Proteina G/GPCR
Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.
Sottocategorie di "Proteina G/GPCR"
- recettore 5-HT(1.025 prodotti)
- Recettore dell'adenosina(249 prodotti)
- Recettore adrenergico(3.030 prodotti)
- Recettore della bombesina(35 prodotti)
- Recettore della bradichinina(61 prodotti)
- CXCR(159 prodotti)
- CaSR(34 prodotti)
- Recettore dei cannabinoidi(217 prodotti)
- Colecistochinina(1 prodotti)
- Recettore della dopamina(444 prodotti)
- Recettore dell'endotelina(86 prodotti)
- Recettore GNRH(84 prodotti)
- GPCR19(33 prodotti)
- GRK(33 prodotti)
- GTPase(22 prodotti)
- Recettore del glucagone(196 prodotti)
- Proteina Hedgehog/Smoothened(49 prodotti)
- Recettore dell'istamina(385 prodotti)
- Recettore LPA(21 prodotti)
- Recettore della melatonina(26 prodotti)
- Recettore OX(42 prodotti)
- Recettore degli oppioidi(325 prodotti)
- PAFR(14 prodotti)
- PKA(55 prodotti)
- Recettore S1P(17 prodotti)
- SGLT(31 prodotti)
- Recettore Sigma(46 prodotti)
Mostrare 19 più sottocategorie
Trovati 5984 prodotti di "Proteina G/GPCR"
Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Antidepressant agent 4
Antidepressant agent 4: orally active, has antidepressant, anxiolytic, and nootropic effects.Formula:C19H38ClN5O2SColore e forma:SolidPeso molecolare:436.06Urocortin III (human)
CAS:Urocortin III, a human peptide, binds CRF-R2, affecting insulin via somatostatin feedback with K i values 13.5-100+ nM.Formula:C185H307N53O50S2Colore e forma:SolidPeso molecolare:4137.93Pasireotide ditrifluoroacetate
Pasireotide is a stable cyclohexapeptide somatostatin mimic.Formula:C62H68F6N10O13Purezza:98%Colore e forma:SolidPeso molecolare:1275.25HAEGTFT
CAS:HAEGTFT is the first N-terminal 1-7 residues of GLP-1 peptide.Formula:C33H47N9O12Purezza:98%Colore e forma:SolidPeso molecolare:761.7817-trifluoromethylphenyl trinor Prostaglandin F2α
CAS:A number of 17-phenyl trinor prostaglandin F2α (17-phenyl trinor PGF2α) derivatives have been approved for the treatment of glaucoma.Formula:C24H31F3O5Colore e forma:SolidPeso molecolare:456.502Piperulin A
CAS:Piperulin A effectively inhibits platelet-activating factor receptor (PAFR) by specifically blocking its binding to isolated rabbit platelet plasma membranes,Formula:C23H28O6Colore e forma:SolidPeso molecolare:400.46PEN (human)
CAS:PEN (human) is an Endogenous peptide GPR83 agonist. ProSAAS-derived neuropeptide.Formula:C97H159N27O32Purezza:98%Colore e forma:SolidPeso molecolare:2215.49Kisspeptin-10, human
CAS:Kisspeptin-10, human is an effective vasoconstrictor and inhibitor of angiogenesis.Formula:C63H83N17O14Purezza:98%Colore e forma:SolidPeso molecolare:1302.462L-threo Lysosphingomyelin (d18:1)
CAS:L-threo Lysosphingomyelin, a natural S1P receptor agonist, has EC50s: 19.3 nM (hS1P1), 131.8 nM (hS1P3), 313.3 nM (hS1P2).Formula:C23H49N2O5PColore e forma:SolidPeso molecolare:464.62PD 142893
CAS:PD 142893 is a functional endothelin-stimulated vasoconstriction antagonist.Formula:C50H65N7O10Purezza:98%Colore e forma:SolidPeso molecolare:924.09Cortistatin-8 acetate
<p>Cortistatin-8 acetate: synthetic corticosteroid analog, GHS-R antagonist; doesn't affect acyl GH release or hesperidin response.</p>Formula:C49H72N12O11S2Purezza:99.01%Colore e forma:SoildPeso molecolare:1069.3Ref: TM-TP2236L
1mg229,00€5mg560,00€10mg800,00€25mg1.216,00€50mg1.644,00€100mg2.213,00€500mg4.436,00€Septide
