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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

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Trovati 5378 prodotti di "Proteina G/GPCR"

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  • Glucagon receptor antagonists-1
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    Glucagon receptor antagonists-1

    CAS:
    <p>Glucagon receptor antagonist -1 is a highly effective glucagon receptor antagonist.</p>
    Formula:C29H34FNO2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:447.58

    Ref: TM-T11413

  • TRV045
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    TRV045

    CAS:
    <p>TRV045 is a selective agonist of the sphingosine-1-phosphate (S1P) subtype 1 receptor and does not impact lymphocyte trafficking. It possesses antiepileptic properties.</p>
    Formula:C18H18N4O3
    Colore e forma:Solid
    Peso molecolare:338.36

    Ref: TM-T203071

  • ABT 724 trihydrochloride
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    ABT 724 trihydrochloride

    CAS:
    <p>ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.</p>
    Formula:C17H22Cl3N5
    Purezza:99.91%
    Colore e forma:Solid
    Peso molecolare:402.75

    Ref: TM-T22019

  • GR231118
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    GR231118

    CAS:
    <p>Potent NPY Y1 antagonist &amp; Y4 agonist; inhibits rat appetite; binds to NPFF receptors (Ki: 43-73 nM).</p>
    Formula:C110H170N34O24
    Purezza:98%
    Colore e forma:Lyophilized Powder
    Peso molecolare:2352.77

    Ref: TM-TP2022

  • Logo CymitQuimica
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    CAP-100

    <p>CAP-100 is a monoclonal antibody targeting CCR7. It neutralizes the ligand binding site and signaling of CCR7. This compound effectively inhibits migration, extravasation, homing, and survival in chronic lymphocytic leukemia (CLL) samples induced by CCR7. CAP-100 can mediate potent tumor cell killing through host immune mechanisms and exhibits favorable toxicity profiles in related hematopoietic cell subsets. It is involved in research on antitumor activity and diseases like chronic lymphocytic leukemia (CLL).</p>
    Colore e forma:Odour Liquid

    Ref: TM-T9901A-961

  • Zalospirone
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    Zalospirone

    CAS:
    <p>Zalospirone is a 5-HT1A receptor agonist that can be used to study anxiety disorders and major depressive disorder.</p>
    Formula:C24H29N5O2
    Purezza:98.41% - 99.82%
    Colore e forma:Solid
    Peso molecolare:419.52

    Ref: TM-T68172

  • (Rac)-Norcisapride
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    (Rac)-Norcisapride

    CAS:
    <p>Norcisapride, a 5-HT3 and 5-HT4 agonist, treats GI, orofacial, and ENT disorders.</p>
    Formula:C14H20ClN3O3
    Purezza:99.32%
    Colore e forma:Soild
    Peso molecolare:313.78

    Ref: TM-T68116L

  • Logo CymitQuimica
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    Endolide F

    Endolide F (Compound 2) is a proline-containing lactone that serves as a moderate antagonist of the arginine vasopressin V1A receptor.
    Formula:C25H32N4O6
    Peso molecolare:484.23218

    Ref: TM-TN11172

  • Cetirizine D8 dihydrochloride
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    Cetirizine D8 dihydrochloride

    CAS:
    <p>Cetirizine D8 dihydrochloride is a deuterated H1-antihistamine with long-acting effects.</p>
    Formula:C21H26Cl2N2O3
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:433.4

    Ref: TM-T19234

  • Logo CymitQuimica
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    Myristoylated ARF6 (2-13)

    <p>Myristoylated ARF6 (2-13) inhibits the MyD88–ARNO–ARF6 signaling axis by inactivating ARF6.</p>
    Formula:C74H128N16O18
    Peso molecolare:1528.95925

    Ref: TM-TP3490

  • NTRC-824
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    NTRC-824

    CAS:
    <p>NTRC-824: NTS2 antagonist, 150x more selective than NTS1; IC50: 38 nM, Ki: 202 nM; nonpeptide, neurotensin-like.</p>
    Formula:C25H26F3N3O6S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:553.55

    Ref: TM-T16358

  • (Iso)-RJW100
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    (Iso)-RJW100

    CAS:
    <p>Potent LRH-1/NR5A2 and SF-1/NR5A1 agonist; pEC50: 6.4 (LRH-1), 7.2 (SF-1).</p>
    Formula:C28H34O
    Purezza:99.79%
    Colore e forma:Soild
    Peso molecolare:386.57

    Ref: TM-T64363

  • IRL-1038 acetate
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    IRL-1038 acetate

    <p>IRL-1038 acetate is a potent ETB endothelin receptor antagonist.</p>
    Formula:C70H96N14O17S2
    Purezza:97.51%
    Colore e forma:Soild
    Peso molecolare:1469.73

    Ref: TM-TP2262L

  • Ki16198
    Targetmol
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    Ki16198

    CAS:
    <p>Ki16198, a methyl ester derivative of Ki16425, blocks LPA1/3, weak on LPA2; inactive on LPA4/5/6. Ki values: 0.34 μM (LPA1), 0.93 μM (LPA3).</p>
    Formula:C24H25ClN2O5S
    Purezza:98.09%
    Colore e forma:Solid
    Peso molecolare:488.98

    Ref: TM-T6347

  • I-BOP
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    I-BOP

    CAS:
    <p>I-BOP is an agonist (KD=0.61 nM) at the thromboxane A2 receptor (TP).</p>
    Formula:C23H29IO5
    Colore e forma:Solid
    Peso molecolare:512.384

    Ref: TM-T35585

  • Enuvaptan
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    Enuvaptan

    CAS:
    <p>Enuvaptan is a vasopressin receptor antagonist and has the potential for research into renal and cardiovascular diseases.</p>
    Formula:C21H15ClF6N8O3
    Colore e forma:Solid
    Peso molecolare:576.84

    Ref: TM-T39611

  • Mirtazapine N-oxide
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    Mirtazapine N-oxide

    CAS:
    <p>Mirtazapine N-oxide, a mirtazapine metabolite, is produced by CYP1A2 and CYP3A4 in human liver.</p>
    Formula:C17H19N3O
    Colore e forma:Solid
    Peso molecolare:281.359

    Ref: TM-T37430

  • Guanylate cyclase-IN-1
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    Guanylate cyclase-IN-1

    CAS:
    <p>Guanylate cyclase-IN-1 (Example 46) is a specific inhibitor of guanylate cyclase, employed in research related to cardiovascular diseases.</p>
    Formula:C20H17FN8O
    Colore e forma:Solid
    Peso molecolare:404.409

    Ref: TM-T38770

  • [bAla8]-Neurokinin A(4-10)
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    [bAla8]-Neurokinin A(4-10)

    CAS:
    [bAla8]-Neurokinin A(4-10) is a neurokinin 2 (NK2) receptor agonist.
    Formula:C35H56N8O10S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:780.94

    Ref: TM-TP1100

  • Xanthine amine congener trihydrochloride
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    Xanthine amine congener trihydrochloride

    CAS:
    <p>Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.</p>
    Formula:C21H29ClN6O4
    Purezza:98.81%
    Colore e forma:Solid
    Peso molecolare:464.95

    Ref: TM-T23535L