; similar human/rodent CCR2 potency, less rodent CCR5 effect.</p>Formula:C25H36F3N5O3Purezza:98%Colore e forma:SolidPeso molecolare:511.58L 662025
CAS:<p>L 662025 is a PAF receptor antagonist.</p>Formula:C23H27N3O6Purezza:98%Colore e forma:SolidPeso molecolare:441.48S1P1 agonist 6 hemicalcium
CAS:<p>Compound I (S1P1 agonist 6 hemicalcium) is an S1P1 agonist that diminishes autoimmune activity by inhibiting lymphocyte trafficking, and serves as an</p>Formula:C25H26F3NO3CaPurezza:98%Colore e forma:SolidPeso molecolare:465.51L-749329
CAS:<p>L-749329 is a ligand of ET(A) and ET(B) endothelin receptor.</p>Formula:C28H29NO8SPurezza:98%Colore e forma:SolidPeso molecolare:539.6GSK726701A
CAS:<p>GSK726701A is a new type of prostaglandin E2 receptor 4 (EP4) partial agonist (pEC50: 7.4).</p>Formula:C24H22FNO5Purezza:98%Colore e forma:SolidPeso molecolare:423.43Prostaglandin E1 ethanolamide
CAS:<p>Prostaglandin E1 ethanolamide, an analog of Prostaglandin E1 (PGE1), can potentially inhibit the GLI2-induced expression of target genes such as Gli1 and Ptch1, thereby reducing tumor growth [1].</p>Formula:C22H39NO5Colore e forma:SolidPeso molecolare:397.55NKP608
CAS:NKP608 is a NK-1 receptor antagonist with anticancer and anxiolytic activities.Formula:C31H24ClF6N3O2Purezza:99.88% - 99.88%Colore e forma:SolidPeso molecolare:619.99GYKI-46903 HCl
CAS:<p>GYKI-46903 is a noncompetitive 5-HT3 receptor antagonist.</p>Formula:C17H21ClFNO2Colore e forma:SolidPeso molecolare:325.81S1PR1-MO-1
CAS:<p>S1PR-MO-1 is a modulator of sphingosine-1-phosphate receptor and is used to study hyperproliferative inflammatory diseases.</p>Formula:C25H29N3O3Purezza:98%Colore e forma:SolidPeso molecolare:419.52LY 53857
CAS:<p>LY 53857 is a potent and selective antagonist of 5-HT2 serotonin receptor.</p>Formula:C27H36N2O7Colore e forma:SolidPeso molecolare:500.5925-HT2C agonist-3
CAS:<p>5-HT2C agonist-3 ((+)-19), a selective 5-HT2C agonist (EC 50: 24 nM, Ki: 78 nM), exhibits antipsychotic-like activity by blocking amphetamine-induced</p>Formula:C19H23ClFNO2Purezza:98%Colore e forma:SolidPeso molecolare:351.84AJ-76 hydrochloride
CAS:<p>AJ-76 hydrochloride ((+)-AJ 76 hydrochloride) serves as a dopamine autoreceptor antagonist, exhibiting pK i values of 6.95 for hD3, 6.67 for hD4, 6.37 for hD2S, 6.21 for hD2L, and 6.07 for rD2 receptors, indicating its binding affinity strength across these receptor types.</p>Formula:C15H24ClNOColore e forma:SolidPeso molecolare:269.81L 640035
CAS:L 640035 inhibits human platelet aggregation which is induced by arachidonic acid, collagen, and the prostaglandin-endoperoxide analog of U44069.Formula:C15H12O3SPurezza:98%Colore e forma:SolidPeso molecolare:272.32GS-6201
CAS:<p>GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor.</p>Formula:C21H21F3N6O2Purezza:99.74% - 99.78%Colore e forma:SolidPeso molecolare:446.43BU-E 75
CAS:<p>BU-E 75 is an agonist of the histamine H2.</p>Formula:C21H24F2N6Colore e forma:SolidPeso molecolare:398.45Emicerfont
CAS:<p>Emicerfont is an antagonist of the corticotropin-releasing factor type 1 receptor (IC50: 66 nM).</p>Formula:C22H24N6O2Purezza:98%Colore e forma:SolidPeso molecolare:404.46Binedaline
