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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

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Trovati 5352 prodotti di "Proteina G/GPCR"

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  • Logo CymitQuimica
    Targetmol
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    Urocortin II, human TFA

    <p>hUcn II, a CRF family member, targets CRF2 receptor, has time-linked stress regulation effects, showing mild motor suppression and delayed anxiolytic action.</p>
    Formula:C196H340F3N63O56S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:4564.3

    Ref: TM-TP1557

  • Triazolomethylindole-3-acetic acid
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    Triazolomethylindole-3-acetic acid

    CAS:
    <p>Triazolomethylindole-3-acetic acid is a metabolite of Rizatriptan, which acts as an agonist for the serotonin (5-HT) receptor subtypes 5-HT1B and 5-HT1D.</p>
    Formula:C13H12N4O2
    Colore e forma:Solid
    Peso molecolare:256.26

    Ref: TM-T203624

  • FSLLRY-NH2
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    FSLLRY-NH2

    CAS:
    <p>PAR2 antagonist; counters taxol effects, PKC in mice; inhibits ERK, collagen in fibroblasts; lessens dermatophyte itch in mice.</p>
    Formula:C39H60N10O8
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:796.97

    Ref: TM-TP1904

  • β-MSH, human
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    β-MSH, human

    CAS:
    <p>beta-MSH, human is an endogenous peptide hormone and neurotransmitter by POMC, an agonist of MC4-R (melanocortin 4 receptor).</p>
    Formula:C118H174N34O35S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:2660.92

    Ref: TM-TP1004

  • TAK-615
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    TAK-615

    CAS:
    <p>TAK-615 is commonly used to study pulmonary fibrosis and is a negative allosteric modulator of LPA1 receptors.</p>
    Formula:C25H22FNO4
    Purezza:99.73%
    Colore e forma:Solid
    Peso molecolare:419.44

    Ref: TM-T9699

  • PG 931 acetate
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    PG 931 acetate

    <p>PG 931 acetate is a potent agonist of melanocortin 4 (MC4) receptors.</p>
    Formula:C61H89N15O13
    Purezza:98.74%
    Colore e forma:Solid
    Peso molecolare:1240.45

    Ref: TM-TP1953L

  • ABT-702
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    ABT-702

    CAS:
    <p>ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.</p>
    Formula:C22H19BrN6O
    Purezza:99.57%
    Colore e forma:Soild
    Peso molecolare:463.33

    Ref: TM-T4668L

  • Tecastemizole
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    Tecastemizole

    CAS:
    <p>Tecastemizole (R 43512) is a selective antagonist of H1 receptor and a major metabolite of astemizole with anti-inflammatory effects.</p>
    Formula:C19H21FN4
    Purezza:99.70%
    Colore e forma:Solid
    Peso molecolare:324.4

    Ref: TM-T26253

  • Logo CymitQuimica
    Targetmol
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    ALD1613

    <p>ALD1613 is a potent neutralizing monoclonal antibody targeting adrenocorticotropic hormone (ACTH). It neutralizes ACTH-induced signaling and inhibits cyclic adenosine monophosphate accumulation in ACTH-stimulated Y1 (mouse adrenal cell line) via all five melanocortin receptors. ALD1613 significantly reduces plasma corticosterone levels in wild-type rats and is applicable in studies involving elevated ACTH-related conditions.</p>
    Colore e forma:Odour Liquid

    Ref: TM-T9901A-967

  • Kassinin
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    Kassinin

    CAS:
    <p>Kassinin is a peptide derived from the Kassina frog. It belongs to tachykinin family of neuropeptides.</p>
    Formula:C59H95N15O18S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1334.54

    Ref: TM-TP1738

  • GLP-1R agonist 19
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    GLP-1R agonist 19

    CAS:
    <p>GLP-1R agonist 19 (M3190) is a potent, selective GLP-1 receptor agonist that demonstrates excellent plasma and liver microsomal stability, along with low hERG toxicity [1].</p>
    Formula:C94H136FN21O25
    Colore e forma:Solid
    Peso molecolare:1979.21

    Ref: TM-T86507

  • Bay 55-9837
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    Bay 55-9837

    CAS:
    <p>Selective VPAC2 agonist; EC50: 0.4 nM (VPAC2), 100 nM (VPAC1), &gt;1000 nM (PAC1). Enhances insulin secretion, reduces HIV-1 replication.</p>
    Formula:C167H270N52O46
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3742.29

    Ref: TM-TP2071

  • Hydroxybupropion
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    Hydroxybupropion

    CAS:
    <p>Hydroxybupropion is the major active metabolite of Bupropion and an antagonist of nACh receptor. Hydroxybupropion inhibits norepinephrine uptake (IC50 = 1.7 μM).</p>
    Formula:C13H18ClNO2
    Purezza:99.73%
    Colore e forma:Off-White Solid
    Peso molecolare:255.74

    Ref: TM-T11588

  • LE 300
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    LE 300

    CAS:
    <p>LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.</p>
    Formula:C20H22N2
    Purezza:97.91% - 98.79%
    Colore e forma:Solid
    Peso molecolare:290.4

    Ref: TM-T22921

  • Sulamserod
    Targetmol
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    Sulamserod

    CAS:
    <p>Sulamserod (RS 100302) is a potent 5-HT4 receptor antagonist with antiarrhythmic activity for the study of atrial fibrillation and cardiovascular related</p>
    Formula:C19H28ClN3O5S
    Purezza:98.76%
    Colore e forma:Solid
    Peso molecolare:445.96

    Ref: TM-T13021

  • Dipivefrin
    Targetmol
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    Dipivefrin

    CAS:
    <p>Dipivefrin is a prodrug of epinephrine, and is used to treat open-angle glaucoma.</p>
    Formula:C19H29NO5
    Colore e forma:Solid
    Peso molecolare:351.44

    Ref: TM-T0103L

  • Fabesetron
    Targetmol
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    Fabesetron

    CAS:
    <p>Fabesetron (FK1052): oral dual antagonist for 5-HT3/5-HT4 receptors. Aids in managing acute and delayed chemo-induced emesis.</p>
    Formula:C18H19N3O
    Colore e forma:Solid
    Peso molecolare:293.37

    Ref: TM-T38692

  • Logo CymitQuimica
    Targetmol
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    (D-Ala2)-GRF (1-29) amide (human)

    CAS:
    (D-Ala2)-GRF (1-29) amide (human) is a potent superagonist of Growth Hormone-Releasing Factor (GRF), demonstrating an exceptionally high Growth Hormone (GH)-
    Formula:C149H246N44O42S
    Peso molecolare:3357.88

    Ref: TM-T83549

  • Sch 202596
    Targetmol
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    Sch 202596

    CAS:
    <p>Sch 202596 is a selective non-peptide antagonist of GAL-1 receptor.</p>
    Formula:C25H22Cl2O12
    Colore e forma:Solid
    Peso molecolare:585.34

    Ref: TM-T28705

  • Lys-[Des-Arg9]Bradykinin
    Targetmol
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    Lys-[Des-Arg9]Bradykinin

    CAS:
    Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.
    Formula:C50H73N13O11
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1032.21

    Ref: TM-TP1918