CAS:Septide is an NK1 receptor agonist acting at a site distinct from substance P.Formula:C39H53N7O7SPurezza:98%Colore e forma:SolidPeso molecolare:763.95Prostaglandin J2
CAS:PGJ2, a PGD2 metabolite, is a DP agonist (Ki: 0.9 nM hDP, 6.6 nM hCRTH2), induces cAMP (EC50: 1.2 nM), oxidative stress, neuronal apoptosis, and neurotoxicity.Formula:C20H30O4Colore e forma:SolidPeso molecolare:334.45SHU 9119
CAS:SHU 9119 is a potent antagonist for human MC3R/MC4R and partial agonist for MC5R with IC50 values of 0.23, 0.06, 0.09 nM.Formula:C54H71N15O9Purezza:98%Colore e forma:SolidPeso molecolare:1074.258[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P
CAS:Broad-spectrum inverse agonist; potent at ghrelin receptor (EC50=5.2 nM); blocks other neuropeptide receptors; induces apoptosis; inhibits tumor growth.Formula:C79H109N19O12Purezza:98%Colore e forma:SolidPeso molecolare:1516.85Stressin I
Potent CRF1 agonist; Ki: 1.5 nM (CRF1), 224 nM (CRF2). Boosts ACTH, enhances stool frequency after i.p. administration.Formula:C203H337N57O56Purezza:98%Colore e forma:SolidPeso molecolare:4472.24Hydroxybupropion
CAS:Hydroxybupropion is the major active metabolite of Bupropion and an antagonist of nACh receptor. Hydroxybupropion inhibits norepinephrine uptake (IC50 = 1.7 μM).Formula:C13H18ClNO2Purezza:99.73%Colore e forma:Off-White SolidPeso molecolare:255.74Ref: TM-T11588
1mg89,00€5mg204,00€10mg331,00€25mg545,00€50mg777,00€100mg1.063,00€1mL*10mM (DMSO)232,00€PACAP-38 (16-38), human, mouse, rat
CAS:PACAP-38 (16-38), human, mouse, rat demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal NPY and catecholamine productionFormula:C123H215N39O28SPurezza:98%Colore e forma:SolidPeso molecolare:2720.33CB2R probe 1
CAS:<p>CB2R Probe 1, a cannabinoid 2 receptor (CB2R) fluorescent probe, exhibits both safety and environmental friendliness, boasting a dissociation constant (K i) of</p>Formula:C36H42N4O4Colore e forma:SolidPeso molecolare:594.74Neuropeptide S(Rat)
CAS:Potent endogenous neuropeptide S receptor (NSPR) agonist (EC50 = 3.2 nM).Formula:C95H160N34O27Purezza:98%Colore e forma:SolidPeso molecolare:2210.52Sch 202596
CAS:Sch 202596 is a selective non-peptide antagonist of GAL-1 receptor.Formula:C25H22Cl2O12Colore e forma:SolidPeso molecolare:585.34ELA-11(human)
CAS:Apelin receptor agonist with high affinity (Ki = 14 nM). Blocks cAMP production and promotes β-arrestin activation; derived from ELA-32.Formula:C58H90N16O13S2Purezza:98%Colore e forma:SolidPeso molecolare:1283.57Clozapine N-oxide dihydrochloride
CAS:Clozapine N-oxide dihydrochloride is a derivative of Clozapine and an agonist of DREADDs.Formula:C18H21Cl3N4OPurezza:98.11%Colore e forma:SolidPeso molecolare:415.74α1A-AR Degrader 9c
CAS:α1A-AR Degrader 9c is a potent, selective, and reversible PROTAC degrader targeting the α1A adrenergic receptor (α1A-AR) with a DC50 of 2.86 μM.Formula:C38H43N11O11Purezza:98%Colore e forma:SolidPeso molecolare:829.8212-epi Leukotriene B4
CAS:LTB4 is made enzymatically (12(R)-specific) and non-enzymatically (6-trans-12-epi mix). 12-epi LTB4 has low receptor activity.Formula:C20H32O4Colore e forma:SolidPeso molecolare:336.472GLP-1 receptor agonist 9 citrate
<p>GLP-1 receptor agonist 9 citrate is an agonist of GLP-1.</p>Formula:C38H39ClFN3O12Purezza:98.76%Colore e forma:SolidPeso molecolare:784.18Isobutyryl-L-carnitine
