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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

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Trovati 5352 prodotti di "Proteina G/GPCR"

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  • LY83583
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    LY83583

    CAS:
    <p>LY83583 is a soluble guanylate cyclase competitive inhibitor with IC50 of 2 µM.</p>
    Formula:C15H10N2O2
    Purezza:99.54% - 99.80%
    Colore e forma:Solid
    Peso molecolare:250.25

    Ref: TM-T21576

  • Logo CymitQuimica
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    Anti-TSHR Antibody (M22)

    <p>Anti-TSHR Antibody (M22) is a humanized IgG1 monoclonal antibody targeting the thyroid-stimulating hormone receptor (TSHR). This antibody is capable of inhibiting the interaction between TSH and TSHR.</p>
    Colore e forma:Odour Liquid

    Ref: TM-T9901A-942

  • Fabesetron
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    Fabesetron

    CAS:
    <p>Fabesetron (FK1052): oral dual antagonist for 5-HT3/5-HT4 receptors. Aids in managing acute and delayed chemo-induced emesis.</p>
    Formula:C18H19N3O
    Colore e forma:Solid
    Peso molecolare:293.37

    Ref: TM-T38692

  • Logo CymitQuimica
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    α-CGRP(human) TFA

    <p>α-CGRP(human) TFA is a 37-amino acid regulatory neuropeptide that is extensively located within the central and peripheral nervous system, functioning as a</p>
    Formula:C165H268F3N51O51S2
    Colore e forma:Solid
    Peso molecolare:3903.33

    Ref: TM-T75788

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    NI-203

    <p>NI-203 is a monoclonal antibody inhibitor that targets amylin and shows potential for research in type 2 diabetes.</p>
    Colore e forma:Odour Liquid

    Ref: TM-T9901A-993

  • Pellotine
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    Pellotine

    CAS:
    <p>Pellotine is an alkaloid isolated from Lophophora. It acts as an inverse agonist of the 5-HT7 receptor (5-HT7 receptor), with an EC50 of 291 nM. Pellotine shows strong affinity for the 5-HT1DR and 5-HT6R, with Ki values of 117 nM and 170 nM, respectively. Additionally, Pellotine reduces intracellular cAMP levels, thereby decreasing neuronal excitability and neurotransmitter release.</p>
    Formula:C13H19NO3
    Colore e forma:Solid
    Peso molecolare:237.295

    Ref: TM-TN9164

  • 5-MeO-pyr-T
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    5-MeO-pyr-T

    CAS:
    <p>5-MeO-pyr-T (5-Methoxy pyrrolidinyltryptamine) acts as a 5-HT1AR agonist, exhibiting Ki values of 0.577 μM and 373 μM for 5-HT1AR and 5-HT2AR, respectively. It inhibits the reuptake of 5-HT and triggers its release. Additionally, 5-MeO-pyr-T can induce reduced motor activity.</p>
    Formula:C15H20N2O
    Colore e forma:Solid
    Peso molecolare:244.33

    Ref: TM-T203568

  • Logo CymitQuimica
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    Bay 55-9837 TFA

    <p>Bay 55-9837 TFA is a VPAC2 agonist with a 0.65 nM Kd, potential for type 2 diabetes research.</p>
    Formula:C150H240F3ClN44O44
    Colore e forma:Solid
    Peso molecolare:3456.22

    Ref: TM-T75825

  • Cyclosomatostatin Acetate
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    Cyclosomatostatin Acetate

    <p>Cyclosomatostatin Acetate is an effective antagonist of the somatostatin receptor.Cyclosomatostatin Acetate inhibits SSTR1 signaling and decreases cell</p>
    Formula:C46H61N7O8
    Purezza:98.83%
    Colore e forma:Solid
    Peso molecolare:840.02

    Ref: TM-T21567L

  • Logo CymitQuimica
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    (3R,5R,6S)-Atogepant

    <p>(3R,5R,6S)-Atogepant (MK-8031) is a CGRP antagonist enantiomer used in migraine research.</p>
    Formula:C29H23F6N5O3
    Colore e forma:Solid
    Peso molecolare:603.52

    Ref: TM-T73703

  • Bradykinin (1-3)
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    Bradykinin (1-3)

    CAS:
    <p>Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.</p>
    Formula:C16H28N6O4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:368.43

    Ref: TM-TP1780

  • TRV045
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    TRV045

    CAS:
    <p>TRV045 is a selective agonist of the sphingosine-1-phosphate (S1P) subtype 1 receptor and does not impact lymphocyte trafficking. It possesses antiepileptic properties.</p>
    Formula:C18H18N4O3
    Colore e forma:Solid
    Peso molecolare:338.36

    Ref: TM-T203071

  • M40
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    M40

    CAS:
    <p>Potent, non-selective galanin receptor antagonist (Ki values are 1.82 and 5.1 nM at GAL1 and GAL2 respectively) that inhibits galanin (1-29) binding in rat</p>
    Formula:C94H145N23O24
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1981.33

    Ref: TM-TP1992

  • ABT 724 trihydrochloride
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    ABT 724 trihydrochloride

    CAS:
    <p>ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.</p>
    Formula:C17H22Cl3N5
    Purezza:99.91%
    Colore e forma:Solid
    Peso molecolare:402.75

    Ref: TM-T22019

  • GR231118
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    GR231118

    CAS:
    <p>Potent NPY Y1 antagonist &amp; Y4 agonist; inhibits rat appetite; binds to NPFF receptors (Ki: 43-73 nM).</p>
    Formula:C110H170N34O24
    Purezza:98%
    Colore e forma:Lyophilized Powder
    Peso molecolare:2352.77

    Ref: TM-TP2022

  • (Rac)-Norcisapride
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    (Rac)-Norcisapride

    CAS:
    <p>Norcisapride, a 5-HT3 and 5-HT4 agonist, treats GI, orofacial, and ENT disorders.</p>
    Formula:C14H20ClN3O3
    Purezza:99.32%
    Colore e forma:Soild
    Peso molecolare:313.78

    Ref: TM-T68116L

  • Parstatin(human)
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    Parstatin(human)

    CAS:
    Cell-permeable PAR1-derived peptide; inhibits endothelial migration, proliferation (IC50 ~3μM), induces apoptosis, and has cardioprotective effects.
    Formula:C191H330N64O53S3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:4467.29

    Ref: TM-TP1965

  • Logo CymitQuimica
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    20-SOLA

    <p>20-SOLA is the first water-soluble 20-HETE antagonist with oral bioavailability. It significantly improves blood pressure changes and kidney damage associated with the streptozotocin (STZ) diabetic mouse model. Additionally, 20-SOLA acts as a GPR75 receptor blocker. This compound is useful in research related to cardiovascular pathology.</p>
    Formula:C33H62O9
    Peso molecolare:602.43938

    Ref: TM-T208783

  • Bombinakinin M acetate
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    Bombinakinin M acetate

    <p>Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial smooth muscle bradykinin receptors and is</p>
    Formula:C102H163N31O26
    Purezza:99.80%
    Colore e forma:Solid
    Peso molecolare:2239.58

    Ref: TM-TP2075L

  • (2R,2R)-PF-07258669
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    (2R,2R)-PF-07258669

    CAS:
    <p>(2R,2R)-PF-07258669' is an antagonist for the MC4R (melanocortin 4 receptor), primarily studied for its role in regulating appetite and energy expenditure.</p>
    Formula:C25H27FN6O2
    Colore e forma:Solid
    Peso molecolare:462.52

    Ref: TM-T88749