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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

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Trovati 5378 prodotti di "Proteina G/GPCR"

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  • Nolomirole
    Targetmol
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    Nolomirole

    CAS:
    <p>Nolomirole is a dopamine receptor agonist that reduces symptoms of congestive heart failure caused by monoclinine.</p>
    Formula:C19H27NO4
    Colore e forma:Solid
    Peso molecolare:333.42

    Ref: TM-T33711

  • J-115814
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    J-115814

    CAS:
    <p>J-115814 is a potent feeding stimulant.</p>
    Formula:C29H38ClN5O3S
    Colore e forma:Solid
    Peso molecolare:572.16

    Ref: TM-T32246

  • Hemopressin (human, mouse)
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    Hemopressin (human, mouse)

    CAS:
    <p>Endogenous peptide, inhibits ep24.15/24.16/ACE with Ki of 27.76/3.43/1.87 μM. Lowers blood pressure, CB1 inverse agonist, reduces pain in vivo.</p>
    Formula:C50H79N13O12
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1054.26

    Ref: TM-TP1900

  • Logo CymitQuimica
    Targetmol
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    TRPV1/CB2 agonist 1

    <p>TRPV1/CB2 agonist 1 (compound 41) is a dual agonist targeting hTRPV1 and CB2 receptors, with an EC50 value of 26.8 μM for hTRPV1. It is applicable in research related to the nervous system.</p>
    Colore e forma:Odour Solid

    Ref: TM-T200749

  • Alprostadil ethyl ester
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    Alprostadil ethyl ester

    CAS:
    <p>Alprostadil ethyl ester is a biochemical used in the treatment of scleroderma.</p>
    Formula:C22H38O5
    Colore e forma:Solid
    Peso molecolare:382.53

    Ref: TM-T29908

  • N-Nitroso Atenolol
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    N-Nitroso Atenolol

    CAS:
    <p>N-Nitroso Atenolol is a derivative of Atenolol. At concentrations ranging from 0.1 to 1 mM, it induces DNA fragmentation in rat hepatocytes.</p>
    Formula:C14H21N3O4
    Colore e forma:Solid
    Peso molecolare:295.33

    Ref: TM-T203130

  • Logo CymitQuimica
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    PSB-1114 triethylamine

    <p>PSB-1114 triethylamine is a potent, enzymatically stable, P2Y2 receptor agonist with a 134 nM EC50, exhibiting greater than 50-fold selectivity over P2Y4 (EC50</p>
    Formula:C10H15F2N3O13P3S·xC6H15N
    Purezza:98%
    Colore e forma:Solid

    Ref: TM-T78080

  • Pobilukast
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    Pobilukast

    CAS:
    <p>Pobilukast (SKF 104353) is a cysteinyl leukotriene receptor antagonist that can be used to study limiting myocardial injury in MI/R rats.</p>
    Formula:C26H34O5S
    Purezza:99.65% - 99.84%
    Colore e forma:Solid
    Peso molecolare:458.61

    Ref: TM-T68130

  • AGN 191976
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    AGN 191976

    CAS:
    <p>AGN 191976 is a novel thromboxane A2-mimetic.</p>
    Formula:C21H32O6
    Colore e forma:Solid
    Peso molecolare:380.481

    Ref: TM-T29722

  • Norisoboldine hydrochloride
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    Norisoboldine hydrochloride

    CAS:
    <p>Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.</p>
    Formula:C18H20ClNO4
    Colore e forma:Solid
    Peso molecolare:349.81

    Ref: TM-T75433

  • d[Leu4,Lys8]-VP
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    d[Leu4,Lys8]-VP

    CAS:
    <p>Vasopressin V1B agonist; Ki: 0.16nM V1B, 64nM oxytocin; weak antidiuretic/vasopressor; minimal oxytocic action.</p>
    Formula:C47H67N11O11S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1026.2

    Ref: TM-TP1927

  • Kisspeptin 234
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    Kisspeptin 234

    CAS:
    <p>Kisspeptin receptor antagonist; blocks kisspeptin-10 effects on IP (IC50 = 7 nM) and GnRH release.</p>
    Formula:C63H78N18O13
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1295.42

    Ref: TM-TP1896

  • Logo CymitQuimica
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    20-SOLA

    <p>20-SOLA is the first water-soluble 20-HETE antagonist with oral bioavailability. It significantly improves blood pressure changes and kidney damage associated with the streptozotocin (STZ) diabetic mouse model. Additionally, 20-SOLA acts as a GPR75 receptor blocker. This compound is useful in research related to cardiovascular pathology.</p>
    Formula:C33H62O9
    Peso molecolare:602.43938

    Ref: TM-T208783

  • CB2 receptor agonist 2
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    CB2 receptor agonist 2

    CAS:
    <p>CB2 receptor agonist 2 (ZINC72105556): potent, Ki=8.5 nM, high selectivity for CB2.</p>
    Formula:C30H36N2O4
    Purezza:99.75%
    Colore e forma:Solid
    Peso molecolare:488.62

    Ref: TM-T22009

  • CAY10606
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    CAY10606

    CAS:
    <p>CAY10606 has a wide range of applications in life science related research.</p>
    Formula:C22H18ClNO3
    Colore e forma:Solid
    Peso molecolare:379.84

    Ref: TM-T37353

  • Proglumide hemicalcium
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    Proglumide hemicalcium

    CAS:
    Proglumide hemicalcium is a antagonist of nonpeptide and orally active cholecystokinin (CCK)-A/B receptors, has antiepileptic and antioxidant activities.
    Formula:C18H28CaN2O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:376.51

    Ref: TM-T12544

  • IRL-3630
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    IRL-3630

    CAS:
    <p>IRL 3460 is an enantiomer.</p>
    Formula:C31H40N4O6S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:596.74

    Ref: TM-T25541

  • Azepexole hydrochloride
    Targetmol
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    Azepexole hydrochloride

    CAS:
    <p>Azepexole hydrochloride (4H-Oxazolo[4,5-d]azepin-2-amine, 6-ethyl-5,6,7,8-tetrahydro-, hydrochloride (1:1)) is a potent α2-Adrenoceptor agonist with anaesthetic</p>
    Formula:C9H16ClN3O
    Purezza:99.88% - 99.89%
    Colore e forma:Soild
    Peso molecolare:217.7

    Ref: TM-T21787L

  • Misoprostol acid
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    Misoprostol acid

    CAS:
    <p>Misoprostol acid is an active metabolite of Misoprostol,can be used for non-steroidal anti-inflammatory drug-induced (NSAID) gastric ulcers.</p>
    Formula:C21H36O5
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:368.51

    Ref: TM-T12047

  • Octodrine
    Targetmol
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    Octodrine

    CAS:
    <p>Octodrine (2-Amino-6-methylheptane) is primarily used as a pharmaceutical intermediate for Octamylamine; it also functions as a local anesthetic and vasoconstrictor.</p>
    Formula:C8H19N
    Purezza:99.98%
    Colore e forma:Clear Colorless To Light Yellow Liquid
    Peso molecolare:129.24

    Ref: TM-T0043