CAS:Isobutyryl-L-carnitine is a member of the class of compounds known as acylcarnitines. Isobutyryl-L-carnitine is a product of the acyl-CoA dehydrogenases.Formula:C11H21NO4Purezza:98%Colore e forma:SolidPeso molecolare:231.29GLP-1 (9-36) amide
CAS:GLP-1 (9-36) amide is an antagonist at the human GLP-1 receptor.Formula:C140H214N36O43Purezza:97%Colore e forma:SolidPeso molecolare:3089.41HAEGTFTSD acetate(926018-45-3 free base)
HAEGTFTSD acetate is the first N-terminal 1-9 residues of GLP-1 peptide.The GLP-1 (7-36) amide is a product of the preproglucagon gene, which is secreted fromFormula:C42H61N11O19Purezza:98%Colore e forma:SolidPeso molecolare:1024.01[Ala11,D-Leu15]-Orexin B(human)
CAS:OX2 receptor agonist with 400x selectivity vs OX1. EC50: 0.13 nM (OX2), 52 nM (OX1).Formula:C120H206N44O35SPurezza:98%Colore e forma:SolidPeso molecolare:2857.28Methdilazine
CAS:Methdilazine: oral antibiotic, histamine antagonist, fights mycobacterium (MIC 5-15 μg/mL) for infectious disease research.Formula:C18H20N2SColore e forma:SolidPeso molecolare:296.43Adrenomedullin (16-31), human TFA
Human adrenomedullin (16-31) TFA, fragment 16-31, binds CGRP1 receptor, raises rat blood pressure, not cats’.Formula:C84H130F3N25O23S2Colore e forma:SolidPeso molecolare:1979.21Maceneolignan H
CAS:Maceneolignan H, a neolignane from Myristica fragrans, selectively blocks CCR3 (EC50=1.4μM) with allergy research potential.Formula:C24H30O7Colore e forma:SolidPeso molecolare:430.49TGR5 agonist 2
TGR5 agonist 2 (compound 19) serves as a highly potent agonist of TGR5, demonstrating an EC50 value of 0.27 µM [1].Formula:C29H50NNaO6SColore e forma:SolidPeso molecolare:563.77Amylin (8-37), human
CAS:Human-derived Amylin (8-37) is a vasodilator in rat arteries and forms aggregates linked to type II diabetes.Formula:C138H216N42O45Colore e forma:SolidPeso molecolare:3183.495Danshenol B
Danshenol B is a natural product that can be used as a reference standard.Formula:C22H26O4Colore e forma:SolidPeso molecolare:354.446Zicronapine fumarate
CAS:Zicronapine fumarate, an antipsychotic, targets D1/D2 & 5-HT2A receptors; may treat neuropsychiatric conditions.Formula:C26H31ClN2O4Colore e forma:SolidPeso molecolare:470.99Ghrelin receptor full agonist-2
CAS:Ghrelin receptor full agonist-2 is a highly potent Ghrelin receptor full agonist.Formula:C26H28ClN5O5SColore e forma:SolidPeso molecolare:558.05Angiopeptin
CAS:Angiopeptin is a synthetic octapeptide analog of somatostatin; suppresses accelerated transplant atherosclerosis in rabbit heart arteries.Formula:C54H71N11O10S2Colore e forma:SolidPeso molecolare:1098.34α-MSH TFA
CAS:α-Melanocyte-stimulating hormone (α-MSH) is a 13-amino acid peptide hormone produced by post-translational processing of proopiomelanocortin (POMC) in theFormula:C79H110F3N21O21SColore e forma:SolidPeso molecolare:1778.93SR142948A
CAS:SR142948A is a selective and reversible non-peptide neurotensin receptor antagonist blocking hypothermia and analgesic effects, NMDA-induced dopamine release.Formula:C39H52ClN5O6Purezza:98%Colore e forma:SolidPeso molecolare:722.31PACAP (6-38), human, ovine, rat TFA
PACAP (6-38) is a PACAP receptor blocker with IC50s of 30, 600, 40 nM for type I, VIP1, and VIP2 receptors.Formula:C184H301N56FO47SPurezza:98%Colore e forma:SolidPeso molecolare:4138.76Amitraz
