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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

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Trovati 5352 prodotti di "Proteina G/GPCR"

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  • Quipazine
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    Quipazine

    CAS:
    <p>Quipazine: 5-HT agonist, Ki 1.4 nM at 5-HT3R, anti-SARS-CoV-2 (EC50 31.64 μM), for neurological research.</p>
    Formula:C13H15N3
    Colore e forma:Solid
    Peso molecolare:213.28

    Ref: TM-T73341

  • Brefonalol
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    Brefonalol

    CAS:
    <p>Brefonalol is a vasodilating beta-adrenergic receptor blocker.</p>
    Formula:C22H28N2O2
    Colore e forma:Solid
    Peso molecolare:352.47

    Ref: TM-T30586

  • Raclopride tartrate
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    Raclopride tartrate

    CAS:
    <p>Raclopride is a selective antagonist on D2 dopamine receptor ( D2 Ki: 1.8 nm, D3 Ki: 3.5 nm, D4 Ki: 2400, D1 Ki: 18000 nM).</p>
    Formula:C19H26Cl2N2O9
    Colore e forma:Solid
    Peso molecolare:497.32

    Ref: TM-T7635L

  • RU 24969 succinate
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    RU 24969 succinate

    CAS:
    <p>RU 24969 succinate, a 5-HT receptor agonist, exhibits K i values of 0.38 nM for 5-HT 1B and 2.5 nM for 5-HT 1A, indicating its affinity towards these receptors. It reduces fluid consumption and enhances forward locomotion. This compound is utilized in neurological disease research.</p>
    Formula:C18H22N2O5
    Colore e forma:Solid
    Peso molecolare:346.38

    Ref: TM-T71502

  • Midaglizole
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    Midaglizole

    CAS:
    <p>Midaglizole, an α2-adrenoceptor blocker, raises blood pressure and lowers glucose.</p>
    Formula:C16H17N3
    Colore e forma:Solid
    Peso molecolare:251.33

    Ref: TM-T68098

  • Cangrelor free acid
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    Cangrelor free acid

    CAS:
    <p>Cangrelor, a reversible P2Y12 inhibitor for IV use, was approved in June 2015; it rapidly blocks ADP-induced platelet aggregation.</p>
    Formula:C17H25Cl2F3N5O12P3S2
    Colore e forma:Solid
    Peso molecolare:776.36

    Ref: TM-T70335

  • Eltoprazine dihydrochloride
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    Eltoprazine dihydrochloride

    CAS:
    <p>Eltoprazine dihydrochloride, a drug developed for aggression, is now studied for L-DOPA-induced dyskinesia in Parkinson's.</p>
    Formula:C12H18Cl2N2O2
    Purezza:99.64%
    Colore e forma:Solid
    Peso molecolare:293.19

    Ref: TM-T7746

  • 4-Methylhistamine hydrochloride
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    4-Methylhistamine hydrochloride

    CAS:
    <p>Compound with imidazole ring &amp; amine group; inhibits copper enzymes, affects gene expression.</p>
    Formula:C6H12ClN3
    Purezza:95%
    Colore e forma:Solid
    Peso molecolare:161.633

    Ref: TM-T50049

  • Butyrophenone
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    Butyrophenone

    CAS:
    <p>Butyrophenone (NSC-8463) is a chemical compound. Some of its derivatives are used to treat various psychiatric disorders.</p>
    Formula:C10H12O
    Purezza:99.84%
    Colore e forma:Colourless To Yellow Liquid
    Peso molecolare:148.2

    Ref: TM-T20324

  • BCTC
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    BCTC

    CAS:
    <p>BCTC is a potent TRPV1 antagonist that inhibits capsaicin-induced and acid-induced activation of rat TRPV1 (IC50 of 35 and 6 nM, respectively)</p>
    Formula:C20H25ClN4O
    Purezza:99.21%
    Colore e forma:Solid
    Peso molecolare:372.89

    Ref: TM-T7102

  • Ibutamoren
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    Ibutamoren

    CAS:
    <p>Ibutamoren (MK-677) is a drug which acts as a potent, orally active growth hormone secretagogue, mimicking the GH stimulating action of the endogenous hormone ghrelin. It also alters the metabolism of body fat and so may have an application in the treatment of obesity.</p>
    Formula:C27H36N4O5S
    Purezza:97.59%
    Colore e forma:Solid
    Peso molecolare:528.66

    Ref: TM-T20095

  • GBR 12935
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    GBR 12935

    CAS:
    <p>GBR-12935: selective dopamine inhibitor, used in Parkinson's research.</p>
    Formula:C28H34N2O
    Colore e forma:Solid
    Peso molecolare:414.58

    Ref: TM-T1871L

  • M 1145 acetate
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    M 1145 acetate

    <p>M1145 acetate: chimeric peptide, selective GAL2 agonist, Ki=6.55 nM; &gt;90x affinity vs GAL1, 76x vs GalR3. Enhances galanin signal.</p>
    Formula:C130H209N37O34
    Purezza:99.1%
    Colore e forma:Solid
    Peso molecolare:2834.28

    Ref: TM-TP1991L

  • Loxapine hydrochloride
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    Loxapine hydrochloride

    CAS:
    <p>Loxapine hydrochloride, an oral anti-psychotic, inhibits dopamine and blocks 5-HT receptors.</p>
    Formula:C18H19Cl2N3O
    Colore e forma:Solid
    Peso molecolare:364.27

    Ref: TM-T61381

  • Brompheniramine
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    Brompheniramine

    CAS:
    <p>Brompheniramine, an alkylamine antihistamine, targets H1 receptors (Kd=6.06nM) and has anticholinergic/depressant qualities. Blocks Ca/Na/hERG channels.</p>
    Formula:C16H19BrN2
    Colore e forma:Solid
    Peso molecolare:319.24

    Ref: TM-T60843

  • GSK 789472 hydrochloride
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    GSK 789472 hydrochloride

    CAS:
    <p>GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.</p>
    Formula:C15H22ClN3O
    Purezza:99.89%
    Colore e forma:Solid
    Peso molecolare:295.81

    Ref: TM-T22817

  • Neuropeptide EI, rat acetate
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    Neuropeptide EI, rat acetate

    <p>Neuropeptide EI, rat acetate Displays functional MCH-antagonist and MSH-agonist activity in different behavioral paradigms.</p>
    Formula:C65H102N16O25
    Purezza:95.55%
    Colore e forma:Solid
    Peso molecolare:1507.6

    Ref: TM-TP1578L

  • CYM 50358 hydrochloride (1314212-39-9 free base)
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    CYM 50358 hydrochloride (1314212-39-9 free base)

    CAS:
    <p>CYM50358 HCl is an S1P4 antagonist.</p>
    Formula:C20H19Cl3N2O2
    Purezza:99.57%
    Colore e forma:Solid
    Peso molecolare:425.73

    Ref: TM-T25282

  • N-ACETYLTRYPTAMINE
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    N-ACETYLTRYPTAMINE

    CAS:
    <p>N-ACETYLTRYPTAMINE is a partial agonist for melatonin receptors in the retina. Also used for determination of serotonin N-acetyl transferase.</p>
    Formula:C12H14N2O
    Purezza:98.79%
    Colore e forma:Powder
    Peso molecolare:202.25

    Ref: TM-T8600

  • GR 125743
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    GR 125743

    CAS:
    <p>GR 125743 is a novel antagonist of 5-HT1B/1D receptor.</p>
    Formula:C25H28N4O2
    Purezza:99.76%
    Colore e forma:Solid
    Peso molecolare:416.52

    Ref: TM-T8737