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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

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Trovati 5378 prodotti di "Proteina G/GPCR"

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  • Gastrin I, rat
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    Gastrin I, rat

    CAS:
    <p>Gastrin I, rat is a peptide hormone that effectively stimulates gastric acid secretion.</p>
    Formula:C94H128N22O31S2
    Colore e forma:Solid
    Peso molecolare:2126.3

    Ref: TM-T38203

  • Dotanoc
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    Dotanoc

    CAS:
    <p>Dotanoc is a ligand to make gallium Ga 68-DOTANOC, which is a gallium Ga 68-radiolabeled analog of somatostatin.</p>
    Formula:C69H94N14O17S2
    Colore e forma:Solid
    Peso molecolare:1455.71

    Ref: TM-T24014

  • [Ala2] Endothelin-3, human
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    [Ala2] Endothelin-3, human

    CAS:
    <p>[Ala2] Endothelin-3, a linear ET-3 analog with Ala replacing Cys, stimulates endothelial cell migration.</p>
    Formula:C120H166N26O32S4
    Colore e forma:Solid
    Peso molecolare:2613.02

    Ref: TM-T76305

  • Logo CymitQuimica
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    Selepressin acetate

    <p>Selepressin acetate is a useful organic compound for research related to life sciences and the catalog number is T73654.</p>
    Formula:C48H77N13O13S2
    Colore e forma:Solid
    Peso molecolare:1108.33

    Ref: TM-T73654

  • Sufotidine
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    Sufotidine

    CAS:
    <p>Sufotidine (AH 25352X) is a highly selective competitive H2 receptor antagonist.</p>
    Formula:C20H31N5O3S
    Purezza:99.03% - 99.92%
    Colore e forma:Solid
    Peso molecolare:421.56

    Ref: TM-T68146

  • Neuropeptide W-30 (rat)
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    Neuropeptide W-30 (rat)

    CAS:
    <p>Neuropeptide W-30 (rat) acts as a crucial stress mediator within the central nervous system, influencing the hypothalamus-pituitary-adrenal (HPA) axis and sympathetic outflow. It serves as an endogenous ligand for the two related orphan G-protein-coupled receptors (GPCRs), GPR7 and GPR8. NPW-30 binds and activates both GPR7 and GPR8 at comparable effective doses [1] [2] [3].</p>
    Formula:C165H249N49O38S
    Colore e forma:Solid
    Peso molecolare:3559.11

    Ref: TM-TP2611

  • MLGFFQQPKPR-NH2
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    MLGFFQQPKPR-NH2

    CAS:
    <p>MLGFFQQPKPR-NH2 is a reversed Substance P peptide. Substance P is a neuropeptide [1] .</p>
    Formula:C63H98N18O13S
    Colore e forma:Solid
    Peso molecolare:1347.63

    Ref: TM-T76451

  • Substance P (4-11)
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    Substance P (4-11)

    CAS:
    Substance P (4-11), a C-terminal fragment of Substance P, acts as a highly selective agonist for NK1 receptors, demonstrating specificity in its interaction.
    Formula:C46H67N11O10S
    Colore e forma:Solid
    Peso molecolare:966.16

    Ref: TM-T76455

  • Tamuzimod
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    Tamuzimod

    CAS:
    <p>Tamuzimod, an effective immunomodulator, exhibits modulatory activity on S1P Receptors with EC50 values below 1 μM [1] [2].</p>
    Formula:C21H13Cl3F3N5O3
    Colore e forma:Solid
    Peso molecolare:546.71

    Ref: TM-T74747

  • Ro60-0175
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    Ro60-0175

    CAS:
    <p>Ro60-0175 is a selective 5-HT2B and 5-HT2C serotonin receptor agonist, often used as fumarate.</p>
    Formula:C11H12ClFN2
    Purezza:97.09%
    Colore e forma:Solid
    Peso molecolare:226.68