CAS:Amitraz (NSC 324552): white monoclinic crystals, mp 86-87°C, water-insoluble, used as acaricide and in canine demodectic mange.Formula:C19H23N3Purezza:99.88%Colore e forma:White/Pale Yellow Crystalline SolidPeso molecolare:293.41Mosapride citrate dihydrate
CAS:<p>Mosapride Citrate, a 5-HT4 agonist, boosts gut movement by enhancing acetylcholine release.</p>Formula:C27H35ClFN3O11Purezza:98%Colore e forma:SolidPeso molecolare:632.04KwFwLL-NH2
CAS:KwFwLL-NH2 is a hexapeptide that serves as a ligand for the ghrelin receptor (ghrelin receptor). This compound acts as a specific inverse agonist for the ghrelin receptor, exhibiting moderate potency (EC50=45.6 nM).Formula:C49H66N10O6Colore e forma:SolidPeso molecolare:891.11Adrenomedullin (1-50), rat
CAS:Rat adrenomedullin (1-50) is a 50-AA peptide; induces arterial vasodilation by activating CGRP1 receptors.Formula:C248H381N77O75S5Purezza:98%Colore e forma:SolidPeso molecolare:5729.5β-CGRP (mouse)
β-CGRP (mouse), a calcitonin gene-related peptide, induces vasodilation and is applicable in research areas including cardiovascular, pro-inflammatory, migraine, and metabolic studies.Formula:C165H265N49O55S2Colore e forma:SolidPeso molecolare:3879.29Neuropeptide Y(29-64)
CAS:Neuropeptide Y(29-64) is a 36 amino acid peptide, a fragment of Neuropeptide Y.Formula:C189H284N54O58SPurezza:98%Colore e forma:SolidPeso molecolare:4272.7Adenosine receptor agonist 1
<p>Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.</p>Formula:C12H14ClN5O2SeColore e forma:SolidPeso molecolare:374.68Y1 receptor antagonist 1 formic
H 409-22 isomer formic, a formate salt of Y1 receptor antagonist 1, is an antagonist of the neuropeptide Y1 receptor (neuropeptide Y1 receptor). This compound effectively blocks the actions of the receptor, playing a crucial role in modulating physiological responses.Formula:C29H35N5O5Colore e forma:SolidPeso molecolare:533.62cAC 253 acetate
<p>cAC 253 acetate (TP2135 Free base) is an amylin antagonist. cAC 253 acetate inhibits 125I-adrenomedullin binding, with an IC50 of 25 nM.</p>Formula:C128H206N42O42S2Purezza:98.16% - 99.99%Colore e forma:SoildPeso molecolare:3069.39BA 1
CAS:Potent BB1, BB2, and BB3 agonist; IC50: 0.26, 1.55, 2.52 nM. Boosts glucose transport in myocytes, promotes cancer cell growth in vitro.Formula:C57H76N14O11Purezza:98%Colore e forma:SolidPeso molecolare:1133.32(S)-V-0219 hydrochloride
(S)-V-0219 hydrochloride, a GLP-1R PAM, triggers calcium in hGLP-1R HEK cells, lowers glucose in mice, and reduces fasting hunger.Formula:C20H26ClF3N4O2Colore e forma:SolidPeso molecolare:446.8915(S)-15-methyl Prostaglandin E2
CAS:15(S)-15-methyl PGE2: A stable PGE2 analog; strong antiulcer with double PGE2 affinity; excels PGE1 in uterine contraction.Formula:C21H34O5Colore e forma:SolidPeso molecolare:366.49Cortistatin-14 acetate
<p>Cortistatin-14 acetate, a neuropeptide have structural similarity to somatostatin-14, binds and exerts its function via the somatostatin receptors (sst1-sst5).</p>Formula:C83H118N20O20S2Purezza:98.24% - 99.63%Colore e forma:SoildPeso molecolare:1780.08Senktide TFA
Senktide TFA is a potent and selective neurokinin 3 (NK3) receptor agonist with an EC50 of 0.5-3 nM, while showing significantly weaker activity on NK1 receptors (EC50=35 µM). It is a promising candidate for research in neurological disorders.Colore e forma:Odour SolidCYM5442 hydrochloride
