CymitQuimica logo
Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

Mostrare 18 più sottocategorie

Trovati 5337 prodotti di "Proteina G/GPCR"

Ordinare per
Purezza (%)
0
100
|
0
|
50
|
90
|
95
|
100
prodotti per pagina.
  • Rocavorexant
    Targetmol
    + Info

    Rocavorexant

    CAS:
    <p>Rocavorexant is an antagonist of the orexin-1 receptor (orexin-1 receptor), exhibiting a pIC50 value of 9.1 for human OX1 and a pIC50 of 6.0 for human OX2.</p>
    Formula:C18H19F3N8O
    Colore e forma:Solid
    Peso molecolare:420.392

    Ref: TM-T206374

  • Netupitant metabolite Monohydroxy Netupitant
    Targetmol
    + Info

    Netupitant metabolite Monohydroxy Netupitant

    CAS:
    <p>Monohydroxy Netupitant is a highly selective antagonist of NK1 receptor, and is Netupitant metabolite.</p>
    Formula:C30H32F6N4O2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:594.59

    Ref: TM-T12211

  • TM38837
    Targetmol
    + Info

    TM38837

    CAS:
    <p>CB1 antagonist 4 is an inverse agonist of cannabinoid receptor 1 (CB1) with an IC50 of 0.4 nM. It can reduce body weight, improve plasma inflammatory markers, and enhance glucose homeostasis [1].</p>
    Formula:C27H20Cl2F3N7O
    Colore e forma:Solid
    Peso molecolare:586.40

    Ref: TM-T86011

  • DSP-1053 benzenesulfonate
    Targetmol
    + Info

    DSP-1053 benzenesulfonate

    CAS:
    <p>DSP-1053: Benzylpiperidine-based, potent SERT inhibitor (Ki=1.02nM), partial 5-HT1A receptor agonist (Ki=5.05nM), antidepressant.</p>
    Formula:C32H38BrNO7S
    Colore e forma:Solid
    Peso molecolare:660.62

    Ref: TM-T72220

  • Delmadinone acetate
    Targetmol
    + Info

    Delmadinone acetate

    CAS:
    <p>Delmadinone acetate is an orally active compound used to control estrus and ovulation in both female and male pets. It induces adrenal suppression by inhibiting the pituitary release of ACTH.</p>
    Formula:C23H27ClO4
    Colore e forma:Solid
    Peso molecolare:402.911

    Ref: TM-T206595

  • Metrazoline
    Targetmol
    + Info

    Metrazoline

    CAS:
    <p>Metrazoline (o-Methyl-tracizoline) acts as a ligand for adrenergic receptors (low affinity) and imidazoline I2 receptors.</p>
    Formula:C14H16N2O4
    Colore e forma:Solid
    Peso molecolare:276.288

    Ref: TM-T204804

  • Teoprolol
    Targetmol
    + Info

    Teoprolol

    CAS:
    <p>Teoprolol is a blocker of β-adrenergic receptor.</p>
    Formula:C23H30N6O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:454.52

    Ref: TM-T13124

  • A3AR antagonist 5
    Targetmol
    + Info

    A3AR antagonist 5

    CAS:
    <p>A3AR antagonist 5 (Compound 16) acts as a selective antagonist for the human adenosine A3 receptor (human adenosine A3 receptor), with an affinity expressed as a pC value of 4.542 μM.</p>
    Formula:C18H16N2O2S
    Colore e forma:Solid
    Peso molecolare:324.40

    Ref: TM-T200493

  • PAR-2-IN-2
    Targetmol
    + Info

    PAR-2-IN-2

    CAS:
    <p>PAR-2-IN-2 (compound P-596) is an inhibitor of protease-activated receptor 2 (PAR-2), with an IC50 of 10.79 μM for SLIGKV and an IC50 greater than 200 μM for trypsin.</p>
    Formula:C25H20F3N5O2
    Colore e forma:Solid
    Peso molecolare:479.454

    Ref: TM-T204647

  • (Rac)-BI 703704
    Targetmol
    + Info

    (Rac)-BI 703704

    CAS:
    <p>(Rac)-BI 703704 is a potent activator of soluble guanylyl cyclase (sGC).</p>
    Formula:C32H37N3O4S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:559.72