    Ref: TM-T39161

  • Logo CymitQuimica
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    Utreglutide

    CAS:
    <p>Utreglutide is a potent glucagon-like peptide 1 (GLP-1) receptor agonit [1] .</p>
    Formula:C191H298N46O58
    Colore e forma:Solid
    Peso molecolare:4166.67

    Ref: TM-T76237

  • Neuropeptide Y (18-36) (porcine)
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    Neuropeptide Y (18-36) (porcine)

    CAS:
    <p>"Neuropeptide Y (18-36) (porcine) is a NPY heart receptor blocker, halts I-NPY binding, aids in heart failure research."</p>
    Formula:C112H174N36O27
    Colore e forma:Solid
    Peso molecolare:2456.8

    Ref: TM-T76357

  • LY 344864 racemate
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    LY 344864 racemate

    CAS:
    <p>LY 344864 racemate is a 5-HT1F receptor agonist.</p>
    Formula:C21H22FN3O
    Purezza:99.75%
    Colore e forma:Soild
    Peso molecolare:351.42

    Ref: TM-T2344L

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    ANQ-11125 TFA

    <p>ANQ-11125 TFA is a motilin antagonist with a pKd of 8.24, inhibiting motilide contractions in rabbits.</p>
    Formula:C88H126F3N19O23
    Colore e forma:Solid
    Peso molecolare:1875.05

    Ref: TM-T75861

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    K-(D-1-Nal)-FwLL-NH2 TFA

    <p>K-(D-1-Nal)-FwLL-NH2 TFA: potent ghrelin inverse agonist; Ki=4.9 nM (COS7), 31 nM (HEK293T); blocks Gq/G13 signaling.</p>
    Formula:C53H68F3N9O8
    Colore e forma:Solid
    Peso molecolare:1016.16

    Ref: TM-T75948

  • Logo CymitQuimica
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    Human growth hormone-releasing factor TFA

    <p>Human growth hormone-releasing factor TFA is a hypothalamic peptide that promotes GH secretion by targeting pituitary GHRHR.</p>
    Formula:C217H359F3N72O68S
    Colore e forma:Solid
    Peso molecolare:5153.67

    Ref: TM-T75713

  • Logo CymitQuimica
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    Ecnoglutide

    CAS:
    <p>Ecnoglutide (XW003) is a glucagon-like peptide 1 (GLP-1) receptor agonist [1] .</p>
    Formula:C194H304N48O61
    Colore e forma:Solid
    Peso molecolare:4284.76

    Ref: TM-T76234

  • Logo CymitQuimica
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    HPP-9

    <p>HPP-9, a Proteolysis-Targeting Chimera (PROTAC) derived from Hedgehog Pathway Inhibitor-1 (HPI-1) with a pIC50 value of 6.71, is designed to degrade BET</p>
    Formula:C49H52N6O11
    Colore e forma:Solid
    Peso molecolare:900.97

    Ref: TM-T79907

  • Logo CymitQuimica
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    dCNP

    <p>dCNP binds to NPR-B/C receptors (NPR-B/C receptor), initiating the cGMP signaling pathway and regulating vascular function. It exhibits anti-hypoxic effects by downregulating hypoxia-related genes such as HIF1α and HIF2α. Additionally, dCNP inhibits tumor stroma induction, demonstrating antifibrotic properties. It also enhances immune response by upregulating CTL, NK cells, and conventional type 1 dendritic cells in tumors.</p>
    Formula:C141H248N38O36S3
    Colore e forma:Solid
    Peso molecolare:3147.91

    Ref: TM-TP3063

  • Corazonin
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    Corazonin

    CAS:
    <p>Corazonin, a neuropeptide in insects, regulates caste identity and behavior, mainly in workers/foragers.</p>
    Formula:C62H83N17O19
    Colore e forma:Solid
    Peso molecolare:1370.42

    Ref: TM-T76183