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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

Mostrare 18 più sottocategorie

Trovati 5745 prodotti di "Proteina G/GPCR"

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  • Opaganib
    Targetmol
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    Opaganib

    CAS:
    Opaganib (ABC294640) is an orally active and specific sphingosine kinase-2 (SphK2) inhibitor (IC50: 60 μM).
    Formula:C23H25ClN2O
    Purezza:98.86% - 99.85%
    Colore e forma:Solid
    Peso molecolare:380.91

    Ref: TM-T6750

  • BETP
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    BETP

    CAS:
    BETP is an agonist of GLP-1 receptor (EC50s: 0.66 and 0.755 μM for human and rat GLP-1 receptor).
    Formula:C20H17F3N2O2S
    Purezza:98.51%
    Colore e forma:Solid
    Peso molecolare:406.42

    Ref: TM-TQ0124

  • Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
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    Sar-[D-Phe8]-des-Arg9-Bradykinin acetate

    Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant to
    Formula:C49H70N12O13
    Purezza:99.93%
    Colore e forma:Solid
    Peso molecolare:1035.15

    Ref: TM-TP1917L1

  • Preladenant
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    Preladenant

    CAS:
    <p>Preladenant (SCH-420814) is an orally bioavailable antagonist of the adenosine A2A receptor (Ki: 1.1 nM) and has &gt;1000-fold selectivity over all other adenosine</p>
    Formula:C25H29N9O3
    Purezza:98.02% - 99.68%
    Colore e forma:Solid
    Peso molecolare:503.56

    Ref: TM-T4290

  • AM1241
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    AM1241

    CAS:
    <p>AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.</p>
    Formula:C22H22IN3O3
    Purezza:98.937% - 99.1%
    Colore e forma:Solid
    Peso molecolare:503.33

    Ref: TM-T6755

  • [Sar9] Substance P acetate(77128-75-7 free base)
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    [Sar9] Substance P acetate(77128-75-7 free base)

    [Sar9]-Substance P acetate, an NK-1 receptor agonist, mimics SP's effect on progesterone metabolism.
    Formula:C66H104N18O15S
    Purezza:96.67%
    Colore e forma:Solid
    Peso molecolare:1421.71

    Ref: TM-TP1862L

  • Ponesimod
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    Ponesimod

    CAS:
    <p>Ponesimod (ACT-128800) is an orally available sphingosine-1-phosphate receptor 1 (S1PR1, S1P1) agonist with potential immunomodulating activity.</p>
    Formula:C23H25ClN2O4S
    Purezza:99.42% - 99.96%
    Colore e forma:Solid
    Peso molecolare:460.97

    Ref: TM-T3258

  • HCGRP-(8-37) acetate
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    HCGRP-(8-37) acetate

    <p>HCGRP-(8-37) acetate is a human calcitonin gene-related peptide (hCGRP) fragment acetate and also an antagonist of CGRP receptor.</p>
    Formula:C141H234N44O40
    Purezza:99.29%
    Colore e forma:Solid
    Peso molecolare:3185.64

    Ref: TM-TP1134L

  • Ibrolipim
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    Ibrolipim

    CAS:
    <p>Ibrolipim (NO-1886) attenuates high glucose-induced endothelial dysfunction in cultured human umbilical vein endothelial cells via PI3K/Akt pathway.</p>
    Formula:C19H20BrN2O4P
    Purezza:98.04%
    Colore e forma:Solid
    Peso molecolare:451.25

    Ref: TM-T7832

  • Amitriptyline
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    Amitriptyline

    CAS:
    <p>Amitriptyline: a tricyclic antidepressant used for depression and neuropathic pain.</p>
    Formula:C20H23N
    Purezza:98.24% - 99.64%
    Colore e forma:Crystals Solid
    Peso molecolare:277.4

    Ref: TM-T22240

  • Siramesine
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    Siramesine

    CAS:
    Siramesine (Lu 28-179)(Lu 28-179) is a selective sigma-2 receptor agonist, which has been shown to trigger cell death of cancer cells and to exhibit a potent
    Formula:C30H31FN2O
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:454.58

    Ref: TM-T4620

  • [Sar9,Met(O2)11]-Substance P acetate
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    [Sar9,Met(O2)11]-Substance P acetate

    <p>[Sar9,Met(O2)11]-Substance P acetate is an NK1 agonist, raising MAP and HR equally to septide but with unique timing and behaviors.</p>
    Formula:C66H106N18O18S
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:1471.75

    Ref: TM-TP1369L

  • BD 1008 dihydrobromide
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    BD 1008 dihydrobromide

    CAS:
    <p>BD 1008 dihydrobromide: selective σ1 receptor antagonist (Ki=2 nM), high σ1 and moderate σ2 affinity.</p>
    Formula:C15H24Br2Cl2N2
    Purezza:97.81%
    Colore e forma:Solid
    Peso molecolare:463.08

    Ref: TM-T21788

  • Almotriptan
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    Almotriptan

    CAS:
    Almotriptan (LAS 31416), a triptan and 5-HT1B/1D agonist, treats migraines by constricting cranial vessels and altering blood flow.
    Formula:C17H25N3O2S
    Purezza:99.85%
    Colore e forma:Light Yellow Or White Power
    Peso molecolare:335.46

    Ref: TM-T21231

  • [Lys5,MeLeu9,Nle10]-NKA(4-10)
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    [Lys5,MeLeu9,Nle10]-NKA(4-10)

    CAS:
    Highy selective and potent NK2 receptor agonist (IC50 = 6.1 nM). Induces contraction of the rat fundus and bladder (EC50 values are 117 and 10 nM respectively).
    Formula:C39H65N9O9
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:803.99

    Ref: TM-TP1883

  • FAUC 346
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    FAUC 346

    CAS:
    FAUC 346 is a highly selective D3 partial agonist with EC50 of 1.5 nM.
    Formula:C24H29N3O2S
    Purezza:99.46%
    Colore e forma:Solid
    Peso molecolare:423.57

    Ref: TM-T9081

  • Neuropeptide S (Mouse) acetate
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    Neuropeptide S (Mouse) acetate

    Neuropeptide S (Mouse) acetate is a bioactive peptide.
    Formula:C95H160N34O29
    Purezza:98.25%
    Colore e forma:Solid
    Peso molecolare:2242.5

    Ref: TM-TP1981L

  • S26131
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    S26131

    CAS:
    <p>S26131 (N-[2-[7-[3-[8-(2-acetamidoethyl)naphthalen-2-yl]oxypropoxy]naphthalen-1-yl]ethyl]acetamide) behaves as an antagonist on MT1 and MT2 receptors with Ki of</p>
    Formula:C31H34N2O4
    Purezza:99.77%
    Colore e forma:Solid
    Peso molecolare:498.61

    Ref: TM-T16834

  • PU02
    Targetmol
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    PU02

    CAS:
    <p>PU02 (6-[(1-Naphthalenylmethyl)thio]-9H-purine) is a potent and selective antagonist of 5-HT3 receptor.</p>
    Formula:C16H12N4S
    Purezza:99.35%
    Colore e forma:Solid
    Peso molecolare:292.36

    Ref: TM-T8445

  • MIPS521
    Targetmol
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    MIPS521

    CAS:
    MIPS521 ({2-Amino-4-[3,5-bis(trifluoromethyl)phenyl]thiophen-3-yl}(4-chlorophenyl)methanone) is a positive allosteric modulator of the A1R.
    Formula:C19H10ClF6NOS
    Purezza:99.76%
    Colore e forma:Solid
    Peso molecolare:449.8

    Ref: TM-T9330