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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

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Trovati 5352 prodotti di "Proteina G/GPCR"

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  • [Ala11,D-Leu15]-Orexin B(human)
    Targetmol
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    [Ala11,D-Leu15]-Orexin B(human)

    CAS:
    <p>OX2 receptor agonist with 400x selectivity vs OX1. EC50: 0.13 nM (OX2), 52 nM (OX1).</p>
    Formula:C120H206N44O35S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:2857.28

    Ref: TM-TP1975

  • Logo CymitQuimica
    Targetmol
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    ATMW-2

    <p>ATMW-2 is an antagonist engineered using NeuralGenThesis (NGT) technology, specifically targeting the melanocortin 2 receptor (MC2R).</p>
    Formula:C27H29ClN2O4
    Colore e forma:Solid
    Peso molecolare:480.98

    Ref: TM-T203063

  • Moperone
    Targetmol
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    Moperone

    CAS:
    <p>Moperone (R 1658) is an antagonist of both the D2 dopamine receptor (D2 dopamine receptor) and the D3 dopamine receptor (D3 dopamine receptor), with IC50 values for each of 1.0 nM.</p>
    Formula:C22H26FNO2
    Colore e forma:Solid
    Peso molecolare:355.45

    Ref: TM-T203131

  • Dexbrompheniramine
    Targetmol
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    Dexbrompheniramine

    CAS:
    <p>Dexbrompheniramine: oral H1 antagonist, antihistamine for hay fever and urticaria research.</p>
    Formula:C16H19BrN2
    Colore e forma:Solid
    Peso molecolare:319.24

    Ref: TM-T75276

  • 7-Methyl DMT
    Targetmol
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    7-Methyl DMT

    CAS:
    <p>7-Methyl DMT (7-TMT) acts as a 5-HT2 receptor agonist. Structurally, it is a tryptamine derivative and serves as an analytical reference for the psychoactive substance DOM. It is also applicable in research related to neurological disorders.</p>
    Formula:C13H18N2
    Colore e forma:Solid
    Peso molecolare:202.3

    Ref: TM-T203196

  • 15(S)-15-methyl Prostaglandin D2
    Targetmol
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    15(S)-15-methyl Prostaglandin D2

    CAS:
    <p>15(S)-15-methyl PGD2 is a stable PGD2 analog that induces vasoconstriction, raises blood pressure, and shows strong antifertility effects.</p>
    Formula:C21H34O5
    Colore e forma:Solid
    Peso molecolare:366.49

    Ref: TM-T36153

  • Methdilazine
    Targetmol
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    Methdilazine

    CAS:
    <p>Methdilazine: oral antibiotic, histamine antagonist, fights mycobacterium (MIC 5-15 μg/mL) for infectious disease research.</p>
    Formula:C18H20N2S
    Colore e forma:Solid
    Peso molecolare:296.43

    Ref: TM-T75313

  • Maceneolignan H
    Targetmol
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    Maceneolignan H

    CAS:
    <p>Maceneolignan H, a neolignane from Myristica fragrans, selectively blocks CCR3 (EC50=1.4μM) with allergy research potential.</p>
    Formula:C24H30O7
    Colore e forma:Solid
    Peso molecolare:430.49

    Ref: TM-T75499

  • Methamnetamine hydrochloride
    Targetmol
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    Methamnetamine hydrochloride

    CAS:
    <p>Methamnetamine (PAL-1046) hydrochloride is a psychoactive substance derived from phenethylamine, known to cause excessive serotonin release.</p>
    Formula:C14H18ClN
    Colore e forma:Solid
    Peso molecolare:235.75

    Ref: TM-T203312

  • δ8-THC acetate
    Targetmol
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    δ8-THC acetate

    CAS:
    <p>Delta8-THC acetate (Delta8-tetrahydrocannabinol) is a psychoactive cannabinoid that binds to the cannabinoid receptor 1 (CB1 receptor) and exhibits anti-nausea, appetite-stimulating, and anti-inflammatory effects. It may also offer neuroprotective benefits and has potential applications in research on anxiety and depression.</p>
    Formula:C23H32O3
    Colore e forma:Solid
    Peso molecolare:356.5

    Ref: TM-T203037

  • SBI-810
    Targetmol
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    SBI-810

