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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

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Trovati 5352 prodotti di "Proteina G/GPCR"

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  • EP4 receptor antagonist 3
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    EP4 receptor antagonist 3

    CAS:
    <p>EP4 receptor antagonist 3 from patent WO2010019796 A1 targets EP4 for research on pain, arthritis, and cancer.</p>
    Formula:C26H21F3N2O3S
    Colore e forma:Solid
    Peso molecolare:498.52

    Ref: TM-T38595

  • JNJ-40929837 succinate
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    JNJ-40929837 succinate

    CAS:
    <p>JNJ-40929837 succinate is a selective, orally active inhibitor of LTA 4 H (leukotriene A 4 hydrolase). This compound effectively inhibits aminopeptidase activity, leading to the accumulation of Pro-Gly-Pro in serum, and can be utilized in asthma research [1].</p>
    Formula:C22H24N4O2S·xC4H6O4
    Colore e forma:Solid

    Ref: TM-T86771

  • Logo CymitQuimica
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    BIM-23190 hydrochloride

    <p>BIM-23190 hydrochloride, somatostatin analog, SSRT2/5 agonist, Ki: 0.34 nM (SSTR2), 11.1 nM (SSTR5). Used in cancer, acromegaly research.</p>
    Colore e forma:Liquid

    Ref: TM-T37109

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    HS024 TFA

    <p>HS024, a selective MC4 receptor antagonist, exhibits affinity with Ki values of 0.29, 3.29, 5.45, and 18.6 nM for MC4, MC5, MC3, and MC1 receptors, respectively</p>
    Formula:C60H80F3N19O12S2
    Colore e forma:Solid
    Peso molecolare:1380.52

    Ref: TM-T75852

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    GLP-1(28-36)amide TFA

    <p>GLP-1(28-36)amide TFA, a nonapeptide cleavage product of GLP-1, shows antioxidant properties with anti-diabetic and cardioprotective effects.</p>
    Formula:C56H86F3N15O11
    Colore e forma:Solid
    Peso molecolare:1202.37

    Ref: TM-T76191

  • SB656104
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    SB656104

    CAS:
    <p>SB656104 is a bioactive chemical.</p>
    Formula:C25H30ClN3O3S
    Colore e forma:Solid
    Peso molecolare:488.04

    Ref: TM-T34546

  • LH-RH (7-10)
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    LH-RH (7-10)

    CAS:
    LH-RH (7-10), a tetrapeptide, is a key LHRH degradation product found in macrophages and pneumocytes.
    Formula:C19H36N8O4
    Colore e forma:Solid
    Peso molecolare:440.54

    Ref: TM-T76353

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    SAR441255

    SAR441255 is a potent unimolecular peptide that acts as a GLP-1/GIP/GCG receptor triagonist, demonstrating balanced activation across all three target receptors
    Colore e forma:Odour Solid

    Ref: TM-T81214

  • Substance P (alligator)
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    Substance P (alligator)

    CAS:
    <p>Substance P from alligator: a neuropeptide with structure Arg-Pro-Arg-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH2.</p>
    Formula:C63H98N20O13S
    Colore e forma:Solid
    Peso molecolare:1375.64

    Ref: TM-T76449

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    Amylin, amide, human TFA

    <p>Amylin, a 37-amino acid human hormone, moderates glucose regulation by reducing glucagon, delaying digestion, and increasing satiety.</p>
    Formula:C167H262F3N51O57S2
    Colore e forma:Solid
    Peso molecolare:4017.3

    Ref: TM-T75787

  • Pramlintide
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    Pramlintide

    CAS:
    <p>Pramlintide, a polypeptide analog of human amylin, is an antidiabetic agent with antineoplastic properties in colorectal cancer.</p>
    Colore e forma:Solid

    Ref: TM-T38998

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    CCZ01048 TFA

    CCZ01048 TFA, α-MSH analog, binds MC1R with 0.31 nM affinity, internalizes in melanoma cells, and is stable for melanoma PET imaging.
    Formula:C73H106F3N21O18
    Colore e forma:Solid
    Peso molecolare:1622.75

    Ref: TM-T76072L

  • Logo CymitQuimica
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    (Phe2,Orn8)-Oxytocin acetate

    <p>(Phe2,Orn8)-Oxytocin acetate: V1 agonist with EC50 of 280 nM for rabbit epididymis contractility.</p>
    Formula:C44H69N13O13S2
    Colore e forma:Solid
    Peso molecolare:1052.23

    Ref: TM-T76630

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    CART(55-102)(rat) TFA

    <p>Rat CART(55-102) TFA suppresses appetite, links to leptin/neuropeptide Y, and may induce anxiety/stress.</p>
    Formula:C228H368F3N65O67S7
    Colore e forma:Solid
    Peso molecolare:5373.2

    Ref: TM-T75900

  • DOTA-JR11
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    DOTA-JR11

    CAS:
    <p>DOTA-JR11 is a somatostatin receptor 2 (SSTR2) antagonist that can be radiolabeled with 68Ga.</p>
    Formula:C74H98ClN19O21S2
    Colore e forma:Solid
    Peso molecolare:1689.27

    Ref: TM-T80157

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    Neuropeptide SF(mouse,rat) TFA

    <p>Neuropeptide SF TFA is a potent agonist for NPFF1 (Ki=48.4 nM) and NPFF2 (Ki=12.1 nM) and enhances ASIC3 current.</p>
    Formula:C42H66F3N13O12
    Colore e forma:Solid
    Peso molecolare:1002.05

    Ref: TM-T75865

  • Relamorelin TFA
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    Relamorelin TFA

    CAS:
    <p>Relamorelin (RM-131) TFA: ghrelin analog, GHSR agonist, 0.42 nM affinity, boosts growth hormone, enhances gastric emptying, potential in motility disorders.</p>
    Formula:C45H51F3N8O7S
    Colore e forma:Solid
    Peso molecolare:905

    Ref: TM-T75262

  • [Lys5,MeLeu9,Nle10]Neurokinin A(4-10)
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    [Lys5,MeLeu9,Nle10]Neurokinin A(4-10)

    CAS:
    <p>'[Lys5,MeLeu9,Nle10]Neurokinin A(4-10)' is a selective NK2R agonist with prokinetic activity for smooth muscle studies.</p>
    Formula:C39H64N8O10
    Colore e forma:Solid
    Peso molecolare:804.97

    Ref: TM-T76426

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    Neuropeptide Y (2-36) (porcine)

    CAS:
    <p>Porcine Neuropeptide Y (2-36) is 97.14% similar to rat/human, an agonist for Y5, Y2, Y1 receptors, used in obesity research.</p>
    Formula:C181H278N54O55
    Colore e forma:Solid
    Peso molecolare:4090.47

    Ref: TM-T76356

  • [D-Glp1,D-Phe2,D-Trp3,6]-LH-RH
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    [D-Glp1,D-Phe2,D-Trp3,6]-LH-RH

    CAS:
    <p>[D-Glp1,D-Phe2,D-Trp3,6]-LH-RH is a synthetic LHRH analog and a GnRH receptor antagonist.</p>
    Formula:C67H84N16O13
    Colore e forma:Solid
    Peso molecolare:1321.48

    Ref: TM-T76350