CAS:CYM 5442 HCl: potent, selective S1P1 agonist (EC50 = 1.35 nM), induces MAPK activation & lymphopenia, brain-penetrant.Formula:C23H28ClN3O4Colore e forma:SolidPeso molecolare:445.94MGV354
MGV354 is a soluble activator of guanylate cyclase(sGC) with EC 50 s of <0.5 nM, and 5 nM in CHO and GTM-3 E cells, respectively [1] [2].Formula:C35H37N5O3Purezza:98%Colore e forma:SolidPeso molecolare:575.7(R)-Preclamol hydrochloride
CAS:(R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.Formula:C14H22ClNOColore e forma:SolidPeso molecolare:255.78Bay 55-9837
CAS:Selective VPAC2 agonist; EC50: 0.4 nM (VPAC2), 100 nM (VPAC1), >1000 nM (PAC1). Enhances insulin secretion, reduces HIV-1 replication.Formula:C167H270N52O46Purezza:98%Colore e forma:SolidPeso molecolare:3742.2919(R)-hydroxy Prostaglandin E1
CAS:19(R)-hydroxy Prostaglandin E1 is an agonist of EP1 and EP3 receptor subtypes and exhibits contractile activity on smooth muscle and is the major prostaglandinFormula:C20H34O6Colore e forma:SolidPeso molecolare:370.486Phoenixin-14 TFA
Phoenixin-14 TFA (PNX-14 TFA) is an endogenous neuropeptide that can modulate GnRH receptor expression and exerts anxiolytic effects.Formula:C75H110N18O20·xC2HF3O2Purezza:99.11%Colore e forma:SolidPeso molecolare:1583.78 (free base)Thioperamide maleate
CAS:Thioperamide maleate (MR-12842 maleate) is an effective and selective antagonist of H3 receptor (Ki = 4.3 nM) for inhibition of [3H]histamine synthesis (Ki = 31Formula:C19H28N4O4SPurezza:98.48%Colore e forma:SolidPeso molecolare:408.522-Furoyl-LIGRLO-amide
CAS:2-Furoyl-LIGRLO-amide TFA is a peptide that acts as a proteinase-activated receptor-2 (PAR2) agonist, and contains a furoyl group addition at its N-terminal.Formula:C36H63N11O8Purezza:98%Colore e forma:SolidPeso molecolare:777.95GRK-IN-1
CAS:<p>4-Amino-5-(bromomethyl)-2-methylpyrimidine used in vitamin B1 analogs and esters synthesis.</p>Formula:C6H10Br3N3Colore e forma:SolidPeso molecolare:363.879GLP-1(7-36), amide acetate
CAS:GLP-1(7-36), amide acetate is a derivative of GLP-1 peptide , activate the GLP-1 receptor, promote insulin secretion,Type 2 diabetes mellitus and obesity.Formula:C151H230N40O47Purezza:99.89%Colore e forma:SolidPeso molecolare:3357.68Pal-Glu(OSu)-OH
CAS:Pal-Glu(OSu)-OH is a Liraglutide side chain, a GLP-1 agonist for type 2 diabetes study.Formula:C25H42N2O7Colore e forma:SolidPeso molecolare:482.618ELA-21 (human)
CAS:Apelin receptor agonist with high affinity for normal/PAH hearts (pKi 9.31/9.46). Blocks cAMP, promotes β-arrestin in vitro. Part of ELA-32.Formula:C112H184N40O25S3Purezza:98%Colore e forma:SolidPeso molecolare:2587.125-HT1AR/5-HT6R ligand-1
5-HT1AR/5-HT6R ligand-1 (Compound PP13) functions as a ligand for the 5-HT receptor, demonstrating high affinity for 5-HT1AR, 5-HT6R, and 5-HT7R with Ki values of 19, 69, and 198 nM, respectively. In HEK293 cells, it inhibits cAMP production with EC50 values of 1535, 488, and 53 nM for these receptors. Additionally, 5-HT1AR/5-HT6R ligand-1 exhibits antiproliferative effects on several cancer cell lines, including 1321N1, U87MG, MCF7, and AsPC-1, with IC50 values of 9.6, 13.6, 19.3, and 14.6 μM, respectively. The compound also shows antagonistic activity towards the dopamine receptor D2R, with a Ki of 1903 nM.Formula:C25H29ClN4O2SColore e forma:SolidPeso molecolare:485.04Apelin-17(human, bovine)