    CAS:
    <p>SBI-810 is a functional selective β-arrestin-biased allosteric modulator of the neurotensin receptor 1 (NTSR1). In the presence of the endogenous ligand neurotensin (NT), SBI-810 regulates NTSR1 signaling through a G protein-specific mechanism. It fully antagonizes NT-induced Gq activation and partially antagonizes NT-induced Gi1 activation, allowing NTSR1 to activate GoA and G12.</p>
    Formula:C27H34N4O2
    Colore e forma:Solid
    Peso molecolare:446.59

    Ref: TM-T203513

  • CB2 receptor agonist 9
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    CB2 receptor agonist 9

    CAS:
    <p>CB2 receptor agonist 9 (Compound 33) is an orally active agonist of cannabinoid receptor 2 (CB2 receptor) with an EC50 of 16.2 nM. It inhibits the expression of TNF-α, IL-1β, and IL-6, demonstrating anti-inflammatory activity in a DSS-induced acute colitis model in mice.</p>
    Formula:C16H23N3O2S
    Colore e forma:Solid
    Peso molecolare:321.44

    Ref: TM-T203517

  • SB656104
    Targetmol
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    SB656104

    CAS:
    <p>SB656104 is a bioactive chemical.</p>
    Formula:C25H30ClN3O3S
    Colore e forma:Solid
    Peso molecolare:488.04

    Ref: TM-T34546

  • (±)-9-Nor-9α-hydroxy Hexahydrocannabinol
    Targetmol
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    (±)-9-Nor-9α-hydroxy Hexahydrocannabinol

    CAS:
    <p>(±)-9-Nor-9α-hydroxy Hexahydrocannabinol is a cannabinoid-structured compound that exhibits potent cannabinoid-like activity in both dogs and mice.</p>
    Formula:C20H30O3
    Colore e forma:Solid
    Peso molecolare:318.45

    Ref: TM-T203604

  • N-Nitroso Atenolol
    Targetmol
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    N-Nitroso Atenolol

    CAS:
    <p>N-Nitroso Atenolol is a derivative of Atenolol. At concentrations ranging from 0.1 to 1 mM, it induces DNA fragmentation in rat hepatocytes.</p>
    Formula:C14H21N3O4
    Colore e forma:Solid
    Peso molecolare:295.33

    Ref: TM-T203130

  • NF 340
    Targetmol
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    NF 340

    CAS:
    <p>P2Y11 antagonist</p>
    Formula:C37H30N4Na4O15S4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:990.87

    Ref: TM-T23064

  • Dalcotidine
    Targetmol
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    Dalcotidine

    CAS:
    <p>Dalcotidine (KU 1257), a histamine H2/H9 blocker, inhibits acid secretion; Ki=0.040, KB=0.041, aids ulcer healing, may lower relapse.</p>
    Formula:C18H29N3O2
    Purezza:99.11%
    Colore e forma:Solid
    Peso molecolare:319.44

    Ref: TM-T31195

  • Logo CymitQuimica
    Targetmol
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    (S)-V-0219 hydrochloride

    <p>(S)-V-0219 hydrochloride, a GLP-1R PAM, triggers calcium in hGLP-1R HEK cells, lowers glucose in mice, and reduces fasting hunger.</p>
    Formula:C20H26ClF3N4O2
    Colore e forma:Solid
    Peso molecolare:446.89

    Ref: TM-T74265

  • Logo CymitQuimica
    Targetmol
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    GLI1-IN-3

    <p>GLI1-IN-3 (Compound 11a) is a triterpenoid-like compound that inhibits Hedgehog signaling in cancer cells with GLI1 overexpression. It suppresses the proliferation of non-small cell lung cancer and prostate cancer cell lines with excessive Hh signaling activation. Additionally, GLI1-IN-3 reduces the expression of GLI1 protein and its target genes associated with tumor progression and proliferation in A549 and DU-145 cancer cells.</p>
    Colore e forma:Odour Solid

    Ref: TM-T206757

  • Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate
    Targetmol
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    Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate

    CAS:
    <p>Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate is an NPR-A agonist and ANP hormone. Carperitide increases cGMP levels and reduces the heart's workload.</p>
    Formula:C129H207N45O41S3
    Purezza:99.78%
    Colore e forma:Soild
    Peso molecolare:3140.5

    Ref: TM-TP1219