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Proteina G/GPCR

Proteina G/GPCR

Gli inibitori dei GPCR/proteine G sono composti che bersagliano i recettori accoppiati alle proteine G (GPCR) e le proteine G associate, che svolgono ruoli critici nella trasmissione dei segnali dall'esterno all'interno delle cellule. Questi inibitori sono essenziali per studiare le vie di segnalazione mediate dai GPCR, coinvolte in numerosi processi fisiologici, tra cui la percezione sensoriale, la risposta immunitaria e la neurotrasmissione. Gli inibitori dei GPCR sono anche importanti nello sviluppo di farmaci, poiché molti agenti terapeutici prendono di mira questi recettori. Presso CymitQuimica, offriamo una vasta gamma di inibitori dei GPCR/proteine G di alta qualità per supportare le tue ricerche in farmacologia, biologia cellulare e campi correlati.

Sottocategorie di "Proteina G/GPCR"

Mostrare 18 più sottocategorie

Trovati 5378 prodotti di "Proteina G/GPCR"

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  • [Sar4] Substance P (4-11)


    <p>'[Sar4] Substance P (4-11) is a C-terminus fragment and agonist of Substance P.'</p>
    Formula:C44H65N11O10S
    Colore e forma:Solid
    Peso molecolare:940.12
  • Zalospirone

    CAS:
    <p>Zalospirone is a 5-HT1A receptor agonist that can be used to study anxiety disorders and major depressive disorder.</p>
    Formula:C24H29N5O2
    Purezza:98.41% - 99.82%
    Colore e forma:Solid
    Peso molecolare:419.52
  • SR 142948 dihydrochloride


    <p>SR 142948 dihydrochloride is a selective oral non-peptide NT antagonist, IC50 &lt;4 nM, with brain penetration and potential for psychiatric research.</p>
    Formula:C39H53Cl2N5O6
    Colore e forma:Solid
    Peso molecolare:758.77
  • Atrial natriuretic factor (1-28) (rat) TFA


    <p>ANP (1-28), rat (TFA) inhibits Ang II-induced endothelin-1 secretion; main circulating ANP form in rats.</p>
    Formula:C130H206N45F3O41S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3176.43
  • α-MSH acetate


    <p>α-MSH acetate is an endogenous neuromodulatory peptide derived from POMC and an agonist of MC4R (melanocortin receptor 4).</p>
    Purezza:99.71%
    Colore e forma:Odour Solid
  • GLP-1R agonist 29


    <p>GLP-1R agonist 29 (Compound 20) is a GLP-1R agonist that induces hGLP-1R-mediated cAMP stimulation with an EC50 of 0.018 nM. It exhibits favorable pharmacokinetic properties and shows good in vivo exposure, with an AUC0-∞,sc of 77688 ng·h/mL.</p>
    Colore e forma:Odour Solid
  • (D-Phe7)-α-MSH

    CAS:
    <p>(D-Phe7)-α-MSH is an α-MSH analogue [1] .</p>
    Formula:C77H109N21O19S
    Colore e forma:Solid
    Peso molecolare:1664.88
  • PACAP-Related Peptide (PRP), human


    <p>PRP, human: 29-amino-acid PACAP precursor segment, synthesized for biological/structural research.</p>
    Formula:C139H229N41O42
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3146.57
  • Cortistatin-8 acetate


    <p>Cortistatin-8 acetate: synthetic corticosteroid analog, GHS-R antagonist; doesn't affect acyl GH release or hesperidin response.</p>
    Formula:C49H72N12O11S2
    Purezza:99.01%
    Colore e forma:Soild
    Peso molecolare:1069.3
  • TAK-615

    CAS:
    <p>TAK-615 is commonly used to study pulmonary fibrosis and is a negative allosteric modulator of LPA1 receptors.</p>
    Formula:C25H22FNO4
    Purezza:99.73%
    Colore e forma:Solid
    Peso molecolare:419.44
  • ABT-702

    CAS:
    <p>ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.</p>
    Formula:C22H19BrN6O
    Purezza:99.57%
    Colore e forma:Soild
    Peso molecolare:463.33
  • AMTG-DA1


    <p>AMTG-DA1 is a ligand for the gastrin-releasing peptide receptor (GRPR), and it can be utilized in cancer research.</p>
    Formula:C101H149IN22O25
    Colore e forma:Solid
    Peso molecolare:2197.0109
  • GR 64349

    CAS:
    <p>Potent NK2 agonist, EC50=3.7 nM in rat colon; &gt;1000x selectivity over NK1, &gt;300x over NK3; effective in vivo.</p>
    Formula:C42H68N10O11S
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:921.12
  • RVD-Hpα

    CAS:
    <p>N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.</p>
    Formula:C65H105N19O17
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:1424.66
  • GW-328267

    CAS:
    <p>GW-328267 is an agonist of the adenosine A2 receptor.</p>
    Formula:C21H26N10O4
    Colore e forma:Solid
    Peso molecolare:482.5
  • Nolomirole

    CAS:
    <p>Nolomirole is a dopamine receptor agonist that reduces symptoms of congestive heart failure caused by monoclinine.</p>
    Formula:C19H27NO4
    Colore e forma:Solid
    Peso molecolare:333.42
  • Fsh receptor-binding inhibitor fragment(bi-10)

    CAS:
    <p>FSH antagonist bi-10 suppresses ovulation, induces follicular atresia, and may help in ovarian cancer by downregulating FSHR/ERβ.</p>
    Formula:C42H67N13O19
    Colore e forma:Solid
    Peso molecolare:1058.06
  • Peptide 401

    CAS:
    Peptide 401: AMP from bee/wasp venom, triggers histamine release, reduces paw swelling.
    Formula:C110H192N40O24S4
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:2587.22
  • α-Helical CRF(9-41)

    CAS:
    <p>Corticotropin-releasing factor receptor antagonist (Ki values are 17, 5 and 0.97 at human CRF1, rat CRF2α and mouse CRF2β receptors respectively).</p>
    Formula:C166H274N46O53S2
    Purezza:98%
    Colore e forma:Solid
    Peso molecolare:3827
  • SGLT1/2-IN-2

    CAS:
    <p>SGLT1/2-IN-2 is a chemical compound with robust dual inhibitory properties, exhibiting potent activities against SGLT1 (IC50 = 96 nM) and SGLT2 (IC50 = 1.3 nM).</p>
    Formula:C23H26F2O7
    Colore e forma:Solid
    Peso molecolare:452.451