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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

Mostrare 18 più sottocategorie

Trovati 5352 prodotti di "Proteina G/GPCR"

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  • LY 78335
    Targetmol
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    LY 78335

    CAS:
    <p>LY 78335 (1-(2,3-Dichlorophenyl)ethanamine hydrochloride) is a phenylethanolamine-N-methyltransferase (PNMT) inhibitor.</p>
    Formula:C8H10Cl3N
    Purezza:99.30% - 99.81%
    Colore e forma:Solid
    Peso molecolare:226.53

    Ref: TM-T22956

  • Alloxazine
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    Alloxazine

    CAS:
    <p>Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.</p>
    Formula:C10H6N4O2
    Purezza:99.75%
    Colore e forma:Solid
    Peso molecolare:214.18

    Ref: TM-T22234

  • Taprenepag
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    Taprenepag

    CAS:
    <p>Taprenepag (CP-544326) (CP-544326) is a potent and selective prostaglandin E2 receptor agonist (EC50 = 2.8 nM).</p>
    Formula:C24H22N4O5S
    Purezza:98.89% - 99.15%
    Colore e forma:Solid
    Peso molecolare:478.52

    Ref: TM-T3174

  • Talnetant hydrochloride
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    Talnetant hydrochloride

    CAS:
    <p>Talnetant (SB 223412) hydrochloride, an NK3 antagonist, selectively binds hNK-3 at 1.4 nM, much less to hNK-2, none to hNK-1 at 100 μM.</p>
    Formula:C25H23ClN2O2
    Colore e forma:Solid
    Peso molecolare:418.92

    Ref: TM-T62199

  • Arformoterol Tartrate
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    Arformoterol Tartrate

    CAS:
    <p>Arformoterol Tartrate ((R,R)-Formoterol tartrate) is the tartrate salt of arformoterol.</p>
    Formula:C23H30N2O10
    Purezza:99.98%
    Colore e forma:Solid
    Peso molecolare:494.49

    Ref: TM-T22245

  • BP 897
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    BP 897

    CAS:
    <p>BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.</p>
    Formula:C26H31N3O2
    Purezza:99.44%
    Colore e forma:Solid
    Peso molecolare:417.54

    Ref: TM-T9100

  • Jatrorrhizine
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    Jatrorrhizine

    CAS:
    <p>Jatrorrhizine (neprotin) is a protoberberine alkaloid isolated from Enantia chlorantha (Annonaceae) and other species.</p>
    Formula:C20H20NO4
    Purezza:97.18% - 99.06%
    Colore e forma:Solid
    Peso molecolare:338.38

    Ref: TM-T3933

  • Guanabenz Acetate
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    Guanabenz Acetate

    CAS:
    <p>Guanabenz Acetate (Wytensin) is a specific agonist of adrenergic receptor.</p>
    Formula:C8H8Cl2N4·C2H4O2
    Purezza:99% - 99.66%
    Colore e forma:White Solid From Acetonitrile White Solid
    Peso molecolare:291.13

    Ref: TM-T6522

  • Haloperidol decanoate
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    Haloperidol decanoate

    CAS:
    <p>Haloperidol decanoate (KD 16), an antipsychotic, treats schizophrenia and mood disorders as an intramuscular ester.</p>
    Formula:C31H41ClFNO3
    Purezza:99.57% - 99.72%
    Colore e forma:Solid
    Peso molecolare:530.11

    Ref: TM-T25487

  • Bretylium tosylate
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    Bretylium tosylate

    CAS:
    <p>Bretylium tosylate is an inhibitor of the presynaptic release of vasoconstrictor neurotransmitters, a available antiarrhythmic drug for ventricular arrhythmias.</p>
    Formula:C18H24BrNO3S
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:414.36

    Ref: TM-T7386

  • SB-222200
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    SB-222200

    CAS:
    <p>SB-222200 is a selective, reversible, and competitive antagonist of the human NK-3 receptor(Ki=4.4 nM).</p>
    Formula:C26H24N2O
    Purezza:97.13%
    Colore e forma:Solid
    Peso molecolare:380.48

    Ref: TM-T16849

  • Talastine HCl
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    Talastine HCl

    CAS:
    <p>Talastine is an antihistamine drug.</p>
    Formula:C19H22ClN3O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:343.86

    Ref: TM-T24851

  • KB-5492 anhydrous
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    KB-5492 anhydrous

    CAS:
    <p>KB 5492 is an agent of anti-ulcer. It preventing cysteamine-induced duodenal ulcers by stimulating duodenal HCO3- secretion.</p>
    Formula:C27H34N2O10
    Colore e forma:Solid
    Peso molecolare:546.57

    Ref: TM-T24254

  • Dasotraline
    Targetmol
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    Dasotraline

    CAS:
    <p>Dasotraline: a triple reuptake inhibitor targeting DA, NE, and 5-HT with IC50 values of 4, 6, 11 nM. Possible new antidepressant class.</p>
    Formula:C16H15Cl2N
    Colore e forma:Solid
    Peso molecolare:292.2

    Ref: TM-T60607

  • Lys-[Des-Arg9]Bradykinin,TFA
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    Lys-[Des-Arg9]Bradykinin,TFA

    <p>Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and &gt; 30000 nM at human B1 and B2</p>
    Formula:C54H75F6N13O15
    Purezza:97.35%
    Colore e forma:Solid
    Peso molecolare:1260.24

    Ref: TM-TP1918L

  • HS024
    Targetmol
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    HS024

    CAS:
    <p>HS024 is a highly potent melanocortin MC4 receptor antagonist, increases food intake, and blocks α-MSH- and MTII-induced hypotension and bradycardia in rats.</p>
    Formula:C58H79N19O10S2
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:1266.5

    Ref: TM-TP1898

  • Regadenoson hydrate
    Targetmol
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    Regadenoson hydrate

    CAS:
    <p>Regadenoson is an A2A adenosine receptor agonist, a coronary vasodilator commonly used in pharmacologic stress testing.</p>
    Formula:C15H20N8O6
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:408.37

    Ref: TM-T26054

  • Fipamezole HCl
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    Fipamezole HCl

    CAS:
    <p>Fipamezole HCl, a α2-adrenoceptor antagonist, is used potentially for the treatment of dyskinesia associated with Parkinson's disease.</p>
    Formula:C14H16ClFN2
    Colore e forma:Solid
    Peso molecolare:266.74

    Ref: TM-T27321

  • BQ-123
    Targetmol
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    BQ-123

    CAS:
    <p>BQ-123 is a selective endothelin A receptor (ETA) antagonist with IC50 of 7.3 nM. Phase 2.</p>
    Formula:C31H42N6O7
    Purezza:99.22% - ≥95%
    Colore e forma:Solid
    Peso molecolare:610.7

    Ref: TM-T6792

  • Metadoxine
    Targetmol
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    Metadoxine

    CAS:
    <p>Metadoxine (Metadoxil) is a neurotransmitter stimulant.</p>
    Formula:C8H11NO3·C5H7NO3
    Purezza:99.19%
    Colore e forma:Off-White Powder
    Peso molecolare:298.29

    Ref: TM-T3269