    Ref: TM-T12661

  • SGL5213
    Targetmol
    + Info

    SGL5213

    CAS:
    <p>SGL5213 is a potent oral SGLT1 inhibitor (IC50: 29 nM) with potential for treating type 2 diabetes.</p>
    Formula:C37H55N3O8
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:669.85

    Ref: TM-T12892

  • PF-07258669
    Targetmol
    + Info

    PF-07258669

    CAS:
    <p>PF-07258669 is a selective melanocortin 4 receptor (MC4) antagonist used in the study of cachexia and loss of appetite.</p>
    Formula:C25H27FN6O2
    Purezza:99.9%
    Colore e forma:Solid
    Peso molecolare:462.52

    Ref: TM-T69526

  • Vofopitant dihydrochloride
    Targetmol
    + Info

    Vofopitant dihydrochloride

    CAS:
    <p>Vofopitant dihydrochloride (GR 205171A) is a tachykinin NK1 receptor antagonist and a potential compound for the treatment of pathologic vomiting.</p>
    Formula:C21H25Cl2F3N6O
    Purezza:98.99%
    Colore e forma:Solid
    Peso molecolare:505.36

    Ref: TM-T13329L

  • SB-423562
    Targetmol
    + Info

    SB-423562

    CAS:
    <p>SB-423562 is a calcium-sensing receptor (CaSR) antagonist and can be used in studies about osteoporosis.</p>
    Formula:C26H32N2O4
    Purezza:99.22%
    Colore e forma:Solid
    Peso molecolare:436.54

    Ref: TM-T12846

  • BQ-788
    Targetmol
    + Info

    BQ-788

    CAS:
    <p>BQ-788 is an ETB receptor antagonist with potential hypertensive activity that inhibits exogenous ET-1-induced elevation of coronary perfusion pressure.</p>
    Formula:C34H51N5O7
    Purezza:98.81%
    Colore e forma:Solid
    Peso molecolare:641.8

    Ref: TM-T10595

  • Dersimelagon
    Targetmol
    + Info

    Dersimelagon

    CAS:
    <p>Dersimelagon (MT-7117) is an orally active, selective melanocortin 1 receptor (MC1R) agonist.Cost-effective and quality-assured.</p>
    Formula:C36H45F4N3O5
    Purezza:97.35% - 98.23%
    Colore e forma:Solid
    Peso molecolare:675.75

    Ref: TM-T25310

  • BMS-986141
    Targetmol
    + Info

    BMS-986141

    CAS:
    <p>BMS-986141(UDM-003183) is a selective and potent protease-activated receptor-4 (PAR-4) antagonist with oral activity and an IC50 value of 0.4 nM.BMS-98614</p>
    Formula:C27H23N5O5S2
    Purezza:98.43% - 99.26%
    Colore e forma:Solid
    Peso molecolare:561.63

    Ref: TM-T63966

  • SB-224289 hydrochloride
    Targetmol
    + Info

    SB-224289 hydrochloride

    CAS:
    <p>SB-224289 hydrochloride (SB-224289A) is a selective antagonist of 5-HT1B receptor, with anxiolytic effect.</p>
    Formula:C32H33ClN4O3
    Purezza:97.82% - 98.99%
    Colore e forma:Solid
    Peso molecolare:557.08

    Ref: TM-T12841

  • Vofopitant
    Targetmol
    + Info

    Vofopitant

    CAS:
    <p>Vofopitant (GR 205171) is a potent NK1 receptor antagonist with anxiolytic and antiemetic activity for the study of post-traumatic stress disorder (PTSD).</p>
    Formula:C21H23F3N6O
    Purezza:97.86%
    Colore e forma:Solid
    Peso molecolare:432.44

    Ref: TM-T13329

  • Treprostinil diethanolamine
    Targetmol
    + Info

    Treprostinil diethanolamine

    CAS:
    <p>Treprostinil diethanolamine (UT-15C) is a potent agonist of EP2, DP1 and IP, with values of 3.6, 4.4, 32.1, 212, 826, 2505 and 4680 nM for EP2, DP1, IP, EP1,</p>
    Formula:C27H45NO7
    Purezza:99.86%
    Colore e forma:Solid
    Peso molecolare:495.65

    Ref: TM-T63349