CAS:Binedaline is a selective norepinephrine reuptake inhibitor with Ki value of 25 nM.Formula:C19H23N3Purezza:98%Colore e forma:SolidPeso molecolare:293.41L-736380
CAS:<p>L-736380, a CCK-B antagonist, reduces gastric acid (ID50: 0.064mg/kg) and blocks [(125)I]CCK-8S in mouse brains (ED50: 1.7mg/kg).</p>Formula:C25H29N9O2Colore e forma:SolidPeso molecolare:487.56LBT 999
CAS:<p>LBT 999 is used as a dopamine reuptake inhibitor.</p>Formula:C20H26FNO2Colore e forma:SolidPeso molecolare:331.42Capeserod HCl
CAS:<p>Capeserod HCl, a 5-hydroxytriptamine 4 (5-HT4) receptor agonist, is used potentially for the treatment of Alzheimer's disease.</p>Formula:C23H26Cl2N4O4Purezza:98%Colore e forma:SolidPeso molecolare:493.38GSA-10
CAS:<p>GSA-10 is a potent Smoothened (Smo) receptor agonist with an EC50 of 1.2 μM.</p>Formula:C26H30N2O5Purezza:99.71%Colore e forma:SolidPeso molecolare:450.53(S)-Bexicaserin
CAS:<p>(S)-Bexcaserin (compound 2) serves as a 5-HT2C receptor agonist, presenting research possibilities in obesity and psychiatric disorders [1].</p>Formula:C15H19F2N3OPurezza:98%Colore e forma:SolidPeso molecolare:295.33Droxicam
CAS:<p>Droxicam (Droxicamum) is a non-steroidal anti-inflammatory compound and can be used for research on the relief of inflammation and pain in musculoskeletal</p>Formula:C16H11N3O5SPurezza:99.04%Colore e forma:SolidPeso molecolare:357.34Casopitant mesylate
CAS:<p>Casopitant mesylate (GW679769B): Selective, brain-permeable NK1 receptor blocker, oral antiemetic.</p>Formula:C31H39F7N4O5SPurezza:98%Colore e forma:SolidPeso molecolare:712.72TAK-441
CAS:TAK-441: oral Hedgehog signal blocker, potent anticancer, IC50=4.4 nM, reduces Gli1 mRNA & tumor growth.Formula:C28H31F3N4O6Purezza:99.82%Colore e forma:SolidPeso molecolare:576.56Anti-inflammatory agent 49
CAS:<p>Compound SC9, an anti-inflammatory agent, serves as a potent and selective inhibitor of the Drp1-Fis1 interaction, mitigating FIS1-mediated mitochondrial</p>Formula:C21H22N8O3SPurezza:99.56% - 99.74%Colore e forma:SolidPeso molecolare:466.52AY 77
CAS:<p>AY 77: Potent, selective PAR2 agonist, favors Ca2+ (ec50=40nM) & ERK1/2 (ec50=2μM), boosts breast cancer cell migration.</p>Formula:C21H32N4O4Purezza:99.7%Colore e forma:SolidPeso molecolare:404.5GV150013
CAS:<p>GV150013 is an antagonist of cholecystokinin-2 (CCK2) receptor.</p>Formula:C33H34N4O3Purezza:99.93%Colore e forma:SolidPeso molecolare:534.65WAY-639889
CAS:<p>WAY-639889 is a small molecule compound with selective and potent inhibitory effects on neuropeptide Y-5 receptors.</p>Formula:C25H27N5OPurezza:99.73%Colore e forma:SolidPeso molecolare:413.51PAOPA
CAS:dopamine D2 receptor modulatorFormula:C11H18N4O3Purezza:>99.99%Colore e forma:SolidPeso molecolare:254.29Ertugliflozin L-pyroglutamic acid
CAS:<p>Ertugliflozin is a potent oral hSGLT2 inhibitor (IC50: 0.877 nM) for type 2 diabetes treatment studies.</p>Formula:C27H32ClNO10Purezza:99.88% - 99.94%Colore e forma:SolidPeso molecolare:566Calindol hydrochloride
CAS:<p>Calindol (hydrochloride) is a positive allosteric modulator (PAM) of calcimimetic calcium-sensing receptor (CaSR) with an EC50 of 132 nM.</p>Formula:C21H21ClN2Purezza:99.47%Colore e forma:SolidPeso molecolare:336.86GW 833972A
