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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

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Trovati 5378 prodotti di "Proteina G/GPCR"

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  • SCH-23390 hydrochloride
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    SCH-23390 hydrochloride

    CAS:
    <p>SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).</p>
    Formula:C17H19Cl2NO
    Purezza:98% - 99.83%
    Colore e forma:Solid
    Peso molecolare:324.24

    Ref: TM-T4369

  • Idazoxan hydrochloride
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    Idazoxan hydrochloride

    CAS:
    <p>Idazoxan hydrochloride (RX 781094) is a benzodioxane-linked imidazole. It has alpha-2 adrenoceptor antagonist activity.</p>
    Formula:C11H12N2O2·HCl
    Purezza:99.42% - 99.84%
    Colore e forma:Solid
    Peso molecolare:240.69

    Ref: TM-T0115

  • Clozapine N-Oxide
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    Clozapine N-Oxide

    CAS:
    View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.
    Formula:C18H19ClN4O
    Purezza:98.65% - 99.94%
    Colore e forma:Solid
    Peso molecolare:342.82

    Ref: TM-T4494

  • SB-334867 free base
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    SB-334867 free base

    CAS:
    <p>SB-334867 free base (SB334867A free base) is a selective orexin-1 (OX1) receptor antagonist.</p>
    Formula:C17H13N5O2
    Purezza:99.67% - >99.99%
    Colore e forma:Solid
    Peso molecolare:319.32

    Ref: TM-T6140

  • Bay 59-3074
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    Bay 59-3074

    CAS:
    <p>Bay 59-3074 is a CB1/CB2 receptor partial agonist (Ki: 48.3/45.5 nM).</p>
    Formula:C18H13F6NO4S
    Purezza:97.68% - 99.69%
    Colore e forma:Solid
    Peso molecolare:453.36

    Ref: TM-T3699

  • RS 504393
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    RS 504393

    CAS:
    RS 504393 is a highly selective CCR2 chemokine receptor antagonist (IC50s: 89 nM and > 100 μM for human recombinant CCR2 and CCR1).
    Formula:C25H27N3O3
    Purezza:98.64% - 99.62%
    Colore e forma:Solid
    Peso molecolare:417.5

    Ref: TM-T5384

  • 2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base)
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    2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base)

    <p>2-Furoyl-LIGRLO-amide TFA(729589-58-6 free base) is a potent and selective protease-activated receptor 2 (PAR2) agonist.</p>
    Formula:C38H64F3N11O10
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:891.98

    Ref: TM-TP1378

  • Rimcazole dihydrochloride
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    Rimcazole dihydrochloride

    CAS:
    <p>Rimcazole dihydrochloride: a σ receptor antagonist, hydrochloride salt, blocks dopamine uptake.</p>
    Formula:C21H28ClN3
    Purezza:99.63%
    Colore e forma:Solid
    Peso molecolare:357.92

    Ref: TM-T23234

  • Galanin (1-16), mouse, porcine, rat
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    Galanin (1-16), mouse, porcine, rat

    CAS:
    <p>Galanin (1-16), mouse, porcine, rat is a hippocampal galanin receptor agonist(Kd = 3 nM) with high biological activity on locus coeruleus neurons.</p>
    Formula:C78H116N20O21
    Purezza:98.65%
    Colore e forma:White Powder
    Peso molecolare:1669.88

    Ref: TM-TP1380

  • (±)-Ibipinabant
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    (±)-Ibipinabant

    CAS:
    <p>(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.</p>
    Formula:C23H20Cl2N4O2S
    Purezza:99.28% - 99.83%
    Colore e forma:Solid
    Peso molecolare:487.4

    Ref: TM-T4654

  • Pimozide
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    Pimozide

    CAS:
    <p>Pimozide: antipsychotic that blocks type 2 dopamine, alpha-adrenergic, and 5-HT2 receptors, reducing tics and delusions.</p>
    Formula:C28H29F2N3O
    Purezza:99.63% - >99.99%
    Colore e forma:Solid
    Peso molecolare:461.55

    Ref: TM-T2546

  • BML-190
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    BML-190

    CAS:
    <p>BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体，其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki&gt; 2 μM)。</p>
    Formula:C23H23ClN2O4
    Purezza:97.70%
    Colore e forma:Solid
    Peso molecolare:426.89

    Ref: TM-T6417

  • γ-L-Glutamyl-L-alanine
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    γ-L-Glutamyl-L-alanine

    CAS:
    <p>γ-L-Glutamyl-L-alanine, composed of gamma-glutamate and alanine, is the substrate of CRF21 (gamma-Glutamylcyclotransferase, GGCT).</p>
    Formula:C8H14N2O5
    Purezza:99.49%
    Colore e forma:Solid
    Peso molecolare:218.21

    Ref: TM-T7507

  • Ditolylguanidine
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    Ditolylguanidine

    CAS:
    <p>Ditolylguanidine (Di-o-tolylguanidine) is an agonist of sigma receptor (σ1/σ2 receptor).</p>
    Formula:C15H17N3
    Purezza:98.42%
    Colore e forma:White To Pinkish Solid Powder
    Peso molecolare:239.32

    Ref: TM-T5969

  • Bevantolol hydrochloride
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    Bevantolol hydrochloride

    CAS:
    <p>Bevantolol hydrochloride (NC-1400 hydrochloride) is a β1-adrenoceptor antagonist that treatment angina pectoris and hypertension.</p>
    Formula:C20H28ClNO4
    Purezza:99.49%
    Colore e forma:Solid
    Peso molecolare:381.9

    Ref: TM-T8143

  • Neurokinin A(4-10) TFA(97559-35-8 free base)
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    Neurokinin A(4-10) TFA(97559-35-8 free base)

    <p>Neurokinin A(4-10) TFA(97559-35-8 free base) is a tachykinin NK2 receptor agonist[1].</p>
    Formula:C36H55F3N8O12S
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:880.93

    Ref: TM-TP1385

  • Ziprasidone mesylate
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    Ziprasidone mesylate

    CAS:
    <p>Ziprasidone mesylate (CP-88059), an oral 5-HT &amp; dopamine blocker, binds D2, 5-HT2A, 5-HT1A with Ki values: 4.8, 0.42, 3.4 nM.</p>
    Formula:C22H25ClN4O4S2
    Colore e forma:Solid
    Peso molecolare:509.04

    Ref: TM-T63504

  • Bavisant dihydrochloride hydrate
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    Bavisant dihydrochloride hydrate

    CAS:
    Bavisant dihydrochloride (JNJ31001074AAC) is an oral H3 receptor antagonist for ADHD treatment. Phase 2 trials show no significant benefits at 10 mg/day.
    Formula:C19H31Cl2N3O3
    Colore e forma:Solid
    Peso molecolare:420.38

    Ref: TM-T10462L

  • (+)-PD 128907 hydrochloride
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    (+)-PD 128907 hydrochloride

    CAS:
    <p>(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .</p>
    Formula:C14H20ClNO3
    Purezza:97.76%
    Colore e forma:Solid
    Peso molecolare:285.77

    Ref: TM-T7553

  • 1-[(5-methylisoxazol-3-yl)methyl]piperazine
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    1-[(5-methylisoxazol-3-yl)methyl]piperazine

    CAS:
    <p>1-[(5-methylisoxazol-3-yl)methyl]piperazine (Piperazine, 1-[(5-methyl-3-isoxazolyl)methyl]- (9CI)) is a P2Y12 inhibitor.</p>
    Formula:C9H15N3O
    Purezza:95%
    Colore e forma:Solid
    Peso molecolare:181.23

    Ref: TM-T8582