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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

Mostrare 18 più sottocategorie

Trovati 5352 prodotti di "Proteina G/GPCR"

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  • Urocortin (rat) acetate
    Targetmol
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    Urocortin (rat) acetate

    <p>Urocortin (rat) acetate: CRF receptor agonist; Ki=13nM (hCRF1), 1.5nM (rCRF2α), 0.97nM (mCRF2β); neuropeptide.</p>
    Purezza:97.76%
    Colore e forma:Soild

    Ref: TM-TP1020L

  • Indacaterol maleate
    Targetmol
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    Indacaterol maleate

    CAS:
    <p>Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.</p>
    Formula:C28H32N2O7
    Purezza:99.03% - 99.67%
    Colore e forma:Solid
    Peso molecolare:508.56

    Ref: TM-T1239

  • Lafutidine
    Targetmol
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    Lafutidine

    CAS:
    <p>Lafutidine (FRG-8813) is a newly developed histamine H(2)-receptor antagonist, which can inhibit gastric acid secretion.</p>
    Formula:C22H29N3O4S
    Purezza:98.55%
    Colore e forma:Yellowish White Crystalline Powder
    Peso molecolare:431.55

    Ref: TM-T0081

  • Rimonabant
    Targetmol
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    Rimonabant

    CAS:
    <p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>
    Formula:C22H21Cl3N4O
    Purezza:98% - 99.91%
    Colore e forma:White Or Almost White Crystalline Powder
    Peso molecolare:463.79

    Ref: TM-T1519L

  • 2-Bromo-6-methoxynaphthalene
    Targetmol
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    2-Bromo-6-methoxynaphthalene

    CAS:
    <p>2-Bromo-6-methoxynaphthalene was used in the synthesis of nabumetone [4-(6-methoxy-2-naphthalenyl)-2-butanone] by Heck reaction.</p>
    Formula:C11H9BrO
    Purezza:98.51%
    Colore e forma:White To Off-White Powder
    Peso molecolare:237.09

    Ref: TM-T0663

  • Amiselimod hydrochloride
    Targetmol
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    Amiselimod hydrochloride

    CAS:
    <p>Amiselimod hydrochloride (MT-1303 hydrochloride) is a sphingosine 1-phosphate receptor-1 (S1P1) modulator.</p>
    Formula:C19H31ClF3NO3
    Purezza:99.55%
    Colore e forma:Solid
    Peso molecolare:413.9

    Ref: TM-T10305

  • Prucalopride
    Targetmol
    + Info

    Prucalopride

    CAS:
    <p>Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is &gt;290x more specific for these receptors.</p>
    Formula:C18H26ClN3O3
    Purezza:>99.99%
    Colore e forma:Solid
    Peso molecolare:367.87

    Ref: TM-T2542

  • Clonidine hydrochloride
    Targetmol
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    Clonidine hydrochloride

    CAS:
    <p>Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.</p>
    Formula:C9H10Cl3N3
    Purezza:99.16% - 99.86%
    Colore e forma:Solid
    Peso molecolare:266.55

    Ref: TM-T1247

  • Methyldopa
    Targetmol
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    Methyldopa

    CAS:
    <p>Methyldopa (MK-351), an alpha-adrenergic agonist (selective for α2-adrenergic receptors) psychoactive medicine, is served as an antihypertensive or</p>
    Formula:C10H13NO4
    Purezza:98.95% - 99.86%
    Colore e forma:Less Or Almost Colorless Crystals Or White To Yellowish-White Fine
    Peso molecolare:211.21

    Ref: TM-T0505

  • CYM 50769
    Targetmol
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    CYM 50769

    CAS:
    <p>CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).</p>
    Formula:C24H17ClN2O3
    Purezza:98% - 99.08%
    Colore e forma:Solid
    Peso molecolare:416.86

    Ref: TM-T22702

  • Fluparoxan hydrochloride
    Targetmol
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    Fluparoxan hydrochloride

    CAS:
    <p>Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental</p>
    Formula:C10H11ClFNO2
    Purezza:99.98%
    Colore e forma:Soild
    Peso molecolare:231.65

    Ref: TM-T77565

  • Fluvoxamine maleate
    Targetmol
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    Fluvoxamine maleate

    CAS:
    <p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>
    Formula:C19H25F3N2O6
    Purezza:99.92% - 99.94%
    Colore e forma:White Crystalline Powder
    Peso molecolare:434.41

    Ref: TM-T1077

  • Levosulpiride
    Targetmol
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    Levosulpiride

    CAS:
    <p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>
    Formula:C15H23N3O4S
    Purezza:98.20% - 99.88%
    Colore e forma:White Crystalline Powder
    Peso molecolare:341.43

    Ref: TM-T1211

  • PF429242 dihydrochloride
    Targetmol
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    PF429242 dihydrochloride

    CAS:
    <p>PF429242 dihydrochloride can reversibly inhibit S1P (IC50 of 175 nM).</p>
    Formula:C25H37Cl2N3O2
    Purezza:99.68%
    Colore e forma:Solid
    Peso molecolare:482.49

    Ref: TM-T12437

  • Roxatidine Acetate hydrochloride
    Targetmol
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    Roxatidine Acetate hydrochloride

    CAS:
    <p>Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.</p>
    Formula:C19H29ClN2O4
    Purezza:99.49%
    Colore e forma:Solid
    Peso molecolare:384.9

    Ref: TM-T0157

  • NF-56-EJ40 hydrochloride
    Targetmol
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    NF-56-EJ40 hydrochloride

    CAS:
    <p>NF-56-EJ40 HCl is a selective human SUCNR1 antagonist, IC50 = 25 nM, Ki = 33 nM; low rat SUCNR1 activity, Ki = 17.4 nM.</p>
    Formula:C27H31Cl2N3O3
    Purezza:99.33%
    Colore e forma:Soild
    Peso molecolare:516.46

    Ref: TM-T12216L

  • Diphenylpyraline hydrochloride
    Targetmol
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    Diphenylpyraline hydrochloride

    CAS:
    <p>Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.</p>
    Formula:C19H23NO·HCl
    Purezza:98.72%
    Colore e forma:Solid
    Peso molecolare:317.85

    Ref: TM-T0059

  • Salmeterol
    Targetmol
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    Salmeterol

    CAS:
    <p>Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.</p>
    Formula:C25H37NO4
    Purezza:99.2% - 99.9%
    Colore e forma:Solid
    Peso molecolare:415.57

    Ref: TM-T12829

  • Aripiprazole
    Targetmol
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    Aripiprazole

    CAS:
    <p>Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.</p>
    Formula:C23H27Cl2N3O2
    Purezza:99.43% - 99.62%
    Colore e forma:Colourless Flake Crystalline Solid
    Peso molecolare:448.39

    Ref: TM-T1566

  • Naluzotan hydrochloride
    Targetmol
    + Info

    Naluzotan hydrochloride

    CAS:
    <p>Naluzotan hydrochloride, a hERG K+ blocker (IC50: 3800 nM) and potent 5-HT1A agonist (IC50: ~20 nM, Ki: ~5.1 nM), is used in anxiety and depression studies.</p>
    Formula:C23H39ClN4O3S
    Purezza:99.96%
    Colore e forma:Solid
    Peso molecolare:487.1

    Ref: TM-T68113