CAS:<p>GW 833972A: selective CB2 agonist; reduces neural depolarization and citric acid cough in animals.</p>Formula:C18H14Cl2F3N5OPurezza:99.93%Colore e forma:SoildPeso molecolare:444.24Clazosentan
CAS:Clazosentan (Ro 61-1790) is a selective ET_A receptor antagonist that inhibits ET-1 vasoconstriction and prevents cerebral vasospasm.Formula:C25H23N9O6SPurezza:95.39% - >99.99%Colore e forma:SolidPeso molecolare:577.57Didesmethyl cariprazine
CAS:<p>Didesmethyl cariprazine, Cariprazine's active metabolite, treats schizophrenia/bipolar with D3/D2 affinity; half-life 1-3 weeks.</p>Formula:C19H28Cl2N4OPurezza:99.52%Colore e forma:SolidPeso molecolare:399.36PSB-603
CAS:<p>PSB-603 is a selective antagonist of Adenosine A2B receptor(Ki = 0.553 nM) with anti-inflammatory effects.</p>Formula:C24H25ClN6O4SPurezza:97.13%Colore e forma:SolidPeso molecolare:529.01Lotiglipron
CAS:<p>Lotiglipron (PF-07081532) is a GLP-1R agonist that lowers blood glucose and may be used in the study of type 2 diabetes mellitus (T2DM) and excess obesity.</p>Formula:C31H31ClN4O5Purezza:98.3%Colore e forma:SolidPeso molecolare:575.05INT-777
CAS:<p>INT-777 (S-EMCA) is a potent TGR5 agonist with an EC50 of 0.82 μM.</p>Formula:C27H46O5Purezza:99.89%Colore e forma:SolidPeso molecolare:450.65CCR3 antagonist 1
CAS:<p>CCR3 antagonist 1 is a potent CCR3 antagonist, used for the research of inflammatory and immunologic diseases.</p>Formula:C19H21Cl2N3O4S2Purezza:98.28%Colore e forma:SolidPeso molecolare:490.42Talibegron hydrochloride
CAS:<p>Talibegron hydrochloride: β3 adrenoceptor agonist, pD2 3.72, relaxes rat arteries, reduces leptin in mice.</p>Formula:C18H22ClNO4Purezza:99.82%Colore e forma:SolidPeso molecolare:351.83Deriglidole
CAS:<p>Deriglidole (SL 86-0715), an alpha2 receptor inhibitor, blocks colistin/Idazoxan but not prazosin/α2-adrenergic receptors.</p>Formula:C16H21N3Purezza:97.31% - 98.23%Colore e forma:SolidPeso molecolare:255.36Adomeglivant
CAS:<p>Adomeglivant (LY2409021) is a potent and selective glucagon receptor antagonist. Which is used in clinical trial for type 2 diabetes mellitus.</p>Formula:C32H36F3NO4Purezza:99.91%Colore e forma:SolidPeso molecolare:555.63LGD-6972
CAS:<p>LGD-6972 is an antagonist of glucagon receptor.</p>Formula:C43H46N2O5SPurezza:98.8% - 99.62%Colore e forma:SolidPeso molecolare:702.9Selatogrel
CAS:<p>Selatogrel (ACT-246475) is a P2Y12 receptor antagonist with antithrombotic activity and inhibits platelet aggregation.</p>Formula:C28H39N6O8PPurezza:98.43%Colore e forma:SolidPeso molecolare:618.62WAY-607695
CAS:<p>WAY-607695 is a potential 5-HT1A receptor agonist.</p>Formula:C13H12FNO2Purezza:99.82%Colore e forma:SolidPeso molecolare:233.24SB 216641 hydrochloride
CAS:<p>SB 216641 hydrochloride (SB-216641A) is a 5-HT1B/D receptor antagonist with anxiolytic properties.</p>Formula:C28H31ClN4O4Purezza:98.06% - 99.23%Colore e forma:SolidPeso molecolare:523.02(±)-Prenalterol
CAS:<p>(±)-Prenalterol (H 80/62) is an agonist of beta-2- and beta-1-adrenergic receptors and is used to study chronic congestive heart failure.</p>Formula:C12H19NO3Purezza:99.73%Colore e forma:SolidPeso molecolare:225.28