CAS:Endogenous apelin receptor agonist. Potently inhibits forskolin-stimulated cAMP accumulation (pIC50 = 9.94).Formula:C96H156N34O20SPurezza:98%Colore e forma:SolidPeso molecolare:2138.56Donetidine
CAS:Donetidine is a histamine H2 receptor antagonist used to treat digestive disorders.Formula:C20H25N5O3SPurezza:99.32%Colore e forma:SolidPeso molecolare:415.51MM 07
CAS:Biased agonist for apelin/G protein pathway, enhances eNOS and cell growth, reduces apoptosis, improves heart function, and dilates vessels.Formula:C67H106N22O14S3Purezza:98%Colore e forma:SolidPeso molecolare:1539.9BAY-747
CAS:BAY-747: oral, brain-penetrant sGC stimulator; improves rat memory, cognition, lowers blood pressure, aids Duchenne muscular dystrophy.Formula:C22H26F2N4O2Colore e forma:SolidPeso molecolare:416.46LAS190792
CAS:LAS190792 (AZD8999) is a dual muscarinic antagonist/β2-agonist, pIC50s (M1-M5, β1-β3): 8.9-5.6; used as a bronchodilator.Formula:C39H43ClN4O9S2Colore e forma:SolidPeso molecolare:811.36GLP-1(9-36)amide TFA
GLP-1(9-36)amide TFA, a DPP-4 metabolite of GLP-1(7-36) amide, antagonizes human pancreatic GLP-1 receptor.Formula:C142H215F3N36O45Colore e forma:SolidPeso molecolare:3203.43BMS-604992 dihydrochloride
CAS:BMS-604992 dihydrochloride is a selective GHSR agonist with high affinity (Ki=2.3 nM) and potent activity (EC50=0.4 nM), stimulating rodent appetite.Formula:C24H33Cl2N7O5Colore e forma:SolidPeso molecolare:570.47Galanin (1-29)(rat, mouse)
CAS:Non-selective galanin agonist; Ki: GAL1-0.98, GAL2-1.48, GAL3-1.47 nM. Anticonvulsant, stops full seizures in rats.Formula:C141H211N43O41Purezza:98%Colore e forma:White Lyophilized PowderPeso molecolare:3164.499Pexopiprant
CAS:Pexopiprant, a potent oral antagonist of the prostaglandin D2 receptor 2 (DP2) with a K i value less than 100nM, is a valuable compound for asthma research.Formula:C21H17Cl2F2NO4Colore e forma:SolidPeso molecolare:456.27NPC 567
CAS:NPC 567 is an antagonist of the bradykinin receptor.Formula:C60H87N19O13Purezza:98%Colore e forma:SolidPeso molecolare:1282.48NSC380324
NSC380324 is a P2Y12 receptor antagonist with antiplatelet properties, which can be employed in research on atherosclerotic cardiovascular diseases.Formula:C31H24N4O4Colore e forma:SolidPeso molecolare:516.55L-770644
CAS:L-770644 is an agonist of B3 adrenergic receptor.Formula:C30H37N7O4SColore e forma:SolidPeso molecolare:591.72VU0453379 hydrochloride
VU0453379 hydrochloride: selective CNS-penetrant GLP-1R PAM, EC50 1.3 μM.Formula:C26H35ClN4O2Colore e forma:SolidPeso molecolare:471.03Neuropeptide Y (13-36), amide, human
CAS:Neuropeptide Y (13-36), amide, human is a neuropeptide Y receptor agonist.Formula:C134H207N41O36SPurezza:98%Colore e forma:SolidPeso molecolare:3000.4Neuropeptide Y (22-36)
CAS:Neuropeptide Y (22-36) is a 15-amino acid fragment of NPY, which is abundant in the mammalian brain and involved in multiple physiological functions.Formula:C85H139N29O21Purezza:98%Colore e forma:SolidPeso molecolare:1903.19Cagrilintide acetate
.Cagrilintide is a long-acting amylin analog,treat diabetes and obesity by reducing appetite through activation of the AMY3R and calcitonin receptor.Formula:C196H316N54O61S2Purezza:99.88%Colore e forma:SolidPeso molecolare:4469.06Sarafotoxin S6b
CAS:non-selective endothelin receptor agonistFormula:C110H163N27O34S5Purezza:98%Colore e forma:SolidPeso molecolare:2567.96P2Y14R antagonist 3
