CymitQuimica logo
Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

Mostrare 18 più sottocategorie

Trovati 5352 prodotti di "Proteina G/GPCR"

Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
prodotti per pagina.
  • (R)-Propranolol hydrochloride
    Targetmol
    + Info

    (R)-Propranolol hydrochloride

    CAS:
    <p>(R)-Propranolol hydrochloride (Dexpropranolol hydrochloride) is the less active enantiomer of the anti-adrenoceptor (β-adrenoceptor) antagonist propranolol.</p>
    Formula:C16H22ClNO2
    Purezza:98.63% - 99.01%
    Colore e forma:Solid
    Peso molecolare:295.8

    Ref: TM-T20898

  • Capromorelin Tartrate
    Targetmol
    + Info

    Capromorelin Tartrate

    CAS:
    <p>Capromorelin Tartrate (CP 424391-18) is a potent, orally active growth hormone secretagogue receptor (GHSR) agonist (Ki: 7 nM for hGHS-R1a).</p>
    Formula:C32H41N5O10
    Purezza:97.69%
    Colore e forma:Solid
    Peso molecolare:655.7

    Ref: TM-TQ0022

  • Vanoxerine dihydrochloride
    Targetmol
    + Info

    Vanoxerine dihydrochloride

    CAS:
    <p>Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)</p>
    Formula:C28H34Cl2F2N2O
    Purezza:98.16% - 98.35%
    Colore e forma:White Solid
    Peso molecolare:523.49

    Ref: TM-T7153

  • Pramipexole dihydrochloride hydrate
    Targetmol
    + Info

    Pramipexole dihydrochloride hydrate

    CAS:
    <p>Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.</p>
    Formula:C10H17N3S·2HCl·H2O
    Purezza:99.68%
    Colore e forma:White To Off-White Crystalline Powder
    Peso molecolare:302.26

    Ref: TM-T6951

  • Sultopride hydrochloride
    Targetmol
    + Info

    Sultopride hydrochloride

    CAS:
    <p>Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.</p>
    Formula:C17H27ClN2O4S
    Purezza:≥95%
    Colore e forma:White Or Yellowish Powder
    Peso molecolare:390.93

    Ref: TM-T7180

  • SHU 9119 acetate
    Targetmol
    + Info

    SHU 9119 acetate

    <p>SHU 9119 acetate: hMC3R &amp; hMC4R antagonist, hMC5R partial agonist. IC50: MC3R 0.23nM, MC4R 0.06nM, MC5R 0.09nM.</p>
    Formula:C56H75N15O11
    Purezza:99.8%
    Colore e forma:Solid
    Peso molecolare:1134.29

    Ref: TM-T16879L

  • TGR5 Receptor Agonist
    Targetmol
    + Info

    TGR5 Receptor Agonist

    CAS:
    TGR5 is a potent TGR5(GPCR19) agonist.
    Formula:C18H14Cl2N2O2
    Purezza:99.77% - ≥95%
    Colore e forma:Solid
    Peso molecolare:361.22

    Ref: TM-T1824

  • Metoclopramide
    Targetmol
    + Info

    Metoclopramide

    CAS:
    <p>Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.</p>
    Formula:C14H22ClN3O2
    Purezza:99.75%
    Colore e forma:Solid
    Peso molecolare:299.80

    Ref: TM-T4616

  • GR-73632
    Targetmol
    + Info

    GR-73632

    CAS:
    <p>Potent and selective tachykinin NK1 receptor agonist (EC50 = 2 nM in guinea pig vas deferens).</p>
    Formula:C40H59N7O6S
    Purezza:99.68%
    Colore e forma:Solid
    Peso molecolare:766

    Ref: TM-TP1572

  • Naftopidil dihydrochloride
    Targetmol
    + Info

    Naftopidil dihydrochloride

    CAS:
    <p>Naftopidil dihydrochloride (KT-611 2HCl) is a selective 5-HT1A and α1-adrenergic receptor antagonist with IC50 of 0.1 μM and 0.2 μM, respectively.</p>
    Formula:C24H28N2O3·2HCl
    Purezza:99.76%
    Colore e forma:White Solid
    Peso molecolare:465.41

    Ref: TM-T6600

  • 5-Iodotubercidin
    Targetmol
    + Info

    5-Iodotubercidin

    CAS:
    <p>5-Iodotubercidin (NSC-113939) is a potent adenosine kinase inhibitor with IC50 of 26 nM.</p>
    Formula:C11H13IN4O4
    Purezza:99.98%
    Colore e forma:Tan Solid
    Peso molecolare:392.15

    Ref: TM-T6745

  • Zotepine
    Targetmol
    + Info

    Zotepine

    CAS:
    <p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>
    Formula:C18H18ClNOS
    Purezza:99.78%
    Colore e forma:Solid
    Peso molecolare:331.86

    Ref: TM-T19680

  • Exo-1
    Targetmol
    + Info

    Exo-1

    CAS:
    <p>Exo-1 (Methyl 3-(4-fluorobenzoyl)-6-methyl-2-pyridinecarboxylate) is a synthetic compound that has been shown to affect the metabolism of various nutrients, as</p>
    Formula:C15H12FNO3
    Purezza:99.45%
    Colore e forma:Solid
    Peso molecolare:273.26

    Ref: TM-T9200

  • Mebhydrolin
    Targetmol
    + Info

    Mebhydrolin

    CAS:
    <p>Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.</p>
    Formula:C19H20N2
    Purezza:99.3% - ≥98%
    Colore e forma:Solid
    Peso molecolare:276.38

    Ref: TM-T7085

  • Fexofenadine
    Targetmol
    + Info

    Fexofenadine

    CAS:
    <p>Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.</p>
    Formula:C32H39NO4
    Purezza:99.35%
    Colore e forma:White To Off-White Solid
    Peso molecolare:501.66

    Ref: TM-T21390

  • Idalopirdine Hydrochloride
    Targetmol
    + Info

    Idalopirdine Hydrochloride

    CAS:
    <p>Idalopirdine Hydrochloride (Lu AE58054 Hydrochloride) is an in-vivo binding affinity and effect, in-vitro selectivity and potency of 5-HT(6)R antagonist (Ki: 0.</p>
    Formula:C20H20ClF5N2O
    Purezza:99.77%
    Colore e forma:Solid
    Peso molecolare:434.83

    Ref: TM-T22936

  • Dimemorfan phosphate
    Targetmol
    + Info

    Dimemorfan phosphate

    CAS:
    <p>Dimemorfan phosphate (3,17-dimethylmorphinan) is a sigma 1 receptor agonist. Dimemorfan phosphate is used as a potent antitussive.</p>
    Formula:C18H25N·H3O4P
    Purezza:99.65%
    Colore e forma:Solid
    Peso molecolare:353.4

    Ref: TM-T5027

  • TG6-10-1
    Targetmol
    + Info

    TG6-10-1

    CAS:
    <p>TG6-10-1 is an EP2 antagonist.</p>
    Formula:C23H23F3N2O4
    Purezza:99.66% - ≥95%
    Colore e forma:Solid
    Peso molecolare:448.43

    Ref: TM-T2428

  • BAR501
    Targetmol
    + Info

    BAR501

    CAS:
    <p>BAR501是高效选择性的 GPBAR1激动剂(EC50:1 μM)。</p>
    Formula:C26H46O3
    Purezza:99.29% - 99.68%
    Colore e forma:Solid
    Peso molecolare:406.64

    Ref: TM-T4083

  • ANP(1-28) Acetate (human, porcine)
    Targetmol
    + Info

    ANP(1-28) Acetate (human, porcine)

    CAS:
    <p>Carperitide acetate: 28-amino acid hormone from human heart, counters cardiac injury/stretch, reduces endothelin-1.</p>
    Formula:C129H207N45O41S3
    Purezza:98.24%
    Colore e forma:Solid
    Peso molecolare:3140.5

    Ref: TM-TP1220L