P2Y14R antagonist 3 (compound A) is an orally active P2Y14R antagonist with an IC50 of 23.60 nM and a Kd of 7.26 μM. It mitigates lung injury in mice induced by Lipopolysaccharides (LPS) and can be utilized in the study of inflammatory diseases.Formula:C26H25N5O5Colore e forma:SolidPeso molecolare:487.51Navafenterol saccharinate
CAS:AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).Formula:C45H47N7O9S3Colore e forma:SolidPeso molecolare:926.09Pramlintide TFA
Pramlintide TFA, a polypeptide analogue of human amylin and an antidiabetic agent, exhibits antineoplastic properties in colorectal cancer [1].Formula:C173H268N51F3O55S2Colore e forma:SolidPeso molecolare:4063.4GIP/GLP-1 dual receptor agonist-1
CAS:Compound 4: GIP/GLP-1 agonist for metabolic/fatty liver disease research.Colore e forma:SolidTaspoglutide
CAS:Taspoglutide is a long-acting glucagon-like peptide 1 (GLP-1) receptor agonist(EC50 value of 0.06 nM),and for treatment of type 2 diabetesFormula:C152H232N40O45Purezza:98%Colore e forma:SolidPeso molecolare:3339.763[Asu1,6-Arg8]Vasopressin
CAS:[Asu1,6-Arg8]Vasopressin, a vasopressin agonist, boosts cAMP and ACTH release in cultured rat pituitary cells.Formula:C48H68N14O12Colore e forma:SolidPeso molecolare:1033.14LSN3160440
CAS:LSN3160440 is a GLP-1R allosteric modulator and PPI stabilizer aiding inactive GLP-1 attachment.Formula:C27H27Cl2N3OColore e forma:SolidPeso molecolare:480.43Urocortin II, human
Human urocortin (hUcn) II is a new member of the corticotropin-releasing-factor (CRF) family. It selectively binds to the CRF2 receptor.Formula:C194H339N63O54SPurezza:98%Colore e forma:SolidPeso molecolare:4450.28D[LEU4,LYS8]-VP TFA
<p>D[LEU4,LYS8]-VP TFA: V1b receptor agonist; K_i: 0.16 nM (rat), 0.52 nM (human), 1.38 nM (mouse); weak antidiuretic/vasopressor/oxytocic.</p>Formula:C49H68F3N11O13S2Colore e forma:SolidPeso molecolare:1140.25Latanoprost lactone diol
CAS:Latanoprost lactone diol, a key intermediate for synthesizing Latanoprost (a prostaglandin F2α analogue), lowers IOP by activating FP receptors.Formula:C18H24O4Purezza:98%Colore e forma:White Or Almost White Crystalline PowderPeso molecolare:304.38Etelcalcetide
CAS:Etelcalcetide (AMG 416), a synthetic peptide CaSR activator, treats secondary hyperparathyroidism in hemodialysis patients.Formula:C38H73N21O10S2Purezza:98%Colore e forma:SolidPeso molecolare:1048.2615(S)-HpEPE
CAS:15(S)-HpEPE, a monohydroperoxy fatty acid, forms when 15-lipoxygenase acts on EPA, with expected biological activities akin to 15(S)-HpETE.Formula:C20H30O4Colore e forma:SolidPeso molecolare:334.456Amylin (8-37) (human)
CAS:Amylin (8-37) (human) is a fragment of human IAPP with a hairpin structure.Formula:C138H215N41O46Colore e forma:SolidPeso molecolare:3184.43Apelin-36(rat, mouse)
CAS:Endogenous APJ agonist from adipocytes; binds APJ tightly, inhibits cAMP, regulates heart function and fluid balance, blocks some HIV strains.Formula:C185H304N68O43SPurezza:98%Colore e forma:SolidPeso molecolare:4200.93
![[D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1931.webp&w=3840&q=75)
![[Ala11,D-Leu15]-Orexin B(human)](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1975.webp&w=3840&q=75)
![[Asu1,6-Arg8]Vasopressin](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT76510.webp&w=3840&q=75)
